Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65941 productos de "Derivados de Quinazolina y Quinolina"
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Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Fórmula:C14H16N2·HClPureza:99.74%Forma y color:SolidPeso molecular:248.75Anagrelide
CAS:Anagrelide (Xagrid) is a Platelet-reducing Agent.Fórmula:C10H7Cl2N3OPureza:99.53% - >99.99%Forma y color:SolidPeso molecular:256.09Maprotiline
CAS:Maprotiline blocks norepinephrine uptake, has antidepressant properties, and fights cancer by inducing apoptosis and inhibiting ERK and CRABP1.Fórmula:C20H23NForma y color:SolidPeso molecular:277.4Tacrine hydrochloride (hydrate)
CAS:Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.Fórmula:C13H14N2·XHCl·XH2OPureza:99.01% - 99.89%Forma y color:SolidPeso molecular:234.72Tacrine
CAS:Tacrine (CS 12602) is an indirect cholinergic agonist and centrally acting anticholinesterase. It is approved for the treatment of Alzheimer's disease.Fórmula:C13H14N2Pureza:99.97%Forma y color:SolidPeso molecular:198.26Clomifene (Clomiphene) EP Impurity A HCl (Clomiphene USP Related Compound A)
CAS:Fórmula:C26H29NO·HClPeso molecular:371.52 36.46Regorafenib
CAS:Regorafenib (BAY 73-4506) is a multi-targeted receptor tyrosine kinase inhibitor that inhibits RET, C-RAF, VEGFR2, c-Kit, VEGFR1, and PDGFRβ and is orallyFórmula:C21H15ClF4N4O3Pureza:98% - 99.95%Forma y color:SolidPeso molecular:482.82Nirmatrelvir
CAS:<p>PF-07321332 is a potent and orally active inhibitor of SARS-CoV 3C-like protease (3CLPRO) .</p>Fórmula:C23H32F3N5O4Pureza:98.66% - 99.93%Forma y color:SolidPeso molecular:499.53Efavirenz
CAS:Efavirenz (DMP 266) is an HIV-1 inhibitor, affecting reverse transcriptase and various cytochrome P450 enzymes.Fórmula:C14H9ClF3NO2Pureza:99.2% - 99.84%Forma y color:White To Slightly Pink Crystalline PowderPeso molecular:315.67JNJ0966
CAS:<p>JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).</p>Fórmula:C16H16N4O2S2Pureza:99.46% - 99.62%Forma y color:SolidPeso molecular:360.45Tosedostat
CAS:Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.Fórmula:C21H30N2O6Pureza:98.14% - 99.4%Forma y color:SolidPeso molecular:406.474-Bromo Riluzole
CAS:Producto controlado<p>Applications 4-Bromo Riluzole is an impurity of Riluzole (R510000); a benzothiazole derivative that is used to treat amyotrophic lateral sclerosis.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Ahamed, A., et al.: J. Pharm. Res., 3, 1028 (2010); Satyanarayana, B., et al.: ARKIVOC, no vol., 109 (2008)<br></p>Fórmula:C8H4BrF3N2OSForma y color:NeatPeso molecular:313.09Tadalafil Ketolactam (>90%)
CAS:Producto controlado<p>Stability Hygroscopic, Unstable in Solution<br>Applications Tadalafil Ketolactam is a Tadalafil (T004500) impurity.<br></p>Fórmula:C22H19N3O6Pureza:>90%Forma y color:NeatPeso molecular:421.40284,6-dimethyl-N-(pyridin-2-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Pureza:95.0%Peso molecular:269.3699951171875Dibenzazepine-10,11-dione
CAS:Producto controlado<p>Applications Dibenzazepine-10,11-dione is an impurity of Oxcarbazepine (O869250). Dibenzazepine-10,11-dione is used as a reagent in the preparation of bifunctional dipolar electroluminescent template for optoelectronic applications.<br>References Chen, C.-T. et al.: Chem. Comm., 31, 3980 (2005); Heckendorn, R. et al.: Helv, Chim. Acta, 70, 1955 (1987);<br></p>Fórmula:C14H9NO2Forma y color:NeatPeso molecular:223.23Levosimendan Triazene Impurity
CAS:<p>Stability Light Sensitive<br>Applications Levosimendan Triazene is an impurity of Levosimendan (L378000); a positive inotropic agent with vasodilating activity. Also cardiotonic.<br>References Sandell, E.-P., et al.: J. Cardiovasc. Pharmacol., 26, S57 (1995); Pagel, P.S., et al.: Cardiovasc. Drug Rev., 14, 286 (1996)<br></p>Fórmula:C22H23N7O2Forma y color:NeatPeso molecular:417.46N,O-Bis(trimethylsilyl)trifluoroacetamide (~90%)
CAS:Producto controlado<p>Applications Used as a reactant in the preparation of pyrimidinone ribosides and analogs that show anti-tumor properties.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Driscoll, J.S. et al.: J. Med. Chem., 34, 3280 (1991); Pan, L. et al.: J. Pharm. Biomed. Anal., 52, 589 (2010);<br></p>Fórmula:C8H18F3NOSi2Pureza:~90%Forma y color:Colourless To Light YellowPeso molecular:257.403-(4-((1H-IMIDAZOL-1-YL)METHYL)PHENYL)-N-(TERT-BUTYL)THIOPHENE-2-SULFONAMIDE
CAS:Pureza:95.0%Peso molecular:375.510009765625[2-(2-Methyl-1H-indol-3-yl)ethyl](pyridin-3-ylmethyl)amine dihydrochloride
CAS:Pureza:95.0%Peso molecular:338.2799987792969Bisnortilidine
CAS:Producto controlado<p>Applications A metabolite of Tilidine (T440300(M)), which is a controlled substance (opiate) and a analgesic. Tilidine is used in clinical trial in comparison with Nefopam. Tilidine is one of the most widely used narcotics in Germany and Belgium.<br>References Hengy, H., et al.: J. Pharm. Sci., 67, 1765 (1978); Cordonnier, J., et al.: J. Anal. Toxicol., 11, 144 (1987); Hajda, J., et al.: J. Clin. Pharmacol., 42, 1257 (2002); Vollmer, K.-O., et al.: Arzneim.-Forsch., 20, 990 (1970); Abeloos, J., et al.: Acta Anaesthesiol. Belg., 34, 283 (1983); Van Cauwenberge, H., et al.: Int. J. Clin. Pharmacol. Res., 12, 1 (1992)<br></p>Fórmula:C15H19NO2Forma y color:NeatPeso molecular:245.32(S)-(-)-Carvedilol
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications The optically active isomer of Carvedilol (C184625), a nonselective ß-adrenergic blocker with a1-blocking activity. An antihypertensive used in the treatment of congestive heart failure.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990),<br></p>Fórmula:C24H26N2O4Forma y color:Off White SolidPeso molecular:406.47(E)-2-((1-Acetyl-3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)-N-methylbenzamide (Axitinib Impurity)
CAS:Pureza:97%Forma y color:SolidPeso molecular:428.51N-Ethyl-N-methyl-3-vinylphenyl Carbamate
CAS:Producto controlado<p>Impurity Rivastigmine USP Related Compound F<br>Stability Light Sensitive<br>Applications A related compound of Rivastigmine (R541000), a cholinesterase inhibitor. Rivastigmine USP Related Compound F.<br></p>Fórmula:C12H15NO2Forma y color:White SolidPeso molecular:205.25
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