CAS 401904-75-4

Carotegrast

CAS : 401904-75-4

Carotegrast

Formule : C₂₇H₂₄Cl₂N₄O₅

Degré de pureté : ≥95%

Masse moléculaire : 555.41

Ref: 54-OR1108208

Carotegrast

CAS : 401904-75-4

Carotegrast is a drug that has been approved for the treatment of HIV infection. It is a prodrug that is hydrolyzed in vivo to carotegravir and piperazine. Carotegravir inhibits the HIV-1 protease, blocking the processing of viral proteins, which prevents new virus particles from being released. The activity of carotegravir has been shown in vitro and in clinical trials to be similar to that of other protease inhibitors such as saquinavir and ritonavir. Piperazine, a piperazine compound, has antiviral properties and may help to prevent HIV-1 replication by inhibiting reverse transcriptase activity. Carotegrast is effective against a wide range of HIV-1 subtypes and strains, including multidrug resistant isolates. This drug also has an excellent safety profile with no significant adverse events reported during clinical trials.

Formule : C₂₇H₂₄Cl₂N₄O₅

Degré de pureté : Min. 95%

Masse moléculaire : 555.4 g/mol

Ref: 3D-BRA90475

Carotegrast

CAS : 401904-75-4

Carotegrast is a selective α4 integrin antagonist, blocking the interaction between α4β1/α4β7 integrins and their ligands.

Formule : C₂₇H₂₄Cl₂N₄O₅

Couleur et forme : Yellow Solid

Masse moléculaire : 555.41

Ref: TM-T14876