récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
940 produits trouvés pour "récepteur 5-HT"
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2-Methyl-N,N-dimethyltryptamine
CAS :<p>2-Methyl-N,N-dimethyltryptamine (2,N,N-TMT, compound 15) exhibits binding affinity for the serotonin (5-HT) receptor, with a pA2 value of 6.04. It plays a significant role in neurological disease research.</p>Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.31,8-Cineole
CAS :<p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>Formule :C10H18ODegré de pureté :97.44% - 97.44%Couleur et forme :SolidMasse moléculaire :154.25LY 344864 racemate
CAS :<p>LY 344864 racemate is a 5-HT1F receptor agonist.</p>Formule :C21H22FN3ODegré de pureté :99.75%Couleur et forme :SoildMasse moléculaire :351.42Dipentylone hydrochloride
CAS :<p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>Formule :C14H20ClNO3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :285.77JPC0323
<p>JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target properties, acceptable plasma exposure, and adequate</p>Formule :C22H43NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.585-HT6R antagonist 1
<p>Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability</p>Formule :C17H22F2N6ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.394-Hydroxy MPT
CAS :<p>4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.</p>Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.324-hydroxy DiPT hydrochloride
CAS :<p>4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.</p>Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.847-Methyl DMT
CAS :<p>7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.</p>Formule :C13H18N2Couleur et forme :SolidMasse moléculaire :202.3PZ-1922
<p>PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.</p>Degré de pureté :98%Couleur et forme :Odour Solid5-MeO-MET
CAS :<p>5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.</p>Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.3225N-NBOMe hydrochloride
CAS :<p>25N-NBOMe hydrochloride is a derivative of 2C-N and acts as an agonist for the 5-HT2A and 5-HT2C receptors, with Ki values of 0.144 nM and 1.06 nM, respectively. It has minimal effect on the release of preloaded neurotransmitters from recombinant dopamine, serotonin, and norepinephrine transporters.</p>Formule :C18H23ClN2O5Couleur et forme :SolidMasse moléculaire :382.844-Bromo-2,5-DMMA
CAS :<p>4-Bromo-2,5-DMMA (Compound 2) demonstrates affinity for the 5-HT2 binding site and has an ED50 of 0.82 mg/kg in rat discrimination experiments.</p>Formule :C12H18BrNO2Couleur et forme :SolidMasse moléculaire :288.18Alosetron-d3
CAS :<p>Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Formule :C17H18N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.3725E-NBOMe hydrochloride
CAS :<p>25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.</p>Formule :C20H28ClNO3Couleur et forme :SolidMasse moléculaire :365.89Galanin (1-15) (porcine, rat)
CAS :<p>N-terminal galanin fragment used to mediate central cardiovascular effects</p>Formule :C72H105N19O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1556.725-HT2A receptor agonist-6
CAS :<p>5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.</p>Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.36MRS7925
<p>MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosis</p>Formule :C20H26IN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.36Peptide 401
CAS :<p>Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.</p>Formule :C110H192N40O24S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2587.22Desmethyl Mirtazapine (hydrochloride)
CAS :<p>Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.</p>Formule :C16H18ClN3Couleur et forme :SolidMasse moléculaire :287.794-Iodoamphetamine hydrochloride
CAS :<p>4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.</p>Formule :C9H13ClINCouleur et forme :SolidMasse moléculaire :297.56Methamnetamine hydrochloride
CAS :<p>Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.</p>Formule :C14H18ClNCouleur et forme :SolidMasse moléculaire :235.755-HT1AR agonist 2
<p>5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.</p>Formule :C31H31N5O3Couleur et forme :SolidMasse moléculaire :521.614-fluoro MBZP
CAS :<p>4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.</p>Formule :C12H17FN2Couleur et forme :SolidMasse moléculaire :208.28LEK 8804
CAS :<p>LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.</p>Formule :C19H19N3OCouleur et forme :SolidMasse moléculaire :305.375-HT6 agonist 1
<p>Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting platelet</p>Formule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37Tabernanthalog
CAS :<p>TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.</p>Formule :C14H18N2ODegré de pureté :99.82% - 99.89%Couleur et forme :SoildMasse moléculaire :230.31Xylamidine
CAS :<p>Xylamidine is a biochemical.</p>Formule :C19H24N2O2Couleur et forme :SolidMasse moléculaire :312.41Minaprine
CAS :<p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>Formule :C17H22N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.386-Fluoro-N,N-diethyltryptamine
CAS :<p>6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.</p>Formule :C14H19FN2Couleur et forme :SolidMasse moléculaire :234.31FFN246
CAS :<p>FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and</p>Formule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27BMY-14802
CAS :<p>BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.</p>Formule :C18H22F2N4ODegré de pureté :99.84%Couleur et forme :SoildMasse moléculaire :348.394-Chloromethamphetamine hydrochloride
CAS :<p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>Formule :C10H15Cl2NCouleur et forme :SolidMasse moléculaire :220.14SB 258585
CAS :<p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>Formule :C18H22IN3O3SDegré de pureté :99.8%Couleur et forme :SoildMasse moléculaire :487.36p-MPPF
CAS :<p>p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.</p>Formule :C25H27FN4O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :434.51Asenapine citrate
CAS :<p>Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).</p>Formule :C23H24ClNO8Couleur et forme :SolidMasse moléculaire :477.89BIMU 8
CAS :<p>BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.</p>Formule :C19H27ClN4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :378.9Tiflucarbine
CAS :<p>Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of soluble</p>Formule :C16H17FN2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :288.38SB 699551
CAS :<p>SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.</p>Formule :C34H45N3ODegré de pureté :99.83%Masse moléculaire :511.74Eletriptan
CAS :<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Formule :C22H26N2O2SCouleur et forme :SolidMasse moléculaire :382.52DOAM
CAS :<p>DOAM is an antagonist of the 5-HT2 receptor.</p>Formule :C16H27NO2Couleur et forme :SolidMasse moléculaire :265.39rac Desmethyl Citalopram Hydrochloride
CAS :<p>rac Desmethyl Citalopram Hydrochloride is a 5-hydroxy tryptamine uptake inhibitor with IC50 value of 0.013 μM.</p>Formule :C19H20ClFN2ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :346.83Naratriptan D3 Hydrochloride
CAS :<p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>Formule :C17H26ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.94Nemifitide diTFA
CAS :<p>Nemifitide diTFA is a synthetic pentapeptide with antidepressant properties, resembling MIF, that crosses the blood-brain barrier.</p>Formule :C37H45F7N10O10Degré de pureté :99.78% - 99.84%Couleur et forme :SolidMasse moléculaire :922.8LP 12 hydrochloride
CAS :<p>LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).</p>Formule :C32H40ClN3OCouleur et forme :SolidMasse moléculaire :518.14Minesapride
CAS :<p>Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.</p>Formule :C21H31ClN4O5Degré de pureté :99.85% - 99.88%Couleur et forme :SolidMasse moléculaire :454.95MR33317
<p>MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.</p>Formule :C22H28ClN3O2Masse moléculaire :401.187PF-03382792
CAS :<p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>Formule :C23H32FN3O4Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :433.524-Hydroxy MET
CAS :<p>4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.</p>Formule :C13H18N2OCouleur et forme :SolidMasse moléculaire :218.3Antipsychotic agent-2
<p>Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.</p>Formule :C22H26FN5OCouleur et forme :SolidMasse moléculaire :395.47Ethylpropyltryptamine
CAS :<p>Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.</p>Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35(R)-Citalopram oxalate
CAS :<p>(R)-Citalopram oxalate is a weak selective serotonin reuptake inhibitor (SSRI) that antagonises its S-isomer (escitalopram), anticonvulsant and antidepressant</p>Formule :C22H23FN2O5Degré de pureté :99.76%Couleur et forme :White SolidMasse moléculaire :414.43SC-53116
CAS :<p>SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.</p>Formule :C16H22ClN3O2Couleur et forme :SolidMasse moléculaire :323.82SB 216641
CAS :<p>SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety disorders and depression.</p>Formule :C28H30N4O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :486.56R 50595
CAS :<p>R 50595 is a selective non-competitive cisapride antagonist.</p>Formule :C30H35Cl2F2N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.52Litoxetine HCl
<p>Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.</p>Formule :C16H20ClNODegré de pureté :99.56% - 99.75%Couleur et forme :SoildMasse moléculaire :277.79Spiroxatrine
CAS :<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Formule :C22H25N3O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :379.45Altanserin
CAS :<p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>Formule :C22H22FN3O2SCouleur et forme :SolidMasse moléculaire :411.49Setiptiline maleate
CAS :<p>Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.</p>Formule :C23H23NO4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :377.43SB-269970 hydrochloride
CAS :<p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits >50-fold selectivity</p>Formule :C18H28N2O3S·HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :388.95Clozapine-d8
CAS :<p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>Formule :C18H19ClN4Couleur et forme :SolidMasse moléculaire :334.87Asenapine hydrochloride
CAS :<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Formule :C17H17Cl2NOCouleur et forme :SolidMasse moléculaire :322.23Cefaclor
CAS :<p>Cefaclor (Panoral) is a cephalosporin antibiotic.</p>Formule :C15H14ClN3O4SDegré de pureté :99.03% - 99.98%Couleur et forme :SolidMasse moléculaire :367.81(R)-Praziquantel-d11
CAS :<p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>Formule :C19H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.47WAY-100635
CAS :<p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>Formule :C25H34N4O2Degré de pureté :98.972%Couleur et forme :SolidMasse moléculaire :422.56Quetiapine-d4 hemifumarate
CAS :<p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>Formule :C25H29N3O6SDegré de pureté :98%Couleur et forme :White SolidMasse moléculaire :503.61Aripiprazole (D8)
CAS :<p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>Formule :C23H27Cl2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.44Nefazodone
CAS :<p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>Formule :C25H32ClN5O2Degré de pureté :99.85%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :470.015-HT3 antagonist 5
CAS :<p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>Formule :C16H13N3O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :279.29Asenapine
CAS :<p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>Formule :C17H16ClNODegré de pureté :99.64%Couleur et forme :CoaMasse moléculaire :285.77Ziprasidone amino acid
CAS :<p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>Formule :C21H23ClN4O2SCouleur et forme :SolidMasse moléculaire :430.954,4-Diphenylbutylamine hydrochloride
CAS :<p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>Formule :C16H20ClNCouleur et forme :SolidMasse moléculaire :261.79Thioridazine
CAS :<p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>Formule :C21H26N2S2Couleur et forme :SolidMasse moléculaire :370.57SB-277011 hydrochloride
CAS :<p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>Formule :C28H31ClN4ODegré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :475.03Agomelatine-d6
CAS :<p>Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.</p>Formule :C15H17NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :249.34Ziprasidone D8
CAS :<p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>Formule :C21H21ClN4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.993-Hydroxy agomelatine D3
CAS :<p>3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).</p>Formule :C15H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.32Olanzapine D3
CAS :<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Formule :C17H20N4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.45Levomepromazine
CAS :<p>Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.</p>Formule :C19H24N2OSDegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :328.47Flibanserin-d4
CAS :<p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>Formule :C20H21F3N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :394.43Tegaserod
CAS :<p>Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).</p>Formule :C16H23N5ODegré de pureté :99.20% - 99.89%Couleur et forme :SolidMasse moléculaire :301.39Paliperidone Palmitate
CAS :<p>Paliperidone: atypical antipsychotic, dopamine & serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>Formule :C39H57FN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :664.89Clothiapine
CAS :<p>Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.</p>Formule :C18H18ClN3SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :343.87BW 723C86
CAS :<p>BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.</p>Formule :C16H19ClN2OSDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :322.855-HT2B antagonist-1
CAS :<p>Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.</p>Formule :C11H14BrN5Degré de pureté :99.965%Couleur et forme :SolidMasse moléculaire :296.171-Phenylbiguanide HCl
CAS :<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Formule :C8H12ClN5Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :213.67Agomelatine (L(+)-Tartaric acid)
CAS :<p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>Formule :C19H23NO8Couleur et forme :SolidMasse moléculaire :393.39Granisetron
CAS :<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.41Eplivanserin (mixture)
CAS :<p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387SB-200646A
CAS :<p>SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.</p>Formule :C15H15ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.763-Hydroxy agomelatine
CAS :<p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>Formule :C15H17NO3Couleur et forme :SolidMasse moléculaire :259.3Sumatriptan
CAS :<p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>Formule :C14H21N3O2SDegré de pureté :99.93%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :295.4cis-(Z)-Flupentixol dihydrochloride
CAS :<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Formule :C23H27Cl2F3N2OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :507.44Alosetron D3 Hydrochloride
CAS :<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Formule :C17H19ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.83Cariprazine D6
CAS :<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Formule :C21H26D6Cl2N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :433.45Dehydroaripiprazole
CAS :<p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>Formule :C23H25Cl2N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :446.37Fluvoxamine
CAS :<p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>Formule :C15H21F3N2O2Couleur et forme :SolidMasse moléculaire :318.33Vilazodone-d8
CAS :<p>Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.</p>Formule :C26H27N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :449.57LY310762
CAS :<p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>Formule :C24H27FN2O2·HClDegré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :430.94Chlorprothixene
CAS :<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86Cyclopiazonic acid
CAS :<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Formule :C20H20N2O3Degré de pureté :99.27% - 99.80%Couleur et forme :SolidMasse moléculaire :336.38m-Chlorophenylbiguanide hydrochloride
CAS :<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Formule :C8H11Cl2N5Degré de pureté :99.43% - 99.87%Couleur et forme :SolidMasse moléculaire :248.11Piperacetazine
CAS :<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Piboserod hydrochloride
CAS :<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Formule :C22H32ClN3O2Couleur et forme :SolidMasse moléculaire :405.96SB 204741
CAS :<p>SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.</p>Formule :C14H14N4OSDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :286.35Buclizine dihydrochloride
CAS :<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Formule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95Tandospirone citrate
CAS :<p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>Formule :C27H37N5O9Degré de pureté :97.84% - 99.90%Couleur et forme :SolidMasse moléculaire :575.61NGB 2904
CAS :<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Formule :C28H29Cl2N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :494.46Zacopride hydrochloride
CAS :<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.265-Benzyloxygramine
CAS :<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Formule :C18H20N2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :280.36N-Desmethylclozapine
CAS :<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.84F 4PP oxalate
CAS :<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formule :C22H26FNO·C2H2O4Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :429.49Sarpogrelate
CAS :<p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>Formule :C24H31NO6Couleur et forme :SolidMasse moléculaire :429.51Spiperone hydrochloride
CAS :<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Formule :C23H27ClFN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.93Harmine hydrochloride
CAS :<p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>Formule :C13H13ClN2ODegré de pureté :99.61% - >99.99%Couleur et forme :Yellow To Slightly Green Crystalline PowderMasse moléculaire :248.71Ondansetron
CAS :<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Formule :C18H19N3ODegré de pureté :99.92%Couleur et forme :White To Yellow CrystalsMasse moléculaire :293.36SB 242084 dihydrochloride
CAS :<p>SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.</p>Formule :C21H21Cl3N4O2Couleur et forme :SolidMasse moléculaire :467.78S1RA hydrochloride
CAS :<p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki ></p>Formule :C20H24ClN3O2Degré de pureté :98% - 99.84%Couleur et forme :SolidMasse moléculaire :373.87SKF-83566
CAS :<p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>Formule :C17H18BrNODegré de pureté :95.00% - 99.82%Couleur et forme :SolidMasse moléculaire :332.23Dasotraline hydrochloride
CAS :<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66ML 10302
CAS :<p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>Formule :C15H21ClN2O3Couleur et forme :SolidMasse moléculaire :312.79SAX-187
CAS :<p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87L-745870 trihydrochloride
CAS :<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21Rotigotine-
CAS :<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Zotepine
CAS :<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Metoclopramide
CAS :<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.80Desvenlafaxine succinate hydrate
CAS :<p>Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).</p>Formule :C20H33NO7Degré de pureté :99.26%Couleur et forme :White Crystalline PowdeMasse moléculaire :399.48Harmine
CAS :<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Formule :C13H12N2ODegré de pureté :98.29% - 99.92%Couleur et forme :Off-White SolidMasse moléculaire :212.25Rotigotine Hydrochloride
CAS :<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.93Ramosetron hydrochloride
CAS :<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formule :C17H18ClN3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :315.8Pergolide mesylate
CAS :<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Formule :C20H30N2O3S2Degré de pureté :99.70%Couleur et forme :White To Off-White SolidMasse moléculaire :410.59Trazodone
CAS :<p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>Formule :C19H22ClN5ODegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.861-(1-Naphthyl) piperazine hydrochloride
CAS :<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Formule :C14H17ClN2Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :248.75A-582941 dihydrochloride
CAS :<p>A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial</p>Formule :C17H22Cl2N4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :353.29Sertindole
CAS :<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Formule :C24H26ClFN4ODegré de pureté :99.87% - 99.92%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :440.94Rizatriptan benzoate
CAS :<p>Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraine</p>Formule :C22H25N5O2Degré de pureté :99% - 99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47PU02
CAS :<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Formule :C16H12N4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :292.36Cinitapride
CAS :<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Formule :C21H30N4O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :402.49Lurasidone hydrochloride
CAS :<p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.</p>Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14Sarpogrelate hydrochloride
CAS :<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formule :C24H32ClNO6Degré de pureté :99.73%Couleur et forme :Colorless LiquidMasse moléculaire :465.97Clozapine N-Oxide
CAS :<p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>Formule :C18H19ClN4ODegré de pureté :98.43% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82Flibanserin hydrochloride
CAS :<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Formule :C20H22ClF3N4OCouleur et forme :SolidMasse moléculaire :426.875-HT1A modulator 2 hydrochloride
CAS :<p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>Formule :C11H16ClNODegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :213.7MK 212 hydrochloride
CAS :<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Formule :C8H11ClN4·HClDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :235.12Eptapirone
CAS :<p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>Formule :C16H23N7O2Degré de pureté :99.39% - 99.65%Couleur et forme :SolidMasse moléculaire :345.4Brexpiprazole HCl
CAS :<p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>Formule :C25H27N3O2S·xHClDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :433.6Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formule :C35H47FN10O8Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :754.85Brexpiprazole
CAS :<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.578-Hydroxy-DPAT hydrobromide
CAS :<p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>Formule :C16H26BrNODegré de pureté :98.90% - 99.09%Couleur et forme :SolidMasse moléculaire :328.29Ansofaxine hydrochloride
CAS :<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Geissoschizine methyl ether
CAS :<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Formule :C22H26N2O3Degré de pureté :99.24% - 99.68%Couleur et forme :SolidMasse moléculaire :366.45Tropisetron
CAS :<p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>Formule :C17H20N2O2Degré de pureté :99.68%Couleur et forme :White SolidMasse moléculaire :284.35Sevoflurane
CAS :<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formule :C4H3F7ODegré de pureté :98%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05SB399885
CAS :<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35LY334370
CAS :<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Formule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42Lurasidone
CAS :<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formule :C28H36N4O2SDegré de pureté :99.78% - 99.91%Couleur et forme :SolidMasse moléculaire :492.68Eltoprazine
CAS :<p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>Formule :C12H16N2O2Couleur et forme :SolidMasse moléculaire :220.27Perospirone
CAS :<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57ARC-239
CAS :<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formule :C24H29N3O3Couleur et forme :SolidMasse moléculaire :407.51VUF 10166
CAS :<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Formule :C13H15ClN4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :262.74(S)-Amisulpride
CAS :<p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>Formule :C17H27N3O4SDegré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :369.48Puerarin
CAS :<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Formule :C21H20O9Degré de pureté :98.90% - 99.21%Couleur et forme :Yellow Brown Fine PowderMasse moléculaire :416.38Nelotanserin
CAS :<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formule :C18H15BrF2N4O2Degré de pureté :98.42% - 99.88%Couleur et forme :SolidMasse moléculaire :437.24S 14506 HCl
CAS :<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Formule :C24H26FN3O2Couleur et forme :SolidMasse moléculaire :407.48RU 24969 free base
CAS :<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.29Azaphen
CAS :<p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>Formule :C16H21Cl2N5ODegré de pureté :97.62%Couleur et forme :SolidMasse moléculaire :370.28Alosetron (Hydrochloride(1:X))
CAS :<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Formule :C17H18ClN4OCouleur et forme :SolidMasse moléculaire :329.11691(E)-3,4,5-Trimethoxycinnamic acid
CAS :<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Formule :C12H14O5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :238.24Loxapine hydrochloride
CAS :<p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>Formule :C18H19Cl2N3OCouleur et forme :SolidMasse moléculaire :364.27Cinanserin
CAS :<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Formule :C20H24N2OSCouleur et forme :SolidMasse moléculaire :340.48Serotonin hydrochloride
CAS :<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Formule :C10H13ClN2ODegré de pureté :98.05% - 99.93%Couleur et forme :White To Cream PowderMasse moléculaire :212.676WAY-100635 Monomaleate
CAS :<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Formule :C25H34N4O2·C4H4O4Degré de pureté :98.44% - 99.46%Couleur et forme :SolidMasse moléculaire :538.64Piboserod
CAS :<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Almotriptan Malate
CAS :<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55Risperidone hydrochloride
CAS :<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Formule :C23H28ClFN4O2Couleur et forme :SolidMasse moléculaire :446.95Ocaperidone
CAS :<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Formule :C24H25FN4O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :420.48Phenylbiguanide
CAS :<p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>Formule :C8H11N5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.21Sumatriptan hydrochloride
CAS :<p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>Formule :C14H22ClN3O2SCouleur et forme :SolidMasse moléculaire :331.86Escitalopram Oxalate
CAS :<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43BRL-15572 hydrochloride
CAS :<p>BRL-15572 hydrochloride: selective h5-HT1D antagonist with high affinity; useful for studying h5-HT1D responses.</p>Formule :C25H28Cl2N2OCouleur et forme :SolidMasse moléculaire :443.414i
CAS :<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74SB 242084
CAS :<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Formule :C21H19ClN4O2Degré de pureté :99.75% - ≥98%Couleur et forme :SolidMasse moléculaire :394.85PNU 22394 hydrochloride
CAS :<p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>Formule :C13H17ClN2Degré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :236.74Amitriptyline
CAS :<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4Pirenperone
CAS :<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formule :C23H24FN3O2Degré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :393.45Quipazine
CAS :<p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>Formule :C13H15N3Couleur et forme :SolidMasse moléculaire :213.28SR 57227 hydrochloride
CAS :<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Formule :C10H14ClN3·HClDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :248.15Ramosetron
CAS :<p>Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。</p>Formule :C17H17N3ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :279.34F-15599
CAS :<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Formule :C19H21ClF2N4ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :394.857-Amino-4-(trifluoromethyl)coumarin
CAS :<p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>Formule :C10H6F3NO2Degré de pureté :97.31% - 97.84%Couleur et forme :Yellow PowderMasse moléculaire :229.16Tiprenolol
CAS :<p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>Formule :C13H21NO2SDegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :255.38BMY 7378 dihydrochloride
CAS :<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42Tandospirone hydrochloride
CAS :<p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>Formule :C21H30ClN5O2Couleur et forme :SolidMasse moléculaire :419.95γ-Mangostin
CAS :<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Formule :C23H24O6Degré de pureté :98.55% - 99.08%Couleur et forme :SolidMasse moléculaire :396.43Xanthotoxol
CAS :<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Formule :C11H6O4Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :202.16TG6-10-1
CAS :<p>TG6-10-1 is an EP2 antagonist.</p>Formule :C23H23F3N2O4Degré de pureté :99.66% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43Cariprazine
CAS :<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formule :C21H32Cl2N4ODegré de pureté :99.68% - 99.87%Couleur et forme :SolidMasse moléculaire :427.41PRX-07034 hydrochloride
CAS :<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formule :C21H29Cl2N3O4SDegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :490.44Aripiprazole monohydrate
CAS :<p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>Formule :C23H29Cl2N3O3Couleur et forme :SolidMasse moléculaire :466.4MDL 100009
CAS :<p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>Formule :C22H28FNO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :373.46
