Caséine Kinase
Les caséine kinases sont une famille de kinases protéiques sérine/thréonine qui régulent divers processus cellulaires, y compris la réparation de l'ADN, les rythmes circadiens et la transduction du signal. Ces kinases sont impliquées dans la phosphorylation de nombreuses protéines et sont associées à des maladies telles que le cancer, les troubles neurodégénératifs et les syndromes métaboliques. Chez CymitQuimica, nous proposons une sélection d'inhibiteurs de la caséine kinase pour soutenir vos recherches sur la transduction du signal, la régulation du cycle cellulaire et le développement thérapeutique.
130 produits trouvés pour "Caséine Kinase"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
HDAC/CK2-IN-1
CAS :<p>HDAC/CK2-IN-1 (compound 38) acts as an inhibitor of HDAC1 (IC 50 = 1.46 μM), HDAC6 (IC 50 = 0.66 μM), and CK2 (IC 50 = 3.67 μM). It demonstrates promising antiproliferative effects on various cell lines, including Jurkat, MCF-7, HCT-116, and HL-60.</p>Formule :C15H18Br4N4O2Couleur et forme :SolidMasse moléculaire :605.95CK2-IN-4
CAS :<p>CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.</p>Formule :C18H11N3O4SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :365.36CK2α-IN-1
CAS :<p>CK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 µM and a Ki of 1.6 µM.CK2α-IN-1 exhibits potential anticancer activity and can</p>Formule :C16H11N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.34CK1-IN-2
CAS :<p>CK1-IN-2 (compound Nr.4) is a potent CK1 inhibitor p38a, and is used in DUX4 overexpression-associated diseases, such as muscular dystrophy.</p>Formule :C17H12FN3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :309.29PI-828
CAS :<p>PI-828 (LY 294002), a PI3K inhibitor, researches PI3K function and aids stem cell differentiation into mesoderm.</p>Formule :C19H18N2O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :322.36XL413 xHCl
CAS :<p>BMS-863233 HCl is an ATP-competitive Cdc7 inhibitor (IC50: 3.4 nM) that is potent and selective.BMS-863233 HCl inhibited CK2 and PIM1 with IC50 values of 215</p>Formule :C14H12ClN3O2·xHClDegré de pureté :99.37% - 99.67%Couleur et forme :SolidMasse moléculaire :326.18BioE-1115
CAS :<p>BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).</p>Formule :C19H18FN3O2Degré de pureté :97.54%Couleur et forme :SolidMasse moléculaire :339.36Casein kinase 1δ-IN-1
CAS :<p>Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ.</p>Formule :C11H7N3OSDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :229.26Ac-VDVAD-CHO
CAS :<p>Ac-VDVAD-CHO is an inhibitor of caspase-2 and caspase-3 (IC50: 46 nM for caspase-2 and 15 nM for caspase-3) [1].</p>Formule :C23H37N5O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :543.57ON 108600
CAS :<p>ON 108600 is a chemical inhibitor targeting CK2 (Casein Kinase 2), TNIK, and DYRK1, demonstrating IC50 values of 0.016 μM and 0.007 μM for DYRK1A and DYRK1B, 0.</p>Formule :C22H14Cl2N2O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :537.39Casein kinase 1δ-IN-5
CAS :<p>Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects in</p>Formule :C16H11F3N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.33Casein kinase 1δ-IN-10
CAS :<p>Casein kinase 1δ-IN-10 is an inhibitor of casein kinase 1δ (CK1δ).</p>Formule :C21H17N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :359.38TID43
CAS :<p>TID43, a CK2 inhibitor, exhibits potent inhibition with an IC50 value of 0.3 μM. It is applicable in anti-angiogenic research [1].</p>Formule :C10H3I4NO4Couleur et forme :SolidMasse moléculaire :708.755XL413 hydrochloride
CAS :<p>XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7. XL413 hydrochloride also inhibits CK2 and PIM1.</p>Formule :C14H13Cl2N3O2Degré de pureté :98.81% - 99.8%Couleur et forme :SolidMasse moléculaire :326.18Casein kinase 1δ-IN-4
CAS :<p>"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."</p>Formule :C16H12N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :320.37Casein Kinase II Inhibitor IV
CAS :<p>Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.</p>Formule :C24H23N5O3Degré de pureté :99.65% - 99.75%Couleur et forme :SolidMasse moléculaire :429.47Casein kinase 1δ-IN-13
CAS :Casein kinase1δ-IN-13 (compound 401) is an inhibitor of Casein kinase1δ. It is utilized in the research of neurodegenerative diseases.Formule :C15H13N3O2SCouleur et forme :SolidMasse moléculaire :299.35Casein kinase 1δ-IN-28
CAS :<p>Casein kinase1δ-IN-28 (Compound 4) is an inhibitor of CK1ε, with an IC50 of 0.0146 μM. The human liver microsome metabolism rate for Casein kinase1δ-IN-28 is 52%.</p>Formule :C23H23FN6Couleur et forme :SolidMasse moléculaire :402.467CK1δ-IN-6
CAS :<p>CK1δ-IN-6 (Compound 303) is an inhibitor of Casein kinase 1δ, with potential applications in Alzheimer's disease research.</p>Formule :C23H17N3O4Couleur et forme :SolidMasse moléculaire :399.399WAY-606344
CAS :<p>WAY-606344 (Compound 97) is an inhibitor of Casein kinase 1δ and shows potential for Alzheimer's disease research.</p>Formule :C14H8ClN3O2Couleur et forme :SolidMasse moléculaire :285.685
