Endocrinologie/Hormones
Les inhibiteurs en endocrinologie/hormonaux sont des composés qui bloquent l'action des hormones ou interfèrent avec les voies de signalisation hormonales. Ces inhibiteurs sont essentiels pour étudier la régulation des systèmes endocriniens et pour développer des traitements pour les maladies liées aux hormones, telles que le diabète, les troubles de la thyroïde et les cancers hormonodépendants. En modulant l'activité hormonale, ces inhibiteurs peuvent aider à élucider les interactions complexes au sein du système endocrinien. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité en endocrinologie/hormonaux pour soutenir vos recherches en endocrinologie, pharmacologie et sciences médicales.
Sous-catégories appartenant à la catégorie "Endocrinologie/Hormones"
- Récepteur des androgènes(229 produits)
- Annexine A(16 produits)
- Aromatase(23 produits)
- Récepteur d'œstrogène/progestatif(66 produits)
- GPR(1 produits)
- Récepteur des glucocorticoïdes(165 produits)
- LHRH(2 produits)
- Récepteur opioïde(327 produits)
- Récepteur de prostaglandine(122 produits)
- RAAS(89 produits)
- Réductase(51 produits)
- Somatostatine(57 produits)
- Récepteur des hormones thyroïdiennes (THR)(33 produits)
- Récepteur de la vasopressine(48 produits)
Affichez 6 plus de sous-catégories
3420 produits trouvés pour "Endocrinologie/Hormones"
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LY2623091
CAS :LY2623091, a mineralocorticoid receptor antagonist, is utilized in treating refractory hypertension. It demonstrates CYP3A4-dependent clearance and exhibits synergistic effects when combined with CYP3A4 inhibitors.Formule :C30H30FN5O3Couleur et forme :SolidMasse moléculaire :527.59pTH (1-37) (human)
CAS :pTH (1-37) human fragment boosts cAMP, alkaline phosphatase, growth, and BMD, potential for osteoporosis research.Formule :C195H316N58O54S2Couleur et forme :SolidMasse moléculaire :4401.08BIBS 39
CAS :BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.Formule :C32H36N4O3Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :524.65β-Lipotropin (61-69)
CAS :β-Lipotropin (61-69) is a potent opioid agonist [1] [2] .Formule :C45H66N10O15SMasse moléculaire :1019.13PL-017 TFA
PL-017 TFA: μ opioid agonist, IC50 5.5 nM, long-lasting analgesia in rats.Formule :C31H38F3N5O7Masse moléculaire :649.66(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat)
CAS :'(Tyr36)-pTH-Related Protein (1-36) (human, mouse, rat), a peptide, functions as a ligand for parathyroid hormone (PTH) receptors [1].'Formule :C194H303N59O53Masse moléculaire :4309.85PROTAC ERα Degrader-10
CAS :PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.Formule :C45H49N5O4Masse moléculaire :723.9Kalata B7
CAS :Kalata B7, a cyclotide isolated from Oldenlandia affinis DC (Rubiaceae), possesses membrane-permeating capabilities and acts as a partial agonist of oxytocin- and vasopressin V1a-receptors [1] [2].Formule :C128H196N36O40S6Masse moléculaire :3071.53Acetalin-3
CAS :Acetalin-3 (Ac-RFMWMT-NH2) is a hexapeptide that acts as a μ opioid receptor antagonist, displaying high affinity for μ and κ3 opioid receptors, weak affinity for κ1 receptors, and no affinity for κ2 receptors [1].Formule :C42H61N11O8S2Masse moléculaire :912.13Axelopran sulfate
CAS :Axelopran sulfate is used in Oral Therapies for Opioid-induced Bowel Dysfunction in Patients with Chronic Noncancer Pain.Formule :C26H41N3O8SCouleur et forme :SolidMasse moléculaire :555.68ErSO
CAS :ErSO is a selective activator of anticipatory unfolded protein response (UPR) via ERα receptor. ErSO can be used in studies about anti-cancer.Formule :C22H13F6NO3Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :453.33Ref: TM-T39980
500mgÀ demander1mg71,00€5mg161,00€1mL*10mM (DMSO)172,00€10mg250,00€25mg411,00€50mg577,00€100mg772,00€N-Acetylthyroxine
CAS :N-Acetylthyroxine is a kind of Thyroxine analogue for the treatment of diagnosing and treating diabetes.Formule :C17H13I4NO5Couleur et forme :SolidMasse moléculaire :818.91Gridegalutamide
CAS :Gridegalutamide exhibits anti-androgen and anti-tumor activities.Formule :C41H45F3N8O5SCouleur et forme :SolidMasse moléculaire :818.91Isomer-Turosteride
Isomer-Turosteride, a novel 5α-reductase inhibitor, reduces prostate DHT and has anticancer properties without raising T levels.Formule :C27H45N3O3Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :459.67Latanoprost acid
CAS :Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to reduce intraocular pressure.Formule :C23H34O5Degré de pureté :97.96%Couleur et forme :Pale Yellow OilMasse moléculaire :390.51Ref: TM-T15718
1mg54,00€5mg138,00€1mL*10mM (DMSO)152,00€10mg215,00€25mg429,00€50mg637,00€100mg874,00€200mg1.161,00€Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,
Degré de pureté :99.89%Couleur et forme :SoildA 779
CAS :A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.Formule :C39H60N12O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :872.97CIMBA hydrochloride
CIMBA hydrochloride is a selective antagonist of the G protein-coupled estrogen receptor (GPER). It can be utilized in research related to cholesterol gallstone disease in women.Couleur et forme :Odour SolidTyr-W-MIF-1
CAS :Tyr-W-MIF-1, an opioid tetrapeptide, exhibits both opiate and antiopiate activities, and has been demonstrated to induce analgesia [1] [2] [5].Formule :C27H32N6O5Masse moléculaire :520.58SR-29065
CAS :SR-29065 is a REV-ERBα agonist that represses BMAL1 transcription and is used to study circadian regulation, cancer, and autoimmune disease mechanisms.Formule :C24H24F6N2O2SDegré de pureté :97.24% - 98.42%Couleur et forme :Odour SolidMasse moléculaire :518.52XOMA-213
XOMA-213 (LFA-102; X213) is a human monoclonal antibody (mAb) that specifically targets the PRLR/Prolactin Receptor. It inhibits hPRL-dependent growth of BaF3/hPRLR cells with an EC50 of 0.5 μg/mL. In models such as the Nb2-11-luc xenograft mouse and the DMBA-induced rat breast cancer model, XOMA-213 effectively suppresses PRLR signaling and tumor growth. This compound is applicable in research focused on breast cancer, hyperprolactinemia, and prostate cancer.Nesvacumab
CAS :Nesvacumab (REGN910) is a fully human monoclonal antibody targeting Angiopoietin 2 (Ang2), which can be used for studying advanced solid tumors.Degré de pureté :98.7% (SDS-PAGE); 95.7% (SEC-HPLC) - 99.11% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :144.84 kDa3-Iodothyronamine hydrochloride
CAS :3-Iodothyronamine hydrochloride, Thyroid hormone derivative, activates TAAR1, induces hypothermia, for endocrine/metabolic research.Formule :C14H15ClINO2Couleur et forme :SolidMasse moléculaire :391.63UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Formule :C84H142N32O23Degré de pureté :95.92%Couleur et forme :SolidMasse moléculaire :1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS :is a ketone and a building block.
Formule :C38H57N7O8Degré de pureté :96.94%Couleur et forme :SolidMasse moléculaire :739.9OX04528
CAS :OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may be useful in cancer research.Formule :C16H13F6NO2Degré de pureté :99.74%Couleur et forme :SoildMasse moléculaire :365.27CTOP acetate
CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.Formule :C52H71N11O13S2Degré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :1122.32BMS-903452
CAS :BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe for liver cells.Formule :C21H19Cl2FN4O4SDegré de pureté :98.69% - 99.76%Couleur et forme :SolidMasse moléculaire :513.37Ref: TM-T67791
1mg95,00€5mg207,00€1mL*10mM (DMSO)244,00€10mg295,00€25mg444,00€50mg600,00€100mg810,00€200mg1.063,00€Nociceptin (1-13), amide
CAS :Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrainFormule :C61H100N22O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1381.59Alunacedase alfa
CAS :Alunacedase alfa (APN-01) is an angiotensin-converting enzyme 2 with antiviral activity.Degré de pureté :99.1% (SDS-PAGE); 99.9% (SEC-HPLC) - 99.1% (SDS-PAGE); 99.9% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :85.03 kDaDuP 747 HCl
CAS :DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.Formule :C24H29Cl3N2O2Degré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :483.86Urotensin II, mouse TFA (9047-55-6 free base)
Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It is a potent vasoconstrictor.Formule :C78H101N18F3O21S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1747.88SNC 80
CAS :SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Formule :C28H39N3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :449.63NH-3
CAS :NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.Formule :C28H27NO6Degré de pureté :97.79% - 99.40%Couleur et forme :SolidMasse moléculaire :473.52Ref: TM-T40548
1mg207,00€1mL*10mM (DMSO)467,00€5mg520,00€10mg750,00€25mg1.144,00€50mg1.521,00€100mg2.062,00€500mg4.159,00€GPCR agonist-2
CAS :GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.Formule :C10H10N2O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :222.215(R)-15-methyl Prostaglandin D2
CAS :15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor agonist.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.49β-Endorphin (6-31), human
CAS :β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.Formule :C131H218N34O40Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2909.38BPR1M97
CAS :BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.Formule :C18H18Cl2N2ODegré de pureté :98.78% - 99.95%Couleur et forme :SolidMasse moléculaire :349.25LY255582
CAS :LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,Formule :C22H35NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.52DPDPE
CAS :DPDPE is selective δ-opioid receptor agonist peptide.Formule :C30H39N5O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :645.79Deltorphin
CAS :Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.Formule :C44H62N10O10S2Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :955.15[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway ofFormule :C31H43N5O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.65β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formule :C141H221N33O42SDegré de pureté :96.52%Couleur et forme :SolidMasse moléculaire :3082.52[Orn5]-URP acetate
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.Formule :C50H66N10O12S2Degré de pureté :98.4300%Couleur et forme :SolidMasse moléculaire :1063.25AT-121 hydrochloride
CAS :AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.Formule :C24H39ClN4O3SDegré de pureté :97.28% - >99.99%Couleur et forme :SolidMasse moléculaire :499.11Dermorphin
CAS :Dermorphin is agonist of μ-opioid receptor (MOR) agonist.Formule :C40H50N8O10Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :802.87[Orn8]-Urotensin II acetate
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.Formule :C65H87N13O20S2Degré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :1434.59[(pF)Phe4]Nociceptin(1-13)NH2 acetate
[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.
Formule :C63H103FN22O17Degré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :1459.63(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS :(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].Formule :C48H74N12O12S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1075.3Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFormule :C46H66N10O12S2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :1015.21Ref: TM-T20166L
1mg175,00€5mg394,00€10mg590,00€25mg1.060,00€50mg1.591,00€100mg2.387,00€200mg3.580,00€
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