Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
573 produits trouvés pour "Canal calcique"
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Devapamil
CAS :Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.Formule :C26H36N2O3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :424.58Lercanidipine
CAS :Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.Formule :C36H41N3O6Degré de pureté :99.92%Couleur et forme :White To Light Yellow SolidMasse moléculaire :611.73Acetylcholine chloride
CAS :Acetylcholine Chloride is the chloride salt form of acetylcholine, a synthetic, quaternary amino alcohol with cholinergic properties.Formule :C7H16ClNO2Degré de pureté :98.02% - ≥95%Couleur et forme :White Crystalline PowderMasse moléculaire :181.661-EBIO
CAS :1-EBIO (1-EBIO) is a calium channel agonist.Formule :C9H10N2ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :162.19Cinnarizine
CAS :Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Formule :C26H28N2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :368.51Brompheniramine maleate
CAS :Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Cilnidipine
CAS :Cilnidipine (FRC-8653)(FRC8653) is a dual L- and N-type calcium channel blocker and displays antihypertensive, sympatholytic and neuroprotective activity.Formule :C27H28N2O7Degré de pureté :99.83% - 99.96%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :492.52Amlodipine Besylate
CAS :Amlodipine Besylate(Amlodipine benzenesulfonate) is a long-lasting calcium channel blocker.Formule :C26H31ClN2O8SDegré de pureté :96.67% - 99.92%Couleur et forme :White PowderMasse moléculaire :567.05CRAC intermediate 1
CAS :CRAC intermediate 1 (5-(S)-Fluorowillardiine) is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.Formule :C10H7F2N3ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :223.18Carboxyamidotriazole Orotate
CAS :Carboxyamidotriazole Orotate (L-651582 Orotate) is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signalingFormule :C22H16Cl3N7O6Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :580.76Ebselen
CAS :Ebselen is a selenium compound with anti-inflammatory and antioxidant properties, mimicking glutathione peroxidase to protect against ROS damage.Formule :C13H9NOSeDegré de pureté :98.99% - 99.94%Couleur et forme :White SolidMasse moléculaire :274.18Ranolazine dihydrochloride
CAS :Ranolazine 2HCl, an antianginal, treats arrhythmia by inhibiting sodium current without changing blood pressure or heart rate.Formule :C24H35Cl2N3O4Degré de pureté :99.30% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :500.46Ethaverine hydrochloride
CAS :Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Formule :C24H30ClNO4Degré de pureté :99.66% - 99.90%Couleur et forme :SolidMasse moléculaire :431.96Ref: TM-T0369
2mg44,00€5mg63,00€10mg102,00€25mg167,00€50mg250,00€100mg358,00€200mg530,00€1mL*10mM (DMSO)85,00€Dantrolene sodium
CAS :Dantrolene sodium treats spasticity by disrupting muscle contraction; not central in action, grouped with central relaxants.Formule :C14H9N4NaO5Degré de pureté :98% - 99.87%Couleur et forme :CoaMasse moléculaire :336.23Catharanthine tartrate
CAS :Catharanthine tartrate (Catharanthine hemitartrate) is an alkaloid from periwinkle that inhibits voltage-gated L-type calcium channels and has antitumor effect.Formule :C25H30N2O8Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :486.51Diltiazem hydrochloride
CAS :Diltiazem hydrochloride (RG 83606 HCl) is a benzothiazepine calcium channel blocking agent with vasodilating action.Formule :C22H27ClN2O4SDegré de pureté :98% - 99.65%Couleur et forme :Odorless White PowderMasse moléculaire :450.98Ethosuximide
CAS :Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied byFormule :C7H11NO2Degré de pureté :98.87% - 99.72%Couleur et forme :Crystals From Acetone And Ether SolidMasse moléculaire :141.17Flufenamic acid
CAS :Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.Formule :C14H10F3NO2Degré de pureté :98.68%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :281.23BMS-195270
CAS :BMS-195270 is a bio-active chemical.Formule :C15H9ClF3N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :355.7L-Ascorbic acid
CAS :L-Ascorbic acid (Vitamin C) is a natural product that is a potent reducing agent and antioxidant.Formule :C6H8O6Degré de pureté :99.85% - 99.89%Couleur et forme :Crystals (Usually Plates Sometimes Needles Mon°Clinic System) Taste Almost Odorless (Ntp 1992)Masse moléculaire :176.12Nicardipine hydrochloride
CAS :Nicardipine hydrochloride is a potent calcium channel blocker used to dilate cerebral and coronary vessels.Formule :C26H30ClN3O6Degré de pureté :99.58% - 99.89%Couleur et forme :Yellow SolidMasse moléculaire :515.99Levamlodipine
CAS :Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers.Formule :C20H25ClN2O5Degré de pureté :97.21%Couleur et forme :White Crystal PowderMasse moléculaire :408.88Cav 2.2 blocker 1
CAS :Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.Formule :C25H29ClN2O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :424.96Ref: TM-T10690
1mg48,00€5mg105,00€10mg173,00€25mg323,00€50mg494,00€100mg740,00€200mg973,00€1mL*10mM (DMSO)111,00€Butamben
CAS :Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Formule :C11H15NO2Degré de pureté :99.43%Couleur et forme :Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Masse moléculaire :193.24Gabapentin
CAS :Gabapentin (Neurontin) is an Anti-epileptic Agent.Formule :C9H17NO2Degré de pureté :99.55% - 99.91%Couleur et forme :White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidMasse moléculaire :171.24Synta66
CAS :Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.Formule :C20H17FN2O3Degré de pureté :99.57% - 99.84%Couleur et forme :SolidMasse moléculaire :352.36Ref: TM-T13047
2mg34,00€5mg50,00€10mg80,00€25mg147,00€50mg227,00€100mg339,00€200mg482,00€1mL*10mM (DMSO)55,00€Clevidipine
CAS :Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for bloodFormule :C21H23Cl2NO6Degré de pureté :99.40%Couleur et forme :PowderMasse moléculaire :456.32Ca2+ channel agonist 1
CAS :Ca2+ channel agonist 1 activates N-type Ca2+ channels and inhibits Cdk2 (EC50: 14.23 μM/3.34 μM) for motor nerve issues.Formule :C19H26N6ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :354.45Ref: TM-T10659
1mg92,00€5mg178,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.071,00€1mL*10mM (DMSO)207,00€Flunarizine dihydrochloride
CAS :Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.99%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Fendiline hydrochloride
CAS :Fendiline hydrochloride (Fendiline HCl) is a non-selective blocker of calcium channel.Formule :C23H26ClNDegré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :351.91Azelnidipine
CAS :Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker.Formule :C33H34N4O6Degré de pureté :99.78%Couleur et forme :Light Yellowish PowderMasse moléculaire :582.65Ref: TM-T0121
2mg34,00€5mg49,00€10mg64,00€25mg103,00€50mg167,00€100mg260,00€200mg385,00€1mL*10mM (DMSO)59,00€Nifedipine
CAS :Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent.Formule :C17H18N2O6Degré de pureté :99.39% - 99.49%Couleur et forme :Yellow Crystals Physical Description Odorless Yellow Crystals Or Powder Tasteless (Ntp 1992)Masse moléculaire :346.33Minocycline hydrochloride
CAS :Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.Formule :C23H28ClN3O7Degré de pureté :99.28% - >99.99%Couleur et forme :Bright Yellow-Orange Amorphous Solid Crystalline YellowMasse moléculaire :493.94Levetiracetam
CAS :Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onsetFormule :C8H14N2O2Degré de pureté :99.67% - 99.86%Couleur et forme :White Crystalline PowderMasse moléculaire :170.21Norverapamil hydrochloride
CAS :Norverapamil HCl, a Verapamil metabolite, blocks L-type calcium channels and inhibits P-gp function.Formule :C26H37ClN2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :477.04Ref: TM-T16339
1mg34,00€5mg105,00€10mg177,00€25mg299,00€50mg447,00€100mg602,00€200mg842,00€1mL*10mM (DMSO)110,00€Flavoxate hydrochloride
CAS :Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Formule :C24H26ClNO4Degré de pureté :99.78%Couleur et forme :White SolidMasse moléculaire :427.92Manidipine dihydrochloride
CAS :Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Formule :C35H40Cl2N4O6Degré de pureté :99.76% - 99.86%Couleur et forme :SolidMasse moléculaire :683.62Amlodipine
CAS :Amlodipine (UK-48340) is a synthetic dihydropyridine and a calcium channel blocker with antihypertensive and antianginal properties.Formule :C20H25ClN2O5Degré de pureté :99.33% - 99.60%Couleur et forme :Solid PowderMasse moléculaire :408.88Topiramate
CAS :Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36TPC2-A1-P
CAS :TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).Formule :C20H21BrF3NO3Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :460.29Ref: TM-T36806
1mg92,00€5mg225,00€10mg374,00€25mg710,00€50mg1.153,00€100mg1.755,00€1mL*10mM (DMSO)226,00€Verapamil hydrochloride
CAS :Verapamil hydrochloride (Verapamil HCl) is a calcium channel blocker that is a class IV anti-arrhythmia agent.Formule :C27H39ClN2O4Degré de pureté :98.7% - 99.98%Couleur et forme :White To Off-White PowderMasse moléculaire :491.06Caldaret HCl
CAS :Caldaret HCl is an intracellular Ca2+ modulator that regulates calcium homeostasis at the sarcoplasmic reticulum and cell membrane, and can be used to study acute myocardial infarction and heart failure.Formule :C11H17ClN2O3SDegré de pureté :98.99%Couleur et forme :SoildMasse moléculaire :292.78Trimethadione
CAS :Trimethadione (3,5,5,-Trimethyloxazolidine-2,4-dione) is a dione-type anticonvulsant with antiepileptic activity.Formule :C6H9NO3Degré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :143.14Nilvadipine
CAS :Nilvadipine (FK235), a calcium channel blocker (CCB), is utilized for treatment of hypertension.Formule :C19H19N3O6Degré de pureté :99.86% - 99.93%Couleur et forme :Yellow PrismsMasse moléculaire :385.37Tetracaine hydrochloride
CAS :Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.Formule :C15H25ClN2O2Degré de pureté :99.72% - 99.94%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :300.82Cinepazide maleate
CAS :Cinepazide maleate (MD-67350), a maleate salt form of cinepazide, is a vasodilator.
Formule :C22H31N3O5·C4H4O4Degré de pureté :99.9% - 99.97%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :533.57Bupivacaine hydrochloride
CAS :Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Formule :C18H28N2O·HClDegré de pureté :99.89% - 99.9%Couleur et forme :SolidMasse moléculaire :324.89Nisoldipine
CAS :Nisoldipine (BAY-k 5552) is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.Formule :C20H24N2O6Degré de pureté :98.79% - 99.57%Couleur et forme :SolidMasse moléculaire :388.41Cromolyn sodium
CAS :Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.Formule :C23H14Na2O11Degré de pureté :99.4% - 99.95%Couleur et forme :Colorless Crystals From Ethanol + Ether White Crystalline PowderMasse moléculaire :512.33Lacidipine
CAS :Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.Formule :C26H33NO6Degré de pureté :99.98%Couleur et forme :White-To-Off-White Crystalline SolidMasse moléculaire :455.54BX430
CAS :BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonistFormule :C15H15Br2N3ODegré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :413.115,5-Dimethyloxazolidine-2,4-dione
CAS :5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Formule :C5H7NO3Degré de pureté :99.12%Couleur et forme :Drypowder PelletslargecrystalsMasse moléculaire :129.11CRAC intermediate 2
CAS :CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.Formule :C11H7F6N3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :295.18GSK-7975A
CAS :GSK-7975A is a potent and orally available inhibitor of CRAC channel.Formule :C18H12F5N3O2Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :397.3Ref: TM-T15423
1mg42,00€2mg55,00€5mg88,00€10mg130,00€25mg250,00€50mg378,00€100mg570,00€500mg1.189,00€1mL*10mM (DMSO)87,00€Nitrendipine
CAS :Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.Formule :C18H20N2O6Degré de pureté :99% - 99.55%Couleur et forme :SolidMasse moléculaire :360.36Ref: TM-T0119
1g414,00€10mg35,00€25mg52,00€50mg67,00€100mg113,00€200mg172,00€500mg268,00€1mL*10mM (DMSO)52,00€Caloxin 2A1 TFA
Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.Formule :C66H92F3N19O24Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :1592.55Strontium ranelate
CAS :Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.Formule :C12H6N2O8S·2SrDegré de pureté :98.97%Couleur et forme :Crystalline SolidMasse moléculaire :513.49Nimodipine
CAS :Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.Formule :C21H26N2O7Degré de pureté :99.64% - 99.79%Couleur et forme :SolidMasse moléculaire :418.44GV-58
CAS :GV-58 agonizes N/P-Q-type Ca2+ channels (EC50: 7.21/8.81 μM) with 20x less inhibition on CDK kinases.Formule :C18H26N6OSDegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :374.5Ref: TM-T11517
1mg49,00€5mg137,00€10mg205,00€25mg409,00€50mg592,00€100mg827,00€500mg1.648,00€1mL*10mM (DMSO)150,00€Penfluridol
CAS :Penfluridol (TLP-607) is a highly potent antipsychotic.Formule :C28H27ClF5NODegré de pureté :98.9% - 99.87%Couleur et forme :Off-White To White Crystalline PowderMasse moléculaire :523.97Felodipine
CAS :Felodipine (CGH-869) is a longlasting 1, 4-dihydropyridine calcium channel repressor.Formule :C18H19Cl2NO4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :384.25Ref: TM-T0145
2mg34,00€5mg50,00€10mg67,00€25mg96,00€50mg123,00€100mg168,00€500mg409,00€1mL*10mM (DMSO)54,00€Boc-LRR-AMC TFA
Boc-LRR-AMC TFA is a fluorogenic protease substrate for detecting trypsin-like activity in the 26S proteasome or 20S proteasome core.Formule :C35H53F3N10O9Degré de pureté :97.70%Couleur et forme :SolidMasse moléculaire :814.85PACAP-38 (31-38), human, mouse, rat TFA
PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.Formule :C49H84F3N17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1176.29Isotachysterol 3
CAS :Isotachysterol 3 boosts calcium transport in gut and bone mobilization in kidneyless rats.Formule :C27H44OCouleur et forme :SolidMasse moléculaire :384.64Nesiritide
CAS :Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.Formule :C143H244N50O42S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3464.04NSC156529
CAS :NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.Formule :C28H21ClS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.05Ryanodine
CAS :Ryanodine: a diterpenoid modulating Ca2+ release via ryanodine receptors; concentration-dependent effects; found in Ryania speciosa; toxic.Formule :C25H35NO9Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :493.553D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS :Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.Formule :C6H8Na8O18P4Couleur et forme :SolidMasse moléculaire :675.93G-Glu-Ser
CAS :G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.Formule :C8H14N2O6Couleur et forme :SolidMasse moléculaire :234.21Elgodipine
CAS :Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formule :C29H33FN2O6Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :524.58NAADP tetrasodium salt
CAS :Ca2+ mobilizing agentFormule :C21H27N6O18P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :744.39D-myo-Inositol-1,3-diphosphate (sodium salt)
CAS :D-myo-Inositol-1,3-phosphate (Ins(1,3)P) is an inositol phosphate involved in cellular signal transduction.
Formule :C6H12Na2O12P2Couleur et forme :SolidMasse moléculaire :384.08Mast cell degranulating peptide (28-49)
CAS :Mast cell degranulating peptide (28-49) is a bee venom depolarizer that can improve the cGMP content of cerebellum tablets in mice.
Formule :C110H196N40O24S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2591.25RyRs activator 5
Compound A-1 (RyRs activator 5) is an efficacious agonist of ryanodine receptors, exhibiting activity against Spodoptera frugiperda [1].Couleur et forme :Odour SolidBTT-266
CAS :BTT-266 is a blocker of voltage-gated calcium channel for pain management.
Formule :C34H28N4O4Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :556.61Cd1a
Cd1a, a β-toxin from the African spider Ceratogyrus darlingi, modulates calcium ion channels and inhibits human calcium ion channels (Ca v 2.2)(IC 50 2.6 μM) asCouleur et forme :Odour Solidω-Conotoxin MVIIC
CAS :Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.Formule :C106H178N40O32S7Degré de pureté :98%Couleur et forme :White Lyophilised SolidMasse moléculaire :2749Fasudil
CAS :Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.Formule :C14H17N3O2SDegré de pureté :99.79% - 99.84%Couleur et forme :SolidMasse moléculaire :291.37Triphenylethylene
CAS :Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C20H16Couleur et forme :White PowderMasse moléculaire :256.34Cavα2δ-IN-1
CAS :Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a KiFormule :C18H27N5OCouleur et forme :SolidMasse moléculaire :329.448Huwentoxin I
CAS :Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.Formule :C161H246N48O44S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3750.36Mipsagargin
CAS :Mipsagargin (G-202) is a new antibiotic that inhibits DNA biosynthesis.Formule :C66H100N6O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1409.52Nesiritide acetate
CAS :Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.Formule :C143H244N50O42S4C2H4O2Couleur et forme :SolidMasse moléculaire :3524.1Cyclic ADP-ribose ammonium
cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.Couleur et forme :LiquidChlorocresol
CAS :Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.Formule :C7H7ClOCouleur et forme :SolidMasse moléculaire :142.58ω-Agatoxin TK
CAS :Selective blocker of CaV2.1 P/Q-type calcium channels.Formule :C215H337N65O70S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5273.02PACAP-38 (31-38), human, mouse, rat
CAS :PACAP-38 (31-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormule :C47H83N17O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1062.27Candidalysin
CAS :Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.Formule :C153H266N38O38S2Couleur et forme :SolidMasse moléculaire :3310.11sFTX-3.3
CAS :sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.Formule :C12H29N7OCouleur et forme :SolidMasse moléculaire :287.412MMK 1
CAS :Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.Formule :C75H123N19O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1610.97Katacalcin
CAS :Katacalcin (PDN 21) is a potent plasma calcium-lowering peptide[1].Formule :C97H154N34O36S2Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :2436.6Kurtoxin
Kurtoxin is a selective Cav3 (T-type) voltage-gated Ca2+ channel gating inhibitor, exhibiting a dissociation constant (Kd) of 15 nM for the Cav3.1 (α1G T-type)Formule :C324H478N94O90S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7386.36SG-094
CAS :SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.
Formule :C30H29NO3Degré de pureté :97.06%Couleur et forme :SoildMasse moléculaire :451.56(±)5(6)-DiHETE
CAS :Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472Sulcardine 2HCl
CAS :Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.Formule :C24H35Cl2N3O4SDegré de pureté :99.33% - 99.76%Couleur et forme :SoildMasse moléculaire :532.523Ethacrynic acid D5
CAS :Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.Formule :C13H12Cl2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.17ω-Conotoxin GVIA
CAS :Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.Formule :C120H182N38O43S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3037UK-59811 hydrochloride
CAS :UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.Formule :C22H30BrClN2O5Couleur et forme :SolidMasse moléculaire :517.85Ziconotide
CAS :Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.Formule :C102H172N36O32S7Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :2639.131-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS :1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(
Formule :C5H10ClNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :151.59
