Sérine protéase
Les inhibiteurs de protéases à sérine sont des composés qui ciblent et inhibent les protéases à sérine, un groupe d'enzymes caractérisées par un résidu de sérine dans leur site actif. Ces protéases sont impliquées dans de nombreux processus physiologiques, notamment la digestion, la réponse immunitaire, la coagulation sanguine et l'inflammation. Les inhibiteurs de protéases à sérine sont essentiels pour étudier les maladies où ces enzymes sont dysrégulées, telles que les maladies cardiovasculaires, le cancer et les affections inflammatoires. Chez CymitQuimica, nous proposons des inhibiteurs de protéases à sérine pour soutenir vos recherches en enzymologie, mécanismes des maladies et interventions thérapeutiques.
55 produits trouvés pour "Sérine protéase"
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TAO Kinase inhibitor 2
CAS :<p>TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.</p>Formule :C25H24N2O3Degré de pureté :98.58%Couleur et forme :SoildMasse moléculaire :400.47BAY-85-8501
CAS :BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Formule :C22H17F3N4O3SDegré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :474.46Ref: TM-T12613L
1mg96,00€2mg128,00€5mg212,00€10mg314,00€25mg565,00€50mg792,00€100mg1.093,00€1mL*10mM (DMSO)220,00€C1 Esterase Inhibitor (Human)
C1 Esterase Inhibitor (Human) is a glycoprotein derived from human plasma and acts as a serine protease inhibitor. It inactivates enzymes like C1r, C1s, and mannose-binding lectin-associated serine proteases (MASP) through covalent binding. This compound possesses anti-inflammatory properties and is utilized to prevent angioedema attacks associated with hereditary angioedema.Couleur et forme :Odour LiquidRecombinant Trypsin
Recombinant Trypsin is a serine protease that hydrolyzes proteins at the carboxyl side of lysine or arginine.Activated Protein C (390-404), human
CAS :Human Activated Protein C (390-404) peptide derived from serine protease, suppresses APC anticoagulation.Formule :C91H130N22O23Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1900.14α-Methyl-DL-aspartic acid
CAS :α-Methyl-DL-aspartic acid specifically inhibits argininosuccinate synthase (ASS), the rate-limiting enzyme in 1-citrulline-to-1-arginine recycling.Formule :C5H9NO4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :147.13Lonodelestat TFA
Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.Formule :C73H112F3N15O21Couleur et forme :SolidMasse moléculaire :1592.75Protease Inhibitor Library
A unique collection of 343 protease and proteasome inhibitors for research in chemical genomics, and drug screening;Couleur et forme :Odour SolidRef: TM-L1100
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderDansyl-Glu-Gly-Arg-Chloromethylketone
CAS :Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activatedFormule :C26H36ClN7O7SCouleur et forme :SolidMasse moléculaire :626.12Ala-Phe-Pro-pNA TFA
Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.Couleur et forme :Odour SolidSFTI-1
CAS :SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.Formule :C67H104N18O18S2Couleur et forme :SolidMasse moléculaire :1513.78α 1 Antichymotrypsin, Human Plasma
CAS :Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.Couleur et forme :SolidTilpisertib fosmecarbil TFA
CAS :Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.Formule :C37H37ClF3N8O9PCouleur et forme :SolidMasse moléculaire :861.16Roseltide rT1
CAS :Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.Formule :C110H177N31O31S6Couleur et forme :SolidMasse moléculaire :2622.16KKI-5
CAS :<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Formule :C35H55N11O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :773.88Tiprelestat
CAS :<p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>Formule :C254H416N72O75S10Couleur et forme :SolidMasse moléculaire :5999.09MeOSuc-AAPA-CMK
MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].Formule :C20H31ClN4O8Couleur et forme :SolidMasse moléculaire :490.94Suc-AAP-Abu-pNA
CAS :Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Formule :C25H34N6O9Couleur et forme :SolidMasse moléculaire :562.57Chymotrypsinogen
CAS :Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .Couleur et forme :SolidPhosphorylase Kinase β-Subunit Fragment (420-436)
CAS :Phosphorylase Kinase β-Subunit Fragment (420-436) is a peptide fragment (430-436) derived from the β-Subunit of phosphorylase kinase.Formule :C79H131N31O25SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1947.14
