Signalisation du cytosquelette
Les inhibiteurs de la signalisation du cytosquelette sont des composés qui perturbent les voies de signalisation régulant le cytosquelette, essentiel pour la forme, la motilité, la division des cellules et le transport intracellulaire. Ces inhibiteurs sont utilisés pour étudier la dynamique des protéines du cytosquelette, telles que l'actine et la tubuline, et leur rôle dans des processus comme la migration cellulaire, l'adhésion et la métastase du cancer. Les inhibiteurs de la signalisation du cytosquelette sont précieux dans la recherche en biologie cellulaire, en cancérologie et en neurobiologie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs de la signalisation du cytosquelette de haute qualité pour soutenir vos recherches dans ces domaines.
1381 produits trouvés pour "Signalisation du cytosquelette"
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BRD9876
CAS :<p>BRD9876 is a selective inhibitor of MM1S growth.</p>Formule :C16H14N2Degré de pureté :97.81%Couleur et forme :SolidMasse moléculaire :234.3Phorbol 12-myristate 13-acetate
CAS :<p>Phorbol 12-myristate 13-acetate (PMA) belongs to the phorbol ester group of natural products and is an activator of PKC, SphK, and NF-κB.</p>Formule :C36H56O8Degré de pureté :98.55% - >99.99%Couleur et forme :White To Off-White SolidMasse moléculaire :616.83Afuresertib hydrochloride
CAS :<p>Afuresertib hydrochloride is an inhibitor of Akt kinase (Kis of 0.08/2/2.6 nM for Akt1/Akt2/Akt3 respectively)</p>Formule :C18H18Cl3FN4OSDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :463.8Pyrintegrin
CAS :<p>Pyrintegrin: β1-integrin agonist, boosts embryonic stem cell survival, and podocyte protection, improves cell-matrix adhesion.</p>Formule :C23H25N5O3SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :451.54Uprosertib
CAS :<p>Uprosertib (GSK2141795) is a potent, selective Akt broad-spectrum inhibitor for Akt1/Akt2/Akt3.Cost-effective and quality-assured.</p>Formule :C18H16Cl2F2N4O2Degré de pureté :95.62% - 99.73%Couleur et forme :SolidMasse moléculaire :429.25TN-16
CAS :<p>TN-16 is a microtubule polymerization inhibitor (IC50 :0.4-1.7 μM)</p>Formule :C19H18N2O2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :306.36VER-49009
CAS :<p>VER-49009 (CCT 129397) is a potent Hsp90 inhibitor(IC50 of 25 nM and Kd of 78 nM).</p>Formule :C19H18ClN3O4Degré de pureté :99.36% - 99.99%Couleur et forme :SolidMasse moléculaire :387.82Leukadherin-1
CAS :<p>Leukadherin-1 boosts CD11b/CD18 adhesion, lowers leukocyte movement, cuts inflammation.</p>Formule :C22H15NO4S2Degré de pureté :98.49% - 98.93%Couleur et forme :SolidMasse moléculaire :421.49Gap 27
CAS :<p>Gap 27 is a peptide(Ser-Arg-Pro-Thr-Glu-Lys-Thr-Ile-Phe-Ile-Ile) derived from connexin 43 that is a selective gap junction blocker.</p>Formule :C60H101N15O17Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :1304.53Midostaurin
CAS :<p>PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.</p>Formule :C35H30N4O4Degré de pureté :97.61% - >99.99%Couleur et forme :SolidMasse moléculaire :570.64Cyclo(RGDyK) trifluoroacetate
CAS :<p>Cyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with IC50 of 20 nM.</p>Formule :C31H43F6N9O12Degré de pureté :95.28% - ≥95%Couleur et forme :SolidMasse moléculaire :847.72Recilisib sodium
CAS :<p>Recilisib (ON 01210.Na) is a radioprotective agent altering cancer cell cycles and preventing radiation-induced apoptosis.</p>Formule :C16H13ClNaO4SCouleur et forme :SolidMasse moléculaire :359.78AT7867
CAS :<p>AT7867 inhibits Akt1/2/3 & p70S6K/PKA (IC50: 32/17/47 nM & 85/20 nM), minimal effect beyond AGC kinases.</p>Formule :C20H20ClN3Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :337.85Vindesine sulfate
CAS :<p>Vindesine sulfate, a vinca alkaloid derived from vinblastine, binds to spindle microtubules, causing cell death.</p>Formule :C43H57N5O11SDegré de pureté :97.51%Couleur et forme :Amorphous SolidMasse moléculaire :8522',4'-DIHYDROXYCHALCONE
CAS :<p>2',4'-DIHYDROXYCHALCONE (2',4'-DHC) as a compound with Hsp90 inhibitory and antifungal effects</p>Formule :C15H12O3Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :240.25Spastazoline
CAS :<p>Spastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM ).</p>Formule :C20H30N8Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :382.51PU-H54
CAS :<p>PU-H54 is a purine-derived Grp94 inhibitor targeting the S2 subpocket's unique binding region.</p>Formule :C18H19N5SDegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :337.44TB500
CAS :<p>TB-500 is a synthesised peptide, essentially a short-chain version of the naturally occurring Thymosin Beta-4.</p>Formule :C38H68N10O14Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :889.01Smurf1-IN-A01
CAS :<p>Smurf1-IN-A01 is a potent Smurf1 inhibitor enhancing BMP-2, with a Kd of 3.664 nM, preventing Smad1/5 degradation.</p>Formule :C22H20ClF3N4O3SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :512.93TNIK-IN-2
CAS :<p>TNIK-IN-2 is an inhibitor Traf2- and Nck-interacting protein kinase (TNIK, IC50 = 1.33 μM)) which is a downstream signal protein of the Wnt/β-catenin pathway.</p>Formule :C22H19N3O3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :373.4Milnacipran ((1S-cis) hydrochloride)
CAS :<p>Milnacipran (1S-cis) hydrochloride (Levomilnacipran Hydrochloride) is a serotonin-norepinephrine reuptake inhibitor (SNRI), treatment of fibromyalgia.</p>Formule :C15H23ClN2ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :282.81AKT-IN-1
CAS :<p>AKT-IN-1 (AZD-26) is an allosteric AKT inhibitor (IC50: 1.04 μM).</p>Formule :C22H21N3ODegré de pureté :98.63%Couleur et forme :SolidMasse moléculaire :343.422-hydroxy Flutamide
CAS :<p>2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer</p>Formule :C11H11F3N2O4Degré de pureté :99.45% - 99.82%Couleur et forme :SolidMasse moléculaire :292.21NRX-252262
CAS :<p>NRX-252262 is a potent enhancer of the interaction between β-Catenin, and its cognate E3 ligase, SCFβ-TrCP, induces mutant β-catenin degradation(EC50：3.8 nM)</p>Formule :C23H17Cl2F3N2O4SDegré de pureté :98.94% - 99.87%Couleur et forme :SolidMasse moléculaire :545.36Dynasore
CAS :<p>Dynasore, a cell-permeable dynamin inhibitor, blocks GTPase of dynamin 1/2 and Drp1 (IC50: 15 μM) without affecting other small GTPases.</p>Formule :C18H14N2O4Degré de pureté :95.85% - 99.22%Couleur et forme :SolidMasse moléculaire :322.31HSP27 inhibitor J2
CAS :<p>HSP27 inhibitor J2 (J2) (J2) is a HSP27 inhibitor, inhibits a production of HSP27 giant polymers, thereby having an effect of inhibiting a chaperone function of</p>Formule :C13H12O4SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :264.3KBU2046
CAS :<p>KBU2046: oral anti-metastasis compound, enhances survival, targets chaperone complexes, not a typical HSP90 inhibitor.</p>Formule :C15H11FO2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :242.24Albendazole sulfoxide
CAS :Albendazole sulfoxide (Ricobendazole) is a metabolite of Albendazole, an anthelmintic.Formule :C12H15N3O3SDegré de pureté :97.29%Couleur et forme :White To Off-White PowderMasse moléculaire :281.33Onalespib
CAS :<p>Onalespib (AT13387) is an oral Hsp90 inhibitor with anticancer potential, disrupting tumor cell growth and survival.</p>Formule :C24H31N3O3Degré de pureté :98.05% - 99.66%Couleur et forme :SolidMasse moléculaire :409.52Capivasertib
CAS :<p>Capivasertib (AZD5363) is a broad-spectrum AKT inhibitor with inhibitory activity against Akt1, Akt2, and Akt3 (IC50=3/7/7 nM) with oral activity.</p>Formule :C21H25ClN6O2Degré de pureté :97.59% - 99.6%Couleur et forme :SolidMasse moléculaire :428.92TR-14035
CAS :<p>TR-14035 (MDK-1191) is a dual antagonist of α4β7/α4β1 integrins (IC50s: 7/87nM).</p>Formule :C24H21Cl2NO5Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :474.33Staurosporine
CAS :<p>Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-Fgr</p>Formule :C28H26N4O3Degré de pureté :99.24% - 99.82%Couleur et forme :Off-White PowderMasse moléculaire :466.53CK-869
CAS :<p>CK-869 is an Actin-Related Protein 2/3 (ARP2/3) complex inhibitor(IC50 of 7 μM),and is useful tools for the investigation of the Arp2/3 complex.</p>Formule :C17H16BrNO3SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :394.28Fingolimod
CAS :<p>Fingolimod (FTY-720A) is an antagonist of sphingosine 1-phosphate (S1P) (IC50 of 0.033 nM in K562 and NK cells).</p>Formule :C19H33NO2Degré de pureté :99.53% - 99.6%Couleur et forme :SolidMasse moléculaire :307.47Aficamten
CAS :<p>Aficamten is a Next-Generation Cardiac Myosin Inhibitor for the Treatment of Hypertrophic Cardiomyopathy.</p>Formule :C18H19N5O2Degré de pureté :99.19% - 99.57%Couleur et forme :SolidMasse moléculaire :337.38Cyclo(-RGDfK) TFA
CAS :<p>Cyclo(-RGDfK) is a selective αvβ3 integrin inhibitor(IC50 : 0.94 nM).</p>Formule :C29H42F3N9O9Degré de pureté :98.99% - 99.54%Couleur et forme :SolidMasse moléculaire :717.69Degrasyn
CAS :<p>Degrasyn (WP1130) inhibits DUBs (USP5, UCH-L1, USP9x, USP14, UCH37) and Bcr/Abl without affecting the 20S proteasome.</p>Formule :C19H18BrN3ODegré de pureté :98.32% - 99.98%Couleur et forme :SolidMasse moléculaire :384.27CWHM-12
CAS :<p>CWHM-12 is a potent inhibitor of αV integrins (IC50s of 0.2/0.8/1.5/1.8 nM for αvβ8/αvβ3/αvβ6/αvβ1).</p>Formule :C26H32BrN5O6Degré de pureté :98.05% - 99.83%Couleur et forme :SolidMasse moléculaire :590.47AZ13705339 hemihydrate
<p>AZ13705339 hemihydrate: potent PAK1 inhibitor (IC50: 0.33 nM), also binds PAK1/2 (Kd: 0.28/0.32 nM), for cancer research.</p>Formule :C33H36FN7O3SH2OCouleur et forme :SolidMasse moléculaire :638.77Pre-084
CAS :<p>Pre-084 is a high affinity, selective σ1 agonist.</p>Formule :C19H28ClNO3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :353.88D-ERYTHRO-SPHINGOSINE
CAS :<p>D-erythro-Sphingosine (trans-4-Sphingenine) is a protein kinase C (PKC) inhibitor. D-erythro-Sphingosine (Erythrosphingosine) is also a PP2A activator</p>Formule :C18H37NO2Degré de pureté :98% - 99.85%Couleur et forme :SolidMasse moléculaire :299.49Mps1-IN-3 hydrochloride
<p>Mps1-IN-3 HCl: potent Mps1 inhibitor (IC50: 50 nM), hampers glioblastoma growth, enhances vincristine efficacy in vivo.</p>Formule :C26H32ClN7O4SCouleur et forme :SolidMasse moléculaire :574.09PF-04929113 Mesylate
CAS :<p>PF-04929113 Mesylate (SNX-5422 Mesylate), a prodrug of SNX-2112, is an orally available Hsp90 inhibitor (Kd: 41 nM) and also induces Her-2 degradation (IC50: 37</p>Formule :C26H34F3N5O7SDegré de pureté :99% - 99.46%Couleur et forme :SolidMasse moléculaire :617.63Danegaptide Hydrochloride
CAS :<p>Danegaptide Hydrochloride (GAP-134 (Hydrochloride)) (GAP-134 Hydrochloride) is a selective modifier of the gap junction protein.</p>Formule :C14H18ClN3O4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :327.76GPRP acetate (67869-62-9 free base)
CAS :<p>GPRP acetate (Pefabloc FG) is fibrinogen-related peptides, which inhibit the interaction of fibrinogen with the platelet membrane glycoprotein IIbIIIa complex.</p>Formule :C20H35N7O7Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :485.53FRAX597
CAS :<p>FRAX597 is an effective, ATP-competitive inhibitor of group I PAKs, and for PAK1(IC50=8 nM), PAK2(IC50=13 nM), and PAK3 (IC50=19 nM).</p>Formule :C29H28ClN7OSDegré de pureté :97.34% - 99.85%Couleur et forme :SolidMasse moléculaire :558.1Nocodazole
CAS :<p>Nocodazole: synthetic microtubule polymerization blocker, also impedes Abl with low IC50; binds to beta-tubulin.</p>Formule :C14H11N3O3SDegré de pureté :98% - 99.91%Couleur et forme :Physical Description White Powder (Ntp 1992)Masse moléculaire :301.32SB-743921 hydrochloride
CAS :<p>SB-743921 hydrochloride (SB743921 HCl) is an effective inhibitor of kinesin spindle protein, KSP, (Ki =0.1 nM).</p>Formule :C31H34Cl2N2O3Degré de pureté :95.58% - 99.70%Couleur et forme :SolidMasse moléculaire :553.52DTHIB
CAS :<p>DTHIB robustly inhibits the HSF1 cancer gene signature and prostate cancer cell proliferation.</p>Formule :C13H9ClFN3O3Degré de pureté :98.86% - 99.29%Couleur et forme :SolidMasse moléculaire :309.68Wiskostatin
CAS :<p>Wiskostatin selectively inhibits N-WASP, key in actin polymerization, linked to Wiskott-Aldrich Syndrome.</p>Formule :C17H18Br2N2ODegré de pureté :99.84% - 99.97%Couleur et forme :White SolidMasse moléculaire :426.15KY-02327
CAS :<p>KY-02327: Stabilized KY-02061 analog, inhibits Dvl-CXXC5, activates Wnt/β-catenin, and promotes osteoblast differentiation.</p>Formule :C20H27N3O4Degré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :373.45HSP70-IN-1
CAS :<p>HSP70-IN-1 is a heat shock protein (HSP) inhibitor and inhibits the growth of Kasumi-1 cells (IC50: 2.3 μM).</p>Formule :C24H28N6O2SDegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :464.58Benproperine phosphate
CAS :<p>Benproperine phosphate (Pirexyl phosphate) is a cough suppressant.</p>Formule :C21H30NO5PDegré de pureté :99.84%Couleur et forme :PowderMasse moléculaire :407.44Rebastinib
CAS :<p>DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,</p>Formule :C30H28FN7O3Degré de pureté :99.53% - 99.79%Couleur et forme :SolidMasse moléculaire :553.59Tau protein (592-597), Human TFA
<p>Tau protein (592-597), Human (TFA) is a peptide fragment of human Tau protein.</p>Formule :C36H63F3N10O11Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :868.94Cilengitide
CAS :<p>Cilengitide (EMD 121974) is a potent integrin inhibitor for the αvβ3/5 receptor (IC50: 4.1/79 nM, in cell-free assays); ~10-fold selectivity against gpIIbIIIa.</p>Formule :C27H40N8O7Degré de pureté :98% - 99.8%Couleur et forme :SolidMasse moléculaire :588.66ZIP acetate(863987-12-6 free base)
<p>ZIP acetate inhibits PKMζ (protein kinase Mζ), affecting LTP maintenance and spatial memory, with an IC50 of 1-2.5 μM.</p>Formule :C92H158N30O19Degré de pureté :94.68%Couleur et forme :SolidMasse moléculaire :1988.43NSC45586
CAS :<p>NSC45586 is a protein phosphatase PHLPP inhibitor, which is selective for PHLPP1 and PHLPP2.</p>Formule :C20H18N6NaO3Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :413.4BIO-1211
CAS :<p>BIO-1211 is a more potent inhibitor of α4β1 (VLA-4, IC50 = 4 nM) over α4β7(IC50 = 2 μM).</p>Formule :C36H48N6O9Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :708.8Fasudil hydrochloride
CAS :<p>Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.</p>Formule :C14H18ClN3O2SDegré de pureté :99.54% - ≥95%Couleur et forme :White SolidMasse moléculaire :327.83PRE-084 hydrochloride
CAS :<p>PRE-084 hydrochloride is a selective agonist of σ1(IC50:44 nM, in the sigma receptor assay).</p>Formule :C19H28ClNO3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :353.88GNF-2
CAS :<p>GNF-2 is a highly selective non-ATP competitive inhibitor of Bcr-Abl.</p>Formule :C18H13F3N4O2Degré de pureté :98.17% - ≥95%Couleur et forme :SolidMasse moléculaire :374.32Tetradecyltrimethylammonium bromide
CAS :<p>Tetradecyltrimethylammonium bromide (MitMAB) is a Dynamin GTPase activity inhibitor and a cationic surfactant with asymmetrical structure.</p>Formule :C17H38BrNDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :336.39TRC051384 HCl
CAS :<p>TRC051384 is an inducer of heat shock protein Hsp70, activating heat shock factor-1 and enhancing Hsp72 expression in neurons and glial cells.</p>Formule :C25H32ClN5O4Degré de pureté :97.55%Couleur et forme :SolidMasse moléculaire :502.01Enzastaurin
CAS :<p>Enzastaurin (LY317615) (LY317615) is an effective PKCβ selective inhibitor (IC50: 6 nM), 6- to 20-fold selectivity against PKCα/γ/ε.</p>Formule :C32H29N5O2Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :515.6Daphnetin
CAS :<p>Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),</p>Formule :C9H6O4Degré de pureté :97.47% - 99.8%Couleur et forme :SolidMasse moléculaire :178.14S-trityl-L-Cysteine
CAS :<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Formule :C22H21NO2SDegré de pureté :97.02%Couleur et forme :Almost White To Light Yellow Granular PowderMasse moléculaire :363.47Suprafenacine
CAS :<p>Suprafenacine (N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide) is a cell-permeable microtubule destabilizer that induces</p>Formule :C16H18N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :282.34MK2-IN-1 hydrochloride
CAS :<p>MK2-IN-1 hydrochloride (MK 25) selectively inhibits MK2 with IC50 of 0.11 μM, non-ATP competitive.</p>Formule :C27H26Cl2N4O2Degré de pureté :97.32%Couleur et forme :SolidMasse moléculaire :509.43Irigenin
CAS :<p>Irigenin mediates its antimetastatic effect by specifically and selectively blocking the α9β1 and α4β1 integrin binding sites on the C-C loop of the Extra</p>Formule :C18H16O8Degré de pureté :99.50% - 99.85%Couleur et forme :SolidMasse moléculaire :360.31FRAX486 HCL(1232030-35-1 free base)
<p>FRAX486 HCL is a potent p21-activated kinase (PAK) inhibitor with IC50 values of 14, 33, 39 and 575 nM for PAK1, PAK2, PAK3 and PAK4 respectively.</p>Formule :C25H24Cl3FN6ODegré de pureté :98.85% - 99.82%Couleur et forme :SolidMasse moléculaire :549.86Sovilnesib
CAS :<p>Sovilnesib is a kinesin-like protein KIF18A inhibitor. Sovilnesib can be used for the cancer research.</p>Formule :C26H34F2N6O4SDegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :564.65HM03 trihydrochloride
CAS :<p>HM03 trihydrochloride is a potent and selective inhibitor of HSPA5, also known as Bip or Grp78. It exhibits anticancer activity.</p>Formule :C26H30Cl4N4O2Couleur et forme :SolidMasse moléculaire :572.35Arg-Gly-Asp TFA (99896-85-2(free base))
<p>Arg-Gly-Asp TFA (RGD, 99896-85-2) is a tripeptide that promotes cell adhesion and integrin binding.</p>Formule :C14H23F3N6O8Degré de pureté :99.2% - ≥98%Couleur et forme :SolidMasse moléculaire :460.36Clanfenur
CAS :<p>Clanfenur belongs to a new group of substituted benzoylphenylureas. The drug shows both in vitro and in vivo antitumour activity.</p>Formule :C16H15ClFN3O2Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :335.76Carotegrast methyl
CAS :<p>Carotegrast methyl (AJM300), an orally-active small molecule, can antagonize the α4 integrin receptor. It is a specific and dual α4β1/α4β7 integrin antagonist.</p>Formule :C28H26Cl2N4O5Degré de pureté :99.26% - 99.72%Couleur et forme :SolidMasse moléculaire :569.44Taurochenodeoxycholic acid sodium
CAS :<p>Sodium taurochenodeoxycholate: induces apoptosis, anti-inflammatory, boosts insulin, stimulates α2-cells, increases [Ca(2+)](c).</p>Formule :C26H44NNaO6SDegré de pureté :98.23% - 99.45%Couleur et forme :White To Off-White PowderMasse moléculaire :521.68GMB-475
CAS :<p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>Formule :C43H46F3N7O7SDegré de pureté :98.78% - >99.99%Couleur et forme :SolidMasse moléculaire :861.93MitoBloCK-10
CAS :<p>MitoBloCK-10 inhibits Tim44-Hsp70 binding; first to reduce PAM complex activity.</p>Formule :C12H8FN3O3SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :293.27PF-562271 besylate
CAS :<p>PF-562271 besylate: potent, ATP-competitive FAK inhibitor, IC50 1.5 nM, 10x less effective on Pyk2, highly selective vs other kinases.</p>Formule :C21H20F3N7O3S·C6H6O3SDegré de pureté :97.65% - 99.01%Couleur et forme :SolidMasse moléculaire :665.66Chelerythrine
CAS :<p>1.</p>Formule :C21H18NO4Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :348.37GW406108X(Z/E)
CAS :<p>GW406108X(Z/E) is a mixture of different configurations of GW406108X, which is an inhibitor of Kinesin-12 and ULK1 .</p>Formule :C20H11Cl2NO4Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :400.21Teprenone
CAS :<p>Teprenone (Geranylgeranylacetone) is a anti-ulcer drug, and works as an inducer of heat shock proteins (HSPs).</p>Formule :C23H38ODegré de pureté :99.1% - 99.96%Couleur et forme :SolidMasse moléculaire :330.55Go 6983
CAS :<p>Go 6983 is a PKC inhibitor with IC50 values of 7, 7, 6, 10, and 60 nM for PKCα, PKCβ, PKCγ, PKCδ, and PKCζ, respectively. High-Quality, Low-Cost!</p>Formule :C26H26N4O3Degré de pureté :98.41% - 99.85%Couleur et forme :SolidMasse moléculaire :442.51PF-04691502
CAS :<p>PF-04691502 is a potent and selective inhibitor of PI3K and mTOR kinases with antitumor activity.</p>Formule :C22H27N5O4Degré de pureté :96.27% - ≥95%Couleur et forme :SolidMasse moléculaire :425.48K858 (Racemic)
CAS :<p>K858 Racemic (K858) is a selective mitotic kinesin Eg5 inhibitor which acts in an ATP-noncompetitive manner.</p>Formule :C13H15N3O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :277.34CTX-0294885
CAS :<p>CTX-0294885, a bisanilino pyrimidine, inhibits many kinases; used for Sepharose-based kinase capture.</p>Formule :C22H24ClN7ODegré de pureté :98.73% - ≥95%Couleur et forme :SolidMasse moléculaire :437.931,2-Dimyristoyl-sn-glycerol
CAS :<p>1,2-Dimyristoyl-sn-glycerol (1,2-DMG) is able to increase AChE activity by 35-40% at concentrations of 25 micrograms/ml in the parasite S. mansoni..</p>Formule :C31H60O5Degré de pureté :99.96%Couleur et forme :White Powder With LumpsMasse moléculaire :512.81Olverembatinib dimesylate
CAS :<p>Olverembatinib dimesylate (GZD824 Dimesylate) is a novel orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT) and Bcr-Abl(T315I).</p>Formule :C29H27F3N6O·2CH4O3SDegré de pureté :97.66% - >99.99%Couleur et forme :SolidMasse moléculaire :724.77CW-069
CAS :<p>CW-069 (IC50=75 μM）, an allosteric selective inhibitor of microtubule motor protein HSET, exhibits remarkable specificity over KSP.</p>Formule :C23H21IN2O3Degré de pureté :97.52% - 99.52%Couleur et forme :SolidMasse moléculaire :500.33GRGDSP acetate(91037-75-1 free base)
<p>GRGDSP acetate(91037-75-1 free base) is a synthetic linear RGD peptide and is an integrin inhibitor.</p>Formule :C24H41N9O12Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :647.64Hispidin
CAS :<p>Hispidin is a polyphenol originally, including antioxidant, anti-inflammatory, and cytoprotective properties</p>Formule :C13H10O5Degré de pureté :98.27%Couleur et forme :White Crystalline PowderMasse moléculaire :246.22YS-49
CAS :<p>YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).</p>Formule :C20H20BrNO2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :386.28Grp94 Inhibitor-1
CAS :<p>Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).</p>Formule :C22H28N2O2Degré de pureté :97.02%Couleur et forme :SolidMasse moléculaire :352.47SU6656
CAS :<p>SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, 20 nM, 130 nM, and 170 nM for Src, Yes, Lyn, and Fyn, respectively.</p>Formule :C19H21N3O3SDegré de pureté :98.21% - 98.73%Couleur et forme :SolidMasse moléculaire :371.45AZ3146
CAS :<p>AZ3146 is a selective Mps1 inhibitor with IC50 of ~35 nM.</p>Formule :C24H32N6O3Degré de pureté :97.84% - >99.99%Couleur et forme :SolidMasse moléculaire :452.55FRAX1036
CAS :<p>FRAX-1036 is a effective and selective PAK1 inhibitor.</p>Formule :C28H32ClN7ODegré de pureté :97.66% - 98.67%Couleur et forme :SolidMasse moléculaire :518.05Bisindolylmaleimide I
CAS :<p>Bisindolylmaleimide I (GF109203X) is a potent and highly selective protein kinase C (PKC) inhibitor with a Ki of 14 nM.</p>Formule :C25H24N4O2Degré de pureté :98.19% - 98.75%Couleur et forme :Orange SolidMasse moléculaire :412.48KW-2449
CAS :<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Formule :C20H20N4ODegré de pureté :98.43% - 99.69%Couleur et forme :SolidMasse moléculaire :332.4NVP-BAW2881
CAS :<p>NVP-BAW2881 (BAW2881) is a potent and selective VEGFR inhibitor with activity to inhibit chronic and acute skin inflammation.</p>Formule :C22H15F3N4O2Degré de pureté :98.19% - 99.97%Couleur et forme :SolidMasse moléculaire :424.38
