récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
1025 produits trouvés pour "récepteur 5-HT"
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Tiprenolol
CAS :Tiprenolol is a beta adrenergic receptor antagonist.[1]Formule :C13H21NO2SDegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :255.38Ref: TM-T50081
1mg52,00€1mL*10mM (DMSO)89,00€5mg98,00€10mg146,00€25mg235,00€50mg319,00€100mg447,00€200mg587,00€Geissoschizine methyl ether
CAS :Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formule :C22H26N2O3Degré de pureté :99.24% - 99.68%Couleur et forme :SolidMasse moléculaire :366.45Ref: TM-TN1032
1mg130,00€2mg187,00€5mg319,00€1mL*10mM (DMSO)326,00€10mg485,00€25mg770,00€50mg1.035,00€100mg1.395,00€Tandospirone hydrochloride
CAS :Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.Formule :C21H30ClN5O2Couleur et forme :SolidMasse moléculaire :419.95Vortioxetine
CAS :Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45Ref: TM-T2395
1mL*10mM (DMSO)46,00€10mg48,00€25mg65,00€50mg90,00€100mg117,00€200mg203,00€500mg333,00€1g477,00€γ-Mangostin
CAS :Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Formule :C23H24O6Degré de pureté :98.55% - 99.08%Couleur et forme :SolidMasse moléculaire :396.43Xanthotoxol
CAS :Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formule :C11H6O4Degré de pureté :98.44% - 99.97%Couleur et forme :SolidMasse moléculaire :202.16Tianeptine
CAS :Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formule :C21H25ClN2O4SDegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :436.95Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Aripiprazole monohydrate
CAS :Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formule :C23H29Cl2N3O3Couleur et forme :SolidMasse moléculaire :466.4MDL 100009
CAS :MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formule :C22H28FNO3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :373.46Ref: TM-T22359
1mg99,00€5mg187,00€1mL*10mM (DMSO)222,00€10mg280,00€25mg434,00€50mg585,00€100mg775,00€200mg1.054,00€SB399885
CAS :SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35Ref: TM-T19669
1mg67,00€5mg123,00€1mL*10mM (DMSO)150,00€10mg177,00€25mg291,00€50mg393,00€100mg553,00€200mg743,00€Relenopride hydrochloride
CAS :Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formule :C24H31Cl2FN4O4Couleur et forme :SolidMasse moléculaire :529.43Perospirone
CAS :Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57LY334370
CAS :LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42Clozapine HCl
CAS :Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.Formule :C18H20Cl2N4Couleur et forme :SolidMasse moléculaire :363.29Niaprazine
CAS :Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44Sevoflurane
CAS :Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formule :C4H3F7ODegré de pureté :98%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05Ref: TM-T22425
2mg39,00€5mg54,00€1mL*10mM (DMSO)56,00€10mg75,00€25mg110,00€50mg158,00€100mg226,00€200mg339,00€Piboserod
CAS :Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Ref: TM-T2278
1mg38,00€2mg50,00€5mg84,00€10mg118,00€1mL*10mM (DMSO)120,00€25mg220,00€50mg403,00€100mg582,00€500mg1.198,00€Frovatriptan Succinate
CAS :Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.Formule :C18H25N3O6Couleur et forme :SolidMasse moléculaire :379.41AVN-492
CAS :AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formule :C17H21N5O2SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :359.45Ref: TM-T5179
1mg37,00€2mg50,00€5mg77,00€1mL*10mM (DMSO)85,00€10mg114,00€25mg225,00€50mg335,00€100mg484,00€Methiothepin mesylate
CAS :Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formule :C21H28N2O3S3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :452.65Alprenolol benzoate
CAS :Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formule :C22H29NO4Couleur et forme :SolidMasse moléculaire :371.48lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Naluzotan
CAS :Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formule :C23H38N4O3SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :450.64Dolasetron
CAS :Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formule :C19H20N2O3Degré de pureté :99.84% - 99.86%Couleur et forme :White PowderMasse moléculaire :324.37AC-90179 HCl
CAS :AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formule :C23H31ClN2O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :402.96Escitalopram Oxalate
CAS :Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg90,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€Eltoprazine dihydrochloride
CAS :Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Formule :C12H18Cl2N2O2Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :293.19Indophagolin
CAS :Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Adoprazine hydrochloride
CAS :Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formule :C24H25ClFN3O2Couleur et forme :SolidMasse moléculaire :441.93Nefazodone hydrochloride
CAS :Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formule :C25H33Cl2N5O2Degré de pureté :99% - 99.86%Couleur et forme :White SolidMasse moléculaire :506.47Ref: TM-T3275
5mg47,00€10mg70,00€1mL*10mM (DMSO)77,00€25mg120,00€50mg216,00€100mg325,00€200mg472,00€500mg775,00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formule :C20H23Cl2F2N3O2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :446.32Idalopirdine Hydrochloride
CAS :Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Formule :C20H20ClF5N2ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :434.83Almotriptan Malate
CAS :Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55Anpirtoline free base
CAS :Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formule :C10H13ClN2SCouleur et forme :SolidMasse moléculaire :228.74Naratriptan
CAS :Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formule :C17H25N3O2SDegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :335.47Ref: TM-T8666
1mg39,00€2mg50,00€5mg73,00€1mL*10mM (DMSO)88,00€10mg92,00€25mg166,00€50mg240,00€100mg360,00€SB 204741
CAS :SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formule :C14H14N4OSDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :286.35Ref: TM-T23312
1mg38,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg234,00€50mg439,00€100mg600,00€200mg837,00€Serotonin hydrochloride
CAS :Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formule :C10H13ClN2ODegré de pureté :98.05% - 99.93%Couleur et forme :White To Cream PowderMasse moléculaire :212.676Cerlapirdine hydrochloride
CAS :Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formule :C22H24ClN3O3SCouleur et forme :SolidMasse moléculaire :445.96Cilansetron Hydrochloride
CAS :Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formule :C20H24ClN3O2Couleur et forme :SolidMasse moléculaire :373.88Naratriptan hydrochloride
CAS :Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formule :C17H25N3O2S·HClDegré de pureté :99.17% - 99.93%Couleur et forme :Beige SolidMasse moléculaire :371.93Rizatriptan sulfate
CAS :Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formule :C15H21N5O4SCouleur et forme :SolidMasse moléculaire :367.42Ralmitaront
CAS :Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).Formule :C17H22N4O2Degré de pureté :99.71% - 99.79%Couleur et forme :SolidMasse moléculaire :314.38Ref: TM-T9183
1mg105,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg401,00€25mg668,00€50mg897,00€100mg1.243,00€200mg1.693,00€Mosapride Citrate
CAS :Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formule :C21H25ClFN3O3·C6H8O7Degré de pureté :99.70%Couleur et forme :White PowderMasse moléculaire :614.02Cariprazine
CAS :Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormule :C21H32Cl2N4ODegré de pureté :99.68% - 99.87%Couleur et forme :SolidMasse moléculaire :427.41Ref: TM-T4577
1mg49,00€5mg92,00€1mL*10mM (DMSO)103,00€10mg145,00€25mg281,00€50mg394,00€100mg550,00€200mg780,00€Pipamperone HCl
CAS :Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formule :C21H31ClFN3O2Couleur et forme :SolidMasse moléculaire :411.95Intepirdine
CAS :Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Formule :C19H19N3O2SDegré de pureté :98% - 98.63%Couleur et forme :SolidMasse moléculaire :353.44
