Récepteur de l'histamine
Les récepteurs de l'histamine sont des GPCR qui médiatisent les effets de l'histamine, une amine biogène impliquée dans les réponses immunitaires, la sécrétion d'acide gastrique et la neurotransmission. Il existe quatre sous-types de récepteurs de l'histamine (H1, H2, H3 et H4), chacun jouant des rôles distincts dans les réactions allergiques, la fonction gastrique et l'activité du système nerveux central. Les antagonistes des récepteurs de l'histamine sont largement utilisés dans le traitement des allergies, des ulcères gastriques et du mal des transports. Chez CymitQuimica, nous offrons une sélection complète de modulateurs de récepteurs de l'histamine de haute qualité pour soutenir vos recherches en immunologie, gastroentérologie et neuropharmacologie.
385 produits trouvés pour "Récepteur de l'histamine"
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Triprolidine hydrochloride
CAS :Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formule :C19H23ClN2Couleur et forme :SolidMasse moléculaire :314.852Triprolidine
CAS :Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.Formule :C19H22N2Couleur et forme :SolidMasse moléculaire :278.39GSK189254A
CAS :GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).Formule :C21H25N3O2Degré de pureté :98.71% - 99.858%Couleur et forme :SolidMasse moléculaire :351.44Ref: TM-TQ0066
1mg50,00€1mL*10mM (DMSO)64,00€5mg84,00€10mg114,00€25mg205,00€50mg333,00€100mg477,00€200mg690,00€Osthole
CAS :Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.Formule :C15H16O3Degré de pureté :99.93% - 99.96%Couleur et forme :Fine White PowderMasse moléculaire :244.29Betazole
CAS :Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.Formule :C5H9N3Couleur et forme :SolidMasse moléculaire :111.15Betazole dihydrochloride
CAS :Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.Formule :C5H11Cl2N3Degré de pureté :99.12%Couleur et forme :SolidMasse moléculaire :184.067Ref: TM-T8599
1mg34,00€5mg57,00€1mL*10mM (DMSO)57,00€10mg90,00€25mg167,00€50mg290,00€100mg378,00€200mg538,00€Mequitazine
CAS :Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formule :C20H22N2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :322.47Ciproxifan maleate
CAS :Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormule :C20H22N2O6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :386.4Ref: TM-T2004
1mg40,00€2mg52,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg101,00€25mg205,00€50mg380,00€100mg565,00€Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77Mecamylamine hydrochloride
CAS :Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formule :C11H22ClNDegré de pureté :99.76% - >99.99%Couleur et forme :White SolidMasse moléculaire :203.75JNJ-7777120
CAS :JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.Formule :C14H16ClN3ODegré de pureté :99.83% - 99.96%Couleur et forme :SolidMasse moléculaire :277.75Chlorcyclizine
CAS :CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formule :C18H21ClN2Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :300.83Chlorprothixene
CAS :Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86VUF10460
CAS :VUF10460 is a non-imidazole histamine H4 receptor agonist.Formule :C15H19N5Degré de pureté :99.44% - 99.57%Couleur et forme :SolidMasse moléculaire :269.34Dimaprit dihydrochloride
CAS :Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formule :C6H15N3S·2HClDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :234.19Talastine HCl
CAS :Talastine is an antihistamine drug.Formule :C19H22ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :343.86C-Type Natriuretic Peptide (CNP) (1-22), human
CAS :C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Formule :C93H157N27O28S3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :2197.6Ref: TM-TP1187
500µg84,00€1mg113,00€5mg391,00€10mg623,00€25mg895,00€50mg1.198,00€100mg1.611,00€200mg2.152,00€Tiaramide hydrochloride
CAS :Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Formule :C15H19Cl2N3O3SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :392.3Ref: TM-T28972
1mg66,00€5mg130,00€1mL*10mM (DMSO)137,00€10mg177,00€25mg299,00€50mg447,00€100mg623,00€200mg882,00€Tribenoside
CAS :Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Formule :C29H34O6Degré de pureté :≥98%Couleur et forme :LiquidMasse moléculaire :478.58cicloprofen
CAS :cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formule :C16H14O2Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :238.2812Ref: TM-T8586
1mg58,00€1mL*10mM (DMSO)105,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€Acitazanolast
CAS :Acitazanolast (WP-871) is an anti-allergic drug candidate.Formule :C9H7N5O3Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :233.182-Pyridylethylamine dihydrochloride
CAS :2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Formule :C7H12Cl2N2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :195.09Decloxizine
CAS :Decloxizine is a H1 receptor antagonistFormule :C21H28N2O2Degré de pureté :99.53%Couleur et forme :White Or Similar To White PowderMasse moléculaire :340.46Zotepine
CAS :Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Pemirolast
CAS :Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formule :C10H8N6OCouleur et forme :SolidMasse moléculaire :228.21Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3Antazoline
CAS :Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formule :C17H19N3Degré de pureté :≥95%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :265.35Psoralenoside
CAS :Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Formule :C17H18O9Degré de pureté :99.03% - 99.49%Couleur et forme :SolidMasse moléculaire :366.32Ref: TM-TN1008
1mg90,00€2mg132,00€5mg215,00€1mL*10mM (DMSO)222,00€10mg344,00€25mg568,00€50mg800,00€100mg1.063,00€Betahistine EP Impurity C
CAS :Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formule :C15H19N3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :241.33Dioxopromethazine hydrochloride
CAS :Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formule :C17H20N2O2S·HClDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :352.88Betahistine
CAS :Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formule :C8H12N2Degré de pureté :99.87% - 99.87%Couleur et forme :Yellowish Liquid Liquid LiquidMasse moléculaire :136.19Buclizine dihydrochloride
CAS :Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormule :C28H33ClN2·2HClDegré de pureté :98.05%Couleur et forme :Off-White PowderMasse moléculaire :505.95S 38093
CAS :S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Formule :C17H24N2O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :288.38Ref: TM-T4099
2mg35,00€5mg50,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg124,00€50mg198,00€100mg316,00€200mg442,00€Dioxopromethazine
CAS :Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Formule :C17H20N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :316.42Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Formule :C14H20F6N4O7Degré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :470.32Decloxizine dihydrochloride
CAS :Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Formule :C21H28N2O2·2ClHDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :413.39Histamine Phosphate
CAS :Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Formule :C5H9N·2H3O4PDegré de pureté :>99.99%Couleur et forme :White Crystal PowderMasse moléculaire :307.14Alginic acid
CAS :Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Formule :C14H22O13Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :398.317Betahistine dihydrochloride
CAS :Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formule :C8H14Cl2N2Degré de pureté :99.22% - 99.88%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :209.12Thonzylamine
CAS :Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formule :C16H22N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :286.37Alimemazine hemitartrate
CAS :Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formule :C18H22N2SC4H6O6Degré de pureté :98.16% - 99.69%Couleur et forme :SolidMasse moléculaire :448.53JNJ-5207852
CAS :JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formule :C20H32N2ODegré de pureté :97.19%Couleur et forme :SolidMasse moléculaire :316.48LML134
CAS :LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formule :C19H29N5O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :375.47Ref: TM-T8514
1mg34,00€5mg78,00€1mL*10mM (DMSO)86,00€10mg112,00€25mg203,00€50mg299,00€100mg447,00€200mg600,00€S 38093 HCl
CAS :S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formule :C17H25ClN2O2Degré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :324.85Ref: TM-T4087
1mg37,00€5mg71,00€1mL*10mM (DMSO)71,00€10mg92,00€25mg164,00€50mg225,00€100mg323,00€200mg437,00€Hydroxyzine dihydrochloride
CAS :Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formule :C21H27ClN2O2·2HClDegré de pureté :99.46% - 99.79%Couleur et forme :Oil PowderMasse moléculaire :447.83OXOMEMAZINE
CAS :Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formule :C18H22N2O2SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :330.44Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Bepotastine
CAS :Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Formule :C21H25ClN2O3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :388.89Ref: TM-T7893
2mg34,00€5mg50,00€1mL*10mM (DMSO)56,00€10mg78,00€25mg141,00€50mg205,00€100mg313,00€200mg464,00€Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Levocetirizine Dihydrochloride
CAS :Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Formule :C21H27Cl3N2O3Degré de pureté :99.89%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :461.81
