
Chromatine/Épigénétique
Sous-catégories appartenant à la catégorie "Chromatine/Épigénétique"
2613 produits trouvés pour "Chromatine/Épigénétique"
ADTL-SA1215
CAS :ADTL-SA1215 is a SIRT3 activator with SIRT3 deacetylase activity for the study of triple negative breast cancer.Formule :C26H29I2NO3Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :657.32GSK2879552
CAS :GSK2879552: oral, irreversible LSD1 inhibitor with potential cancer-fighting properties.Formule :C23H28N2O2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :364.48DA-3003-1
CAS :DA-3003-1 (NSC 663284) is a Cdc25 dual specificity phosphatase inhibitor with antitumor activity and inhibits Cdc25B2, Cdc25A, Cdc25B2, and Cdc25C.Formule :C15H16ClN3O3Degré de pureté :99.27% - 99.79%Couleur et forme :SolidMasse moléculaire :321.76PR5-LL-CM01
CAS :PR5-LL-CM01 is a novel protein arginine methyltransferase 5 (PRMT5) inhibitor in colorectal and pancreatic cancers.Formule :C23H27N7Couleur et forme :SolidMasse moléculaire :401.51BAY-850
CAS :BAY-850 is ainhibitor of adenosine triphosphatase family protein 2 that inhibits ovarian cancer growth and metastasis in in vitro and in vivo models.Formule :C38H44ClN5O3Degré de pureté :98% - 98%Couleur et forme :SolidMasse moléculaire :654.24I-BET567
CAS :I-BET567: potent, oral pan-BET inhibitor; pIC50s: 6.9 (BRD4 BD1), 7.2 (BD2); effective in mouse cancer and inflammation models.Formule :C17H18ClN5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :359.81Ref: TM-T9619
1mg89,00€5mg187,00€1mL*10mM (DMSO)205,00€10mg286,00€25mg575,00€50mg863,00€100mg1.269,00€PKC-θ inhibitor
CAS :PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.Formule :C20H25F3N6O3Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :454.45Ref: TM-T5423
1mg101,00€5mg236,00€1mL*10mM (DMSO)259,00€10mg313,00€25mg442,00€50mg580,00€100mg893,00€200mg1.198,00€HDAC-IN-4
CAS :HDAC-IN-4 is a selective HDAC6 and HDAC10 inhibitor (pIC50s: 7.2 and 6.8 in BRET assay) with antitumoral activity.Formule :C20H21N3O2Couleur et forme :SolidMasse moléculaire :335.4SIRT5 inhibitor 3
CAS :SIRT5 inhibitor 3 is potent and competitive by inhibiting SIRT5 deacetylation, with potential in metabolic, cancer, neurodegenerative, cardiovascular .Formule :C22H12FN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.35Protein kinase inhibitor H-7 dihydrochloride
CAS :Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor.Formule :C14H19Cl2N3O2SDegré de pureté :99.81%Couleur et forme :White Crystalline SolidMasse moléculaire :364.29Anti-PARP1 Antibody (8I163)
Anti-PARP1 Antibody (8I163) is a Mouse antibody targeting PARP1. Anti-PARP1 Antibody (8I163) can be used in IHC-P.Couleur et forme :Odour LiquidAnti-PARP Antibody (1W26)
Anti-PARP Antibody (1W26) is a Mouse antibody targeting PARP. Anti-PARP Antibody (1W26) can be used in WB,IHC-P,IP.Couleur et forme :Odour LiquidAnti-PARP1 Antibody (6I459)
Anti-PARP1 Antibody (6I459) is an antibody targeting PARP1. Anti-PARP1 Antibody (6I459) can be used in ELISA, IHC.Couleur et forme :Odour LiquidAnti-PARP1 Antibody (7A800)
Anti-PARP1 Antibody (7A800) is an antibody targeting PARP1. Anti-PARP1 Antibody (7A800) can be used in ELISA, WB, IHC.Couleur et forme :Odour LiquidAnti-PARP1 Antibody (9E313)
Anti-PARP1 Antibody (9E313) is a Mouse antibody targeting PARP1. Anti-PARP1 Antibody (9E313) can be used in IHC-P.Couleur et forme :Odour LiquidNSC 694621
CAS :NSC 694621 is a PCAF inhibitor that forms a covalent bond with Cys574, irreversibly inhibiting its acetyltransferase activity, inhibit proliferation,anticancer.Formule :C13H10N2O2SDegré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :258.3Anti-PARP1 Antibody (8S756)
Anti-PARP1 Antibody (8S756) is an antibody targeting PARP1. Anti-PARP1 Antibody (8S756) can be used in ELISA, WB, IHC, IF, FCM.Couleur et forme :Odour LiquidGintemetostat
CAS :Gintemetostat (KTX-1001) is a potent NSD2 inhibitor (IC50=0.001-0.01μM) for treating NSD2-dysregulated cancers.Formule :C25H26F4N8O2Couleur et forme :SolidMasse moléculaire :546.52(±)-1,2-Diolein
CAS :(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) (1,2-Dioleoyl-rac-glycerol) is a PKC activator. (±)-1,2-Diolein could increases myotubes Ca 2+ influx.Formule :C39H72O5Couleur et forme :SolidMasse moléculaire :620.997-Chloro-4-(piperazin-1-yl)quinoline
CAS :7-Cl-4-(piperazin-1-yl)quinolone: sirtuin inhibitor, serotonin uptake blocker, antimalarial (D10 IC50 1.18µM, K1 IC50 0.97µM).Formule :C13H14ClN3Degré de pureté :99.52%Couleur et forme :Light Yellow SolidMasse moléculaire :247.72AMI-1 free acid
CAS :AMI-1: Potent reversible PRMT inhibitor; IC50: 8.8 μM (hPRMT1), 3.0 μM (yeast-Hmt1p); blocks substrate binding.
Formule :C21H16N2O9S2Degré de pureté :97.8%Couleur et forme :SolidMasse moléculaire :504.49AZ505 ditrifluoroacetate
CAS :AZ505 ditrifluoroacetate is an effective and selective SMYD2 inhibitor (IC50: 0.12 μM).Formule :C33H40Cl2F6N4O8Couleur et forme :SolidMasse moléculaire :805.59XY1
CAS :XY1 is a very close analogue of SGC707 (a potent, selective, and non-competitive inhibitor of PRMT3 with IC50 of 31 nM), It is intended to be used as aFormule :C17H19N3O2Degré de pureté :97.74% - 99%Couleur et forme :SolidMasse moléculaire :297.35AZ960
CAS :AZ960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).Formule :C18H16F2N6Degré de pureté :96.02% - 99.88%Couleur et forme :SolidMasse moléculaire :354.364-(3-Chlorophenyl)-2(3H)-thiazolone
CAS :4-(3-chlorophenyl)-2,3-dihydro-1,3-thiazol-2-one: a thiazole used to make antifungals, antivirals, and anti-inflammatories.Formule :C9H6ClNOSDegré de pureté :95.311%Couleur et forme :SolidMasse moléculaire :211.67UNC0379
CAS :UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.Formule :C23H35N5O2Degré de pureté :94.41% - 99.97%Couleur et forme :SolidMasse moléculaire :413.56WP1066
CAS :WP1066 is a inhibitor of JAK2 (IC50: 2.30 μM) and STAT3 (IC50: 2.43 μM) in HEL cells; shows activity to JAK2, STAT3/5, and ERK1/2, not JAK1 and JAK3.Formule :C17H14BrN3ODegré de pureté :98.92% - 99.73%Couleur et forme :SolidMasse moléculaire :356.22SGC707
CAS :SGC707 is a potent, selective, and cell-active allosteric inhibitor of PRMT3.Formule :C16H18N4O2Degré de pureté :99.75% - 99.89%Couleur et forme :SolidMasse moléculaire :298.34BI-7273
CAS :BI-7273 is an effective, specific, BRD9 BD Inhibitor, which can infiltrate cell.Formule :C20H23N3O3Degré de pureté :97.37% - 99.57%Couleur et forme :SolidMasse moléculaire :353.41TCS PIM-1 1
CAS :TCS PIM-1 1 (SC 204330) is a potent ATP-competitive inhibitor of Pim-1 kinase with an IC50 of 50 nM, selective over MEK1/2 and Pim-2.Formule :C18H11BrN2O2Degré de pureté :97% - 97.98%Couleur et forme :SolidMasse moléculaire :367.2Ref: TM-T2253
1mg34,00€5mg60,00€1mL*10mM (DMSO)92,00€10mg94,00€25mg177,00€50mg269,00€100mg401,00€200mg580,00€Aurothiomalate sodium
CAS :Sodium aurothiomalate (Miochrysin) inhibits PKC-ι, TrxR; used as an anti-rheumatic and has anti-tumor properties.Formule :C4H3AuNa2O4SDegré de pureté :99.66%Couleur et forme :SoildMasse moléculaire :390.07Rucaparib monocamsylate
CAS :Rucaparib monocamsylate (Rucaparib Camsylate) is a PARP inhibitor. Rucaparib Camsylate also displays binding affinity to eight other PARP domains.
Formule :C29H34FN3O5SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :555.665-Ph-IAA
CAS :5-Ph-IAA is a derivative of Indole-3-acetic acid (IAA), which is a plant hormone and acts as an enzyme or prodrug combination for cancer gene therapy.
Formule :C16H13NO2Degré de pureté :99.37% - 99.973%Couleur et forme :SolidMasse moléculaire :251.28PI-1840
CAS :PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.Formule :C22H26N4O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :394.47GSK-J1 sodium salt
CAS :GSK-J1 sodium salt is a potent inhibitor of the H3K27 histone demethylases JMJD3 and UTX.Formule :C22H22N5NaO2Couleur et forme :SolidMasse moléculaire :411.4408CBP/EP300-IN-1
CAS :CBP/EP300-IN-1 is a CBP/EP300 bromodomain inhibitor.Formule :C23H23FN2O5Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :426.44Ref: TM-T7264
1mg46,00€2mg62,00€5mg92,00€1mL*10mM (DMSO)100,00€10mg152,00€25mg250,00€50mg353,00€100mg502,00€200mg682,00€Ro 31-8220
CAS :Ro 31-8220: potent PKC inhibitor (IC50: 5-27 nM). Affects MAPKAP-K1b, MSK1, S6K1, GSK3β (IC50: 3-38 nM), not MKK3/4/6/7.Formule :C25H23N5O2SCouleur et forme :SolidMasse moléculaire :457.55Niraparib hydrochloride
CAS :Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.Formule :C19H21ClN4ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :356.85B2
CAS :B2 (Linazolamide intermediate B impurity 2) promotes inclusion formation in cellular models of Huntington's disease and Parkinson's diseaseFormule :C20H17ClN4O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :396.83Buformin hydrochloride
CAS :Buformin hydrochloride, an oral biguanide antidiabetic, activates AMPK, enhances insulin sensitivity, and inhibits hepatic glucose production.Formule :C6H16ClN5Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :193.68C-7280948
CAS :C-7280948 is a PRMT1 inhibitor.Formule :C14H16N2O2SDegré de pureté :99.55% - ≥95%Couleur et forme :SolidMasse moléculaire :276.35Ref: TM-T2097
5mg46,00€1mL*10mM (DMSO)49,00€10mg66,00€25mg109,00€50mg178,00€100mg268,00€200mg414,00€500mg667,00€AZD1208
CAS :AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency against all three PIM kinases.
Formule :C21H21N3O2SDegré de pureté :97.24% - 99.83%Couleur et forme :SolidMasse moléculaire :379.48Birabresib
CAS :Birabresib (MK-8628) is a synthetic, small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins 2, 3 and 4Formule :C25H22ClN5O2SDegré de pureté :98.3% - 99.36%Couleur et forme :SolidMasse moléculaire :491.99Ref: TM-T6032
2mg46,00€5mg70,00€1mL*10mM (DMSO)74,00€10mg90,00€25mg142,00€50mg222,00€100mg375,00€200mg560,00€500mg893,00€NSC 228155
CAS :NSC 228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and modulate EGFR tyrosine phosphorylation.Formule :C11H6N4O4SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :290.25Ref: TM-T6908
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg63,00€25mg117,00€50mg178,00€100mg334,00€200mg469,00€Aurora kinase inhibitor-3
CAS :Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) is a potent inhibitor of Aurora A kinase (IC50 = 42 nM).1 It is selective for Aurora A over BMX, BTK,Formule :C21H18F3N5ODegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :413.4Ref: TM-T5524
1mg66,00€2mg89,00€5mg152,00€1mL*10mM (DMSO)167,00€10mg236,00€25mg401,00€50mg580,00€100mg797,00€200mg1.099,00€653-47
CAS :653-47 enhances the effects of 666-15 on inhibiting CREB and is a mild CREB inhibitor itself (IC50: 26.3μM).Formule :C20H19ClN2O3Couleur et forme :SolidMasse moléculaire :370.83SNS-314
CAS :SNS-314 inhibits Aurora kinases A and B, blocking cell division in AK-overexpressing tumors.Formule :C18H15ClN6OS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.93Izilendustat hydrochloride
CAS :Izilendustat hydrochloride inhibits prolyl hydroxylase, stabilizing HIF-1α/HIF-2, with potential to treat various HIF-1α diseases.Formule :C22H29Cl2N3O4Couleur et forme :SolidMasse moléculaire :470.39MI-503
CAS :MI-503 is an efficient and selective Menin-MLL inhibitor. MI-503 has a significant inhibitory effect on human MLL leukemia cell line. Cost-effective and quality-assured.Formule :C28H27F3N8SDegré de pureté :99.87% - 99.99%Couleur et forme :SolidMasse moléculaire :564.63Ref: TM-TQ0069
1mg50,00€5mg114,00€1mL*10mM (DMSO)141,00€10mg178,00€25mg334,00€50mg557,00€100mg888,00€PF-CBP1
CAS :PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).Formule :C29H36N4O3Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :488.62Ritlecitinib
CAS :Ritlecitinib (PF-06651600) is an orally available, selective JAK3 inhibitor and does not affect the activity of JAK1/2.Cost-effective and quality-assured.Formule :C15H19N5ODegré de pureté :98.82% - 99.92%Couleur et forme :SolidMasse moléculaire :285.34Ref: TM-T5382
2mg37,00€5mg52,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg205,00€50mg290,00€100mg408,00€200mg595,00€6-Bromo-3-methyl-1,4-dihydroquinazolin-2-one
CAS :CHEMBRDG-BB 7118966 is an inhibitor of Bromodomain-containing protein 4 (human).Formule :C9H9BrN2ODegré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :241.08Ref: TM-T8609
1mg58,00€1mL*10mM (DMSO)107,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€WZ4003
CAS :WZ4003, a highly selective NUAK kinase inhibitor, is with IC50 of 20 nM and 100 nM for NUAK1 and NUAK2, respectively.Formule :C25H29ClN6O3Degré de pureté :99.65% - >99.99%Couleur et forme :SolidMasse moléculaire :496.99Ref: TM-T6291
5mg48,00€1mL*10mM (DMSO)50,00€10mg73,00€25mg111,00€50mg166,00€100mg241,00€200mg358,00€500mg590,00€I-CBP112
CAS :I-CBP112 is a specific and potent acetyl-lysine competitive protein-protein interaction inhibitor targeting the CBP/p300 bromodomains.Formule :C27H36N2O5Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :468.59Ref: TM-T3969
1mg33,00€2mg50,00€5mg92,00€1mL*10mM (DMSO)92,00€10mg161,00€25mg296,00€50mg425,00€100mg583,00€200mg785,00€Paris saponin VII
CAS :Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.Formule :C51H82O21Degré de pureté :99.51% - 99.63%Couleur et forme :SolidMasse moléculaire :1031.18Amifostine sodium
CAS :Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.Formule :C5H15N2NaO3PSCouleur et forme :SolidMasse moléculaire :237.21CM-579 trihydrochloride
CM-579 trihydrochloride: reversible G9a/DNMT inhibitor with IC50s 16 nM (G9a) & 32 nM (DNMT); potent against various cancer cells.Formule :C29H43Cl3N4O3Couleur et forme :SolidMasse moléculaire :602.04NU1025
CAS :NU1025 (NSC-696807) is a potent PARP inhibitor with IC50 of 400 nM.Formule :C9H8N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :176.17Ref: TM-T6912
2mg46,00€5mg67,00€1mL*10mM (DMSO)67,00€10mg98,00€25mg178,00€50mg301,00€100mg475,00€500mg1.063,00€ZINC13466751
CAS :ZINC13466751 is a potent HIF-1α/von Hippel-Lindau interaction inhibitor(IC50 = 2.0 µM).Formule :C20H21N5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :363.41UNC1079
CAS :UNC1079 is an selective L3MBTL3 domain inhibitor
Formule :C28H42N4O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :466.66Senaparib
CAS :Senaparib (IMP4297) is a novel highly potent and selective oral PARP1/2 inhibitor with strong antitumor activity.Formule :C24H20F2N6O3Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :478.45Ref: TM-T9593
1mg46,00€2mg59,00€5mg87,00€1mL*10mM (DMSO)96,00€10mg153,00€25mg274,00€50mg432,00€100mg638,00€A-769662
CAS :A-769662 is an effective, reversible AMPK activator(EC50=0.8 μM).Formule :C20H12N2O3SDegré de pureté :97.52% - 99.58%Couleur et forme :SolidMasse moléculaire :360.39Ref: TM-T2468
2mg37,00€5mg54,00€1mL*10mM (DMSO)56,00€10mg74,00€25mg135,00€50mg244,00€100mg440,00€500mg964,00€BAZ1A-IN-1
CAS :BAZ1A-IN-1, a potent inhibitor, KD 0.52 μM against BAZ1A, is effective in high-BAZ1A cancer cells, not in low-BAZ1A ones.Formule :C16H12N4O3SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :340.36Ref: TM-T9552
1mg84,00€5mg177,00€1mL*10mM (DMSO)195,00€10mg268,00€25mg537,00€50mg803,00€100mg1.099,00€200mg1.468,00€A1874
CAS :A1874 is a nutlin-based and BRD4-degrading PROTAC which induces BRD4 degradation in cells. Effective in inhibiting many cancer cell lines proliferation.
Formule :C58H62Cl3F2N9O7SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :1173.59M1001
CAS :M1001 is a HIF-2α agonist.Formule :C17H17N3O2SDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :327.4Cucurbitacin I
CAS :Cucurbitacin I (JSI-124), a natural compound, is a selective inhibitor of JAK2/STAT3 with anti-cancer activity.Formule :C30H42O7Degré de pureté :96.69% - 99.8%Couleur et forme :SolidMasse moléculaire :514.65KDM4D-IN-1
CAS :KDM4D-IN-1 is a KDM4D inhibitor (IC50: 0.41±0.03 μM).Formule :C11H7N5ODegré de pureté :99.51% - >99.99%Couleur et forme :SolidMasse moléculaire :225.21Ref: TM-T4214
1mg73,00€5mg158,00€1mL*10mM (DMSO)168,00€10mg245,00€25mg495,00€50mg795,00€100mg1.161,00€JNJ-7706621
CAS :JNJ-7706621 is a potent aurora kinase inhibitor, and also inhibits CDK1 and CDK2.Formule :C15H12F2N6O3SDegré de pureté :99.1% - 99.85%Couleur et forme :SolidMasse moléculaire :394.36Ref: TM-T6126
1mg48,00€1mL*10mM (DMSO)94,00€5mg100,00€10mg155,00€25mg268,00€50mg432,00€100mg595,00€200mg833,00€MR837
CAS :MR837 (NSD2-PWWP1 antagonist 3f) is a NSD2-PWWP1 antagonist.Formule :C16H14N2OSDegré de pureté :99.77% - 99.85%Couleur et forme :SolidMasse moléculaire :282.36Ref: TM-T8879
2mg38,00€5mg55,00€1mL*10mM (DMSO)66,00€10mg92,00€25mg138,00€50mg243,00€100mg355,00€200mg502,00€Apabetalone
CAS :Apabetalone (RVX000222) , an effective BET bromodomain inhibitor, has been investigated for the treatment of diabetes, atherosclerosis, and coronary arteryFormule :C20H22N2O5Degré de pureté :98.08% - ≥98%Couleur et forme :SolidMasse moléculaire :370.4PF 477736
CAS :PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (Formule :C22H25N7O2Degré de pureté :97.58% - 99.94%Couleur et forme :SolidMasse moléculaire :419.48BRD4 Inhibitor-24
CAS :BRD4 Inhibitor-24 is a BRD4 small molecule inhibitor with antitumor activity.Formule :C13H14N2O4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :262.26BI-9564
CAS :BI-9564, a specific cell-permeable BRD9 BD inhibitor. The Kd for BRD9 is 5.9 nM, and IC50 for BET family is > 100 μM.
Formule :C20H23N3O3Degré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :353.41EPZ015666
CAS :EPZ015666 (GSK3235025) is an orally available inhibitor of PRMT5 enzymatic activity.Formule :C20H25N5O3Degré de pureté :98% - 99.64%Couleur et forme :SolidMasse moléculaire :383.44CPI-455
CAS :CPI-455 is a specific KDM5 inhibitor.Formule :C16H14N4ODegré de pureté :97.87% - 99.03%Couleur et forme :SolidMasse moléculaire :278.31Ref: TM-T3552
1mg34,00€2mg49,00€5mg70,00€1mL*10mM (DMSO)70,00€10mg105,00€25mg178,00€50mg335,00€100mg505,00€MK-8617
CAS :MK-8617 is an orally available HIF PHD1 3 pan-inhibitor, inhibiting PHD1/2/3 (IC50: 1.0/1.0/14 nM).Formule :C24H21N5O4Degré de pureté :99.38% - >99.99%Couleur et forme :SolidMasse moléculaire :443.45MI-463
CAS :MI-463 is a potent and orally bioavailable inhibitor of the menin-mLL interaction (IC50: 15.3 nM).Formule :C24H23F3N6SDegré de pureté :99.18% - >99.99%Couleur et forme :SolidMasse moléculaire :484.54ASP4132
CAS :ASP4132 is an orally active AMPK activator (EC50 : 18 nM), has anti-cancer activity.Formule :C46H51F3N6O8S2Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :937.06Ref: TM-T8432
1mg50,00€5mg114,00€10mg177,00€1mL*10mM (DMSO)185,00€25mg321,00€50mg482,00€100mg677,00€200mg928,00€LLY-507
CAS :LLY-507 is an effective, cell-active, and specific inhibitor of protein-lysine Methyltransferase SMYD2.Formule :C36H42N6ODegré de pureté :99.58% - 99.93%Couleur et forme :SolidMasse moléculaire :574.76Ref: TM-T6879
1mg42,00€2mg52,00€5mg80,00€1mL*10mM (DMSO)104,00€10mg131,00€25mg289,00€50mg522,00€100mg747,00€PF-06409577
CAS :PF-06409577 is an effective, orally active, and specific allosteric activator of AMPK (EC50: 7 nM, for α1β1γ1).Formule :C19H16ClNO3Degré de pureté :95.17% - 98.21%Couleur et forme :SolidMasse moléculaire :341.79Ref: TM-T4427
1mg34,00€2mg43,00€5mg63,00€1mL*10mM (DMSO)71,00€10mg100,00€25mg200,00€50mg334,00€100mg537,00€200mg762,00€Delgocitinib EtOH
CAS :Delgocitinib (LEO-124249/JTE052) is a selective JAK inhibitor used for reducing skin inflammation and treating chronic dermatitis.Formule :C18H24N6O2Couleur et forme :SolidMasse moléculaire :356.433,6-Dihydroxyflavone
CAS :3,6-Dihydroxyflavone suppresses the epithelial-mesenchymal transition in breast cancer cells by inhibiting the Notch signaling pathway.Formule :C15H10O4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :254.24SETDB1-TTD-IN-1 TFA
SETDB1-TTD-IN-1 TFA: potent, selective SETDB1-TTD inhibitor (Kd: 88 nM), useful for related biological research.Formule :C30H32F3N5O4Couleur et forme :SolidMasse moléculaire :583.6Piribedil hydrochloride
CAS :Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.Formule :C16H19ClN4O2Couleur et forme :SolidMasse moléculaire :334.8ML324
CAS :ML324(IC50=920 nM) is a specific inhibitor of jumonji histone demethylase (JMJD2).Formule :C21H23N3O2Degré de pureté :98.22% - 98.57%Couleur et forme :SolidMasse moléculaire :349.43Ref: TM-T6593
2mg34,00€5mg49,00€10mg74,00€1mL*10mM (DMSO)79,00€25mg122,00€50mg205,00€100mg334,00€200mg494,00€PFI-2 hydrochloride
CAS :PFI-2 hydrochloride ((R)-PFI-2 hydrochloride) is a potent, highly selective, and cell-active inhibitor of the methyltransferase activity of SETD7 (IC50: 2 nM),Formule :C23H26ClF4N3O3SDegré de pureté :99.31% - 99.91%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T4583
1mg38,00€2mg49,00€5mg80,00€10mg111,00€1mL*10mM (DMSO)122,00€25mg200,00€50mg358,00€100mg523,00€500mg1.108,00€Fucosterol
CAS :Fucosterol, from E. stolonifera, has anti-diabetic, anti-adipogenic, anti-cancer properties; it affects PPARα and C/EBPα to control fat cell formation.Formule :C29H48ODegré de pureté :98% - 99.68%Couleur et forme :White PowderMasse moléculaire :412.69BEBT-908
CAS :BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor (IC50 <0.1 μM). BEBT-908 also inhibits HDAC (0.1 μM≤IC50≤1 μM).Formule :C23H25N9O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :507.57Ref: TM-T16529
1mg94,00€5mg222,00€1mL*10mM (DMSO)249,00€10mg334,00€25mg562,00€50mg802,00€100mg1.063,00€200mg1.459,00€4-amino-1,8-Naphthalimide
CAS :4-amino-1,8-Naphthalimide (4-ANI) is a PARP inhibitor with IC50 of 180 nMFormule :C12H8N2O2Degré de pureté :95.13%Couleur et forme :Yellow Solid PowderMasse moléculaire :212.23-methyl-1,2-dihydroquinolin-2-one
CAS :3-methyl-1,2-dihydroquinolin-2-one is the first known micromolar inhibitors of the ATAD2 bromodomain.Formule :C10H9NODegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :159.18Ref: TM-T50035
1mg35,00€1mL*10mM (DMSO)62,00€5mg77,00€10mg103,00€25mg170,00€50mg250,00€100mg354,00€200mg480,00€dencichine
CAS :Dencichine (ODAP) is a neurotoxic agent and a haemostatic agent, which relates to modulation of the coagulation system, and fibrinolytic system.Formule :C5H8N2O5Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :176.13Niraparib tosylate monohyrate
CAS :Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.Formule :C26H30N4O5SDegré de pureté :97.7% - 99.99%Couleur et forme :SolidMasse moléculaire :510.61Ref: TM-T9497
5mg57,00€1mL*10mM (DMSO)66,00€10mg82,00€25mg111,00€50mg137,00€100mg205,00€200mg309,00€500mg515,00€BMS-P5 free base
CAS :BMS-P5 free base is a specific and orally active peptidylarginine deiminase 4 (PAD4) inhibitor.Formule :C27H32N6O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :472.58Ruxolitinib phosphate
CAS :Ruxolitinib phosphate (INCB18424 phosphate) is a JAK1/2 inhibitor with IC50 of 3.3 nM/2.8 nM. Cost-effective and quality-assured.Formule :C17H21N6O4PDegré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :404.36Ref: TM-T3043
5mg49,00€1mL*10mM (DMSO)56,00€10mg62,00€25mg78,00€50mg92,00€100mg138,00€200mg215,00€500mg395,00€1g583,00€COH-SR4
CAS :COH-SR4 (COH-SR4 (Mitochondria uncoupler SR4)) is a uncoupler of mitochondrial oxidative phosphorylation.Formule :C13H8Cl4N2ODegré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :350.03ABBV-744
CAS :ABBV-744 is a BDII-selective BET bromodomain inhibitor that inhibits BRD2/3/4. It is used in the research on inflammatory diseases, cancer, and AIDS.Formule :C28H30FN3O4Degré de pureté :97.03% - >99.99%Couleur et forme :SolidMasse moléculaire :491.55Ref: TM-T4697
1mg44,00€2mg56,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg142,00€25mg284,00€50mg409,00€100mg500,00€200mg718,00€BAY 87-2243
CAS :BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).Formule :C26H26F3N7O2Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :525.53Ref: TM-T2488
1mg34,00€2mg40,00€5mg59,00€1mL*10mM (DMSO)70,00€10mg96,00€25mg200,00€50mg334,00€100mg557,00€IOX2
CAS :IOX2 is a selective HIF PHD inhibitor, active in cells with 21 nM IC50 for PHD2/ELGN-1, not inhibiting FIH at 20uM.Formule :C19H16N2O5Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :352.34Eicosapentaenoic Acid sodium
CAS :EPA sodium, an oral omega-3, demethylates DNA, reactivates tumor suppressors, and induces vasodilation.Formule :C20H29NaO2Couleur et forme :SolidMasse moléculaire :324.434-Phenylbutyric acid
CAS :4-Phenylbutyric acid (Benzenebutyric acid) is a HDAC inhibitor and an endoplasmic reticulum stress (ERS) inhibitor. Cost-effective and quality-assured.Formule :C10H12O2Degré de pureté :98.40% - 99.76%Couleur et forme :SolidMasse moléculaire :164.2

