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Autres inhibiteurs

Autres inhibiteurs

Cette catégorie englobe une grande variété d'inhibiteurs qui ne rentrent pas dans les classifications standard mais qui sont néanmoins cruciaux pour diverses recherches biochimiques et pharmacologiques. Ces inhibiteurs peuvent cibler des voies, des enzymes et des interactions moléculaires uniques ou moins étudiés, fournissant des outils précieux pour des domaines de recherche spécialisés. Chez CymitQuimica, nous offrons une sélection diversifiée d'inhibiteurs de haute qualité ciblant de multiples objectifs biologiques et disciplines de recherche, vous permettant d'explorer de nouvelles avenues thérapeutiques et d'approfondir votre compréhension des processus biologiques complexes.

37902 produits trouvés pour "Autres inhibiteurs"

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  • Nothramicin

    CAS :
    <p>Nothramicin is an anthracycline antibiotic that exhibits antimycobacterial activity.</p>
    Formule :C30H37NO11
    Couleur et forme :Solid
    Masse moléculaire :587.615
  • Cleistanthin

    CAS :
    <p>Cleistanthin, a toxic Cleistanthus collinus compound, has antihypertensive, alpha-antagonist, and diuretic properties; a modified naphthofuran-xylose.</p>
    Formule :C28H28O11
    Couleur et forme :Solid
    Masse moléculaire :540.52
  • Polyoxin K

    CAS :
    <p>Polyoxin K is a nucleoside antifungal antibiotic that exhibits significant effectiveness against rice sheath blight.</p>
    Formule :C22H30N6O13
    Masse moléculaire :586.51
  • ZK168281

    CAS :
    <p>ZK168281 is a 1α,25(OH)2D3 analog, VDR antagonist with 0.1 nM Kd, and blocks receptor CoA interaction.</p>
    Formule :C32H46O5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :510.70
  • RORγt inhibitor 2

    CAS :
    <p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>
    Formule :C31H33F5N2O7S
    Couleur et forme :Solid
    Masse moléculaire :672.66
  • Milbemycin α13

    CAS :
    <p>Milbemycin α13 (Meilingmycin B) is an antibiotic that is effective against nematodes and mites.</p>
    Formule :C37H52O9
    Masse moléculaire :640.80
  • Kri 1314

    CAS :
    Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.
    Formule :C38H51N5O7
    Couleur et forme :Solid
    Masse moléculaire :689.84
  • SLC4011540


    <p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>
    Formule :C24H23ClF3N7OS
    Couleur et forme :Solid
    Masse moléculaire :550
  • Oleuroside

    CAS :
    <p>Oleuroside can protect against mitochondrial dysfunction in models of early Alzheimer's disease and brain ageing.</p>
    Formule :C25H32O13
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :540.51
  • Sulprostone

    CAS :
    <p>EP3 and EP1 receptor agonist</p>
    Formule :C23H31NO7S
    Degré de pureté :98%
    Couleur et forme :White To Off-White Solid
    Masse moléculaire :465.56
  • KCL-440

    CAS :
    <p>RS 57639 is a bioactive chemical.</p>
    Formule :C18H18N2O2
    Couleur et forme :Solid
    Masse moléculaire :294.35
  • SHP2 IN-1

    CAS :
    <p>SHP2 IN-1 is an allergic SHP2 (PTPN11) inhibitor(IC50 : 3 nM).</p>
    Formule :C18H22Cl2N6OS
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :441.38
  • mPGES1-IN-4

    CAS :
    <p>mPGES1-IN-4 (compound 32) is a multi-substituted pyrimidine compound acting as a submicromolar inhibitor of PGE2 production. It primarily exerts its anti-inflammatory effects by inhibiting mPGES-1 and significantly suppresses acute inflammation models in vivo.</p>
    Formule :C27H25F2N3O
    Couleur et forme :Solid
    Masse moléculaire :445.50
  • PI3K-IN-27

    CAS :
    <p>PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.</p>
    Formule :C30H26F2N6O2S
    Couleur et forme :Solid
    Masse moléculaire :572.63
  • Celesticetin B

    CAS :
    <p>Celesticetin B is an antibiotic primarily exhibiting antibacterial activity against Gram-positive microorganisms.</p>
    Formule :C21H38N2O8S
    Couleur et forme :Solid
    Masse moléculaire :478.6
  • Leucomycin U

    CAS :
    <p>Leucomycin U is a macrolide antibiotic. It demonstrates significant activity against Gram-positive bacteria and also exhibits effects on spirochetes, rickettsiae, and chlamydiae.</p>
    Formule :C37H61NO14
    Couleur et forme :Solid
    Masse moléculaire :743.878
  • Gilvusmycin

    CAS :
    <p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>
    Formule :C38H34N6O8
    Couleur et forme :Solid
    Masse moléculaire :702.712
  • 2-Hydroxy-5-iminoazacyclopent-3-ene

    CAS :
    <p>2-Hydroxy-5-iminoazacyclopent-3-ene is a pyrroline-class antibiotic with mild activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C4H6N2O
    Couleur et forme :Solid
    Masse moléculaire :98.103
  • UNC9426

    CAS :
    <p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>
    Formule :C32H34F6N6O
    Degré de pureté :98.051%
    Couleur et forme :Solid
    Masse moléculaire :632.642
  • PPARα/γ agonist 1


    <p>PPARα/γ agonist 1 is a potent and dual PPARα/γ partial agonist which is a promising prototype for the research of dyslipidemia and diabetes.</p>
    Formule :C18H19NO2
    Couleur et forme :Solid
    Masse moléculaire :281.35
  • KCa2 channel modulator 2


    Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.
    Formule :C16H15ClFN5
    Couleur et forme :Solid
    Masse moléculaire :331.78
  • Monamycin G1

    CAS :
    <p>Monamycin G1 is an ester-peptide antibiotic [esterpeptid]. It shows activity against Gram-positive bacteria.</p>
    Formule :C33H54ClN7O8
    Masse moléculaire :712.28
  • TTK inhibitor 3

    CAS :
    <p>TTK inhibitor 3 is a potent and selective TTK (an essential spindle assembly checkpoint enzyme) inhibitor with an IC 50 value of 3.0 nM.</p>
    Formule :C42H49N9O3
    Couleur et forme :Solid
    Masse moléculaire :727.9
  • Coleon-U-quinone

    CAS :
    <p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>
    Formule :C20H24O5
    Couleur et forme :Solid
    Masse moléculaire :344.4
  • Cenicriviroc Sulfone

    CAS :
    <p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>
    Formule :C41H52N4O5S
    Couleur et forme :Solid
    Masse moléculaire :712.94
  • G-4120

    CAS :
    <p>G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.</p>
    Formule :C26H36N8O11S
    Couleur et forme :Solid
    Masse moléculaire :668.68
  • Plasma kallikrein-IN-2


    <p>Plasma kallikrein-IN-2: PKal inhibitor, IC50=0.1 nM. Used in angioedema, diabetic eye disease research.</p>
    Formule :C28H24ClF3N8O3
    Couleur et forme :Solid
    Masse moléculaire :612.99
  • PI3Kβ-IN-1

    CAS :
    <p>PI3Kβ-IN-1 is a selective, orally active PI3Kβ inhibitor (IC50: 2 nM).</p>
    Formule :C25H14F2N8
    Couleur et forme :Solid
    Masse moléculaire :464.43
  • PTP1B-IN-16


    <p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>
    Formule :C26H18ClN3O4S
    Couleur et forme :Solid
    Masse moléculaire :503.96
  • De-N-methylpamamycin-593A

    CAS :
    <p>De-N-methylpamamycin-593A is a 16-membered macrocyclic dilactone known for its ability to induce aerial mycelium formation.</p>
    Formule :C34H59NO7
    Masse moléculaire :593.84
  • ER272

    CAS :
    <p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>
    Formule :C24H34O6
    Couleur et forme :Solid
    Masse moléculaire :418.52
  • XN methyl pyrazole


    <p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>
    Formule :C22H24N2O4
    Couleur et forme :Solid
    Masse moléculaire :380.44
  • CEP-7055

    CAS :
    <p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>
    Formule :C32H35N3O4
    Couleur et forme :Solid
    Masse moléculaire :525.64
  • Tandutinib (MLN518) HCl


    Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.
    Formule :C31H43ClN6O4
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :599.16
  • Cilobamine (free base)

    CAS :
    <p>Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.</p>
    Formule :C17H23Cl2NO
    Couleur et forme :Solid
    Masse moléculaire :328.28
  • AZ0108

    CAS :
    <p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>
    Formule :C24H20F4N6O2
    Couleur et forme :Solid
    Masse moléculaire :500.45
  • Resorcinomycin B

    CAS :
    <p>Resorcinomycin B is an antibiotic found in [Streptoverticillum roseoverticillatum].</p>
    Formule :C13H18N4O5
    Couleur et forme :Solid
    Masse moléculaire :310.306
  • Tembotrione

    CAS :
    <p>Tembotrione is a chemical compound that may reduce the productivity of carrots. It possesses activity that degrades the quality of carrot stems. Additionally, Tembotrione can be used in studies focusing on the overall productivity of carrot cultivation.</p>
    Formule :C17H16ClF3O6S
    Couleur et forme :Solid
    Masse moléculaire :440.82
  • AS1940477

    CAS :
    <p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>
    Formule :C24H22FN5O2
    Couleur et forme :Solid
    Masse moléculaire :431.46
  • Hsp90-IN-16


    <p>Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.</p>
    Formule :C30H26FN3O6
    Couleur et forme :Solid
    Masse moléculaire :543.54
  • NTPDase-IN-3

    CAS :
    <p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>
    Formule :C22H24ClN3OS2
    Couleur et forme :Solid
    Masse moléculaire :446.03
  • Antimalarial agent 9


    <p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>
    Formule :C28H32BrN3O2
    Couleur et forme :Solid
    Masse moléculaire :522.48
  • NS2B/NS3-IN-5


    <p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>
    Formule :C14H9IN2O3S
    Couleur et forme :Solid
    Masse moléculaire :412.2
  • ORP-101

    CAS :
    <p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>
    Formule :C60H84N2O8
    Couleur et forme :Solid
    Masse moléculaire :961.32
  • SLC4101431


    <p>SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.</p>
    Formule :C29H28ClN7OS
    Couleur et forme :Solid
    Masse moléculaire :558.1
  • WAY-855

    CAS :
    <p>WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.</p>
    Formule :C9H11NO4
    Couleur et forme :Solid
    Masse moléculaire :197.19
  • KP 10614

    CAS :
    <p>KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.</p>
    Formule :C23H32O4
    Couleur et forme :Solid
    Masse moléculaire :372.50
  • ZK118182 isopropyl ester

    CAS :
    <p>ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM).</p>
    Formule :C23H37ClO5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :428.99
  • FR 900452

    CAS :
    <p>FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.</p>
    Formule :C22H25N3O3S
    Couleur et forme :Solid
    Masse moléculaire :411.52
  • ADP-2341


    <p>ADP-2341 is a soluble analog of FiVe1.</p>
    Formule :C24H29Cl2N5O3
    Couleur et forme :Solid
    Masse moléculaire :506.43
  • Anticancer agent 16


    <p>Anticancer agent 16 showed good cytotoxic effects on HCT-116 cell line (IC50: 8.55 μM), NCI-H460 cell line (IC50: 5.41 μM) and SKOV3 cell line (IC50: 6.4 μM).</p>
    Formule :C27H33N5O6
    Couleur et forme :Solid
    Masse moléculaire :523.58
  • DMGF

    CAS :
    <p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>
    Formule :C32H22O10
    Couleur et forme :Solid
    Masse moléculaire :566.51
  • DNDI-8219

    CAS :
    <p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>
    Formule :C13H10F3N3O5
    Couleur et forme :Solid
    Masse moléculaire :345.23
  • TSWV-IN-1


    <p>TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.</p>
    Formule :C26H31FO4S2
    Couleur et forme :Solid
    Masse moléculaire :490.65
  • Carmegliptin dihydrochloride

    CAS :
    <p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>
    Formule :C20H30Cl2FN3O3
    Couleur et forme :Solid
    Masse moléculaire :450.38
  • Steroid sulfatase/17β-HSD1-IN-3


    <p>Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).</p>
    Formule :C19H17ClN2O5S
    Couleur et forme :Solid
    Masse moléculaire :420.87
  • di-Val-L-dC

    CAS :
    <p>Di-Val-L-dC, a reverse transcriptase inhibitor, is used potentially for treatment of HBV infection.</p>
    Formule :C19H31N5O6
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :425.48
  • IACS-8779 disodium

    CAS :
    <p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>
    Formule :C21H23N9Na2O10P2S2
    Couleur et forme :Solid
    Masse moléculaire :733.52
  • Antileishmanial agent-4


    <p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>
    Formule :C17H18N4O4
    Couleur et forme :Solid
    Masse moléculaire :342.35
  • Faldaprevir sodium

    CAS :
    <p>Faldaprevir sodium: HCV treatment, inhibits NS3/NS4A protease, P-glycoprotein, CYP3A4, UGT1A1.</p>
    Formule :C40H48BrN6NaO9S
    Couleur et forme :Solid
    Masse moléculaire :891.81
  • Topoisomerase I inhibitor 8

    CAS :
    <p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>
    Formule :C24H21FN2O4
    Couleur et forme :Solid
    Masse moléculaire :420.43
  • Dersimelagon phosphate

    CAS :
    <p>Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.</p>
    Formule :C36H48F4N3O9P
    Couleur et forme :Solid
    Masse moléculaire :773.75
  • AZD2353

    CAS :
    <p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>
    Formule :C22H19ClFN3O3
    Couleur et forme :Solid
    Masse moléculaire :427.86
  • AVE-1330A sodium

    CAS :
    <p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>
    Formule :C7H10N3NaO6S
    Couleur et forme :Solid
    Masse moléculaire :287.23
  • Steroid sulfatase/17β-HSD1-IN-4


    <p>Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).</p>
    Formule :C18H17N3O4S2
    Couleur et forme :Solid
    Masse moléculaire :403.48
  • P2X7 receptor antagonist-1


    <p>P2X7 receptor antagonist-1 is a purinergic P2X7 receptor antagonist with anti-neuroinflammatory effects.</p>
    Formule :C22H20F4N2O3
    Couleur et forme :Solid
    Masse moléculaire :436.4
  • Metocurine chloride

    CAS :
    <p>Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.</p>
    Formule :C40H48Cl2N2O6
    Couleur et forme :Solid
    Masse moléculaire :723.72
  • Cbl-b-IN-1

    CAS :
    <p>Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 &lt;100 nM) with potential anticancer activity for the study of intestinal inflammation.</p>
    Formule :C29H34N6O2
    Degré de pureté :99.68%
    Couleur et forme :Solid
    Masse moléculaire :498.631
  • MSX-3 free acid

    CAS :
    <p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>
    Formule :C21H23N4O7P
    Couleur et forme :Solid
    Masse moléculaire :474.40
  • Guraxetan


    <p>Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.</p>
    Formule :C20H34N4O9
    Couleur et forme :Solid
    Masse moléculaire :474.51
  • Zurletrectinib

    CAS :
    <p>Zurletrectinib is a tyrosine kinase inhibitor with potential as an antineoplastic agent.</p>
    Formule :C19H19F2N7O2
    Couleur et forme :Solid
    Masse moléculaire :415.4
  • 4α-PDD

    CAS :
    <p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>
    Formule :C40H64O8
    Couleur et forme :Solid
    Masse moléculaire :672.93
  • Chitinase-IN-5


    <p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>
    Formule :C20H21ClFN7
    Couleur et forme :Solid
    Masse moléculaire :413.88
  • DWN-12088 HCl

    CAS :
    <p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>
    Formule :C15H21Cl4N3O
    Couleur et forme :Solid
    Masse moléculaire :401.15
  • GZN39838

    CAS :
    <p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>
    Formule :C22H30O6
    Couleur et forme :Solid
    Masse moléculaire :390.47
  • Hexedine

    CAS :
    <p>Hexedine is a biochemical.</p>
    Formule :C22H45N3
    Couleur et forme :Solid
    Masse moléculaire :351.61
  • Anticancer agent 80


    <p>Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).</p>
    Formule :C19H12BrNO5
    Couleur et forme :Solid
    Masse moléculaire :414.21
  • eIF4A3-IN-4


    <p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>
    Formule :C24H20N2O5
    Couleur et forme :Solid
    Masse moléculaire :416.43
  • METTL3-IN-3

    CAS :
    METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor .
    Formule :C26H28BrFN6O2
    Couleur et forme :Solid
    Masse moléculaire :555.44
  • Hetrombopag olamine

    CAS :
    <p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>
    Formule :C29H36N6O7
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :580.63
  • ALK5-IN-7

    CAS :
    <p>ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.</p>
    Formule :C26H28N4O3S
    Couleur et forme :Solid
    Masse moléculaire :476.59
  • Anti-ToCV agent 1


    <p>Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.</p>
    Formule :C22H19FN2O5S
    Couleur et forme :Solid
    Masse moléculaire :442.46
  • Ornoprostil

    CAS :
    <p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>
    Formule :C23H38O6
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :410.54
  • Butaprost

    CAS :
    <p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>
    Formule :C24H40O5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :408.57
  • WS-898


    <p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>
    Formule :C33H25N7OS
    Couleur et forme :Solid
    Masse moléculaire :567.66
  • RS 2135

    CAS :
    <p>RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.</p>
    Formule :C18H21ClN2O2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :332.83
  • PLAP-IN-1

    CAS :
    <p>PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.</p>
    Formule :C25H21Cl2N3O5
    Couleur et forme :Soild
    Masse moléculaire :514.36
  • Odiparcil

    CAS :
    <p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>
    Formule :C15H16O6S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :324.35
  • BILA 1906 BS

    CAS :
    BILA 1906 BS is an inhibitor of substrate analog protease.
    Formule :C41H52N6O4S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :724.95
  • NUCC-555

    CAS :
    <p>NUCC-555 is a first-in-class antagonist of activin. It opens a completely new approach to inhibiting the activity of TGF-beta receptor superfamily members.</p>
    Formule :C25H25N5O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :443.5
  • Fonsartan free acid

    CAS :
    <p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>
    Formule :C26H32N4O5S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :544.69
  • CEP-2563

    CAS :
    <p>CEP-2563 is a prodrug of CEP-751. It also used as an antitumor agent, inhibiting protein kinases.</p>
    Formule :C36H41ClN6O6
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :689.20
  • DLCI-1

    CAS :
    <p>DLCI-1 is a potent and selective oral inhibitor of cytochrome P450 2A6 (CYP2A6), significantly reducing self-administered nicotine doses in both male and female mice.</p>
    Formule :C12H14N2S
    Couleur et forme :Solid
    Masse moléculaire :218.32
  • L-739750

    CAS :
    <p>L-739,750 is an inhibitor (FTI) of peptidomimetic farnesyltransferase.</p>
    Formule :C23H39N3O6S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :517.7
  • MSK-195

    CAS :
    <p>MSK-195 is an effective TRPV1 agonist.</p>
    Formule :C28H40N2O5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :484.63
  • Lp-PLA2-IN-6

    CAS :
    <p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>
    Formule :C25H21F5N4O3
    Couleur et forme :Solid
    Masse moléculaire :520.45
  • 2,4-Diaminoanisole

    CAS :
    <p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>
    Formule :C7H10N2O
    Couleur et forme :Solid
    Masse moléculaire :138.17
  • SID 125240931

    CAS :
    <p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>
    Formule :C19H24N4O3S
    Couleur et forme :Solid
    Masse moléculaire :388.48
  • PAD2-IN-1 hydrochloride


    <p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>
    Formule :C25H30ClFN6O3
    Couleur et forme :Solid
    Masse moléculaire :517
  • HOE-288

    CAS :
    <p>HOE-288 is a converting enzyme (CE) inhibitor.</p>
    Formule :C27H38N2O5
    Couleur et forme :Solid
    Masse moléculaire :470.60
  • Cilengitide hydrochloride

    CAS :
    <p>Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.</p>
    Formule :C27H41ClN8O7
    Couleur et forme :Solid
    Masse moléculaire :625.12
  • UCN-02

    CAS :
    <p>UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.</p>
    Formule :C28H26N4O4
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :482.53
  • rel-MDM2/4-p53-IN-2


    <p>Potent dual MDM2/MDM4 inhibitor &amp; p53 activator; IC50: 70.7 nM (MDM2), 81.4 nM (MDM4); regulates cell cycle, triggers apoptosis, anti-cancer.</p>
    Formule :C25H17Cl3FN3O3
    Couleur et forme :Solid
    Masse moléculaire :532.78
  • MSA-2 dimer

    CAS :
    <p>MSA-2 dimer: selective oral non-nucleotide STING agonist, Kd=145 μM, long-term antitumor effect, non-covalent, higher permeability.</p>
    Formule :C29H28O8S2
    Couleur et forme :Solid
    Masse moléculaire :568.66
  • 16(R)-Iloprost

    CAS :
    <p>Iloprost, a potent prostacyclin analog, binds IP &amp; EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>
    Formule :C22H32O4
    Couleur et forme :Solid
    Masse moléculaire :360.49
  • Anticancer agent 35


    <p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>
    Formule :C15H13N3O3S3
    Couleur et forme :Solid
    Masse moléculaire :379.48
  • Amrubicin HCl

    CAS :
    <p>Amrubicin (SM-5887), an anthracycline, treats lung cancer by inhibiting DNA replication and topoisomerase II, with less cardiac toxicity.</p>
    Formule :C25H25NO9
    Couleur et forme :Solid
    Masse moléculaire :483.47
  • KUS121

    CAS :
    <p>KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.</p>
    Formule :C22H17FN4NaO3S
    Couleur et forme :Solid
    Masse moléculaire :459.45
  • PTP1B-IN-21


    <p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>
    Formule :C22H22O11
    Couleur et forme :Solid
    Masse moléculaire :462.4
  • Antileishmanial agent-6


    <p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>
    Formule :C24H26O8
    Couleur et forme :Solid
    Masse moléculaire :442.46
  • Tubulosine

    CAS :
    <p>Tubulosine is an anticancer agent that inhibits cancer cell growth.</p>
    Formule :C29H37N3O3
    Couleur et forme :Solid
    Masse moléculaire :475.62
  • Antibiotic MA 144M2

    CAS :
    <p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>
    Formule :C42H55NO16
    Couleur et forme :Solid
    Masse moléculaire :829.88
  • Demethoxyviridin

    CAS :
    <p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>
    Formule :C19H14O5
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :322.31
  • MRS2500

    CAS :
    <p>MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.</p>
    Formule :C13H18IN5O8P2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :561.16
  • DI-404

    CAS :
    <p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>
    Formule :C35H45ClN6O6S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :713.29
  • Ranakinin

    CAS :
    <p>Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.</p>
    Formule :C62H95N17O15S
    Couleur et forme :Solid
    Masse moléculaire :1350.59
  • Hypoglycemic agent 1

    CAS :
    <p>Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.</p>
    Formule :C25H24FN5O4
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :477.49
  • Tonantzitlolone

    CAS :
    <p>Tonantzitlolone activates TRPC1/4/5 channels, PKCα/θ, inhibits IRS1/PI3K/AKT, and triggers HSF1 to induce glucose dependence.</p>
    Formule :C26H40O7
    Couleur et forme :Solid
    Masse moléculaire :464.59
  • Calphostin D

    CAS :
    <p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>
    Formule :C30H30O10
    Couleur et forme :Solid
    Masse moléculaire :550.55
  • XR8-89

    CAS :
    <p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>
    Formule :C29H36N4O2S
    Couleur et forme :Solid
    Masse moléculaire :504.69
  • Griseorhodin G

    CAS :
    <p>Griseorhodin G is a quinone antibiotic with antitumor activity.</p>
    Formule :C25H18O12
    Masse moléculaire :510.40
  • Maltophilin

    CAS :
    <p>Maltophilin is a broad-spectrum antifungal antibiotic that exhibits no antibacterial activity against either Gram-positive or Gram-negative bacteria.</p>
    Formule :C29H38N2O6
    Masse moléculaire :510.62
  • Polyoxin J

    CAS :
    <p>Polyoxin J is a nucleoside antifungal antibiotic, notably effective against sheath blight in rice.</p>
    Formule :C17H25N5O12
    Masse moléculaire :491.41
  • Glaucarubin

    CAS :
    <p>Glaucarubin is a bitter lactone naturally found in the fruits of Simaruba glauca. It is employed as an anti-amebic agent in research focused on amebiasis. The compound exhibits good tolerability, with a median lethal dose (LD50) of 1,600 mg/kg in mice and 6,400 mg/kg in rats.</p>
    Formule :C25H36O10
    Masse moléculaire :496.55
  • Lucilactaene

    CAS :
    <p>Lucilactaene exhibits potent antimalarial activity and functions as a P53-transfected tumor cell cycle inhibitor. It effectively halts the cell cycle progression of H1299/TSP53 cells at the G1 phase.</p>
    Formule :C22H27NO6
    Masse moléculaire :401.45
  • Griseolutein A

    CAS :
    <p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C17H14N2O6
    Couleur et forme :Solid
    Masse moléculaire :342.303
  • Saframycin Mx2

    CAS :
    <p>Saframycin Mx2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C29H38N4O8
    Couleur et forme :Solid
    Masse moléculaire :570.634
  • Fleephilone

    CAS :
    <p>Fleephilone is a fungal metabolite isolated from Trichoderma harzianum. It acts as an HIV REV/RRE binding inhibitor, hindering the interaction between REV protein and RRE RNA with an IC50 of 7.6 μM.</p>
    Formule :C24H27NO7
    Couleur et forme :Solid
    Masse moléculaire :441.474
  • Cinnatriacetin A

    CAS :
    <p>Cinnatriacetin A exhibits activity against Gram-positive bacteria.</p>
    Formule :C23H20O5
    Couleur et forme :Solid
    Masse moléculaire :376.402
  • Griseolic acid C

    CAS :
    <p>Griseolic acid C (Dihydrodeoxygriseolic acid) is an antibiotic found in the Streptomyces griseoaurantiacus SANK43894 strain. This compound is a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase [EC 3.1.4.17], with an IC50 of 0.12 μM (enzyme sourced from rat brain tissue).</p>
    Formule :C14H15N5O7
    Couleur et forme :Solid
    Masse moléculaire :365.298
  • Diatretyne Ⅰ

    CAS :
    Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.
    Formule :C8H5NO3
    Couleur et forme :Solid
    Masse moléculaire :163.13
  • Azirinomycin

    CAS :
    <p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C4H5NO2
    Couleur et forme :Solid
    Masse moléculaire :99.088
  • STA-1474

    CAS :
    <p>STA-1474, a soluble prodrug of ganetespib (STA-9090), becomes a strong HSP90 inhibitor effective against canine tumors.</p>
    Formule :C20H21N4O6P
    Couleur et forme :Solid
    Masse moléculaire :444.38
  • SSTR5 antagonist 2 TFA

    CAS :
    <p>Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.</p>
    Formule :C34H36F4N2O7
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :660.65
  • Memnobotrin A

    CAS :
    <p>Memnobotrin A is an antibiotic with inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.</p>
    Formule :C25H33NO5
    Couleur et forme :Solid
    Masse moléculaire :427.53
  • 7-Hydroxyguanine

    CAS :
    <p>7-Hydroxyguanine is an antibiotic that inhibits the growth of L1210 leukemia cells.</p>
    Formule :C5H5N5O2
    Couleur et forme :Solid
    Masse moléculaire :167.126
  • Menoxymycin A

    CAS :
    <p>Menoxymycin A is an antibiotic with cytotoxic properties. It inhibits the growth of KB and N18-RE-105 cells, with IC50 values of 0.86 μM and 0.14 μM, respectively.</p>
    Formule :C24H27NO9
    Couleur et forme :Solid
    Masse moléculaire :473.473
  • Glidobactin C

    CAS :
    <p>Glidobactin C (GlbC) is an antitumor antibiotic with activity against pathogenic fungi and yeasts. It exhibits antifungal properties against Candida albicans and Aspergillus fumigatus, with a minimum inhibitory concentration (MIC) of 0.8 μg/mL. Additionally, Glidobactin C prolongs the survival time of mice inoculated with leukemia P388 cells.</p>
    Formule :C29H48N4O6
    Couleur et forme :Solid
    Masse moléculaire :548.715
  • 2-Hydroxygentamicin C2

    CAS :
    <p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C20H41N5O8
    Couleur et forme :Solid
    Masse moléculaire :479.568
  • CPX-351

    CAS :
    <p>CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.</p>
    Formule :C36H42N4O15
    Degré de pureté :98.95% - 99.763%
    Couleur et forme :Solid
    Masse moléculaire :770.74
  • Neihumicin

    CAS :
    <p>Neihumicin exhibits resistance against the yeast Saccharomyces cerevisiae (ATCC 9763) and the mold Penicillium italicum (Wehmer), but it does not show resistance to bacteria.</p>
    Formule :C19H16N2O2
    Couleur et forme :Solid
    Masse moléculaire :304.342
  • Epithienamycin D

    CAS :
    <p>Epithienamycin D is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C13H16N2O5S
    Couleur et forme :Solid
    Masse moléculaire :312.342
  • Clavalanine

    CAS :
    <p>Clavalanine (Ro 22-5417) is capable of inhibiting various bacteria and fungi.</p>
    Formule :C8H12N2O4
    Couleur et forme :Solid
    Masse moléculaire :200.192
  • Hydranthomycin

    CAS :
    <p>Hydranthomycin is an antibiotic with moderate antifungal activity, exhibiting a minimum inhibitory concentration (MIC) of 25 μg/mL against the rice blast fungus. Additionally, it inhibits the growth of Chlorella (tiny naked algae) and possesses herbicidal properties.</p>
    Formule :C20H20O5
    Couleur et forme :Solid
    Masse moléculaire :340.37
  • Asperenone

    CAS :
    <p>Asperenone is a 15-lipoxygenase (15-LOX) inhibitor with an IC50 of 0.3 mM. Additionally, it acts as a platelet aggregation inhibitor with an IC50 of 0.23 mM. Asperenone also exhibits antifungal properties, inhibiting the growth of pathogenic fungi Ophiostoma crassivaginatum and O. piliferum, and may be utilized in research related to cardiovascular diseases and anti-infective treatments.</p>
    Formule :C20H22O
    Couleur et forme :Solid
    Masse moléculaire :278.388
  • GSK2578999A

    CAS :
    <p>GSK2578999A is a betulin derivative with antitumor activity.</p>
    Formule :C46H62ClNO7
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :776.44
  • Haliangicin A

    CAS :
    <p>Haliangicin A exhibits antifungal activity against filamentous fungi and also affects oomycetes, though it does not possess antibacterial properties.</p>
    Formule :C22H32O5
    Couleur et forme :Solid
    Masse moléculaire :376.49
  • 2-n-Heptyl-4-quinolinol

    CAS :
    <p>2-n-Heptyl-4-quinolinol exhibits activity against Candida albicans, Staphylococcus aureus, Vibrio anguillarum, and Vibrio harveyi.</p>
    Formule :C16H21NO
    Couleur et forme :Solid
    Masse moléculaire :243.34
  • Formadicin A

    CAS :
    <p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>
    Formule :C30H34N4O16
    Couleur et forme :Solid
    Masse moléculaire :706.608
  • BSc5367

    CAS :
    <p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>
    Formule :C20H15N3O2
    Couleur et forme :Soild
    Masse moléculaire :329.35
  • NTPDase-IN-2

    CAS :
    <p>NTPDase-IN-2 inhibits h-NTPDase-2/-8 (IC50: 0.04, 2.27 µM), non-competitive for h-NTPDase-1/-2 (Km: 74 µM); useful in cancer, immune, bacterial research.</p>
    Formule :C24H20FN3OS2
    Couleur et forme :Solid
    Masse moléculaire :449.56
  • Feigrisolide C

    CAS :
    <p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>
    Formule :C21H36O7
    Couleur et forme :Solid
    Masse moléculaire :400.506
  • Deoxyfrenolicin

    CAS :
    <p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>
    Formule :C18H18O6
    Couleur et forme :Solid
    Masse moléculaire :330.332
  • (S)-Butaprost free acid

    CAS :
    <p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>
    Formule :C23H38O5
    Couleur et forme :Solid
    Masse moléculaire :394.54
  • Chitinovorin C

    CAS :
    <p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>
    Formule :C15H20N4O8S
    Couleur et forme :Solid
    Masse moléculaire :416.406
  • Glycotriosyl glutamine

    CAS :
    <p>Glycotriosyl glutamine is a nephritogenoside analog.</p>
    Formule :C23H40N2O18
    Couleur et forme :Solid
    Masse moléculaire :632.57
  • Pyloricidin A2

    CAS :
    <p>Pyloricidin A2 is an antibiotic effective against Helicobacter pylori, produced by Bacillus species HC-70. It exhibits strong anti-Helicobacter pylori activity but shows no activity against other bacteria and yeast.</p>
    Formule :C32H53N5O10
    Couleur et forme :Solid
    Masse moléculaire :667.79
  • Fudecalone

    CAS :
    <p>Fudecalone is produced by the Penicillium strain FO-2030. It completely inhibits the coccidian parasite Eimeria Tenella that is resistant to Monensin.</p>
    Formule :C15H22O3
    Couleur et forme :Solid
    Masse moléculaire :250.33
  • PD-1/PD-L1-IN-16


    <p>PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.</p>
    Formule :C34H30N4O4
    Couleur et forme :Solid
    Masse moléculaire :558.63
  • Phellinsin

    CAS :
    <p>Phellinsin selectively inhibits the activity of chitin synthase I and II, with IC50 values of 76 and 28 μg/mL, respectively. It also exhibits antimicrobial effects against pathogens such as anthracnose, rice blast fungus, Aspergillus fumigatus, and Trichophyton mentagrophytes, with a MIC ranging from 12.5 to 50 μg/mL.</p>
    Formule :C18H14O8
    Couleur et forme :Solid
    Masse moléculaire :358.30
  • LPA5 antagonist 2


    <p>LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.</p>
    Formule :C26H25FN2O4S
    Couleur et forme :Solid
    Masse moléculaire :480.55
  • Mutalomycin

    CAS :
    <p>Mutalomycin is a polyether antibiotic with activity against Gram-positive bacteria, mycoplasma, and coccidia.</p>
    Formule :C41H70O12
    Couleur et forme :Solid
    Masse moléculaire :754.987
  • Epoxyquinomicin A

    CAS :
    <p>Epoxyquinomicin A is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus with MIC values of 3-12.5 µg/mL. Additionally, it shows cytotoxicity in cancer cells L1210, B16, and S180, with an IC50 of 2-8 µg/mL. Furthermore, Epoxyquinomicin A demonstrates anti-inflammatory effects in collagen-induced arthritis.</p>
    Formule :C14H10ClNO6
    Couleur et forme :Solid
    Masse moléculaire :323.685
  • AEP-IN-1


    <p>APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.</p>
    Formule :C18H27N3O3
    Couleur et forme :Solid
    Masse moléculaire :333.43
  • Neuraminidase-IN-7


    <p>Neuraminidase-IN-7, a thiophene, inhibits neuraminidase (IC50 0.03 μM), showing promise for flu research.</p>
    Formule :C21H20N2O6S
    Couleur et forme :Solid
    Masse moléculaire :428.46
  • AS-1940477 hydrobromide

    CAS :
    <p>AS-1940477 hydrobromide is a p38 mitogen-activated protein kinase (MAPK) inhibitor.</p>
    Formule :C24H23BrFN5O2
    Couleur et forme :Solid
    Masse moléculaire :512.38
  • BI-207524

    CAS :
    <p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>
    Formule :C35H36ClN5O5
    Couleur et forme :Solid
    Masse moléculaire :642.14
  • Polyoxin E

    CAS :
    <p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>
    Formule :C17H23N5O13
    Couleur et forme :Solid
    Masse moléculaire :505.39
  • PDE4-IN-5


    <p>PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.</p>
    Formule :C21H28N2O3
    Couleur et forme :Solid
    Masse moléculaire :356.46
  • Micacocidin A

    CAS :
    <p>Micacocidin A is an antibiotic showing excellent activity against Mycoplasma species.</p>
    Formule :C27H37N3O4S3Zn
    Couleur et forme :Solid
    Masse moléculaire :629.20
  • 3-epi-Deoxynegamycin

    CAS :
    <p>3-epi-Deoxynegamycin exhibits antibacterial activity, primarily effective against most Gram-positive bacteria, while its effectiveness is somewhat reduced against Gram-negative bacteria.</p>
    Formule :C9H20N4O3
    Couleur et forme :Solid
    Masse moléculaire :232.28
  • Griseorhodin A

    CAS :
    <p>Griseorhodin A is a quinone antibiotic with activity against Gram-positive bacteria.</p>
    Formule :C25H16O12
    Couleur et forme :Solid
    Masse moléculaire :508.387
  • Melithiazole B

    CAS :
    <p>Melithiazol B is an antibiotic and a potent inhibitor of β-methoxyacrylate (MOA), with both antifungal and cytotoxic properties.</p>
    Formule :C20H24N2O4S2
    Couleur et forme :Solid
    Masse moléculaire :420.546
  • Hypnophilin

    CAS :
    <p>Hypnophilin exhibits multiple activities, including effectiveness against Gram-positive bacteria, Gram-negative bacteria, yeasts, molds, and tumors.</p>
    Formule :C15H20O3
    Couleur et forme :Solid
    Masse moléculaire :248.318
  • Epithienamycin F

    CAS :
    <p>Epithienamycin F is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>
    Formule :C13H18N2O8S2
    Couleur et forme :Solid
    Masse moléculaire :394.421
  • Pluracidomycin C1

    CAS :
    <p>Pluracidomycin C1 is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria and also possesses β-lactamase inhibitory properties.</p>
    Formule :C10H13NO10S2
    Couleur et forme :Solid
    Masse moléculaire :371.341
  • Citrinin hydrate

    CAS :
    <p>Citrinin hydrate is an inhibitor of human rhinovirus (HRV) 3C protease, with an IC50 of 1.0 mM.</p>
    Formule :C13H16O6
    Couleur et forme :Solid
    Masse moléculaire :268.263
  • Piperazinomycin

    CAS :
    <p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>
    Formule :C18H20N2O2
    Couleur et forme :Solid
    Masse moléculaire :296.36
  • Sequoiaflavone

    CAS :
    <p>Sequoiaflavone is a biflavone isolated from Ginkgo biloba.</p>
    Formule :C31H20O10
    Couleur et forme :Solid
    Masse moléculaire :552.48
  • CV 5975

    CAS :
    <p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>
    Formule :C22H31N3O5S
    Couleur et forme :Solid
    Masse moléculaire :449.56
  • Melithiazole A

    CAS :
    <p>Melithiazol A is an antibiotic and a potent β-methoxyacrylate (MOA) inhibitor with antifungal and cytotoxic properties.</p>
    Formule :C20H26N2O4S2
    Couleur et forme :Solid
    Masse moléculaire :422.561
  • Eurystatin A

    CAS :
    <p>Eurystatin A is a prolyl endopeptidase inhibitor, with L-leucine and L-ornithine serving as direct precursors to the L-leucine and L-ornithine components of eurystatins A.</p>
    Formule :C23H38N4O5
    Couleur et forme :Solid
    Masse moléculaire :450.572
  • MCTR1

    CAS :
    <p>MCTR1, a pro-resolving mediator derived from DHA, promotes tissue repair and reduces inflammation by enhancing phagocytosis and decreasing eicosanoids.</p>
    Formule :C32H47N3O9S
    Couleur et forme :Solid
    Masse moléculaire :649.8
  • 20-Deoxysalinomycin

    CAS :
    <p>20-Deoxysalinomycin primarily targets Gram-positive bacteria, with a particular effectiveness against poultry coccidia.</p>
    Formule :C42H70O10
    Couleur et forme :Solid
    Masse moléculaire :735.00
  • 20-Deoxynarasin

    CAS :
    <p>20-Deoxynarasin exhibits activity against Gram-positive bacteria, mycoplasma, coccidia, and viruses, and it also promotes growth.</p>
    Formule :C43H72O10
    Couleur et forme :Solid
    Masse moléculaire :749.03
  • PDE4B/7A-IN-1

    CAS :
    <p>5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.</p>
    Formule :C25H35N3O3
    Couleur et forme :Solid
    Masse moléculaire :425.56
  • EICAR

    CAS :
    <p>EICAR: IMP dehydrogenase inhibitor with anticancer and antiviral properties, failed in leukemia trials, active against various viruses but not SARS.</p>
    Formule :C11H13N3O5
    Couleur et forme :Solid
    Masse moléculaire :267.24
  • A1-Phytoprostane-I

    CAS :
    <p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression &amp; increases phytoalexin synthesis.</p>
    Formule :C18H28O4
    Couleur et forme :Solid
    Masse moléculaire :308.41
  • Z57346765

    CAS :
    <p>Z57346765 is a specific PGK1 inhibitor that inhibits PGK1-dependent cell proliferation by decreasing the metabolic enzyme activity of PGK1 during glycolysis.</p>
    Formule :C17H18N4O
    Degré de pureté :99.85%
    Couleur et forme :Solid
    Masse moléculaire :294.35
  • Latrunculin M

    CAS :
    <p>Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.</p>
    Formule :C21H33NO5S
    Couleur et forme :Solid
    Masse moléculaire :411.55
  • VRT-18858

    CAS :
    <p>VRT-18858 is a metabolite of VX-740.</p>
    Formule :C24H25N5O7
    Couleur et forme :Solid
    Masse moléculaire :495.48
  • Cuevaene A

    CAS :
    <p>Cuevaene A can be isolated from the Streptomyces genus gdmAI-disrupted LZ35 strain. It exhibits moderate activity against Gram-positive bacteria, such as Bacillus subtilis (strain ATCC 11060), and demonstrates moderate activity against fungi, including Fusarium verticillioides (strain S68) and Rhizoctonia solani (strain GXE4).</p>
    Formule :C21H22O5
    Couleur et forme :Solid
    Masse moléculaire :354.396
  • 9(S)-HEPE

    CAS :
    <p>9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.</p>
    Formule :C20H30O3
    Couleur et forme :Solid
    Masse moléculaire :318.45
  • Guanine-7-oxide

    CAS :
    <p>Guanine-7-oxide (Guanine 7-N-oxide) is an antitumor antibiotic with antitumor and anti-Candida albicans activities. It inhibits the replication of viruses such as herpes virus, infectious hematopoietic necrosis virus (IHNV), and infectious pancreatic necrosis virus (IPNV). The compound also demonstrates significant activity against mouse L1210 leukemia cells.</p>
    Formule :C5H5N5O2
    Couleur et forme :Solid
    Masse moléculaire :167.126
  • Mycoversilin

    CAS :
    <p>Mycoversilin is an antibiotic with inhibitory activity against dermatophytes and plant pathogenic fungi, but it does not exhibit activity against yeasts and bacteria. It strongly inhibits protein synthesis.</p>
    Formule :C18H16O8
    Couleur et forme :Solid
    Masse moléculaire :360.315
  • Barixibat

    CAS :
    <p>Barixibat is a bile acid transport inhibitor.</p>
    Formule :C42H55N5O8
    Couleur et forme :Solid
    Masse moléculaire :757.91
  • Chitinovorin A

    CAS :
    <p>Chitinovorin A is a β-lactam antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>
    Formule :C26H41N9O11S
    Couleur et forme :Solid
    Masse moléculaire :687.722
  • FWM-1


    <p>FWM-1 blocks SARS-CoV-2 NSP13, hinders ATP binding, with -328.6 kcal/mol binding energy.</p>
    Formule :C15H11ClN4O4S2
    Couleur et forme :Solid
    Masse moléculaire :410.86
  • Fusarielin A

    CAS :
    <p>Fusarielin A is a natural product found in the genus Fusarium.</p>
    Formule :C25H38O4
    Couleur et forme :Solid
    Masse moléculaire :402.57
  • M-COPA

    CAS :
    <p>M-COPA disrupts Golgi, blocks MET &amp; Arf1 activation, and inhibits angiogenesis via VEGFR &amp; NF-kB pathways.</p>
    Formule :C25H34N2O2
    Couleur et forme :Solid
    Masse moléculaire :394.55