
PDE
Les phosphodiestérases (PDE) sont des enzymes qui hydrolysent les nucléotides cycliques, tels que l'AMPc et le GMPc, en leurs formes inactives, jouant un rôle clé dans la régulation des voies de signalisation intracellulaire. Les inhibiteurs de PDE sont utilisés dans le traitement de diverses affections, notamment les maladies cardiovasculaires, la dysfonction érectile et les troubles respiratoires, en raison de leur capacité à moduler les niveaux de nucléotides cycliques. Chez CymitQuimica, nous proposons une gamme d'inhibiteurs de PDE pour soutenir vos recherches en signalisation cellulaire, pharmacologie et développement thérapeutique.
202 produits trouvés pour "PDE".
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Acetildenafil
CAS :Acetildenafil is an analog of the phosphodiesterase inhibitor sildenafil.Formule :C25H34N6O3Couleur et forme :Off-White To Pale Yelow SolidMasse moléculaire :466.5759PDE4B-IN-6
PDE4B-IN-6 is a highly selective PDE4B inhibitor (IC50=7.42 nM) that exerts anti-inflammatory effects by elevating cAMP and inhibiting TNF-α, used in COPD research.Formule :C22H24F2N2O7Degré de pureté :99.20%Masse moléculaire :466.43Acetildenafil (Standard)
CAS :Acetildenafil (Hongdenafil) (Standard) is the standard substance of Acetildenafil (Hongdenafil), and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Acetildenafil is an analog of the phosphodiesterase inhibitor sildenafil.Formule :C25H34N6O3Masse moléculaire :466.5759Nor-acetildenafil (Standard)
CAS :Nor-acetildenafil (Standard) is the standard substance of Nor-acetildenafil, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Nor-Acetildenafil is a derivative of Acetildenafil, a synthetic phosphodiesterase inhibitor.Formule :C24H32N6O3Masse moléculaire :452.5493Autotaxin modulator 1
CAS :Autotaxin modulator 1 is a new modulator of Autotaxin.Formule :C28H31F6NO3Degré de pureté :99.46%Couleur et forme :White SolidMasse moléculaire :543.5411PF-05180999
CAS :α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is an α-2,3-sialyltransferase inhibitor with anticancer activity.Formule :C19H17F3N8Degré de pureté :99.43% - 99.82%Couleur et forme :SolidMasse moléculaire :414.3871UK 088800 (Standard)
CAS :UK 088800 (Standard) is the standard substance of UK 088800, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. UK 088800 is a bioacitve chemicalFormule :C17H20N4O2Masse moléculaire :312.3663PF-05085727
CAS :PF-05085727 inhibits PDE2A >4,000-fold selectivity over PDE1 and PDE3-11.Formule :C20H18F3N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.399Udenafil (Standard)
CAS :Udenafil (Standard) is the standard substance of Udenafil, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Udenafil is an inhibitor of PDE5 .Formule :C25H36N6O4SMasse moléculaire :516.656Tadalafil-D3
CAS :Tadalafil-D3 is a deuterated compound of Tadalafil. Tadalafil (T1398) has a CAS number of 171596-29-5. Tadalafil (T1398) is a carboline-based compound with vasodilatory activity. Tadalafil (T1398) selectively inhibits the cyclic guanosine monophosphate (cGMP)-specific type 5 phosphodiesterase- (PDE-5)-mediated degradation of cGMP, which is found in the smooth muscle of the corpus cavernosa and corpus spongiosum of the penis. Inhibition of cGMP degradation by tadalafil results in prolonged muscle relaxation, vasodilation, and blood engorgement of the corpus cavernosa, and, so, prolonged penile erection.Formule :C22H19N3O4Masse moléculaire :392.4224DNMDP
CAS :DNMDP is a potent and selective PDE3A inhibitor with anticancer activity. It binds to PDE3A, promoting its interaction with Schlafen 12 (SLFN12).Formule :C15H20N4O3Couleur et forme :Orange SolidMasse moléculaire :304.3443Bay 60-7550
CAS :Bay 60-7550 is a PDE2 inhibitor that exerts positive inotropic effects in the rat heart by increasing PKA-mediated phosphorylation.Formule :C27H32N4O4Degré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :476.5674ALDH7A1 Protein, Human, Recombinant (His)
ALDH7A1 (Aldehyde dehydrogenase 7 family, member A1) is a member of subfamily 7 in the aldehyde dehydrogenase family.Couleur et forme :Transparent LiquidMasse moléculaire :56 kDa (predicted); 56 kDa (reducing conditions)BAY 73-6691 racemate
CAS :BAY 73-6691 racemate (Rac-BAY 73-6691) is a phosphodiesterase 9A (PDE9A) inhibitor, useful for studying Parkinson’s disease.Formule :C15H12ClF3N4OCouleur et forme :White SolidMasse moléculaire :356.73Anti-ALDH7A1 Antibody-FITC (5P692)
Anti-ALDH7A1 Antibody-FITC (5P692) is a FITC-conjugated Rabbit antibody targeting ALDH7A1. Anti-ALDH7A1 Antibody-FITC (5P692) can be used in FCM.Couleur et forme :Odour LiquidAnti-ALDH7A1 Antibody (6G475)
Anti-ALDH7A1 Antibody (6G475) is a Mouse antibody targeting ALDH7A1. Anti-ALDH7A1 Antibody (6G475) can be used in IHC-P.Couleur et forme :Odour LiquidENPP1 Inhibitor C
CAS :ML-354 (VU0099704) is an antagonist with and PAR4 for the study of cardiovascular diseases.Formule :C15H18N6Degré de pureté :99.28%Couleur et forme :Yellow ViscousMasse moléculaire :282.3436Anti-ALDH7A1 Antibody (3P955)
Anti-ALDH7A1 Antibody (3P955) is a Rabbit antibody targeting ALDH7A1. Anti-ALDH7A1 Antibody (3P955) can be used in WB,ELISA,IP.Couleur et forme :Odour LiquidAnti-ALDH7A1 Antibody (5P692)
Anti-ALDH7A1 Antibody (5P692) is a Rabbit antibody targeting ALDH7A1. Anti-ALDH7A1 Antibody (5P692) can be used in FCM,ICC/IF.Couleur et forme :Odour LiquidN-Ethyl tadalafil
CAS :N-Ethyl tadalafil (NEthyl tadalafil) is a PDE inhibitor used in the study of cardiovascular disease.Formule :C23H21N3O4Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :403.43

