
Récepteur adrénergique
Les récepteurs adrénergiques sont des GPCR activés par les catécholamines, telles que l'adrénaline et la noradrénaline. Ces récepteurs sont classés en sous-types alpha et bêta, chacun jouant un rôle clé dans la régulation du rythme cardiaque, de la pression artérielle et de la réponse de lutte ou de fuite. Les modulateurs des récepteurs adrénergiques sont essentiels dans le traitement des maladies cardiovasculaires, de l'asthme et des troubles anxieux. Chez CymitQuimica, nous offrons une large gamme de modulateurs des récepteurs adrénergiques de haute qualité pour soutenir vos recherches en endocrinologie, pharmacologie cardiovasculaire et réponse au stress.
Sous-catégories appartenant à la catégorie "Récepteur adrénergique"
730 produits trouvés pour "Récepteur adrénergique"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
Bevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9Yohimbine hydrochloride
CAS :Yohimbine hydrochloride (Antagonil) is a plant alkaloid with α-2-adrenergic blocking activity, used as a mydriatic and in the treatment of erectile dysfunction
Formule :C21H27ClN2O3Degré de pureté :99.86% - >99.99%Couleur et forme :Very Slightly Yellow NeedlesMasse moléculaire :390.90ACEPROMAZINE MALEATE
CAS :ACEPROMAZINE MALEATE is a dopamine receptor antagonistFormule :C23H26N2O5SDegré de pureté :98.87% - 99.51%Couleur et forme :Off White Or Yellow Crystalline PowderMasse moléculaire :442.53Brimonidine
CAS :Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.Formule :C11H10BrN5Degré de pureté :99.626%Couleur et forme :Yellow SolidMasse moléculaire :292.13Lofexidine
CAS :Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
Formule :C11H12Cl2N2ODegré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :259.13L755507
CAS :L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).Formule :C30H40N4O6SDegré de pureté :99% - 99.75%Couleur et forme :SolidMasse moléculaire :584.73Doxazosin
CAS :Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formule :C23H25N5O5Degré de pureté :99.47% - 99.87%Couleur et forme :SolidMasse moléculaire :451.48Tulobuterol hydrochloride
CAS :Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.Formule :C12H19Cl2NODegré de pureté :99.24% - >99.99%Couleur et forme :Appearance White Crystalline PowderMasse moléculaire :264.19Salbutamol hemisulfate
CAS :Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.Formule :C13H21NO3H2O4SDegré de pureté :99.35%Couleur et forme :White Or Almost White Odourless PowderMasse moléculaire :576.70RS 100329
CAS :RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formule :C20H25F3N4O3Couleur et forme :SolidMasse moléculaire :426.43Dobutamine
CAS :Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formule :C18H23NO3Couleur et forme :SolidMasse moléculaire :301.38Lidamidine Hydrochloride
CAS :Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.Formule :C11H17ClN4OCouleur et forme :SolidMasse moléculaire :256.73Droxidopa hydrochloride
CAS :Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.Formule :C9H12ClNO5Couleur et forme :SolidMasse moléculaire :249.65Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Ref: TM-T2306
1mL*10mM (DMSO)À demander5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48Phentolamine hydrochloride
CAS :Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].Formule :C17H20ClN3OCouleur et forme :SolidMasse moléculaire :317.82Romifidine hydrochloride
CAS :Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.Formule :C9H10BrClFN3Couleur et forme :SolidMasse moléculaire :294.55Norepinephrine bitartrate salt
CAS :Norepinephrine bitartrate salt is an adrenergic neurotransmitter.Formule :C12H17NO9Degré de pureté :97.32% - 99.97%Couleur et forme :SolidMasse moléculaire :319.27Norepinephrine
CAS :Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.Formule :C8H11NO3Degré de pureté :99.66% - 99.84%Couleur et forme :Colorless Microcrystals SolidMasse moléculaire :169.18Bunazosin
CAS :Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].Formule :C19H27N5O3Couleur et forme :SolidMasse moléculaire :373.45Nifenalol
CAS :Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.Formule :C11H16N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :224.26Reboxetine mesylate
CAS :Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).Formule :C19H23NO3·CH4O3SDegré de pureté :99.18% - 99.87%Couleur et forme :Tan Or Off-White Cyrstalline SolidMasse moléculaire :409.5Piribedil hydrochloride
CAS :Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.Formule :C16H19ClN4O2Couleur et forme :SolidMasse moléculaire :334.8Apraclonidine
CAS :Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Formule :C9H10Cl2N4Couleur et forme :SolidMasse moléculaire :245.11Napitane Mesylate
CAS :Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Formule :C23H29NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :431.55Xamoterol
CAS :Xamoterol is a cardiac stimulant.Formule :C16H25N3O5Couleur et forme :SolidMasse moléculaire :339.39Methyldopa hydrate
CAS :Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formule :C10H13NO4H2ODegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :238.24Pimozide
CAS :Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formule :C28H29F2N3ODegré de pureté :99.63% - >99.99%Couleur et forme :SolidMasse moléculaire :461.55Desipramine
CAS :Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.Formule :C18H22N2Couleur et forme :SolidMasse moléculaire :266.38Medetomidine hydrochloride
CAS :Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.Formule :C13H16N2·HClDegré de pureté :99.96%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.74Scopine
CAS :Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.Formule :C8H13NO2Degré de pureté :99.79% - >99.99%Couleur et forme :SolidMasse moléculaire :155.19Ref: TM-T6662
5mg47,00€1mL*10mM (DMSO)50,00€10mg71,00€25mg108,00€50mg166,00€100mg280,00€200mg419,00€500mg672,00€Bevantolol
CAS :Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formule :C20H27NO4Couleur et forme :SolidMasse moléculaire :345.43Eformoterol Hemifumarate
CAS :Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthmaFormule :C19H24N2O4C4H4O4Degré de pureté :99.86% - >99.99%Couleur et forme :White PowderMasse moléculaire :402.4Dexmedetomidine
CAS :Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formule :C13H16N2Degré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :200.28Bretylium tosylate
CAS :Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.Formule :C18H24BrNO3SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :414.36Ref: TM-T7386
2mg42,00€5mg62,00€1mL*10mM (DMSO)67,00€10mg94,00€25mg111,00€50mg140,00€100mg167,00€200mg249,00€Phenylephrine
CAS :Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).Formule :C9H13NO2Degré de pureté :99.5% - 99.89%Couleur et forme :SolidMasse moléculaire :167.21Talinolol
CAS :(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formule :C20H33N3O3Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :363.49Ref: TM-T21640
2mg34,00€5mg52,00€1mL*10mM (DMSO)52,00€10mg92,00€25mg178,00€50mg313,00€100mg535,00€200mg775,00€Isoetharine mesylate salt
CAS :Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formule :C14H25NO6SDegré de pureté :99.35% - 99.75%Couleur et forme :SolidMasse moléculaire :335.42Betaxolol
CAS :Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formule :C18H29NO3Degré de pureté :99.01%Couleur et forme :White Crystalline SolidMasse moléculaire :307.43Droxidopa
CAS :Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formule :C9H11NO5Degré de pureté :97.27% - 99.88%Couleur et forme :SolidMasse moléculaire :213.19Higenamine hydrochloride
CAS :Higenamine HCl is a β2 adrenoreceptor agonist active in fat and muscle tissue.Formule :C16H18ClNO3Degré de pureté :99.44% - 99.80%Couleur et forme :White PowderMasse moléculaire :307.772Amezinium methylsulfate
CAS :Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.Formule :C12H15N3O5SDegré de pureté :99.64% - 99.99%Couleur et forme :SolidMasse moléculaire :313.33Levobetaxolol hydrochloride
CAS :Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.Formule :C18H29NO3·HClDegré de pureté :98.80% - 99.69%Couleur et forme :SolidMasse moléculaire :343.89Meranzin
CAS :Meranzin, a bioactive from TCM CSS, targets alpha 2-adrenoceptor, affects AMPA-ERK1/2–BDNF pathway, and may prevent atherosclerosis and depression.Formule :C15H16O4Degré de pureté :95.08% - 99.3%Couleur et forme :SolidMasse moléculaire :260.29(R)-Propranolol hydrochloride
CAS :(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.Formule :C16H22ClNO2Degré de pureté :98.63% - 99.01%Couleur et forme :SolidMasse moléculaire :295.8Naftopidil dihydrochloride
CAS :Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formule :C24H28N2O3·2HClDegré de pureté :99.76%Couleur et forme :White SolidMasse moléculaire :465.41Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Carbazochrome
CAS :Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.Formule :C10H12N4O3Degré de pureté :98.36%Couleur et forme :Nacarat Crystalline PowderMasse moléculaire :236.23Salmeterol Xinafoate
CAS :Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formule :C36H45NO7Degré de pureté :98% - 98.24%Couleur et forme :White SolidMasse moléculaire :603.75Rilmenidine Phosphate
CAS :Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.Formule :C10H19N2O5PDegré de pureté :99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :278.24Ref: TM-T6641
1mg34,00€5mg67,00€1mL*10mM (DMSO)67,00€10mg93,00€25mg152,00€50mg230,00€100mg363,00€200mg528,00€Terazosin hydrochloride dihydrate
CAS :Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formule :C19H25N5O4·HCl·2H2ODegré de pureté :99.81%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :459.92Levalbuterol tartrate
CAS :Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Formule :C17H27NO9Degré de pureté :99.28% - 99.98%Couleur et forme :SolidMasse moléculaire :389.39Ref: TM-T7164
2mg34,00€5mg50,00€1mL*10mM (DMSO)60,00€10mg88,00€25mg100,00€50mg124,00€100mg177,00€200mg259,00€Rauwolscine hydrochloride
CAS :Rauwolscine HCl, a natural α2-adrenergic antagonist (Ki: 12 nM) & weak 5-HT1A agonist, also blocks 5-HT2B (Ki: 14.3 nM), affects mood/behavior.Formule :C21H27ClN2O3Degré de pureté :99.86% - 99.95%Couleur et forme :White SolidMasse moléculaire :390.9Bucindolol hydrochloride
CAS :Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Formule :C22H26ClN3O2Couleur et forme :SolidMasse moléculaire :399.91Idazoxan hydrochloride
CAS :Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.Formule :C11H12N2O2·HClDegré de pureté :99.42% - 99.84%Couleur et forme :SolidMasse moléculaire :240.69Ref: TM-T0115
2mg34,00€5mg49,00€1mL*10mM (DMSO)52,00€10mg73,00€25mg126,00€50mg177,00€100mg266,00€200mg394,00€Fipamezole HCl
CAS :Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.Formule :C14H16ClFN2Couleur et forme :SolidMasse moléculaire :266.74Tolazoline
CAS :Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formule :C10H12N2Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :160.22Dexmedetomidine hydrochloride
CAS :Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Formule :C13H16N2·HClDegré de pureté :99.94% - 99.94%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :236.74Ref: TM-T6466
5mg39,00€10mg52,00€1mL*10mM (DMSO)52,00€25mg94,00€50mg150,00€100mg215,00€200mg323,00€500mg533,00€Bucindolol
CAS :Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.Formule :C22H25N3O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :363.45CGP 20712 A
CAS :CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formule :C24H29F3N4O8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :590.57Medetomidine
CAS :Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formule :C13H16N2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :200.28Ref: TM-T21492
2mg38,00€5mg57,00€1mL*10mM (DMSO)62,00€10mg77,00€25mg128,00€50mg193,00€100mg290,00€200mg447,00€Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Fenoterol hydrobromide
CAS :Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formule :C17H22BrNO4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :384.27Tamsulosin
CAS :Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.Formule :C20H28N2O5SDegré de pureté :99.93%Couleur et forme :White CrystalsMasse moléculaire :408.51Alfuzosin
CAS :Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formule :C19H27N5O4Degré de pureté :99.64%Couleur et forme :White Crystaline PowderMasse moléculaire :389.45Atipamezole
CAS :Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formule :C14H16N2Degré de pureté :99.88%Couleur et forme :Off-White To Light Yellow Crystal PowderMasse moléculaire :212.29SR59230A hydrochloride
CAS :SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formule :C21H28ClNO2Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :361.91Buflomedil
CAS :Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.Formule :C17H25NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.38DL-Phenylephrine HCl
CAS :DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.Formule :C9H14ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :203.67PF-610355
CAS :PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.
Formule :C34H39N3O6SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :617.76Tulobuterol
CAS :Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.Formule :C12H18ClNOCouleur et forme :Crystalline SolidMasse moléculaire :227.73(RS)-ICI-118551 Hydrochloride
CAS :ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3Formule :C17H27NO2·HClDegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :313.86Amidephrine
CAS :Amidephrine is an adrenergic agent.Formule :C10H16N2O3SCouleur et forme :SolidMasse moléculaire :244.31Isoproterenol sulfate anhydrous
CAS :Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.Formule :C22H36N2O10SDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :520.59Ridazolol HCl
CAS :Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.Formule :C15H19Cl3N4O3Degré de pureté :99.48%Couleur et forme :SoildMasse moléculaire :409.7Amidephrine hydrochloride
CAS :Amidephrine hydrochloride is a biochemical.Formule :C10H17ClN2O3SCouleur et forme :SolidMasse moléculaire :280.77Pardoprunox
CAS :Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27Penbutolol sulfate
CAS :Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.Formule :C18H29NO2H2O4SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :340.47Esmolol hydrochloride
CAS :Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension.Formule :C16H25NO4·HClDegré de pureté :98.72% - 99.48%Couleur et forme :White SolidMasse moléculaire :331.15Atenolol Hydrochloride
CAS :Atenolol Hydrochloride is a selective antagonist of ß1 receptor.Formule :C14H23ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.80Bethanidine sulfate
CAS :Bethanidine sulfate and its ortho-chloro derivative (BW 392C60) are potent adrenergic neuron blockers exhibiting sympathomimetic effects similar to those of bromobenzamine and guanethidine in various animal models, particularly in cats. These compounds inhibit the release of norepinephrine during neural stimulation and enhance the responsiveness of smooth muscle to epinephrine and norepinephrine. Notably, bethanidine sulfate increases the pressor response to tyramine, although this effect diminishes with higher doses. Unlike guanethidine, bethanidine sulfate does not deplete pressor amines in the iris of cats following administration. Additionally, it temporarily suppresses autonomic cholinergic mechanisms and can cause transient neuromuscular paralysis at large doses, contrasting its long-term adrenergic neuron blocking effects.Formule :C20H32N6O4SCouleur et forme :SolidMasse moléculaire :452.57Norreticuline
CAS :Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.Formule :C18H21NO4Couleur et forme :SolidMasse moléculaire :315.36LY 344864
CAS :LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formule :C21H22FN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.42Talsupram hydrochloride
CAS :noradrenalin re-uptake inhibitorFormule :C20H26ClNSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.95Bambuterol
CAS :long acting beta-adrenoceptor agonistFormule :C18H29N3O5Degré de pureté :98%Couleur et forme :Off-White PowderMasse moléculaire :367.44Landiolol
CAS :Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.Formule :C25H39N3O8Degré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :509.59D2343
CAS :D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.Formule :C20H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.43Salmefamol
CAS :Salmefamol is a beta-adrenergic agonist. It may also be used as a bronchodilator.Formule :C19H25NO4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :331.41Efaroxan hydrochloride
CAS :Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.Formule :C13H17ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :252.74Protokylol hydrochloride
CAS :Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.Formule :C18H22ClNO5Couleur et forme :SolidMasse moléculaire :367.83Clonidine
CAS :Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.Formule :C9H9Cl2N3Degré de pureté :99.42% - 99.44%Couleur et forme :Crystals SolidMasse moléculaire :230.09BRL 44408 Maleate Salt
CAS :BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.Formule :C17H21N3O4Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :331.37Butaxamine
CAS :Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.Formule :C15H25NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :267.36Lusaperidone
CAS :Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.Formule :C22H21N3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :359.42IMTPPE
CAS :IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.Formule :C20H27N3O2SCouleur et forme :SolidMasse moléculaire :373.51Abanoquil
CAS :Abanoquil is an antagonist of alpha-1 adrenoceptor.Formule :C22H25N3O4Couleur et forme :SolidMasse moléculaire :395.45Zinterol
CAS :Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).Formule :C19H26N2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :378.49Metoprolol fumarate
CAS :Metoprolol fumarate (CGP 2175C): selective β1-blocker with anti-inflammatory, antitumor, anti-angiogenic effects.Formule :C34H54N2O10Couleur et forme :SolidMasse moléculaire :650.8Clenproperol
CAS :Clenproperol is a β2-adrenergic agonist.Formule :C11H16Cl2N2OCouleur et forme :SolidMasse moléculaire :263.16Isoetharine
CAS :Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.Formule :C13H21NO3Couleur et forme :SolidMasse moléculaire :239.31
