
Récepteur de la dopamine
Les récepteurs de la dopamine sont un groupe de récepteurs couplés aux protéines G (GPCR) qui répondent au neurotransmetteur dopamine, jouant un rôle clé dans la régulation du mouvement, de la motivation, de la récompense et de plusieurs fonctions cognitives. Ces récepteurs sont divisés en familles de type D1 et de type D2, chacune ayant des fonctions et des profils pharmacologiques distincts. Les modulateurs des récepteurs de la dopamine sont largement étudiés pour leurs applications dans le traitement de la maladie de Parkinson, de la schizophrénie, de la dépendance et d'autres troubles neuropsychiatriques. Chez CymitQuimica, nous offrons une large gamme de modulateurs de récepteurs de la dopamine de haute qualité pour soutenir vos recherches en neurosciences, santé mentale et signalisation GPCR.
407 produits trouvés pour "Récepteur de la dopamine"
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Bromopride
CAS :<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formule :C14H22BrN3O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :344.25Oxidopamine hydrobromide
CAS :<p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>Formule :C8H12BrNO3Degré de pureté :98.22% - 99.88%Couleur et forme :Beige To Brown Fine Crystalline PowderMasse moléculaire :250.09NEO 376
CAS :<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formule :C20H24ClN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :357.88GR 103691
CAS :<p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>Formule :C30H35N3O3Degré de pureté :98.94% - 99.29%Couleur et forme :SolidMasse moléculaire :485.62Bromperidol
CAS :<p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>Formule :C21H23BrFNO2Degré de pureté :99.89%Couleur et forme :Tan SolidMasse moléculaire :420.32Quetiapine hemifumarate
CAS :<p>Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.</p>Formule :C46H54N6O8S2Degré de pureté :99.32% - >99.99%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Prochlorperazine Maleate
CAS :<p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>Formule :C28H32ClN3O8SDegré de pureté :99.78%Couleur et forme :Off-White PowderMasse moléculaire :606.09Tiapride hydrochloride
CAS :<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formule :C15H24N2O4S·HClDegré de pureté :99.4% - 99.77%Couleur et forme :SolidMasse moléculaire :364.89L-DOPA
CAS :<p>L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.</p>Formule :C9H11NO4Degré de pureté :98.99% - 99.93%Couleur et forme :Colorless To White Crystals Or Crystalline Powder; Needles From Water SolidMasse moléculaire :197.19Ziprasidone hydrochloride
CAS :<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Formule :C21H22CL2N4OSDegré de pureté :97.97% - 99.82%Couleur et forme :SolidMasse moléculaire :449.4Thioridazine hydrochloride
CAS :<p>Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4</p>Formule :C21H27ClN2S2Degré de pureté :99.55% - 99.957%Couleur et forme :White To Off-White SolidMasse moléculaire :407.04Metoclopramide hydrochloride
CAS :<p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>Formule :C14H22ClN3O2·HClDegré de pureté :99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :336.26Quetiapine
CAS :<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formule :C21H25N3O2SDegré de pureté :99.14% - 99.63%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :383.51Sulpiride
CAS :<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Formule :C15H23N3O4SDegré de pureté :99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Amisulpride
CAS :<p>Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.</p>Formule :C17H27N3O4SDegré de pureté :99.97%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :369.48L-741626
CAS :<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Formule :C20H21ClN2ODegré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :340.85Ziprasidone
CAS :<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formule :C21H21ClN4OSDegré de pureté :99.55%Couleur et forme :Tan SolidMasse moléculaire :412.94Dexpramipexole dihydrochloride
CAS :<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Formule :C10H19Cl2N3SDegré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :284.25Flunarizine dihydrochloride
CAS :<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42Tipepidine hydrochloride
CAS :<p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>Formule :C15H18ClNS2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :311.89Blonanserin
CAS :<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.5Levosulpiride
CAS :<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Formule :C15H23N3O4SDegré de pureté :98.20% - 99.88%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Mefexamide hydrochloride
CAS :<p>Mefexamide hydrochloride is a central stimulant.</p>Formule :C15H25ClN2O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :316.83Ziprasidone hydrochloride monohydrate
CAS :<p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>Formule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12Loxapine succinate
CAS :<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.9Tetrahydropalmatine
CAS :<p>Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic</p>Formule :C21H25NO4Degré de pureté :99.59% - 99.95%Couleur et forme :SolidMasse moléculaire :355.43Talipexole dihydrochloride
CAS :<p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>Formule :C10H17Cl2N3SDegré de pureté :99.89%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Benserazide hydrochloride
CAS :<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Formule :C10H15N3O5·HClDegré de pureté :98.63% - 99.74%Couleur et forme :White Crystalline SolidMasse moléculaire :293.7BP 897 hydrochloride
CAS :<p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>Formule :C26H32ClN3O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :454Pipamperone
CAS :<p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>Formule :C21H30FN3O2Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :375.48Chlorprothixene hydrochloride
CAS :<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Formule :C18H18ClNS·HClDegré de pureté :99.76%Couleur et forme :White PowderMasse moléculaire :352.32Promazine hydrochloride
CAS :<p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>Formule :C17H21ClN2SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :320.88Ro 10-5824 dihydrochloride
CAS :<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Formule :C17H22Cl2N4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :353.29Fosopamine(HCl)
CAS :<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Formule :C9H15ClNO5PDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :283.65Domperidone
CAS :<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formule :C22H24ClN5O2Degré de pureté :98% - 99.82%Couleur et forme :SolidMasse moléculaire :425.91Talquetamab
CAS :<p>Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.</p>Couleur et forme :LiquidMasse moléculaire :144.59 kDaItopride hydrochloride
CAS :<p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9Oxidopamine hydrochloride
CAS :<p>Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.</p>Formule :C8H12ClNO3Degré de pureté :98.34% - 99.85%Couleur et forme :Physical Description Beige Solid (Ntp 1992)Masse moléculaire :205.64Benztropine mesylate
CAS :<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Paliperidone
CAS :<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Bendazol
CAS :<p>Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.</p>Formule :C14H12N2Degré de pureté :98.7% - 99.87%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :208.26Pericyazine
CAS :<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formule :C21H23N3OSDegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :365.49Tetrabenazine
CAS :<p>Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.</p>Formule :C19H27NO3Degré de pureté :98% - 99.91%Couleur et forme :White To Off-White White To Off-White SolidMasse moléculaire :317.42Perphenazine
CAS :<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.99%Couleur et forme :SolidMasse moléculaire :403.97Clozapine
CAS :<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formule :C18H19ClN4Degré de pureté :99.91% - 99.93%Couleur et forme :Yellow Crystals From Acetone-Petroleum Ether SolidMasse moléculaire :326.82Olanzapine
CAS :<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Formule :C17H20N4SDegré de pureté :99.86% - ≥95%Couleur et forme :Yellowish Crystalline PowderMasse moléculaire :312.43Acetophenazine dimaleate
CAS :<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Formule :C31H37N3O10SDegré de pureté :99.39% - 99.48%Couleur et forme :SolidMasse moléculaire :643.71Pramipexole
CAS :<p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>Formule :C10H17N3SDegré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :211.33Iloperidone
CAS :<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.48Dopamine hydrochloride
CAS :<p>Dopamine hydrochloride (ASL279) is a natural catecholamine neurotransmitter, dopamine receptors (D1-5 receptors) (EC50=2.7 nM). High-Quality, Low-Cost!</p>Formule :C8H12ClNO2Degré de pureté :99.47% - 99.72%Couleur et forme :SolidMasse moléculaire :189.64Fluphenazine dihydrochloride
CAS :<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Formule :C22H28Cl2F3N3OSDegré de pureté :99.23%Couleur et forme :Off-White SolidMasse moléculaire :510.44Trifluoperazine dihydrochloride
CAS :<p>Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.</p>Formule :C21H26Cl2F3N3SDegré de pureté :99.57% - 99.96%Couleur et forme :Cream Fine PowderMasse moléculaire :480.43Molindone hydrochloride
CAS :<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formule :C16H24N2O2·HClDegré de pureté :99% - 99.99%Couleur et forme :SolidMasse moléculaire :312.84Droperidol
CAS :<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formule :C22H22FN3O2Degré de pureté :97.16% - 98%Couleur et forme :SolidMasse moléculaire :379.43Spiperone
CAS :<p>Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.</p>Formule :C23H26FN3O2Degré de pureté :99.34% - 99.91%Couleur et forme :SolidMasse moléculaire :395.47Romergoline 2HCl
<p>Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.</p>Formule :C20H24Cl2N4O2Degré de pureté :99.01% - 99.40%Couleur et forme :SoildMasse moléculaire :423.34Haloperidol
CAS :<p>Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.</p>Formule :C21H23ClFNO2Degré de pureté :98.69% - 98.97%Couleur et forme :Crystals SolidMasse moléculaire :375.86Risperidone
CAS :<p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>Formule :C23H27FN4O2Degré de pureté :99.73%Couleur et forme :Crystalline SolidMasse moléculaire :410.48UCM-1306
CAS :<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Formule :C14H14FNO2SDegré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :279.33ONC206
CAS :<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Formule :C23H22F2N4ODegré de pureté :99.38% - 99.81%Couleur et forme :SolidMasse moléculaire :408.44Octodrine
CAS :<p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>Formule :C8H19NDegré de pureté :99.98%Couleur et forme :Clear Colorless To Light Yellow LiquidMasse moléculaire :129.24D5R agonist 1
<p>D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.</p>Couleur et forme :Odour SolidLosulazine
CAS :<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formule :C27H22F4N4O3SDegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :558.55Fenoldopam
CAS :<p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>Formule :C16H16ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.76Preclamol hydrochloride
CAS :<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Formule :C14H22ClNOCouleur et forme :SolidMasse moléculaire :255.78(R)-Preclamol hydrochloride
CAS :<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Formule :C14H22ClNOCouleur et forme :SolidMasse moléculaire :255.78Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Couleur et forme :Odour Solid(-)-GSK598809 hydrochloride
CAS :<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formule :C22H24ClF4N5OSDegré de pureté :98.36%Couleur et forme :SoildMasse moléculaire :517.977-Hydroxy-PIPAT maleate
CAS :<p>7-Hydroxy-PIPAT maleate is a D3R agonist.</p>Formule :C16H22INOCouleur et forme :SolidMasse moléculaire :371.262Quinelorane
CAS :<p>Quinelorane is dextrorotary isomer.</p>Formule :C14H22N4Couleur et forme :SolidMasse moléculaire :246.35Fluphenazine free base
CAS :<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Formule :C22H26F3N3OSCouleur et forme :SolidMasse moléculaire :437.52Moperone
CAS :<p>Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.</p>Formule :C22H26FNO2Couleur et forme :SolidMasse moléculaire :355.45Vanicoside E
CAS :<p>Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .</p>Formule :C53H52O22Couleur et forme :SolidMasse moléculaire :1040.97Dopamine D2 receptor agonist-2
CAS :<p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>Formule :C25H31Cl2N5OSDegré de pureté :98.93%Couleur et forme :SoildMasse moléculaire :520.52ADTN hydrobromide
CAS :<p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>Formule :C10H14BrNO2Couleur et forme :SolidMasse moléculaire :260.13MOR agonist-2
<p>Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.</p>Formule :C37H47Cl2N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :680.71Clomipramine D3
CAS :<p>Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).</p>Formule :C19H23ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :317.87A 77636 hydrochloride
CAS :<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Formule :C20H28ClNO3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :365.89Adrogolide HCl
CAS :<p>Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.</p>Formule :C22H26ClNO4SCouleur et forme :SolidMasse moléculaire :435.96Amisulpride hydrochloride
CAS :<p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>Formule :C17H28ClN3O4SCouleur et forme :SolidMasse moléculaire :405.94DETQ
CAS :<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Formule :C22H25Cl2NO3Couleur et forme :SolidMasse moléculaire :422.34Neuromedin N
CAS :<p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>Formule :C38H63N7O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :745.95Cabergoline
CAS :<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Formule :C26H37N5O2Degré de pureté :97.69% - 99.86%Couleur et forme :White Crystalline SolidMasse moléculaire :451.6ABT 724 trihydrochloride
CAS :<p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>Formule :C17H22Cl3N5Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :402.75LE 300
CAS :<p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>Formule :C20H22N2Degré de pureté :97.91% - 98.79%Couleur et forme :SolidMasse moléculaire :290.4[18F]-Labeled L-dopa precursor
CAS :<p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>Formule :C35H36N2O7Couleur et forme :SolidMasse moléculaire :596.67Secretoneurin, rat
CAS :<p>Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).</p>Formule :C159H252N40O58Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3651.95MLS1082
CAS :<p>MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.</p>Formule :C24H23N3O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :385.46D3R/MOR antagonist 1
<p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>Formule :C22H27Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.38PF-4363467
CAS :<p>PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.</p>Formule :C22H30N2O3SCouleur et forme :SolidMasse moléculaire :402.55ADTN
CAS :<p>ADTN is an agonist of the dopamine receptor.</p>Formule :C10H13NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.22D3R ligand 1
<p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>Formule :C27H37NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.59D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Formule :C25H31ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.98Haloperidol D4
CAS :<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Formule :C21H23ClFNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.89N-0500 HCl
CAS :<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Formule :C15H22ClNO2Degré de pureté :98.85% - 99.54%Couleur et forme :SolidMasse moléculaire :283.79O-2172
CAS :<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Formule :C14H16Cl2O2Couleur et forme :SolidMasse moléculaire :287.18Trimethobenzamide
CAS :<p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>Formule :C21H28N2O5Couleur et forme :SolidMasse moléculaire :388.46ST-836 hydrochloride
CAS :<p>ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .</p>Formule :C23H35ClN4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :451.07Haloperidol (D4')
CAS :<p>Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.</p>Formule :C21H23ClFNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.89Eticlopride hydrochloride
CAS :<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Formule :C17H25ClN2O3·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.31Tiapride-d3
<p>Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.</p>Formule :C15H21D3N2O4SCouleur et forme :SolidMasse moléculaire :331.45Aramisulpride
CAS :<p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>Formule :C17H27N3O4SCouleur et forme :SolidMasse moléculaire :369.48SKF-82958 hydrobromide
CAS :<p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>Formule :C19H21BrClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.73Clomipramine D3 hydrochloride
CAS :<p>Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).</p>Formule :C19H24Cl2N2Couleur et forme :SolidMasse moléculaire :354.33Docosahexaenoic acid ethyl ester
CAS :<p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>Formule :C24H36O2Couleur et forme :SolidMasse moléculaire :356.54Sumanirole maleate
CAS :<p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>Formule :C15H17N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :319.31Pramipexole dihydrochloride
CAS :<p>Pramipexole dihydrochloride could be used to treat Parkinson disease.</p>Formule :C10H18ClN3SDegré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :247.79cis-(Z)-Flupentixol dihydrochloride
CAS :<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Formule :C23H27Cl2F3N2OSDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :507.44PD128907 HCl
CAS :<p>PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.</p>Formule :C14H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :285.77UCSF924
CAS :<p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4(-)-Apomorphine hydrochloride hydrate
CAS :<p>(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.</p>Formule :C17H17NO2HClXH2OCouleur et forme :SolidMasse moléculaire :303.8ABT-724
CAS :<p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>Formule :C17H19N5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :293.37Clozapine N-Oxide
CAS :<p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>Formule :C18H19ClN4ODegré de pureté :98.43% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82SKF-83566
CAS :<p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>Formule :C17H18BrNODegré de pureté :95.00% - 99.82%Couleur et forme :SolidMasse moléculaire :332.23Perospirone hydrochloride
CAS :<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463Alizapride hydrochloride
CAS :<p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>Formule :C16H21N5O2·HClDegré de pureté :99.35% - 99.48%Couleur et forme :CoaMasse moléculaire :351.83GBR 12935
CAS :<p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>Formule :C28H34N2OCouleur et forme :SolidMasse moléculaire :414.58Raclopride tartrate
CAS :<p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>Formule :C19H26Cl2N2O9Couleur et forme :SolidMasse moléculaire :497.32Bisacodyl
CAS :<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Formule :C22H19NO4Degré de pureté :99.45% - 99.78%Couleur et forme :Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMasse moléculaire :361.39BisfluoroModafinil
CAS :<p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>Formule :C15H13F2NO2SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :309.33Nomifensine maleate
CAS :<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Formule :C20H22N2O4Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :354.4OS-3-106
CAS :<p>OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.</p>Formule :C25H30N4O2SDegré de pureté :99.4% - 99.57%Couleur et forme :SolidMasse moléculaire :450.6Glaucine
CAS :<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Formule :C21H25NO4Degré de pureté :99.42% - 99.56%Couleur et forme :SolidMasse moléculaire :355.43SCH-23390 hydrochloride
CAS :<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Xaliproden hydrochloride
CAS :<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Butyrophenone
CAS :<p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>Formule :C10H12ODegré de pureté :99.84%Couleur et forme :Colourless To Yellow LiquidMasse moléculaire :148.29-FLUORENOL
CAS :<p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>Formule :C13H10ODegré de pureté :99.98%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :182.22NGB 2904
CAS :<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Formule :C28H29Cl2N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :494.46DOPEXAMINE
CAS :<p>Dopexamine is a dopaminergic agonist</p>Formule :C22H32N2O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :356.5PD-168077 maleate
CAS :<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Formule :C24H26N4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :450.49ML417
CAS :<p>ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).</p>Formule :C22H25N3O3Degré de pureté :98.4% - 99.42%Couleur et forme :SolidMasse moléculaire :379.453-CPMT
CAS :<p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>Formule :C21H25Cl2NODegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :378.33A-381393
CAS :<p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>Formule :C20H24N4Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :320.43GSK163090
CAS :<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formule :C25H29N5ODegré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :415.53Bromocriptine mesylate
CAS :<p>Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)</p>Formule :C33H44BrN5O8SDegré de pureté :99.85% - 99.96%Couleur et forme :White SolidMasse moléculaire :750.7Nomifensine
CAS :<p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>Formule :C16H18N2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :238.33Mesdopetam
CAS :<p>Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.</p>Formule :C12H18FNO3SCouleur et forme :SolidMasse moléculaire :275.34Propionylpromazine hydrochloride
CAS :<p>Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.</p>Formule :C20H25ClN2OSDegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :376.94Fluoroclebopride
CAS :<p>Fluoroclebopride is a dopamine (DA) D2 receptor ligand.</p>Formule :C20H23ClFN3O2Degré de pureté :99.68% - 99.91%Couleur et forme :SolidMasse moléculaire :391.87Ansofaxine hydrochloride
CAS :<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Cariprazine
CAS :<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formule :C21H32Cl2N4ODegré de pureté :99.68% - 99.87%Couleur et forme :SolidMasse moléculaire :427.41Chlorprothixene
CAS :<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86GSK 789472 hydrochloride
CAS :<p>GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.</p>Formule :C15H22ClN3ODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :295.81Veralipride
CAS :<p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>Formule :C17H25N3O5SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :383.46Cariprazine hydrochloride
CAS :<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Formule :C21H33Cl3N4ODegré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :463.87Pridopidine
CAS :<p>Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.</p>Formule :C15H23NO2SDegré de pureté :95.2% - 99.89%Couleur et forme :SolidMasse moléculaire :281.41D-tetrahydropalmatine
CAS :<p>D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.</p>Formule :C21H25NO4Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :355.43Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Formule :C40H67N7O10Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :805.9Ocaperidone
CAS :<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Formule :C24H25FN4O2Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :420.48Perospirone
CAS :<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57carfenazine
CAS :<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Formule :C24H31N3O2SDegré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :425.59Pergolide
CAS :<p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>Formule :C19H26N2SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :314.49Rotundine
CAS :<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Formule :C21H25NO4Degré de pureté :99.8% - 99.91%Couleur et forme :Off-White SolidMasse moléculaire :355.43Pergolide mesylate
CAS :<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Formule :C20H30N2O3S2Degré de pureté :99.70%Couleur et forme :White To Off-White SolidMasse moléculaire :410.59J-147
CAS :<p>J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.</p>Formule :C18H17F3N2O2Degré de pureté :99.61% - >99.99%Couleur et forme :SolidMasse moléculaire :350.33Zotepine
CAS :<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formule :C18H18ClNOSDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :331.86Rotigotine-
CAS :<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Tavapadon
CAS :<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Formule :C19H16F3N3O3Degré de pureté :99.33% - 99.8%Couleur et forme :SolidMasse moléculaire :391.34Ritanserin
CAS :<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Formule :C27H25F2N3OSDegré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Vanoxerine dihydrochloride
CAS :<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Formule :C28H34Cl2F2N2ODegré de pureté :98.16% - 98.35%Couleur et forme :White SolidMasse moléculaire :523.49Pramipexole dihydrochloride hydrate
CAS :<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Formule :C10H17N3S·2HCl·H2ODegré de pureté :99.68%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :302.26Azaperone
CAS :<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Formule :C19H22FN3ODegré de pureté :98.73%Couleur et forme :White Or Off-White CrystallineMasse moléculaire :327.4SKF38393 hydrobromide
CAS :<p>SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;</p>Formule :C16H18BrNO2Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :336.22FAUC 346
CAS :<p>FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.</p>Formule :C24H29N3O2SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :423.57Sultopride hydrochloride
CAS :<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Formule :C17H27ClN2O4SDegré de pureté :≥95%Couleur et forme :White Or Yellowish PowderMasse moléculaire :390.93Dasotraline
CAS :<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Formule :C16H15Cl2NCouleur et forme :SolidMasse moléculaire :292.2PD 168568
CAS :<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Formule :C22H27N3OCouleur et forme :SolidMasse moléculaire :349.47Alizapride
CAS :<p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>Formule :C16H21N5O2Couleur et forme :SolidMasse moléculaire :315.37BP 897
CAS :<p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>Formule :C26H31N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :417.54Brexpiprazole
CAS :<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57JNJ-37822681
CAS :<p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>Formule :C17H17F5N4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :372.34Rotigotine Hydrochloride
CAS :<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.93Piribedil
CAS :<p>Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.</p>Formule :C16H18N4O2Degré de pureté :99.79% - 99.82%Couleur et forme :SolidMasse moléculaire :298.34Haloperidol hydrochloride
CAS :<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Formule :C21H24Cl2FNO2Couleur et forme :SolidMasse moléculaire :412.33FAUC 213
CAS :<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Formule :C18H19ClN4Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :326.82Metoclopramide
CAS :<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Formule :C14H22ClN3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :299.80Trimethobenzamide hydrochloride
CAS :<p>Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.</p>Formule :C21H29ClN2O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :424.92L-745870 trihydrochloride
CAS :<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21Raclopride
CAS :<p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>Formule :C15H20Cl2N2O3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :347.24Tiapride
CAS :<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Formule :C15H24N2O4SCouleur et forme :SolidMasse moléculaire :328.43Nuciferine
CAS :<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Formule :C19H21NO2Degré de pureté :98.76% - 99.79%Couleur et forme :SolidMasse moléculaire :295.38L-DOPA methyl ester (hydrochloride)
CAS :<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Formule :C10H14ClNO4Degré de pureté :98.69% - 99.81%Couleur et forme :White SolidMasse moléculaire :247.675Zuclopenthixol dihydrochloride
CAS :<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Formule :C22H27Cl3N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :473.89AHN 1-055 hydrochloride
CAS :<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Formule :C21H24ClF2NODegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :379.87L-745870 hydrochloride
CAS :<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Formule :C18H20Cl2N4Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :363.28FAUC-365
CAS :<p>FAUC-365 is a D3 dopamine receptor agonist.</p>Formule :C23H25Cl2N3OSDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :462.44Lurasidone
CAS :<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formule :C28H36N4O2SDegré de pureté :99.78% - 99.91%Couleur et forme :SolidMasse moléculaire :492.68Metergoline
CAS :<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Formule :C25H29N3O2Degré de pureté :99.83% - 99.97%Couleur et forme :SolidMasse moléculaire :403.52(+)-PD 128907 hydrochloride
CAS :<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Formule :C14H20ClNO3Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :285.77Mesdopetam hemitartrate
CAS :<p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>Formule :C28H42F2N2O12S2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :700.77WAY-100635 Monomaleate
CAS :<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Formule :C25H34N4O2·C4H4O4Degré de pureté :98.44% - 99.46%Couleur et forme :SolidMasse moléculaire :538.64Sertindole
CAS :<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Formule :C24H26ClFN4ODegré de pureté :99.87% - 99.92%Couleur et forme :Off-White To Pale Yellow SolidMasse moléculaire :440.94Clebopride malate
CAS :<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Formule :C24H30ClN3O7Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :507.96Fenoldopam mesylate
CAS :<p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>Formule :C16H16ClNO3·CH4O3SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :401.86Flupentixol dihydrochloride
CAS :<p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>Formule :C23H27Cl2F3N2OSDegré de pureté :98.76% - >99.99%Couleur et forme :White Or Off-White SolidMasse moléculaire :507.43GBR 12935 dihydrochloride
CAS :<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Formule :C28H36Cl2N2ODegré de pureté :99.09% - ≥95%Couleur et forme :SolidMasse moléculaire :487.5Decynium 22
CAS :<p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>Formule :C23H23IN2Degré de pureté :99.92%Couleur et forme :Dark Red CrystalsMasse moléculaire :454.35Domperidone monomaleate
CAS :<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Formule :C26H28ClN5O6Couleur et forme :SolidMasse moléculaire :541.98Tetrahydropalmatine hydrochloride
CAS :<p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>Formule :C21H26ClNO4Degré de pureté :98% - 99.59%Couleur et forme :SolidMasse moléculaire :391.888Fluphenazine decanoate
CAS :<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formule :C32H44F3N3O2SDegré de pureté :98.14%Couleur et forme :SolidMasse moléculaire :591.77

