Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(645 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.022 produits)
- BACE(37 produits)
- Bêta-amyloïde(228 produits)
- CaMK(73 produits)
- COX(600 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(372 produits)
- Gamma-sécrétase(61 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(43 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5548 produits trouvés pour "Neuroscience"
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Otenzepad
CAS :Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.Formule :C24H31N5O2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :421.54Ref: TM-T16411
1mg44,00€5mg79,00€10mg114,00€25mg222,00€50mg356,00€100mg572,00€200mg803,00€1mL*10mM (DMSO)87,00€MNI 137
CAS :MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.Formule :C15H9BrN4ODegré de pureté :97.49%Couleur et forme :SolidMasse moléculaire :341.16AQW051
CAS :AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.Formule :C19H22N2ODegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :294.39Ref: TM-T26646
1mg34,00€2mg46,00€5mg66,00€10mg99,00€25mg205,00€50mg313,00€100mg439,00€500mg954,00€1mL*10mM (DMSO)67,00€Itasetron
CAS :Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.
Formule :C16H20N4O2Degré de pureté :98.58% - 99.33%Couleur et forme :SolidMasse moléculaire :300.36Dipraglurant
CAS :Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.Formule :C16H12FN3Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :265.29Ref: TM-T15134
1mg92,00€5mg215,00€10mg313,00€25mg685,00€50mg1.009,00€100mg1.341,00€1mL*10mM (DMSO)260,00€PPI-1019
CAS :PPI-1019 is an APP (β-amyloid A4) inhibitor for the treatment of neurological disorders and the study of Alzheimer's disease (AD).Formule :C36H54N6O5Degré de pureté :95.16% - 98.16%Couleur et forme :SolidMasse moléculaire :650.85Aβ-IN-1
CAS :Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).Formule :C35H49NDegré de pureté :99.1%Couleur et forme :SoildMasse moléculaire :483.77Ensaculin
CAS :Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formule :C26H32N2O5Degré de pureté :99.56% - 99.81%Couleur et forme :SolidMasse moléculaire :452.54CP-810123
CAS :CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.Formule :C14H18N4ODegré de pureté :98.63% - 99.60%Couleur et forme :SolidMasse moléculaire :258.32Nerisopam
CAS :Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Formule :C18H19N3O2Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :309.36Ref: TM-T28159
1mg88,00€5mg190,00€10mg286,00€25mg464,00€50mg672,00€100mg945,00€200mg1.279,00€1mL*10mM (DMSO)256,00€AZD6538
CAS :AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.Formule :C15H6FN5ODegré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :291.24Fengabine
CAS :Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Formule :C17H17Cl2NODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :322.23CP 96021
CAS :"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formule :C29H21FN4OSDegré de pureté :97.81% - 99.62%Couleur et forme :SoildMasse moléculaire :492.57Riluzole hydrochloride
CAS :Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Formule :C8H6ClF3N2OSDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :270.66Lenumlostat
CAS :Lenumlostat is a lysyl oxidase-like protein 2 (LOXL2) inhibitor with inhibitory effects on hLOXL2, hLOXL3 and LOXL2 for the study of fibrotic diseases.Formule :C18H17F4N3O3Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :399.34Ref: TM-T69913
1mg177,00€5mg447,00€10mg672,00€25mg1.341,00€50mg2.088,00€100mg2.988,00€500mg6.004,00€1mL*10mM (DMSO)492,00€Rilapine
CAS :Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formule :C22H20ClN3Degré de pureté :97.76% - 99.20%Couleur et forme :SolidMasse moléculaire :361.87Anpirtoline hydrochloride
CAS :Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formule :C10H14Cl2N2SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :265.20PNU-282987 free base
CAS :PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formule :C14H17ClN2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :264.75Repinotan
CAS :Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.Formule :C21H24N2O4SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :400.49Tedatioxetine
CAS :Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formule :C18H21NSDegré de pureté :99.76% - >99.99%Couleur et forme :SolidMasse moléculaire :283.43LY 272015 hydrochloride
CAS :LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formule :C21H25ClN2O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :372.89BL-1020 Mesylate
CAS :BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formule :C28H45ClN4O11S4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :777.39ADR-851 free base
CAS :ADR-851 free base is an antagonist of the HT3 receptor.Formule :C14H18ClN3O2Degré de pureté :97.88% - 98.39%Couleur et forme :SolidMasse moléculaire :295.77Lirequinil
CAS :Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formule :C26H25ClN2O3Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :448.94Saripidem
CAS :Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formule :C19H20ClN3ODegré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :341.83Femoxetine hydrochloride
CAS :Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formule :C20H26ClNO2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :347.88R 59-022 hydrochloride
CAS :R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.
Formule :C27H27ClFN3OSDegré de pureté :97.7%Couleur et forme :SolidMasse moléculaire :496.04DA-6886
CAS :DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formule :C19H28Cl2N6O2Degré de pureté :99.91% - 99.99%Couleur et forme :SolidMasse moléculaire :443.37AZD 9272
CAS :AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.Formule :C14H6F2N4ODegré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :284.22Faxeladol
CAS :Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formule :C15H23NODegré de pureté :98.77% - 99.67%Couleur et forme :SolidMasse moléculaire :233.35E6801
CAS :E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formule :C17H18ClN5O2S2Degré de pureté :96.32% - 97.24%Couleur et forme :SolidMasse moléculaire :423.94Desformylflustrabromine hydrochloride
CAS :Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.Formule :C17H12INO5Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :437.19Ref: TM-T11004
2mg34,00€5mg50,00€10mg80,00€25mg145,00€50mg225,00€100mg353,00€200mg550,00€1mL*10mM (DMSO)57,00€Ezeprogind disulfate
CAS :Ezeprogind disulfate: neurotrophic inducer targeting neurodegeneration causes like Abeta, tau; for neurological disorder research.Formule :C25H48N6O8S2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :624.81Cianopramine
CAS :Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formule :C20H23N3Degré de pureté :99.92% - 99.92%Couleur et forme :SolidMasse moléculaire :305.42Oxotremorine M iodide
CAS :Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.Formule :C11H19IN2ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :322.19L-838417
CAS :L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormule :C19H19F2N7ODegré de pureté :98.12% - 99.70%Couleur et forme :SolidMasse moléculaire :399.4Masupirdine free base
CAS :Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formule :C21H24BrN3O3SDegré de pureté :98.36% - 99.65%Couleur et forme :SolidMasse moléculaire :478.4Alpidem
CAS :Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formule :C21H23Cl2N3ODegré de pureté :99.56% - 99.97%Couleur et forme :White To Off-White SolidMasse moléculaire :404.33Ref: TM-T26600
1mg58,00€5mg137,00€10mg207,00€25mg371,00€50mg522,00€100mg747,00€500mg1.513,00€1mL*10mM (DMSO)122,00€Teniloxazine
CAS :Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formule :C16H19NO2SDegré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :289.39Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg39,00€5mg52,00€10mg77,00€25mg110,00€50mg166,00€100mg236,00€200mg349,00€1mL*10mM (DMSO)58,00€SCH-900271
CAS :SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.Formule :C14H16N2O4Degré de pureté :98.82% - 99.93%Couleur et forme :SolidMasse moléculaire :276.29Ref: TM-T34573
1mg112,00€5mg261,00€10mg396,00€25mg655,00€50mg888,00€100mg1.251,00€500mg2.493,00€1mL*10mM (DMSO)249,00€Agomelatine hydrochloride
CAS :Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Formule :C15H18ClNO2Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :279.76CT-179
CAS :CT-179 is a potent and selective inhibitor of OLIG2, reduces tumor cell proliferation and induces apoptosis, fpr medulloblastoma and glioblastoma.Formule :C17H22Cl2N6ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :397.3NNC 05-711
CAS :NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formule :C21H23ClN2O3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :386.87RS 42358-197
CAS :RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formule :C19H23ClN2ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :330.85Ref: TM-T20739
1mg158,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€1mL*10mM (DMSO)349,00€MK-3328
CAS :MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.Formule :C14H9FN4ODegré de pureté :99.77% - >99.99%Couleur et forme :SolidMasse moléculaire :268.25Ref: TM-T16094
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€LY266097 hydrochloride
CAS :LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.
Formule :C21H24Cl2N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :407.33Tribendimidine
CAS :Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.Formule :C28H32N6Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :452.59amyloid P-IN-1
CAS :amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer's disease, amyloidosis, osteoarthritis, andFormule :C30H44N2O14Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :656.68CPCCOEt
CAS :CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1bFormule :C13H13NO4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :247.25Divaplon
CAS :Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formule :C17H17N3O2Degré de pureté :97.44% - 98.25%Couleur et forme :SolidMasse moléculaire :295.34Golexanolone
CAS :Golexanolone can be used to study neurological diseases.Formule :C21H31NO2Degré de pureté :99.90% - 99.99%Couleur et forme :SolidMasse moléculaire :329.48GSK233705
CAS :GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.Formule :C24H29BrN2Degré de pureté :99.87% - 99.98%Couleur et forme :SolidMasse moléculaire :425.4ATC 0175
CAS :ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formule :C23H26ClF2N5ODegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :461.93Pimethixene maleate
CAS :Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Formule :C23H23NO4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :409.5ASM-024
CAS :ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.Formule :C15H25N2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :233.37DMCM hydrochloride
CAS :DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formule :C17H19ClN2O4Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :350.8Ref: TM-T11061
1mg34,00€2mg50,00€5mg80,00€10mg105,00€25mg236,00€50mg439,00€100mg620,00€1mL*10mM (DMSO)88,00€RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36Ricasetron
CAS :Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formule :C19H27N3ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :313.44ABP688
CAS :ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used as a PET tracer for clinical imaging.Formule :C15H16N2ODegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :240.3BPDBA
CAS :BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFormule :C19H20Cl2N2ODegré de pureté :99.43% - 99.95%Couleur et forme :SolidMasse moléculaire :363.28LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :99.78% - 99.97%Couleur et forme :SolidMasse moléculaire :379.455HT6-ligand-1
CAS :5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Formule :C20H22BrN3O2SDegré de pureté :99.24% - 99.93%Couleur et forme :SolidMasse moléculaire :448.38Perphenazine dihydrochloride
CAS :Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formule :C21H28Cl3N3OSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :476.895-HT1A modulator 1
CAS :5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formule :C21H25N3O2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :383.51BMY-14802 hydrochloride
CAS :BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formule :C18H23ClF2N4ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :384.85(Z)-Thiothixene
CAS :(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formule :C23H29N3O2S2Degré de pureté :99.21%Couleur et forme :Yellow To Yellow With A Tan Cast PowderMasse moléculaire :443.63Buntanetap
CAS :Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular diseaseFormule :C20H23N3O2Degré de pureté :98.2%Couleur et forme :SolidMasse moléculaire :337.42Ref: TM-T17312
1mg177,00€5mg447,00€10mg713,00€25mg1.333,00€50mg1.935,00€100mg2.520,00€1mL*10mM (DMSO)492,00€CBiPES hydrochloride
CAS :CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.Formule :C21H20ClN3O2SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :413.92Progabide
CAS :Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.Formule :C17H16ClFN2O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :334.77GR 46611
CAS :GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formule :C23H27N3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :377.48Adoprazine
CAS :Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.
Formule :C24H24FN3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :405.46Xanomeline
CAS :Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.Formule :C14H23N3OSDegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :281.42LRRK2-IN-7
CAS :LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, >1000x selectivity vs kinases/channels/CYPs.Formule :C24H26N6ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :414.5Viloxazine
CAS :Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormule :C13H19NO3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :237.29L 663581
CAS :L 663581 is the benzodiazepine receptor partial agonist.Formule :C17H16ClN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :357.79GABAA receptor agent 2 TFA
CAS :Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.Formule :C22H22F3N3O3Couleur et forme :SolidMasse moléculaire :433.42AAK1-IN-3
CAS :AAK1-IN-3: Brain-penetrant AAK1 inhibitor for neuropathic pain research; IC50=11 nM.Formule :C20H20N4Couleur et forme :SolidMasse moléculaire :316.45-HT3-In-1
CAS :5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formule :C16H21ClN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.82VU6007477
CAS :VU6007477 is a brain-penetrant M1 muscarinic receptor PAM (EC50 230 nM) used for research on CNS exposure and seizure-related models.Formule :C24H26N6O2Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :430.5MAO-B-IN-13
CAS :MAO-B-IN-13: a potent, reversible MAO-B inhibitor with BBB penetration, neuroprotective effects; used in Parkinson’s research (IC50=10nM).Formule :C18H19NO3Couleur et forme :SolidMasse moléculaire :297.35PZ-II-029
CAS :PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Formule :C18H15N3O3Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :321.33Ref: TM-T28479
1mg50,00€5mg105,00€10mg167,00€25mg289,00€50mg447,00€100mg685,00€500mg1.378,00€1mL*10mM (DMSO)192,00€MAO-B-IN-27
CAS :MAO-B-IN-27 (Compound 12c), a monoamine oxidase B (MAO-B) inhibitor, exhibits a potent and selective inhibitory effect on hMAO-B, with an IC50 value of 8.9 nM,Formule :C16H17ClF3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.76Gepirone
CAS :Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.Formule :C19H29N5O2Degré de pureté :99.35% - 99.89%Couleur et forme :SolidMasse moléculaire :359.47GR 125487 sulfamate
CAS :GR 125487 sulfamate is a 5-HT4 receptor antagonist.Formule :C19H29FN4O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.58AChE-IN-31
CAS :AChE-IN-31 (compound 1), a non-competitive acetylcholinesterase (AChE) inhibitor, exhibits potential for Alzheimer's disease research [1].Formule :C27H44Na2O9S2Couleur et forme :SolidMasse moléculaire :622.74AAK1-IN-2
CAS :AAK1-IN-2, a potent (IC50=5.8 nM) AAK1 inhibitor, selective & brain-penetrant, is used for neuropathic pain studies.Formule :C20H20N4Couleur et forme :SolidMasse moléculaire :316.4Muscarine tosylate
CAS :Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].Formule :C16H27NO5SCouleur et forme :SolidMasse moléculaire :345.455-HT2A receptor agonist-3
CAS :5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Formule :C21H26BrNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.34MAO-IN-3
CAS :MAO-IN-3 (Compound 5), a reversible and competitive monoamine oxidase (MAO) inhibitor with inhibition constants (K i) of 0.6 μM for MAO A and 0.2 μM for MAO B,Formule :C42H54N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :678.9PQM130
CAS :PQM130 is a Feruloyl-Donepezil Hybrid compound against the neurotoxicity induced by Aβ1-42 oligomer (AβO) and shows anti-inflammatory activity.Formule :C23H27NO4Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :381.46GYKI-46903 HCl
CAS :GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.Formule :C17H21ClFNO2Couleur et forme :SolidMasse moléculaire :325.814-Chloro-L-phenylalanine
CAS :4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases (TPH1 and TPH2).Formule :C9H10ClNO2Degré de pureté :99.76% - 99.96%Couleur et forme :SolidMasse moléculaire :199.63AChE-IN-19
CAS :AChE-IN-19: strong AChE blocker (IC50: 0.56 μM), hinders Aβ clumps, neuro-protective, non-toxic to SH-SY5Y, for Alzheimer's research.Formule :C30H33NO7Couleur et forme :SolidMasse moléculaire :519.59MIN-117
CAS :MIN-117, a SSRI/5-HT receptor antagonist, is potentially used for the treatment of depression.Formule :C25H26Cl3N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :538.85(-)-Bicuculline methochloride
CAS :(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
Formule :C21H20ClNO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :417.842-Methyl-5-HT
CAS :2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.Formule :C11H14N2ODegré de pureté :97.18%Couleur et forme :SolidMasse moléculaire :190.24Ref: TM-T10075
5mg48,00€10mg84,00€25mg177,00€50mg334,00€100mg500,00€500mg1.099,00€1mL*10mM (DMSO)50,00€LY2033298
CAS :LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.Formule :C13H14ClN3O2SDegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :311.79BACE1-IN-1
CAS :BACE1-IN-1 is a high brain penetrant BACE1 inhibitor (IC50s: 32 and 47 nM for human BACE1 and BACE2).Formule :C18H14F3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.33CGP-54626 free base
CAS :CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Formule :C18H28Cl2NO3PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.3
