Derivados de Quinazolina y Quinolina
Las quinazolinas y quinolinas son compuestos heterocíclicos nitrogenados con estructuras aromáticas que desempeñan un papel clave en la síntesis de fármacos con actividad anticancerígena, antimicrobiana y antiinflamatoria. Sus derivados presentan modificaciones estructurales que optimizan su biodisponibilidad y selectividad, lo que permite el desarrollo de nuevos principios activos para diversas aplicaciones terapéuticas. Estos compuestos se utilizan en la fabricación de APIs destinados al tratamiento de cáncer, infecciones, enfermedades neurodegenerativas y cardiovasculares. Además, los derivados de quinazolina y quinolina son esenciales en la investigación de inhibidores enzimáticos y en el diseño de moléculas bioactivas innovadoras. En CymitQuimica disponemos de derivados de quinazolina y quinolina de alta pureza para aplicaciones en síntesis química, desarrollo farmacéutico y biotecnología.
Se han encontrado 65576 productos de "Derivados de Quinazolina y Quinolina"
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Levofloxacin N-oxide
CAS:Producto controlado<p>Impurity Oxifloxacin EP Impurity F<br>Applications Levofloxacin N-oxide is an impurity of Ofloxacin (O245750), which is a fluorinated quinolone antibacterial.<br>References Horstkotter, C., et al.: J. Chromatography Biomed. Sci. Appli., 754, 169 (2001); Monk, J.P., et al.: Drugs, 33, 346 (1987), Drlica, K., Curr. Opin. Microbiol. 2, 504 (1990)<br></p>Fórmula:C18H20FN3O5Forma y color:NeatPeso molecular:377.373,4-Dihydro-7-(4-hydroxybutoxy)-2(1H)-quinolinone
CAS:Fórmula:C13H17NO3Forma y color:NeatPeso molecular:235.283-[(4-Fluorobenzyl)oxy]-2-thiophenecarbohydrazide
CAS:Fórmula:C12H11FN2O2SForma y color:SolidPeso molecular:266.293-Methyl-6-nitro-quinoxaline-2-carboxylic acid benzyl ester
Pureza:95.0%Peso molecular:323.3080139160156Pentoxifylline
CAS:Producto controladoFórmula:C13H18N4O3Forma y color:White To Off-WhitePeso molecular:278.314-(furan-2-yl)-6-(3-methylthiophen-2-yl)pyrimidin-2-amine
CAS:Pureza:95.0%Peso molecular:257.30999755859375Amido Methyl Meloxicam (Meloxicam Impurity)
CAS:Producto controlado<p>Applications Amido Methyl Meloxicam is an impurity of Meloxicam (M216100).<br>References Lazer, E., et al.: J. Med. Chem., 40, 980 (1997),<br></p>Fórmula:C15H15N3O4S2Forma y color:NeatPeso molecular:365.43Cyanuric Acid (1 mg/10 mL in 84:16% ACN:H2O)
CAS:Producto controladoFórmula:C3H3N3O3Forma y color:Single SolutionPeso molecular:129.07Trityl Chloride
CAS:Producto controlado<p>Applications Trityl Chloride is an alkyl halide commonly used in organic synthesis to introduce the trityl protecting group. Trityl Chloride is used in the preparation of S-trityl-L-cysteine (STLC), a tight-binding inhibitor of Eg5 that prevents mitotic progression.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References DeBonis, S. et al.: J. Med. Chem., 51, 1115 (2008); Chadwick, D.J. et al.: J. Chem. Soc. Perk. Trans. Org. Bio-Org. Chem., 1, 102 (1983);<br></p>Fórmula:C19H15ClForma y color:NeatPeso molecular:278.78Saquinavir
CAS:Producto controlado<p>Applications Saquinavir (CAS# 127779-20-8) is a useful research chemical compound.<br></p>Fórmula:C38H50N6O5Forma y color:White To Off-WhitePeso molecular:670.84(S)-1-(2-Amino-5-chlorophenyl)-1-(trifluoromethyl)-3-cyclopropyl-2-propyn-1-ol
CAS:Producto controlado<p>Applications Intermediate in the preparation of Efavirenz (E425000) impurity.<br></p>Fórmula:C13H11ClF3NOForma y color:NeatPeso molecular:289.68(±)-Bifonazole
CAS:<p>Applications (±)-Bifonazole acts as an anti-fungal agent used in the treatment of skin diseases. Causes an increase in Ca2+ concentration and triggers cell death in PC3 human prostate cancer cells.<br>References Cheng, J. et al.: J. Recep. Sign. Transduct., 34, 493 (2014); Chen, Z. et al.: Mol. Pharm., 12, 590 (2015);<br></p>Fórmula:C22H18N2Forma y color:NeatPeso molecular:310.392-Ethyl-2-methyl-succinonitrile
CAS:Producto controlado<p>Applications An intermediate in the preparation of Ethosuximide.<br></p>Fórmula:C7H10N2Forma y color:NeatPeso molecular:122.171-(6,7-Dimethoxyphthalazin-1-yl)piperidin-4-yl ethylcarbamate
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:360.41400146484375(S)-Naproxen Ethyl Ester
CAS:<p>Impurity Naproxen EP Impurity F<br>Applications Naproxen (N377520) ethyl derivative. Naproxen impurity.<br>References Haddock, R., et al.: Xenobiotica, 14, 327 (1984), Jeremy, J., et al.: Drugs, 40, 53 (1990), Wadhwa, L., et al.: Int. J. Pharm., 118, 31 (1995),<br></p>Fórmula:C16H18O3Forma y color:NeatPeso molecular:258.31(S)-O-Desmethyl Naproxen
CAS:Producto controlado<p>Applications A metabolite of Naproxen.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Rettie, A., et al.: Chem. Res. Toxicol., 5, 54 (1992), Tracy, T., et al.: Biochem. Pharmacol., 52, 1305 (1996), Bonnabry, P., et al.: Eur. J. Clin. Pharmacol., 49, 305 (1996), Rao, S., et al.: J. Med. Chem., 43, 2789 (2000), Hutzler, J., et al.: Drug Metab. Dispos., 29, 1029 (2001),<br></p>Fórmula:C13H12O3Forma y color:WhitePeso molecular:216.23Des(methoxycarbonyl) Febantel
CAS:Producto controlado<p>Applications Febantel (F227000) impurity. Anthelmintic.<br>References Wollweber, H., et al.: Arzneim.-Forsch., 34, 531 (1984),<br></p>Fórmula:C18H20N4O4SForma y color:NeatPeso molecular:388.44Asenapine N-β-D-Glucuronide Trifluoroacetic Acid Salt (Mixture of Diastereomers)
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Asenapine N-β-D-Glucuronide is a metabolite of Asenapine (A788000).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Fórmula:C23H25ClNO7·C2F3O2Forma y color:NeatPeso molecular:575.926-Chloro-4-phenyl-1H-quinazolin-2-one
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:256.690002441406253-piperazin-1-yl-6-(2-thienyl)pyridazine
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:246.3300018310547(2S,3R)-Benzyl 6-oxo-2,3-diphenylmorpholine-4-carboxylate
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:387.4352-Deschloro Aripiprazole
CAS:<p>Impurity Aripiprazole EP Impurity D<br>Applications 2-Deschloro Aripiprazole (Aripiprazole EP Impurity D) is an impurity of the antipsychotic agent Aripiprazole (A771000). Aripiprazole impurity B.<br>References Akaike, A., et al.: Brain Res., 418, 262 (1987); Kikuchi, K., et al.: Life Sci., 42, 343 (1988); Caprathe, B., et al.: J. Med. Chem., 34, 2736 (1991); Yamada, S., et al.: J. Pharm. Pharmacol., 49, 206 (1997);<br></p>Fórmula:C23H28ClN3O2Forma y color:WhitePeso molecular:413.94(S)-4-Nitrophenyl 1-Phenyl-3,4-dihydroisoquinoline-2(1H)-carboxylate
CAS:Producto controlado<p>Applications (S)-4-Nitrophenyl 1-Phenyl-3,4-dihydroisoquinoline-2(1H)-carboxylate is a reactant in the synthesis of solifenacin succinate, an antimuscarinic agent.<br>References Niphade, N.C., et. al.: Monatshefte fuer Chemie, 142, 1181 (2011)<br></p>Fórmula:C22H18N2O4Forma y color:NeatPeso molecular:374.392-Chloro-N-(3-chloro-2-methylphenyl)nicotinamide
CAS:<p>Applications An impurity of Clonixine (L488530). Clonixine is a nonsteroidal anti-inflammatory agent used as an analgesic.<br>References Esteve, M.H., et al.: J. High Res. Chromatogr., 13, 445 (1990),<br></p>Fórmula:C13H10Cl2N2OForma y color:Off-WhitePeso molecular:281.144-Bromo Riluzole
CAS:Producto controlado<p>Applications 4-Bromo Riluzole is an impurity of Riluzole (R510000); a benzothiazole derivative that is used to treat amyotrophic lateral sclerosis.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Ahamed, A., et al.: J. Pharm. Res., 3, 1028 (2010); Satyanarayana, B., et al.: ARKIVOC, no vol., 109 (2008)<br></p>Fórmula:C8H4BrF3N2OSForma y color:NeatPeso molecular:313.09N,O-Bis(trimethylsilyl)trifluoroacetamide (~90%)
CAS:Producto controlado<p>Applications Used as a reactant in the preparation of pyrimidinone ribosides and analogs that show anti-tumor properties.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Driscoll, J.S. et al.: J. Med. Chem., 34, 3280 (1991); Pan, L. et al.: J. Pharm. Biomed. Anal., 52, 589 (2010);<br></p>Fórmula:C8H18F3NOSi2Pureza:~90%Forma y color:Colourless To Light YellowPeso molecular:257.40Bisnortilidine
CAS:Producto controlado<p>Applications A metabolite of Tilidine (T440300(M)), which is a controlled substance (opiate) and a analgesic. Tilidine is used in clinical trial in comparison with Nefopam. Tilidine is one of the most widely used narcotics in Germany and Belgium.<br>References Hengy, H., et al.: J. Pharm. Sci., 67, 1765 (1978); Cordonnier, J., et al.: J. Anal. Toxicol., 11, 144 (1987); Hajda, J., et al.: J. Clin. Pharmacol., 42, 1257 (2002); Vollmer, K.-O., et al.: Arzneim.-Forsch., 20, 990 (1970); Abeloos, J., et al.: Acta Anaesthesiol. Belg., 34, 283 (1983); Van Cauwenberge, H., et al.: Int. J. Clin. Pharmacol. Res., 12, 1 (1992)<br></p>Fórmula:C15H19NO2Forma y color:NeatPeso molecular:245.323-Acetyl-2(1H)-pyridinone
CAS:Fórmula:C7H7NO2Pureza:98%Forma y color:Solid, CrystallinePeso molecular:137.1383,5-Dinitrosalicylhydrazide-15N2
CAS:Producto controlado<p>Applications Labelled Nifursol (N458700) metabolite.<br>References Shen, Y. et al.: Faming Zhuanli Shenqing 13 (2009)<br></p>Fórmula:C7H6N215N2O6Forma y color:Light YellowPeso molecular:244.13rac Penbutolol
CAS:<p>Applications A β-adrenoceptor antagonist. Antihypertensive.<br>References Armstrong, D., et al.: Anal. Chem., 66, 1473 (1994), Kato, M., et al.: J. Pharm. Biomed. Anal., 30, 1845 (2003),<br></p>Fórmula:C18H29NO2Forma y color:Off-WhitePeso molecular:291.432-(3-pyridinyl)-5,6-dihydro-1,3-benzothiazol-7(4H)-one
CAS:Pureza:95.0%Peso molecular:230.2899932861328(R)-Bicalutamide
CAS:Producto controlado<p>Applications (R)-Enantiomer of Bicalutamide. Used as an antiandrogen, antineoplastic (hormonal).<br>References Tucker, H., et al.: J. Med. Chem., 31, 954 (1988), Cockshott, I.D., et al.: Eur. Urol., 18, Suppl. 3, 10 (1990), Cockshott, I., et al.: Br. J. Clin. Pharm., 36, 339 (1993), McKillop, D., et al.: Xenobiotica, 25, 623 (1995),<br></p>Fórmula:C18H14F4N2O4SForma y color:WhitePeso molecular:430.376-(Tetrahydro-2H-pyran-4-yloxy)pyridine-2-carboxylic acid
CAS:Pureza:97.0%Forma y color:SolidPeso molecular:223.227996826171884-Hydroxy Nisoldipine
CAS:Producto controlado<p>Applications A metabolite of Nisoldipine<br></p>Fórmula:C20H24N2O7Forma y color:NeatPeso molecular:404.41Tolcapone-d4
CAS:Producto controlado<p>Applications Orally active inhibitor of central and peripheral catechol-O-methyltransferase (COMT). Antiparkinsonian.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Dingemanse, J., et al.: Clin. Pharmacol. Ther., 57, 508 (1995), Keating, K.A., Drugs, 19, 165 (2005),<br></p>Fórmula:C14H7D4NO5Forma y color:NeatPeso molecular:277.27(S)-(-)-Carvedilol
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications The optically active isomer of Carvedilol (C184625), a nonselective ß-adrenergic blocker with a1-blocking activity. An antihypertensive used in the treatment of congestive heart failure.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990),<br></p>Fórmula:C24H26N2O4Forma y color:Off White SolidPeso molecular:406.471-Phenyl-3-(5,6,7,8-tetrahydronaphthalen-2-yl)-1h-pyrazol-5-amine
CAS:Pureza:97%Peso molecular:289.38198852539063-Chloromethyl-5-methylpyridine Hydrochloride
CAS:Producto controlado<p>Applications 3-Chloromethyl-5-methylpyridine is an intermediate in the synthesis of Rupatadine (R701650).<br>References Merlos, M., et al.: Pharmacol. Exp. Therap., 280, 114 (1997), Bell, I., et al.: J. Med. Chem., 41, 2146 (1998),<br></p>Fórmula:C7H8ClN·ClHForma y color:White To BeigePeso molecular:178.06(±)-Mianserin-d3 Hydrochloride (methyl-d3)
CAS:Producto controlado<p>Applications (±)-Mianserin-d3 HCl (methyl-d3) (CAS# 1219804-97-3) is a useful isotopically labeled research compound.<br></p>Fórmula:C18D3H17N2·ClHForma y color:NeatPeso molecular:303.84424-(2-Chloropyrimidin-4-yl)morpholine
CAS:Fórmula:C8H10ClN3OPureza:98%Forma y color:SolidPeso molecular:199.64Decoquinate
CAS:Producto controlado<p>Applications Decoquinate is a quinolone coccidiostat used in veterinary medicine, in particular as animal feed for poultry.<br>References Del Cacho, E. et al.: Int. J. Parasitol., 36, 1515 (2006); Guo, F.C. et al.: Vet. Parasitol., 147, 239 (2007); Davis, J.L. et al.: Vet. Pharmacol. Therap., 9, 1145 (2009);<br></p>Fórmula:C24H35NO5Forma y color:Off-WhitePeso molecular:417.543-[(Dimethylamino)methyl]-1,2,3,9-tetrahydro-9-methyl-4H-carbazol-4-one Hydrochloride
CAS:Producto controlado<p>Impurity Ondansetron EP Impurity A/ Ondansetron USP Related Compound A<br>Applications 3-[(Dimethylamino)methyl]-1,2,3,9-tetrahydro-9-methyl-4H-carbazol-4-one (Ondansetron EP Impurity A) is an impurity of Ondansetron (O655000), an antiemetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Mackinnon, J.W.M., et al.: Eur. J. Cancer Clin. Oncol., 25, 61 (1989);<br></p>Fórmula:C16H20N2O·ClHForma y color:NeatPeso molecular:292.80Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Forma y color:PowderPeso molecular:234.26-fluoro-2-methylquinoline-4-carboxylic acid
CAS:Fórmula:C11H8FNO2Pureza:95.0%Forma y color:Yellow powderPeso molecular:205.1886-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole Hydrochloride
CAS:Producto controlado<p>Impurity Risperidone EP Impurity M; Paliperidone USP Related Compound B<br>Applications 6-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole Hydrochloride (Risperidone EP Impurity M; Paliperidone USP Related Compound B) is a novel antiproliferative agent.<br>References Benaka P. et al.: Invest. New Drugs., 27, 534 (2009);<br></p>Fórmula:C12H13FN2O·ClHForma y color:NeatPeso molecular:256.704'-O-Methylcatechin
CAS:<p>Applications A metabolite of (+)-Catechin, a major polyphenol in many fruits and vegetables.<br>References Heptinstall, S., et al.: J. Cardiovas. Pharmacol., 47, S197 (2006), Gonzalez-Manzano, S., et al.: J. Agric. Food Chem., 57, 1231 (2009), Frank, J., et al.: J. Nut., 139, 58 (2009),<br></p>Fórmula:C16H16O6Forma y color:NeatPeso molecular:304.294-[2-(4-quinolinyl)vinyl]phenol
CAS:Pureza:95.0%Forma y color:Solid, Yellow powderPeso molecular:247.29699707031253-Mercapto-2-methylpropanoic Acid
CAS:Producto controlado<p>Impurity Captopril EP Impurity C<br>Applications 3-Mercapto-2-methylpropanoic Acid (Captopril EP Impurity C) is a useful synthetic intermediate.<br>References Lewis, S.N. et al.: J. Het. Chem., 8, 571-580 (1971)<br></p>Fórmula:C4H8O2SForma y color:NeatPeso molecular:120.17Desamino Chloroimiquimod
CAS:Producto controlado<p>Impurity Imiquimod USP Related Compound C<br>Applications Desamino Chloroimiquimod (Imiquimod USP Related Compound C) is a pharmacologically active compound related to Imiquimod (I475000), an immune response modifier. It stimulates the production of Interferon-a.<br>References Megyeri, K., et al.: Mol. Cell Biol., 15, 2207, (1995), Witt, P.L., et al.: Cancer Res., 53, 5176 (1993), Edwards, L., et al.: Arch. Dermatol., 134, 25 (1998); Gerster, J. et al.: J. Med. Chem., 48, 3481 (2005);<br></p>Fórmula:C14H14ClN3Forma y color:NeatPeso molecular:259.73Aripiprazole-d8 (Butyl-d8)
CAS:Producto controladoFórmula:C232H8H19Cl2N3O2Forma y color:White To Off-WhitePeso molecular:456.43rac Mepindolol
CAS:Producto controlado<p>Applications Mepindolol is a non-selective β-adrenoceptor blocking agent. Mepindolol is used in the treatment of glaucoma.<br>References Luque Otero, M. et al.: Br. J. Clin. Pharmacol., 17, 361 (1984); Beckmann, R. et al.: Arzneim.-Forsch., 36, 811 (1986);<br></p>Fórmula:C15H22N2O2Forma y color:NeatPeso molecular:262.35rac-trans-Ambroxol-d5
CAS:Producto controlado<p>Applications A labelled metabolite of Bromohexine. Ambroxol Hydrochloride is a bronchosecretolytic drug.<br>References Jauch, R., et al.: Arzneim-Forsch., 13, 474 (1963)<br></p>Fórmula:C13H13D5Br2N2OForma y color:NeatPeso molecular:383.13Atrazine
CAS:<p>Applications Selective herbicide. Potential symptoms of overexposure are irritation of eyes and skin; dermatitis, skin sensitization; dyspnea, weakness, incoordination, salivation; hypothermia; liver injury.This compound is a contaminant of emerging concern (CECs)<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Dalgaard-Mikkelsen, S., et al.: Pharmacol. Rev., 14, 225 (1962), Muller, K., et al.: J. Environ. Qual., 31, 309 (2002), Backhaus, T., et al.: Environ. Toxicol. Chem., 23, 258 (2004),<br></p>Fórmula:C8H14ClN5Forma y color:ColourlessPeso molecular:215.683-Chloro Cathinone Hydrochloride
CAS:Producto controlado<p>Applications A metabolite of Bupropion (B689625).<br>References Milena, P., et al.: Eur. Congr. Biopharm. Pharmacokinet., 3rd, 2, 313 (1987),<br></p>Fórmula:C9H11Cl2NOForma y color:NeatPeso molecular:220.15-(1,3-Dioxolan-2-yl)-2-(4-hexyloxybenzoyl)thiophene
CAS:Pureza:97.0%Peso molecular:360.4700012207031Meloxicam
CAS:<p>Applications Preferential cyclooxygenase (COX-2) inhibitor. Sudoxicam and Meloxicam are nonsteroidal anti-inflammatory drugs (NSAIDs) from the enol-carboxamide class.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hawkey, C., et al.: Br. J. Rheumatol., 35, Suppl. 1, 1 (1996), Fleischmann, R., et al.: Expert Opin. Pharmacother., 3, 1501 (2002),<br></p>Fórmula:C14H13N3O4S2Forma y color:Light YellowPeso molecular:351.40Northiaden
CAS:Producto controlado<p>Applications A metabolite of Dothiepin.<br>References Atkinson, H., et al.: Clin. Pharmacokin., 18, 151 (1990), Hagg, S., et al.: Br. J. Clin. Pharmacol., 49, 286 (2000), Fleishaker, J., et al.: Adv. Drug Deliv. Rev., 55, 643 (2003), Katritzky, A., et al.: Bioorg. Med. Chem., 12, 3027 (2004),<br></p>Fórmula:C18H19NSForma y color:NeatPeso molecular:281.42rac-Hesperetin 7-O-Sulfate Sodium Salt
CAS:<p>Applications rac-Hesperetin 7-O-Sulfate Sodium Salt is a metabolite of rac-Hesperetin (H289501); a derivative of Hesperidine (H281185) with potential antihyperglycemic activity.<br>References Zhang, B., et al.: Bioorg. Med. Chem. Lett., 22, 7194 (2012)<br></p>Fórmula:C16H13NaO9SForma y color:NeatPeso molecular:404.322-Ethoxy-5-[(morpholine-4-carbonyl)-amino]-benzenesulfonyl chloride
CAS:Fórmula:C13H17ClN2O5SPureza:98%Forma y color:SolidPeso molecular:348.85-(6-Methoxynaphthalen-2-yl)-1H-pyrazole-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:268.27200317382813-(4-methylphenyl)-1-phenyl-1H-pyrazole-4-carboxylic acid
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:278.31100463867194-[4-[4-(Diphenylmethylene)-1-piperidinyl]-1-hydroxybutyl]-a,a-dimethyl-benzeneacetic Acid
CAS:<p>Applications 4-[4-[4-(Diphenylmethylene)-1-piperidinyl]-1-hydroxybutyl]-α,α-dimethyl-benzeneacetic acid is an impurity of fexofenadine (F322490), the active metabolite of Terfenadine (T114500), a H1-histamine receptor antagonist.<br>References Pratt, E., et al.: Diabet Med., 18, 515 (2001), Mizutani, N., et al.: J. Pharmacol. Sci., 93, 437 (2003), Scadding, G., et al.: Clin. Drug Invest., 25, 153 (2005), Asai, M., et al.: N. Engl. J. Med., 354, 307 (2006),<br></p>Fórmula:C32H37NO3Forma y color:NeatPeso molecular:483.64N-Nitroso Varenicline
CAS:Producto controlado<p>Applications N-Nitroso Varenicline is a derivative of Varenicline (V215635(M)), which is a useful medication for smoking cessation.<br>References Hart, E., et al.: Behavioural Brain Research, 397, 112887 (2021)<br></p>Fórmula:C13H12N4OForma y color:NeatPeso molecular:240.261N-Nitroso Fluoxetine-D5
CAS:Producto controladoFórmula:C17H12D5F3N2O2Forma y color:Colourless To Light YellowPeso molecular:343.362-(1-Nitroso-4-piperidinyl)-1H-benzimidazole
CAS:Producto controladoFórmula:C12H14N4OForma y color:NeatPeso molecular:230.266ABT 199 (>99%)(Venetoclax)
CAS:Producto controlado<p>Applications ABT 199 (>99%) is a potent and selective BCL-2 inhibitor that achieves potent antitumour activity while sparing platelets. It’s practical application is to treat chronic lymphocytic leukaemic cells and estrogen receptor-positive breast cancer.<br>References Davids, M. & Letai, A.: Cancer Cell, 23, 139 (2013); Souers, A.,et al.: Nat. Med., 19, 202 (2013); Vaillant, F., et al.: Cancer Cell, 24, 120 (2013); Vogler, M., et al.: Brit. J. Haematol., 163, 139 (2013);<br></p>Fórmula:C45H50ClN7O7SForma y color:Light Yellow To YellowPeso molecular:868.44(S)-(-)-4’-Hydroxyphenyl Carvedilol
CAS:Producto controlado<p>Applications An optically active metabolite of Carvedilol (C184625), a nonselective ß-adrenergic blocker with α1-blocking activity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., ET AL.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Schaefer, W.H., et al.: Drug Metab. Dispos., 26, 10, 958 (1998),<br></p>Fórmula:C24H26N2O5Forma y color:NeatPeso molecular:422.476-chloro-4-methyl-N-(pyridin-2-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Pureza:95.0%Peso molecular:289.7799987792969(3-Methoxypyridin-4-yl)boronic acid hydrate
CAS:Fórmula:C6H10BNO4Pureza:95.0%Forma y color:SolidPeso molecular:170.964-Demethoxy-4-hydroxy Apixaban
CAS:Producto controlado<p>Applications 4-Demethoxy-4-hydroxy Apixaban is a metabolite of Apixaban (A726700) which is a potent, direct, selective, and orally active inhibitor of coagulation factor Xa.<br>References Luettgen, J.M. et al.: J. Enz. Inhib. Med. Chem., 26, 514 (2011); Glanis, T. et al.: J. Thromb. Thrombol., 31, 310 (2011); barrett, Y.C. et al.: Thromb. Haemos., 105, 181 (2011);<br></p>Fórmula:C24H23N5O4Forma y color:NeatPeso molecular:445.471-(4-Methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
CAS:Pureza:95.0%Peso molecular:309.3210144042969Nevirapine-d3
CAS:Producto controlado<p>Applications Labelled Nevirapine (N391275), a potent (IC50=84nM) and selective non-nucleoside inhibitor of HIV-1 reverse transcriptase. Antiviral.<br>References Hargrave, K.D., et al.: J. Med. Chem., 34, 2231 (1991), Cheeseman, S.H., et al.: Antimicrob. Agents Chemother., 37, 178 (1993), Guay, L.A., et al.: Lancet, 354, 795 (1999),<br></p>Fórmula:C15H11D3N4OForma y color:White To Light BeigePeso molecular:269.328-chloro-2-(3-methylphenyl)quinoline-4-carboxylic acid
CAS:Pureza:95.0%Peso molecular:297.739990234375Pyrazinecarboxylic Acid-d3
CAS:Producto controlado<p>Applications Labelled analogue of Pyrazinecarboxylic Acid, a very potent urate retaining drug. Pyrazinecarboxylic Acid is a metabolite of the antibacterial agent Pyrazinamide (P840600).<br>References Fanelli, G.M. et al.: J. Clin. Invest., 52, 1946 (1973): Fanelli, G.M. et al.: J. Pharmacol. Exp. Therap., 200, 413 (1977); Lacroix, C. et al.: Arzneim.-Forsch., 40, 76 (1990); Kraemer, H.-J. et al.: J. Chrom. B Niomed. Sci. Appl., 706, 319 (1998);<br></p>Fórmula:C5HD3N2O2Forma y color:White To Light YellowPeso molecular:127.12Iso Sildenafil
CAS:Producto controlado<p>Applications Iso Sildenafil is the isomer of Sildenafil methylated at N-2 position of the pyrazolo[4,3-d]pyrimidin-7-one nucleus.<br>References Sheldrick, G., et al.: Acta Crystallogr., A46, 467 (1990), Terrett, N., et al.: Bioorg. Med. Chem. Lett., 6, 1819 (1996),<br></p>Fórmula:C22H30N6O4SForma y color:NeatPeso molecular:474.58O-Desmethyl Mebeverine Acid
CAS:Producto controladoFórmula:C15H23NO3Forma y color:NeatPeso molecular:265.35Astemizole-d3
CAS:Producto controlado<p>Applications Labelled Astemizole. Nonsedating-type histamine H1-receptor antagonist. Potential for combination therapy with antivancer drugs such as doxorubicin in resistant leukemia. Antihistaminic.<br>References Wauquier, A., et al.: Eur. J. Pharmacol., 72, 245 (1981), Laduron, P.M., et al.: Mol. Pharmacol., 21, 294 (1982), Richards, D.M., et al.: Drugs, 28, 38 (1984), Al-Obaid, A.M., et al.: Anal. Profiles Drug Subs., 20, 173 (1991), Ishikawa, M., et al.: Biol. Pharm. Bull., 23, 112 (2000),<br></p>Fórmula:C28H28D3FN4OForma y color:NeatPeso molecular:461.591-(3-Cyano-2-pyridyl)-4-methyl-2-phenylpiperazine
CAS:<p>Applications Used in the preparation of Mirtazapine (M365000) impurities.<br></p>Fórmula:C17H18N4Forma y color:Light Yellow To BrownPeso molecular:278.35Efavirenz Pent-3-ene-1-yne (cis/trans Mixture)
Producto controlado<p>Applications Efavirenz Pen-3-ene-1-yne is an analog of Efavirenz (E425000), a nonnucleoside HIV-1 reverse transcriptase inhibitor and antiviral agent.<br>References Young, S.D., et al.: Antimicrob. Ag. Chemother., 39, 2602 (1995)<br></p>Fórmula:C14H9ClF3NO2Forma y color:NeatPeso molecular:315.67(2S)-1-(2-Chloroacetyl)-2-9-pyrrolidinecarbonitrile
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications (2S)-1-(2-Chloroacetyl)-2-9-pyrrolidinecarbonitrile is a key intermediate for dipeptidyl peptidase IV inhibitor Vildagliptin (V305000).<br>References Singh, S.K., et al.: Beil. J. Org. Chem., 4, 20 (2008);<br></p>Fórmula:C7H9ClN2OForma y color:NeatPeso molecular:172.61Ref: 10-F601898
1gA consultar2gA consultar5gA consultar100mgA consultar250mgA consultar500mgA consultar(5,5’-Bis(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6,6’-dichloro-3-hydroxy-3,3’-biindoline-2,2’-dione)
CAS:<p>Impurity Ziprasidone EP Impurity D<br>Applications (5,5’-Bis(2-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)ethyl)-6,6’-dichloro-3-hydroxy-3,3’-biindoline-2,2’-dione) (Ziprasidone EP Impurity D) is a compound related to Ziprasidone (Z485000), which is a combined serotonin (5HT2) and dopamine (D2) receptor antagonist. Used as an antipsychotic.<br>References Bench, C.J., et al.: Psychopharmacology, 112, 308 (1993), Goldstein, J.M.: Exp. Opin. Invest. Drugs, 4, 291 (1995)<br></p>Fórmula:C42H40Cl2N8O3S2Forma y color:NeatPeso molecular:839.854-CHLORO-2-(3-PYRIDYL)-QUINAZOLINE
CAS:Pureza:95.0%Forma y color:SolidPeso molecular:241.67999267578125Lercanidipine 5-Desmethyl-5-Propyl Ester
CAS:<p>Applications Lercanidipine 5-Desmethyl-5-Propyl Ester is an impurity of the dihydropyridine calcium channel blocker Lercanidipine (L179000).<br></p>Fórmula:C38H45N3O6Forma y color:NeatPeso molecular:639.7804
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