Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol
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Termina el 31 dic( quedan 10 días )
Fadolmidine
CAS:Fadolmidine is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia.Fórmula:C13H14N2OForma y color:SolidPeso molecular:214.26MPV-1306
CAS:MPV-1306 is a metabolite of Dexmedetomidine -- a novel alpha 2-adrenergic receptor agonist.Fórmula:C13H14N2O2Forma y color:SolidPeso molecular:230.26Vacquinol-1
CAS:Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma cell death.Fórmula:C21H21ClN2OPureza:99.92%Forma y color:SolidPeso molecular:352.86Methasquin
CAS:<p>Methasquin is a folic acid antagonist that has been used in the treatment of experimental leukemia; acts by inhibiting the dihydrofolate reductase in the cell.</p>Fórmula:C21H22N6O5Forma y color:SolidPeso molecular:438.44Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Fórmula:C22H31N5Forma y color:SolidPeso molecular:365.52Pyrithione cadmium
CAS:Pyrithione cadmium suppresses tumor growth in vitro and in vivo through inhibition of proteasomal deubiquitinaseFórmula:C10H8CdN2O2S2Forma y color:SolidPeso molecular:364.73Cilengitide hydrochloride
CAS:Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Fórmula:C27H41ClN8O7Forma y color:SolidPeso molecular:625.12Dersalazine
CAS:<p>Dersalazine, a PAF inhibitor, reduces IL-17 to treat colitis in rodents, potentially aiding ulcerative colitis patients.</p>Fórmula:C35H32N6O4Pureza:99.62%Forma y color:SolidPeso molecular:600.67IND 1316
CAS:<p>IND 1316 is an activator of AMP-activated protein kinase (AMPK).</p>Fórmula:C22H17NO3Forma y color:SolidPeso molecular:343.38EPZ033294
CAS:<p>EPZ033294 has potential anticancer and antiproliferative activity.</p>Fórmula:C20H22ClN7OPureza:99.95%Forma y color:SolidPeso molecular:411.89EPZ032597
CAS:EPZ032597 is a novel selective inhibitor of SMYD2 with an IC50 of 16 nM. EPZ032597 has anticancer activity and prevent and treat pancreatic cancerFórmula:C20H23N7OPureza:99.70%Forma y color:SolidPeso molecular:377.44Grp94-IN-2
CAS:<p>Grp94-IN-2 is a inhibitor of Grp94.</p>Fórmula:C22H23ClN2O5Forma y color:SolidPeso molecular:430.88Colterol (free base)
CAS:<p>Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.</p>Fórmula:C12H19NO3Forma y color:SolidPeso molecular:225.28Soyacerebroside II
CAS:<p>Soyacerebroside II is a Ca2+ ionophore; both I and II inhibit IL-18 in PBMCs and modulate immune responses.</p>Fórmula:C40H75NO9Pureza:98%Forma y color:SolidPeso molecular:714.02Nizatidine amide
CAS:Nizatidine amide blocks H2 receptors, reducing stomach acid to treat ulcers and GERD.Fórmula:C11H18N4O3S2Forma y color:SolidPeso molecular:318.42IACS-4759
CAS:<p>IACS-4759 is a novel potent and selective MTH1 inhibitor with excellent cell permeability and good metabolic stability in microsomes.</p>Fórmula:C10H17N3O2Forma y color:SolidPeso molecular:211.26ent-Entecavir
CAS:Ent-Entecavir, an enantiomeric impurity of Entecavir (an oral HBV drug), inhibits HBV replication as a reverse transcriptase inhibitor.Fórmula:C12H15N5O3Forma y color:SolidPeso molecular:277.28JTP 103237
CAS:<p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>Fórmula:C24H29F3N6OForma y color:SolidPeso molecular:474.52MS-049 oxalate salt
CAS:MS-049 oxalate salt is a potent and selective inhibitor of protein arginine methyltransferases (PRMTs) PRMT 4 and PRMT6.Fórmula:C17H26N2O5Forma y color:SolidPeso molecular:338.4Mps1-IN-1 dihydrochloride
CAS:Mps1-IN-1 dihydrochloride, a potent ATP-competitive inhibitor of Mps1 kinase, exhibits an IC50 of 367 nM.Fórmula:C28H35Cl2N5O4SForma y color:SolidPeso molecular:608.58AEG40730 HCl
CAS:<p>AEG40730: A potent, selective IAP inhibitor, induces cIAP1/2 degradation, reduces RIP1 ubiquitination, and depletes XIAP, c-IAP1.</p>Fórmula:C52H70Cl2F6N8O8Forma y color:SolidPeso molecular:1120.0704Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Fórmula:C9H10N4O4·xC4H10N2Forma y color:SolidPeso molecular:562.54CDK8-IN-18
CAS:CDK8-IN-18, also known as ZINC584617986, is a potent and selective inhibitor of CDK8, also modulating CDK19.Fórmula:C18H17N5OForma y color:SolidPeso molecular:319.36Methylsilanol ascorbate
CAS:<p>Methylsilanol ascorbate is a silanol analogue and inhibitor of angiotensin-converting enzyme.</p>Fórmula:C7H12O8SiForma y color:SolidPeso molecular:252.25VER-155008
CAS:<p>VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively.</p>Fórmula:C25H23Cl2N7O4Pureza:97.03% - 99.55%Forma y color:SolidPeso molecular:556.4SG3-179
CAS:SG3-179 is a BET inhibitor.Fórmula:C28H35ClFN7O3SForma y color:SolidPeso molecular:604.14EMD-66684
CAS:EMD-66684 is a non-peptide angiotensin II receptor antagonist.Fórmula:C28H31ClN8O2Forma y color:SolidPeso molecular:547.06KFP-H008
CAS:KFP-H008 is a potassium-competitive acid blocker.Fórmula:C19H18N4O2SForma y color:SolidPeso molecular:366.44KSK213
CAS:KSK213: Strongly inhibits C. trachomatis (EC50=60 nM); non-toxic to commensals/host cells at 25 μM.Fórmula:C28H25N3O2SForma y color:SolidPeso molecular:467.58Verubecestat tosylate
CAS:Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.Fórmula:C25H26N4O4S2Forma y color:SolidPeso molecular:510.627Chlorpromazine Sulfone Hydrochloride
CAS:Chlorpromazine Sulfone Hydrochloride: metabolite of anti-psychotic, may inhibit N-methyltransferase.Fórmula:C17H20Cl2N2O2SForma y color:SolidPeso molecular:387.32F-050
CAS:F-050 inhibits platelet aggregation, potentially treating thrombosis in guinea pigs, rabbits, and rats.Fórmula:C21H20OForma y color:SolidPeso molecular:288.38Olcorolimus
CAS:Olcorolimus blocks specific allergen-induced inflammation, reducing eosinophil, lymphocyte infiltration, and IL-4/IL-5 mRNA expression.Fórmula:C51H81NO12Forma y color:SolidPeso molecular:900.19Fasudil hydrochloride hydrate
CAS:Fasudil HCl hydrate is a ROCK inhibitor that hinders mature CCM development and lowers portal pressure in cirrhotic rats.Fórmula:C28H38Cl2N6O5S2Forma y color:SolidPeso molecular:673.67Delucemine Free Base
CAS:Delucemine Free Base is an NMDA Receptor AntagonistFórmula:C16H17F2NForma y color:SolidPeso molecular:261.31Verubecestat
CAS:<p>Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.</p>Fórmula:C17H17F2N5O3SPureza:92.24% - 99.55%Forma y color:SolidPeso molecular:409.41CVS-1578
CAS:CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Fórmula:C20H30N6O5SForma y color:SolidPeso molecular:466.55GT-2394
CAS:GT-2394 is a histamine H3 receptor agonist.Fórmula:C14H21N3O2Forma y color:SolidPeso molecular:263.34GT-2227
CAS:<p>GT-2227 is a histamine H3 receptor antagonist.</p>Fórmula:C15H24N2Forma y color:SolidPeso molecular:232.36ATM-1001
CAS:ATM-1001 is an inhibitor of the cancer-associated tropomyosin 3.1 (Tpm3.1), suppressing glucose-stimulated insulin secretion (GSIS) from the pancreatic islets.Fórmula:C30H36N4OForma y color:SolidPeso molecular:468.63Paclitaxel Ceribate
CAS:<p>Paclitaxel Ceribate is a mitotic inhibitor used in cancer chemotherapy.</p>Fórmula:C51H57NO18Forma y color:SolidPeso molecular:971.99Pamiparib hydrate
CAS:<p>Pamiparib (BGB-290) is a potent, selective PARP inhibitor that promotes DNA damage and apoptosis in cancer cells.</p>Fórmula:C16H21FN4O4Forma y color:SolidPeso molecular:352.36Cyclanoline (free base)
CAS:Cyclanoline (free base) is an acetylcholinesterase inhibitorFórmula:C20H24NO4Forma y color:SolidPeso molecular:342.41PSI-112
CAS:PSI-112 is a fibrinolysis inhibitor.Fórmula:C35H48N4O3Forma y color:SolidPeso molecular:572.78Vernolepin
CAS:<p>Vernolepin is a natural reversible plant growth inhibitor.</p>Fórmula:C15H16O5Forma y color:SolidPeso molecular:276.28VO-Ohpic trihydrate
CAS:<p>VO-Ohpic trihydrate (VO-Ohpic) is a potent inhibitor of PTEN (phosphatase and tensin homolog) with IC50 of 35 nM.</p>Fórmula:C12H9N2O8V·3H2O·HPureza:>99.99%Forma y color:SolidPeso molecular:415.2Zavondemstat
CAS:Zavondemstat (QC8222 free base) is a KDM4 inhibitor with anticancer and antitumor activity for the study of triple-negative and breast cancers.Fórmula:C26H29N3O3Pureza:99.43% - 99.53%Forma y color:SolidPeso molecular:431.53Acotiamide Methyl Ether
CAS:<p>Acotiamide Methyl Ether is a metabolite enhancing gastric motility, derived from Acotiamide, a drug easing functional dyspepsia symptoms.</p>Fórmula:C22H32N4O5SForma y color:SolidPeso molecular:464.58N-5984 Hydrochloride
CAS:<p>N-5984 Hydrochloride is a beta3-AR agonist.</p>Fórmula:C20H23Cl2NO5Forma y color:SolidPeso molecular:428.31Tomivosertib HCl
CAS:Tomivosertib (eFT508) is a MNK1/2 inhibitor that blocks eIF4E phosphorylation, hindering tumor growth and immune signaling.Fórmula:C17H21ClN6O2Forma y color:SolidPeso molecular:376.845Pemrametostat succinate
CAS:Pemrametostat succinate, an oral PRMT5 inhibitor, strongly curbs tumor growth in vitro and animal studies.Fórmula:C28H38N6O7Forma y color:SolidPeso molecular:570.65CJM-061
CAS:<p>CJM-061 is a Wee1 inhibitor.</p>Fórmula:C28H32N8O4Forma y color:SolidPeso molecular:544.6Famotine
CAS:Famotidine: H2 blocker that reduces stomach acid, treats ulcers and GERD.Fórmula:C16H14ClNOForma y color:SolidPeso molecular:271.74Olmutinib hydrochloride
CAS:Olmutinib is a third-gen EGFR inhibitor for T790M-positive lung cancer, blocking phosphorylation and tumor pathways. Approved in Korea (2016).Fórmula:C26H28Cl2N6O2SForma y color:SolidPeso molecular:559.51ST-115
CAS:ST-115: potent aminopeptidase P2 inhibitor, reduces bradykinin degradation intravenously, boosting its capillary concentration.Fórmula:C21H32FN3O5SForma y color:SolidPeso molecular:457.56Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Fórmula:C29H33FN2O4Pureza:98.77% - 99.93%Forma y color:SolidPeso molecular:492.58NPA101.3
CAS:NPA101.3 is a a Second-Generation RET/VEGFR2 Inhibitor. It is a potential clinical candidate for RET-driven cancers.Fórmula:C29H28N4O4SForma y color:SolidPeso molecular:528.62TPP2a bromide
CAS:<p>TPP2a is a mitochondrial thioredoxin reductase (TrxR) inhibitor.</p>Fórmula:C47H52BrO5PForma y color:SolidPeso molecular:807.81HSP-117 dihydrochloride
CAS:HSP-117 dihydrochloride is a novel tachykinin NK1-receptor antagonist.Fórmula:C23H32Cl2N2OForma y color:SolidPeso molecular:423.42BAY-846
CAS:<p>BAY-846: allosteric MEK inhibitor, long-lasting, highly bioavailable, low brain entry, effective in K-Ras A549 model.</p>Fórmula:C19H13F4IN4O4SForma y color:SolidPeso molecular:596.29L-778123 Dihydrochloride
CAS:L-778123 blocks FPTase/GGPTase-I, halts Ki-Ras prenylation, has acceptable toxicity with radiotherapy in advanced pancreatic cancer.Fórmula:C22H22Cl3N5OForma y color:SolidPeso molecular:478.802Nepaprazole sodium dihydrate
CAS:Nepaprazole sodium dihydrate is a proton pump inhibitor potentially for treatment of gastric ulcers.Fórmula:C18H22N3NaO4SForma y color:SolidPeso molecular:399.44CAM 4750
CAS:<p>CAM 4750 is a nonpeptide tachykinin NK1 receptor antagonist.</p>Fórmula:C30H31ClN4O4Forma y color:SolidPeso molecular:547.05CAM 4515
CAS:<p>CAM 4515 is a nonpeptide tachykinin NK1 receptor antagonist.</p>Fórmula:C29H27N3O4Forma y color:SolidPeso molecular:481.54AZ0108
CAS:<p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>Fórmula:C24H20F4N6O2Forma y color:SolidPeso molecular:500.45MSD-D
CAS:<p>MSD-D is an inhibitor of voltage-gated K(+) (Kv) channels Kv1.5.</p>Fórmula:C20H17N3O2SForma y color:SolidPeso molecular:363.43Voxtalisib
CAS:Voxtalisib (XL765) (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110γ with IC50 of 9 nM; also inhibits DNA-PK and mTOR. Phase 1/2.Fórmula:C13H14N6OPureza:98.21% - 99.69%Forma y color:SolidPeso molecular:270.29MDK80908
CAS:MDK80908 (CAS# 1821380-90-8), a dual PPARα/γ agonist, improves insulin resistance and gluconeogenesis.Fórmula:C21H43NO2SForma y color:SolidPeso molecular:373.64pyimDC
CAS:<p>pyimDC is a novel potent inhibitor of collagen prolyl-4-hydroxylases (CP4H).</p>Fórmula:C10H7N3O4Forma y color:SolidPeso molecular:233.18Derazantinib dihydrochloride
CAS:Derazantinib, a multi-kinase inhibitor targeting FGFR, benefits FGFR2-positive iCCA; its dihydrochloride form is a salt variant.Fórmula:C29H31Cl2FN4OForma y color:SolidPeso molecular:541.49ORP-101
CAS:<p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>Fórmula:C60H84N2O8Forma y color:SolidPeso molecular:961.32LYRM03
CAS:LYRM03, a ubenimex derivative and aminopeptidase inhibitor, suppresses TLR4 to treat LPS-induced ALI in mice.Fórmula:C21H33N3O5Forma y color:SolidPeso molecular:407.510-Oxononadecanedioic acid
CAS:10-Oxononadecanedioic acid: a long-chain linker with two carboxylic ends, forms stable amides with amines using activators like EDC/HATU.Fórmula:C19H34O5Forma y color:SolidPeso molecular:342.47Fipravirimat
CAS:Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.Fórmula:C43H67FN2O4SForma y color:SolidPeso molecular:727.07CDK8-IN-4k
CAS:<p>CDK8-IN-4k is a potent and highly selective CDK8 inhibitor, with no apparent potential for time-dependent CYP3A4 inhibition.</p>Fórmula:C24H23F2N5OForma y color:SolidPeso molecular:435.47PomCapstafin
CAS:PomCapstafin is a prodrug of Capstafin, acting as a potent, selective STAT5b inhibitor.Fórmula:C41H69NO17P2Forma y color:SolidPeso molecular:909.93Vps34-IN-1
CAS:<p>Vps34-IN-1: potent, selective Vps34 inhibitor, 25 nM IC50, spares class I/II PI3Ks.</p>Fórmula:C21H24ClN7OPureza:97.04%Forma y color:SolidPeso molecular:425.91Capstafin
CAS:Capstafin is a highly potent and selective inhibitor of STAT5b.Fórmula:C17H29NO9P2Forma y color:SolidPeso molecular:453.36MeTC7
CAS:<p>MeTC7 is a VDR antagonist with antitumor activity that inhibits PD-L1 and may inhibit the growth of xenografts and transgenic tumors in vivo.</p>Fórmula:C32H48BrN3O4Pureza:99.69%Forma y color:SolidPeso molecular:618.65Miransertib mesylate
CAS:Miransertib mesylate inhibits AKT non-competitively, potentially reducing tumor growth and triggering apoptosis.Fórmula:C29H32N6O6S2Forma y color:SolidPeso molecular:624.73Pipoxolan hydrochloride
CAS:<p>Pipoxolan is an antispasmodic treating GI tract, gallbladder, urogenital, and menstrual cramps, with emerging anticancer properties.</p>Fórmula:C22H26ClNO3Forma y color:SolidPeso molecular:387.9041-Hydroxyvaldecoxib
CAS:1-Hydroxyvaldecoxib is a COX-2 inhibitor.Fórmula:C16H14N2O4SForma y color:SolidPeso molecular:330.36Fenoldopam hydrochloride
CAS:<p>Fenoldopam HCl: D1 dopamine receptor agonist, vasodilator, doesn't cross blood-brain barrier, α2-adrenoceptor antagonist.</p>Fórmula:C16H17Cl2NO3Forma y color:SolidPeso molecular:342.22K-5a2
CAS:K-5a2 is a novel human immunodeficiency virus type 1 (HIV-1) non-nucleoside reverse transcriptase inhibitor (NNRTI).Fórmula:C27H28N6O3S2Forma y color:SolidPeso molecular:548.68GGTI-297
CAS:GGTI-297 is a potent, cell-permeable, and selective peptidomimetic inhibitor of GGTase I compared to Farnesyl Transferase (FTase).Fórmula:C26H31N3O3SForma y color:SolidPeso molecular:465.61UniPR1331
CAS:UniPR1331 is a novel selective antagonist of the Eph-ephrin system.Fórmula:C35H48N2O4Forma y color:SolidPeso molecular:560.77VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Fórmula:C19H16ClN5O6SPureza:98.99% - 99.22%Forma y color:SolidPeso molecular:477.88PF-06427878
CAS:<p>PF-06427878 is an orally active, potent and selective diacylglycerol acyltransferase 2 inhibitor.</p>Fórmula:C26H28N4O5Forma y color:SolidPeso molecular:476.52Berotralstat HCl
CAS:<p>Berotralstat HCl is a selective plasma kallikrein inhibitor, reducing pain and swelling in HAE by blocking bradykinin release.</p>Fórmula:C30H28Cl2F4N6OForma y color:SolidPeso molecular:635.4886GPA512
CAS:<p>GPA512 is a prodrug of aliellalactone, inhibiting STAT3 and preventing the transcription of STAT3 regulated genes.</p>Fórmula:C17H25NO6SForma y color:SolidPeso molecular:371.45Bizine dihydrochloride
CAS:Bizine dihydrochloride is a potent LSD1 inhibitor in vitro, being selective versus monoamine oxidases A/B and the LSD1 homologue, LSD2.Fórmula:C18H25Cl2N3OForma y color:SolidPeso molecular:370.32LASSBio-1829 HCl
CAS:LASSBio-1829 HCl is an orally active IKK2 inhibitor.Fórmula:C25H19ClN4OForma y color:SolidPeso molecular:426.9V-125
CAS:V-125 is an agonist of retinoid X receptors.Fórmula:C23H30N2O2Forma y color:SolidPeso molecular:366.5Indinavir monohydrate
CAS:<p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>Fórmula:C36H49N5O5Forma y color:SolidPeso molecular:631.82BP-5-087
CAS:BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.Fórmula:C36H30F8N2O6SForma y color:SolidPeso molecular:770.69Tofacitinib HCl
CAS:Tofacitinib (tasocitinib, CP-690550) is a JAK inhibitor impacting phosphorylation/activation of STATs with varied IC50 values.Fórmula:C16H21ClN6OForma y color:SolidPeso molecular:348.835UAWJ-247
CAS:UAWJ-247 is a SARS-CoV-2 Main Protease inhibitor (IC50 = 45 nM).Fórmula:C24H28N3NaO8SForma y color:SolidPeso molecular:541.55WNK463
CAS:<p>WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).</p>Fórmula:C21H24F3N7O2Pureza:>99.99% - ≥95%Forma y color:SolidPeso molecular:463.46Milvexian TFA
CAS:Milvexian (BMS-986177/JNJ-70033093) is a factor XIa inhibitor with Ki=44 nM for kallikrein, Ki=35 nM for chymotrypsin, 32% bioavailability.Fórmula:C30H26Cl2F5N9O4Forma y color:SolidPeso molecular:742.49
