
Dynamine
Les inhibiteurs de dynamine ciblent la dynamine, une enzyme GTPase qui joue un rôle crucial dans l'endocytose, le trafic vésiculaire et la cytokinèse. La dynamine est impliquée dans la scission des vésicules à partir des membranes et est essentielle pour la distribution correcte des composants cellulaires pendant la division cellulaire. Inhiber la dynamine peut perturber ces processus, entraînant des défauts de division cellulaire et induisant un arrêt du cycle cellulaire. Les inhibiteurs de dynamine sont précieux pour l'étude de l'endocytose, de la division cellulaire et de la dynamique membranaire. Chez CymitQuimica, nous offrons une gamme d'inhibiteurs de dynamine de haute qualité pour soutenir vos recherches en biologie cellulaire, trafic membranaire et régulation du cycle cellulaire.
23 produits trouvés pour "Dynamine"
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DynaMin inhibitory peptide, myristoylated
CAS :<p>Cell-permeable dynamin inhibitor; blocks its binding to amphiphysin, hindering endocytosis; curbs NMDA receptor internalization.</p>Formule :C61H107N19O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1330.64TAT-P110
CAS :<p>TAT-P110 is a peptide inhibitor that disrupts the interaction between Drp1 and Fis1, effectively reducing pathological changes in various models of neurodegenerative diseases, ischemia, and sepsis without impairing the physiological function of Drp1.</p>Formule :C100H178N44O26Masse moléculaire :2412.76Dynamin inhibitory peptide TFA
<p>Dynamin inhibitory peptide TFA hinders dynamin-amphiphysin interaction and endocytosis, affecting dopamine D3 and GABA A receptors.</p>Formule :C49H81F3N18O16Couleur et forme :SolidMasse moléculaire :1235.27Drp1 peptide inhibitor P110
CAS :<p>Compound P110 (Drp1 peptide inhibitor P110) is a selective Drp1 peptide inhibitor with neuroprotective effects. It inhibits the activation of Drp1, prevents Drp1 mitochondrial translocation induced by MPTP, and alleviates dopamine neuron loss, dopaminergic terminal damage, and behavioral deficits caused by MPTP. This compound is useful for Alzheimer's disease research. Additionally, Compound P110 reduces mitochondrial and organ damage in animal models of Huntington's disease, cerebral ischemia, and myocardial infarction.</p>Formule :C100H179N45O25Couleur et forme :SolidMasse moléculaire :2411.78IIQLPEIVVV TFA
<p>IIQLPEIVVV TFA serves as a specific inhibitor targeting the Drp1-Mff interaction. This compound discriminates between physiological and pathological fission, hindering physiological fission which leads to mitochondrial dysfunction. IIQLPEIVVV TFA is also utilized in research related to Huntington's disease.</p>Formule :C54H95N11O14·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1122.40 (free base)Dynamin IN-2
CAS :<p>Dynamin IN-2 (compound 43) is a Wiskostatin analogue.</p>Formule :C22H21ClN2ODegré de pureté :99.36% - 99.37%Couleur et forme :SoildMasse moléculaire :364.87Anti-Clathrin Heavy Chain Antibody
<p>Anti-Clathrin Heavy Chain Antibody is a human-source antibody expressed in CHO cells, specifically targeting the Clathrin Heavy Chain. For isotype control, please refer to Human IgG1 kappa, Isotype Control.</p>Couleur et forme :Odour LiquidSchaftoside
CAS :<p>Schaftoside (APIGENIN-6-GLUCOSIDE-8-ARABINOSIDE) has antioxidant and anticancer activity.</p>Formule :C26H28O14Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :564.49Mdivi-1
CAS :<p>Mdivi-1 (Mitochondrial division inhibitor 1) is a mitochondrial division inhibitor that inhibits DRP1 and Dynamin I (IC50=1-10 μM).</p>Formule :C15H10Cl2N2O2SDegré de pureté :96.57% - 99.23%Couleur et forme :SolidMasse moléculaire :353.22Dynasore
CAS :<p>Dynasore, a cell-permeable dynamin inhibitor, blocks GTPase of dynamin 1/2 and Drp1 (IC50: 15 μM) without affecting other small GTPases.</p>Formule :C18H14N2O4Degré de pureté :95.85% - 99.22%Couleur et forme :SolidMasse moléculaire :322.31Tetradecyltrimethylammonium bromide
CAS :<p>Tetradecyltrimethylammonium bromide (MitMAB) is a Dynamin GTPase activity inhibitor and a cationic surfactant with asymmetrical structure.</p>Formule :C17H38BrNDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :336.39Trimethyloctadecylammonium bromide
CAS :<p>Trimethyloctadecylammonium bromide is an inhibitor of Dynamin I(IC50 : 1.9 μM) and also inhibits Dynamin Ⅱ.</p>Formule :C21H46N·BrDegré de pureté :99.09%Couleur et forme :Solid SolidMasse moléculaire :392.5Hydroxy-Dynasore
CAS :<p>Hydroxy-Dynasore (Dyngo-4a) , a effective dynamin inhibitor, inhibits withDynI (brain), DynI (rec), and DynII (rec) of IC50 of 0.38 μM, 1.1 μM, and 2.3 μM,</p>Formule :C18H14N2O5Degré de pureté :97.60% - >99.99%Couleur et forme :SolidMasse moléculaire :338.31DNM1 Protein, Human, Recombinant (His)
<p>Microtubule-associated force-producing protein involved in producing microtubule bundles and able to bind and hydrolyze GTP.</p>Couleur et forme :Lyophilized PowderMasse moléculaire :32.2 kDa (predicted)Clathrin-IN-25
CAS :<p>Clathrin-IN-25 is the most effective clathrin terminal domain-amphiphysin inhibitor reported to date.</p>Formule :C19H13KNO5SCouleur et forme :SolidMasse moléculaire :406.47Dynamin IN-1
CAS :<p>Dynamin IN-1 is a potent dynamin inhibitor with an IC 50 value of 1.0 µM .</p>Formule :C23H24N2OCouleur et forme :SolidMasse moléculaire :344.45DRP1i27
CAS :<p>DRP1i27 inhibits human Drp1 at GTPase site, prevents mitochondrial fission, and shields cells from ischemia-reperfusion damage.</p>Formule :C20H26N6OCouleur et forme :SolidMasse moléculaire :366.46Clathrin-IN-2
CAS :<p>Clathrin-IN-2: CME inhibitor, IC50 - 2.3μM; also blocks dyn I GTPase, IC50 - 7.7μM.</p>Formule :C17H18Br2N2OCouleur et forme :SolidMasse moléculaire :426.15Ellipticine quinone
CAS :<p>Ellipticine quinone (NSC-383230) outperforms mdivi-1 in inhibiting Drp1, reduces lung cancer growth, and lessens IR injury by curbing mitochondrial issues.</p>Formule :C15H8N2O2Couleur et forme :SolidMasse moléculaire :248.24Drp1-IN-1
CAS :<p>Drp1-IN-1 (comp A-7) is a Drp1 protein inhibitor (IC50: 0.91 μM).</p>Formule :C22H24N8OSCouleur et forme :SolidMasse moléculaire :448.54

