Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
572 produits trouvés pour "Canal calcique"
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Zegocractin
CAS :Zegocractin (CM-4620) is a calcium-release activated calcium-channel (CRAC channel) inhibitor.Formule :C19H11ClF3N3O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :421.76Ref: TM-TQ0033
1mg119,00€5mg245,00€10mg409,00€25mg677,00€50mg945,00€100mg1.279,00€1mL*10mM (DMSO)268,00€MDK-4025
CAS :MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.Formule :C19H15ClODegré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :294.77Bevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9L-Ascorbic acid sodium salt
CAS :L-Ascorbic acid sodium salt (Vitamin C sodium salt) is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.Formule :C6H7NaO6Degré de pureté :98.73% - 99.75%Couleur et forme :Less Solid PowderMasse moléculaire :198.11SN 6
CAS :SN 6 (SN6) is a selective Na+/Ca2+ exchanger (NCX) inhibitor (IC50s of NCX1: 2.9 μM , NCX2: 16 μM ,NCX3: 8.6 μM)Formule :C20H22N2O5SDegré de pureté :97.28%Couleur et forme :SolidMasse moléculaire :402.46ZSET1446
CAS :ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.Formule :C15H12N2ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :236.27Ref: TM-T8448
1mg50,00€5mg103,00€10mg144,00€25mg281,00€50mg409,00€100mg572,00€200mg772,00€1mL*10mM (DMSO)119,00€Menthol
CAS :Menthol (DL-Menthol) is an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local anesthetic properties.Formule :C10H20ODegré de pureté :99.84% - 99.88%Couleur et forme :White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Masse moléculaire :156.2614-Deoxyandrographolide
CAS :14-Deoxyandrographolide is a bioactive compound of Andrographis paniculata with hepatoprotective efficacy.Formule :C20H30O4Degré de pureté :99.89% - 99.98%Couleur et forme :SolidMasse moléculaire :334.45Cinacalcet metabolite M4
CAS :Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.Formule :C10H12F3NDegré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :203.2Ref: TM-T10814
5mg55,00€10mg74,00€25mg96,00€50mg137,00€100mg170,00€200mg244,00€500mg364,00€1mL*10mM (DMSO)51,00€Tetrandrine
CAS :Tetrandrine (Sinomenine A) is a naturally occurring biphenylisoquinoline alkaloid, a calcium channel inhibitor. Cost-effective and quality-assured.Formule :C38H42N2O6Degré de pureté :99.61% - 99.94%Couleur et forme :White SolidMasse moléculaire :622.75Bupivacaine
CAS :Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channelsFormule :C18H28N2ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.43Apinocaltamide
CAS :Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.Formule :C22H18F3N5ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :425.41(±)-Bay K 8644
CAS :Produit contrôléFormule :C16H15F3N2O4Couleur et forme :NeatMasse moléculaire :356.3Diltiazem
CAS :Diltiazem (CRD 401 free base) is an orally available L-type Ca2+ channel blocker with antihypertensive, antiarrhythmic, and cardioprotective properties that prevent post-reperfusion myocardial injury, angina pectoris, and cardiovascular-related diseases.Formule :C22H26N2O4SDegré de pureté :99.51% - 99.83%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :414.52Equilin
CAS :Equilin (7-Dehydroestrone) is a neurotrophic estrogenic steroid with vasodilatory activity used in the study of hypertension.Formule :C18H20O2Degré de pureté :98.57% - 99.72%Masse moléculaire :268.35HUP30
CAS :HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.Formule :C14H15N3O3SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :305.35Ref: TM-TNU0864
5mg35,00€10mg52,00€25mg96,00€50mg156,00€100mg222,00€200mg310,00€1mL*10mM (DMSO)39,00€Amlodipine maleate
CAS :Amlodipine maleate (Amvaz) is an oral dihydropyridine calcium blocker for hypertension and cancer studies.
Formule :C24H29ClN2O9Degré de pureté :99.4%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :524.95Bupivacaine-d9
CAS :Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.Formule :C18H19D9N2OCouleur et forme :SolidMasse moléculaire :297.48Gabapentin enacarbil
CAS :Gabapentin enacarbil (XP-13512) is a prodrug for the anticonvulsant and analgesic gabapentin, offering sustained dose-proportional exposure and predictable bioavailability.Formule :C16H27NO6Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :329.39Ref: TM-T15366
1mg42,00€5mg88,00€10mg127,00€25mg274,00€50mg439,00€100mg705,00€200mg938,00€1mL*10mM (DMSO)87,00€1-tert-Butyl 3-Ethyl 5-methyl 2-((2-((tert-Butoxycarbonyl)amino)ethoxy)methyl)-4-(2-chlorophenyl)-6-methylpyridine-1,3,5(4H)-tricarboxylate
CAS :Produit contrôléApplications 1-tert-Butyl 3-Ethyl 5-methyl 2-((2-((tert-Butoxycarbonyl)amino)ethoxy)methyl)-4-(2-chlorophenyl)-6-methylpyridine-1,3,5(4H)-tricarboxylate is an intermediate in the synthesis of 3-O-Desethyl-5-O-desmethyl Amlodipine (D291305). 3-O-Desethyl-5-O-desmethyl Amlodipine is an impurity of Amlodipine (A633495), which is a dihydropyridine calcium channel blocker.
References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)Formule :C30H41ClN2O9Couleur et forme :NeatMasse moléculaire :609.1074-(2-Chlorophenyl)-2-methyl-5-oxo-4,4a,5,7,8,10-hexahydro-1H-pyrido[2',3':2,3]azeto[2,1-c][1,4]oxazine-3-carboxylic Acid
Produit contrôléApplications 4-(2-Chlorophenyl)-2-methyl-5-oxo-4,4a,5,7,8,10-hexahydro-1H-pyrido[2',3':2,3]azeto[2,1-c][1,4]oxazine-3-carboxylic Acid is an intermediate in the synthesis of 3-O-Desethyl-5-O-desmethyl Amlodipine (D291305). 3-O-Desethyl-5-O-desmethyl Amlodipine is an impurity of Amlodipine (A633495), which is a dihydropyridine calcium channel blocker.
References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)Formule :C17H17ClN2O4Couleur et forme :NeatMasse moléculaire :348.781Amlodipine besilate impurity G
CAS :Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in theFormule :C17H18ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.78Amlodipine hydrochloride
CAS :Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.Formule :C20H26Cl2N2O5Couleur et forme :SolidMasse moléculaire :445.34Cinepazide
CAS :Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.Formule :C22H31N3O5Couleur et forme :White PowderMasse moléculaire :417.5Topiramate D12
CAS :Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.Formule :C12H21NO8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.44Nifedipine-d6
CAS :Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.
Formule :C17H18N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.37Cinnarizine D8
CAS :Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.Formule :C26H28N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.573Maresin 1
CAS :Maresin 1 is biosynthesized by macrophages (MΦ) and possesses significant anti-inflammatory activity that attenuates LPS-induced lung injury in mice.Formule :C22H32O4Couleur et forme :SolidMasse moléculaire :360.49ORM-10103
CAS :ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nMFormule :C20H16N2O4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :348.35Ref: TM-T12321
1mg43,00€5mg90,00€10mg135,00€25mg278,00€50mg445,00€100mg605,00€200mg817,00€1mL*10mM (DMSO)90,00€R-(-)-Niguldipine hydrochloride
CAS :R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.Formule :C36H40ClN3O6Couleur et forme :SolidMasse moléculaire :646.17Ionomycin calcium
CAS :Ionomycin calcium (SQ23377 calcium) is an effective and selective calcium ionophore, exhibiting high specificity for calcium ions. Cost-effective and quality-assured.
Formule :C41H70CaO9Degré de pureté :98% - 98.11%Couleur et forme :SolidMasse moléculaire :747.07(R)-Lercanidipine Hydrochloride
CAS :Produit contrôléFormule :C36H41N3O6·ClHCouleur et forme :NeatMasse moléculaire :648.19Dehydro Azelnidipine
CAS :Produit contrôléFormule :C33H32N4O6Couleur et forme :Light Yellow To Light GreenMasse moléculaire :580.63N-Desmethyl-N-acetyl Diltiazem
Produit contrôléApplications N-Desmethyl-N-acetyl Diltiazem is a metabolite of Diltiazem (D460620, HCl); a calcium channel blocker with vasodilating activity. Also anti-anginal, anti-hypertensive, and anti-arrhythmic (class IV).
References Sato, et al.: Arzneim.-Forsch., 21, 1338 (1971); Smirnov, S.R.: Eur. J. Pharmacol., 360, 81 (1998); Hansson, L., et al.: Lancet, 356, 359 (2000)Formule :C23H26N2O5SCouleur et forme :NeatMasse moléculaire :442.53Dihydrocinnamyl Cilnidipine
Produit contrôléApplications Dihydrocinnamyl Cilnidipine is a metabolite of Cilnidipine (C441375); a dihydropyridine calcium channel blocker.
References Ikeda, K., et al.: Oyo Yakuri, 44, 433 (1992); Hosono, M., et al.: J. Pharmacobio-Dyn., 15, 547, (1992); Ishii, M.: Japan Pharmacol. Ther., 21, 59 (1993)Formule :C27H30N2O7Couleur et forme :NeatMasse moléculaire :494.54(S)-Lercanidipine Hydrochloride
CAS :Produit contrôléFormule :C36H41N3O6·ClHCouleur et forme :NeatMasse moléculaire :648.19Falipamil
CAS :Produit contrôléApplications Falipamil is a specific bradycardic agent and a calcium channel blocker.
References Boucher, M., et al.: Eur. J. Pharmacol., 306, 93 (1996), Mubagwa, K., et al.: Arch. Int. Pharmacodyn. Ther., 286, 71 (1987), Chaudhry, A., et al.: Development Cardiovascular Medicine, 46, 196 (1985), Ogiwara, Y., et al.: Jpn Heart J., 29, (1988)Formule :C24H32N2O5Couleur et forme :NeatMasse moléculaire :428.523-Desethyl-3-(2-phthalimidoethyl) Phthaloyl Amlodipine
Produit contrôléStability Light and Temperature Sensitive
Applications 3-Desethyl-3-(2-phthalimidoethyl) Phthaloyl Amlodipine is a derivative of Amlodipine (A633495); a dihydropyridine calcium channel blocker where activity mainly resides in the (-)-isomer.
References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)Formule :C36H30ClN3O9Couleur et forme :NeatMasse moléculaire :684.091Halofuginone
CAS :Halofuginone (RU-19110) inhibits prolyl-tRNA synthetase (Ki=18.3 nM), down-regulates Smad3, and blocks TGF-β at 10 ng/ml.Formule :C16H17BrClN3O3Degré de pureté :99.53%Couleur et forme :Off-White SolidMasse moléculaire :414.68Ref: TM-T6856
1mg34,00€5mg82,00€10mg116,00€25mg227,00€50mg344,00€100mg517,00€500mg1.134,00€1mL*10mM (DMSO)92,00€Verapamil
CAS :Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.Formule :C27H38N2O4Degré de pureté :99.61% - 99.93%Couleur et forme :OilMasse moléculaire :454.6Ref: TM-T20656
10mg34,00€25mg49,00€50mg70,00€100mg90,00€200mg136,00€500mg219,00€1mL*10mM (DMSO)52,00€BA 41899
CAS :BA 41899 is a positive inotropic Ca(2+)-sensitizing agent.Formule :C18H16N2O2Couleur et forme :SolidMasse moléculaire :292.33MRS2690
CAS :MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.Formule :C15H24N2O16P2SCouleur et forme :SolidMasse moléculaire :582.37SIM-6080
CAS :SIM-6080 is a calcium channel antagonist. SIM-6080 inhibits the proliferation of rat aortic myocytes.Formule :C29H36F2N2O3Couleur et forme :SolidMasse moléculaire :498.6RS-93522
CAS :RS-93522: Calcium channel antagonist, inhibits phosphodiesterase (IC50=1.6x10^-5M), like milrinone, and has a negative inotropic effect.Formule :C27H30N2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :526.54Ethacrynate Sodium
CAS :Ethacrynate Sodium, a sodium salt, blocks chloride, potassium, and sodium transport mainly in Henle's loop.Formule :C13H12Cl2NaO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.12JTV-519 hemifumarate
CAS :JTV-519 hemifumarate: Ca2+ blocker, SERCA inhibitor, ryanodine receptor partial agonist; antiarrhythmic, cardioprotective.Formule :C54H68N4O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :965.28AJG-049 free base
CAS :AJG-049 free base is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Formule :C27H30N2O2Couleur et forme :SolidMasse moléculaire :414.54Azelnidipine, (S)-
CAS :Azelnidipine, a selective L-type CCB, improves HF severity and cardiac function in HT and HFpEF compared to N-type CCB cilnidipine.Formule :C33H34N4O6Couleur et forme :SolidMasse moléculaire :582.65Hns 32
CAS :Hns 32 possesses antiarrhythmic properties in dog and guinea pig hearts. It also has vasodilator action.Formule :C24H29N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :359.51A 80b
CAS :A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.Formule :C16H17N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.35Methsuximide
CAS :Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].Formule :C12H13NO2Couleur et forme :Crystals From Dilute Alcohol SolidMasse moléculaire :203.243',4'-Dichlorobenzamil HCl
CAS :3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.Formule :C13H12Cl3N7ODegré de pureté :98%Couleur et forme :Yellow SolidMasse moléculaire :388.64BAY-Y-5959
CAS :BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.Formule :C26H24N4O2Couleur et forme :SolidMasse moléculaire :424.49Aladorian
CAS :Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.Formule :C12H13NO4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.3Aprindine hydrochloride
CAS :Aprindine HCl, a Class 1b antiarrhythmic, treats heart arrhythmias, outperforming digoxin in delaying atrial fibrillation. It's effective orally.Formule :C22H31ClN2Couleur et forme :SolidMasse moléculaire :358.95Levamlodipine gentisate
CAS :Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.Formule :C27H31ClN2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :563Cavα2δ1&NET-IN-2
CAS :Cavα2δ1&NET-IN-2 .Formule :C22H26N6O2SCouleur et forme :SolidMasse moléculaire :438.55TDN345
CAS :TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.Formule :C28H34F2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :468.58Nemadipine-A
CAS :Nemadipine A blocks L-type Ca2+ channels, alters C. elegans morphology, boosts TRAIL's cancer kill rate, and lowers Survivin in A549 cells.Formule :C19H18F5NO4Couleur et forme :SolidMasse moléculaire :419.34Ned-K
CAS :Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.Formule :C31H31N5O3Couleur et forme :SolidMasse moléculaire :521.61S-312-d
CAS :S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.Formule :C20H22N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :386.46SB-237376 HCl
CAS :SB-237376 HCl (SB-237376 hydrochloride) is a calcium and potassium channel antagonist used in the treatment of cardiac arrhythmias.Formule :C20H26ClN3O5Degré de pureté :98.70%Couleur et forme :SolidMasse moléculaire :423.89piCRAC-1
CAS :piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel.Formule :C17H10F6N4Couleur et forme :SolidMasse moléculaire :384.28Niguldipine Free Base
CAS :Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.
Formule :C36H39N3O6Degré de pureté :98.97%Couleur et forme :SolidMasse moléculaire :609.71CGP 28392
CAS :CGP 28392 is used as a partial calcium channel agonist.Formule :C18H17F2NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :365.33JTV-519
CAS :K201 (JTV-519) is a Ca2+-dependent blocker and prevents abnormal Ca(2+) leak from the sarcoplasmic reticulum in the ischemic heart and skeletal muscle (SkM) byFormule :C25H33ClN2O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :461.06Ref: TM-T24239
1mg60,00€5mg110,00€10mg155,00€25mg248,00€50mg365,00€100mg545,00€500mg1.188,00€1mL*10mM (DMSO)134,00€TMB 8 (hydrochloride)
CAS :TMB 8 blocks nAChRs (IC50: 390-480 nM), reduces Ca2+ in muscles, hinders rabbit aorta contraction at 50 μM, and inhibits PKC dose-dependently.Formule :C22H38ClNO5Couleur et forme :White SolidMasse moléculaire :431.99Sadopine
CAS :Sadopine is a high-affinity radioligand for DHP receptor in L-type Ca2+ channels, suitable for tissue and membrane labeling.Formule :C30H40F3N3O7SCouleur et forme :SolidMasse moléculaire :643.71Lercanidipine. (R)-
CAS :(R)-Lercanidipine enantiomer: antihypertensive, blocks L-type Ca2+ channels, dilates blood vessels.Formule :C36H41N3O6Couleur et forme :SolidMasse moléculaire :611.73TTA-P2
CAS :TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.Formule :C21H29Cl2FN2O2Couleur et forme :SolidMasse moléculaire :431.37Leconotide
CAS :Leconotide is a calcium channel blocker and antihyperalgesia agent; isolated from the venom of the cone snail, Conus catus.Formule :C107H179N35O36S7Couleur et forme :SolidMasse moléculaire :2756.23IDO1-IN-19
CAS :IDO1-IN-19 (Compound 17) is a potent inhibitor of IDO1 and has potential for cancer disease research.Formule :C25H22F4N2O3Couleur et forme :SolidMasse moléculaire :474.45CXL-1020
CAS :CXL-1020, a HNO prodrug, enhances heart muscle function & relaxation, aiding in heart failure research.Formule :C7H9NO5S2Couleur et forme :SolidMasse moléculaire :251.28PD-217014 HCl
CAS :PD-217014, a GABA analog, blocks (3)H-gabapentin on alpha(2)delta calcium channels (K(i) 18 nmol/l), and is a visceral analgesic.Formule :C11H19NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :197.27Ricinelaidic Acid
CAS :Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.Formule :C18H34O3Couleur et forme :SolidMasse moléculaire :298.46Cavα2δ1&NET-IN-1
CAS :Cavα2δ1&NET-IN-1 .Formule :C23H26N4O2SCouleur et forme :SolidMasse moléculaire :422.54Mci 176
CAS :Mci 176 is a quinazolinone calcium antagonist.Formule :C24H32ClN3O4Couleur et forme :SolidMasse moléculaire :461.98SM-6586
CAS :SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascularFormule :C26H27N5O5Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :489.52UK-52831
CAS :UK-52831, a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.Formule :C22H26Cl2N6O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :525.39PPZ2
CAS :PPZ2 is a novel DAG-activated TRPC3/TRPC6/TRPC7 channels activator.Formule :C22H29N3O2Couleur et forme :SolidMasse moléculaire :367.48Aladorian sodium
CAS :Aladorian sodium is used for Treatment of Cardiovascular Diseases.Formule :C12H13NNaO4SCouleur et forme :SolidMasse moléculaire :290.29Kadethrin
CAS :Kadethrin is a synthetic pyrethroid. It was used as a pesticide.Formule :C23H24O4SDegré de pureté :98%Couleur et forme :Yellow-Brown Viscous Oil SolidMasse moléculaire :396.5N-Salicyloyltryptamine
CAS :N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).Formule :C17H16N2O2Couleur et forme :SolidMasse moléculaire :280.32PAQ
CAS :PAQ protects neurons in Parkinson's models at 10 μM; prevents neuron loss in mice substantia nigra with 25-50 mg/kg doses.Formule :C14H11N3Couleur et forme :SolidMasse moléculaire :221.26YS-035 hydrochloride
CAS :inhibitor of outward K+ currentsFormule :C21H30ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :395.92Ro 18-3981
CAS :Ro 18-3981 inhibits myocardial Ca2+ channels; KD is 1.0 nM, close to IC50 for ICa block (2.3 nM).Formule :C24H33N3O8SCouleur et forme :SolidMasse moléculaire :523.6Azelnidipine, (R)-
CAS :Azelnidipine is an L-type CCB that improves HF severity and cardiac nerve activity in HT and HFpEF compared to cilnidipine.Formule :C33H34N4O6Couleur et forme :SolidMasse moléculaire :582.65SR-33805
CAS :SR-33805: calcium channel blocker for atherosclerosis/heart failure, enhances myocyte function, modulates myofilament phosphorylation.Formule :C32H40N2O5SCouleur et forme :SolidMasse moléculaire :564.74Norbormide
CAS :Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.Formule :C33H25N3O3Degré de pureté :98%Couleur et forme :Crystals From Methylene Chloride + Ether Norbormide Is A Colorless To Off-White Crystalline Powder Used As A Selective Rat Poison (Epa 1998)Masse moléculaire :511.57ORM-10962
CAS :ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55Formule :C27H29N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :459.54Teludipine hydrochloride
CAS :Teludipine hydrochloride is a blocker of lipophilic calcium channel.Formule :C28H39ClN2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :535.07trans-Ned 19
CAS :trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.Formule :C30H31FN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :514.59YM 244769 hydrochloride
CAS :inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)Formule :C26H23ClFN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.93AZD-2066 hydrochloride
CAS :AZD-2066 hydrochloride is an mGlu5 antagonist.Formule :C19H17Cl2N5O2Couleur et forme :SolidMasse moléculaire :418.28Anipamil
CAS :Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.Formule :C34H52N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.79(S)-Lercanidipine hydrochloride
CAS :(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.19Palonidipine HCl
CAS :Palonidipine HCl is a calcium channel antagonist potentially for the treatment of angina pectoris and hypertension.Formule :C29H35ClFN3O6Couleur et forme :SolidMasse moléculaire :576.06TTA-Q6
CAS :TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.Formule :C20H15ClF3N3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :405.8SOCE inhibitor 1
CAS :SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).Formule :C25H22F3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.47Levosemotiadil
CAS :Levosemotiadil（SA 3212） is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to preventFormule :C29H32N2O6SDegré de pureté :98.53% - 98.88%Couleur et forme :SolidMasse moléculaire :536.64
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