
Récepteurs couplés à la protéine G et récepteurs 7-TM
Les récepteurs couplés aux protéines G (GPCRs) et les récepteurs à 7 domaines transmembranaires (7-TM) sont une grande famille de protéines membranaires qui jouent un rôle clé dans la communication cellulaire et la transduction des signaux. Ces récepteurs sont impliqués dans une large gamme de processus physiologiques, notamment la perception sensorielle, la réponse immunitaire et la régulation hormonale. Les GPCRs sont des cibles majeures dans la découverte de médicaments, ce qui les rend essentiels pour la recherche en pharmacologie et en médecine. Chez CymitQuimica, nous offrons une sélection complète de réactifs et de composés de haute qualité liés aux GPCRs et aux récepteurs 7-TM pour soutenir vos recherches et vos efforts de développement de médicaments.
5322 produits trouvés pour "Récepteurs couplés à la protéine G et récepteurs 7-TM"
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Latanoprostene bunod
CAS :<p>LBN is a NO-donating prostaglandin analog for reducing IOP in glaucoma or OHT patients.</p>Formule :C27H41NO8Degré de pureté :99.33% - 99.69%Couleur et forme :SolidMasse moléculaire :507.62Naftifine hydrochloride
CAS :<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Formule :C21H22ClNDegré de pureté :98.75% - 99.84%Couleur et forme :SolidMasse moléculaire :323.86Adenosine A1 receptor activator T62
CAS :<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formule :C15H14ClNOSDegré de pureté :97.83%Couleur et forme :SolidMasse moléculaire :291.8Nepafenac
CAS :<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Formule :C15H14N2O2Degré de pureté :98.94% - 99.43%Couleur et forme :SolidMasse moléculaire :254.28Dexpramipexole dihydrochloride
CAS :<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Formule :C10H19Cl2N3SDegré de pureté :99.75% - 99.88%Couleur et forme :SolidMasse moléculaire :284.25Ranitidine Hydrochloride
CAS :<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Formule :C13H23ClN4O3SDegré de pureté :99.30% - 99.49%Couleur et forme :SolidMasse moléculaire :350.86Volagidemab
CAS :<p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>Degré de pureté :97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)Couleur et forme :LiquidAsenapine Maleate
CAS :<p>Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.</p>Formule :C21H20ClNO5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :401.84Lafutidine
CAS :<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Formule :C22H29N3O4SDegré de pureté :98.55%Couleur et forme :Yellowish White Crystalline PowderMasse moléculaire :431.55Pamabrom
CAS :<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formule :C11H18BrN5O3Degré de pureté :99.84% - >99.99%Couleur et forme :CoaMasse moléculaire :348.2Brompheniramine maleate
CAS :<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Tetrabenazine
CAS :Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.Formule :C19H27NO3Degré de pureté :98% - 99.91%Couleur et forme :White To Off-White White To Off-White SolidMasse moléculaire :317.42NEO 376
CAS :<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formule :C20H24ClN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :357.88Loratadine
CAS :<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Formule :C22H23ClN2O2Degré de pureté :99.71% - 99.98%Couleur et forme :White PowderMasse moléculaire :382.88Bufotenidine hydrochloride(487-91-2 Free base)
CAS :<p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>Formule :C13H19ClN2ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :254.76Talipexole dihydrochloride
CAS :<p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>Formule :C10H17Cl2N3SDegré de pureté :99.89%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Cericlamine
CAS :<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Formule :C12H17Cl2NODegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :262.18N6-Ethyladenosine
CAS :<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formule :C12H17N5O4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :295.29Tropanserin
CAS :<p>Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.</p>Formule :C17H23NO2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :273.37SEP-363856 hydrochloride
CAS :<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formule :C9H14ClNOSDegré de pureté :99.86% - 99.99%Couleur et forme :SolidMasse moléculaire :219.73Cetirizine dihydrochloride
CAS :Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formule :C21H27Cl3N2O3Degré de pureté :99.4% - 99.97%Couleur et forme :SolidMasse moléculaire :461.81Ticagrelor
CAS :<p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>Formule :C23H28F2N6O4SDegré de pureté :98.08% - 99.77%Couleur et forme :SolidMasse moléculaire :522.57PHM-27 (human) acetate
<p>PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.</p>Formule :C137H215F3N34O42SDegré de pureté :99.20%Couleur et forme :SoildMasse moléculaire :3099.44Doxofylline
CAS :<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formule :C11H14N4O4Degré de pureté :99.958% - >99.99%Couleur et forme :SolidMasse moléculaire :266.25Clozapine
CAS :<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formule :C18H19ClN4Degré de pureté :99.91% - 99.93%Couleur et forme :Yellow Crystals From Acetone-Petroleum Ether SolidMasse moléculaire :326.82Efloxate
CAS :<p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>Formule :C19H16O5Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :324.33Triprolidine hydrochloride monohydrate
CAS :Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Formule :C19H25ClN2ODegré de pureté :99.68% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :332.87PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formule :C36H51Cl3N4O7SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :790.24p-MPPI hydrochloride
CAS :<p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Orphenadrine hydrochloride
CAS :<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Formule :C18H23NO·HClDegré de pureté :99.88%Couleur et forme :Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Masse moléculaire :305.85DPTN dihydrochloride
CAS :<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formule :C22H20Cl2N4OSDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :459.39PF-610355 HCl
<p>PF-610355 HCl is a selective and potent β2-adrenergic receptor agonist, a bronchodilator, and for asthma and chronic obstructive pulmonary disease.</p>Formule :C19H22ClN7O6Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :479.87Clomipramine hydrochloride
CAS :<p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>Formule :C19H23ClN2·HClDegré de pureté :99.04% - 99.47%Couleur et forme :White To Slightly Yellow Crystalline PowderMasse moléculaire :351.31Centanafadine hydrochloride
CAS :Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA 38 nM, serotonin 83 nM).Formule :C15H16ClNDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :245.75Mifentidine
CAS :<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Formule :C13H16N4Degré de pureté :98.34% - 99.73%Couleur et forme :SolidMasse moléculaire :228.29PF-04995274
CAS :<p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>Formule :C23H32N2O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :432.51Duloxetine hydrochloride
CAS :<p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>Formule :C18H20ClNOSDegré de pureté :99.93% - >99.99%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :333.88AB928
CAS :<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formule :C23H22N8ODegré de pureté :98.09% - >99.99%Couleur et forme :SolidMasse moléculaire :426.47(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS :<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Formule :C20H29N3O8Degré de pureté :99.72%Couleur et forme :SoildMasse moléculaire :439.46AM095 free acid
CAS :<p>AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).</p>Formule :C27H24N2O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :456.49GR 103691
CAS :<p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>Formule :C30H35N3O3Degré de pureté :98.94% - 99.29%Couleur et forme :SolidMasse moléculaire :485.62Venlafaxine hydrochloride
CAS :<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Formule :C17H28ClNO2Degré de pureté :97.32% - 99.86%Couleur et forme :White Crystalline PowderMasse moléculaire :313.86Mirabegron
CAS :<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formule :C21H24N4O2SDegré de pureté :99.64%Couleur et forme :Light Yellow To Yellow SolidMasse moléculaire :396.51Iloperidone
CAS :<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.482-Bromo-6-methoxynaphthalene
CAS :<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Formule :C11H9BrODegré de pureté :98.51%Couleur et forme :White To Off-White PowderMasse moléculaire :237.09JNJ-39758979
CAS :<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formule :C11H19N5Degré de pureté :98.33% - 99.62%Couleur et forme :SolidMasse moléculaire :221.3Imidazolidinyl urea
CAS :<p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>Formule :C11H16N8O8Degré de pureté :98.6%Couleur et forme :White Fluid Powder With Slight Characteristic OdorMasse moléculaire :388.29Latozinemab
<p>Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.</p>Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :146.28 kDaOzagrel
CAS :<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formule :C13H12N2O2Degré de pureté :97.90% - 99.38%Couleur et forme :White PowderMasse moléculaire :228.25Paliperidone
CAS :<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formule :C23H27FN4O3Degré de pureté :95% - 99.08%Couleur et forme :Off White To Light Orange Coloured SolidMasse moléculaire :426.48Lofepramine
CAS :<p>Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.</p>Formule :C26H27ClN2ODegré de pureté :98.38%Couleur et forme :Crystals From Methanol Or Acetone SolidMasse moléculaire :418.96PF-5190457
CAS :<p>PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).</p>Formule :C29H32N6OSDegré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :512.67L-741626
CAS :<p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>Formule :C20H21ClN2ODegré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :340.85Vilazodone
CAS :<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Formule :C26H27N5O2Degré de pureté :99.61%Couleur et forme :Light Yellow SolidMasse moléculaire :441.52Ondansetron hydrochloride dihydrate
CAS :<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Formule :C18H19N3O·HCl·2H2ODegré de pureté :99.92%Couleur et forme :White Crystal PowderMasse moléculaire :365.86Pramipexole
CAS :<p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>Formule :C10H17N3SDegré de pureté :98% - 99.96%Couleur et forme :SolidMasse moléculaire :211.33Pipamperone
CAS :<p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>Formule :C21H30FN3O2Degré de pureté :99.85%Couleur et forme :White PowderMasse moléculaire :375.48MP-A08
CAS :<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Formule :C27H25N3O4S2Degré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :519.64Azacyclonol
CAS :<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Formule :C18H21NODegré de pureté :99.46%Couleur et forme :Solid PowderMasse moléculaire :267.37Linaclotide
CAS :<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Formule :C59H79N15O21S6Degré de pureté :97.93% - 98.71%Couleur et forme :SolidMasse moléculaire :1526.74Astemizole
CAS :<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Formule :C28H31FN4ODegré de pureté :98.24% - 99.67%Couleur et forme :White Crystals SolidMasse moléculaire :458.57Cinnarizine
CAS :<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Formule :C26H28N2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :368.51CP-809101 hydrochloride
CAS :<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Formule :C15H18Cl2N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :341.24Senktide acetate
<p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>Formule :C42H59N7O13SDegré de pureté :98.26%Couleur et forme :SolidMasse moléculaire :902.02Mepyramine maleate
CAS :<p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>Formule :C21H27N3O5Degré de pureté :99.51% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :401.47Propafenone
CAS :<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Formule :C21H27NO3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :341.44Cisapride
CAS :<p>Cisapride (R 51619), a 5-HT4 agonist, enhances gut peristalsis and gastric emptying, reduces reflux.</p>Formule :C23H29ClFN3O4Degré de pureté :99.77%Couleur et forme :White To Slightly Biege Powder SolidMasse moléculaire :465.95Timonacic
CAS :<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Formule :C4H7NO2SDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :133.17Carbetapentane citrate
CAS :<p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>Formule :C20H31NO3·C6H8O7Degré de pureté :99.46%Couleur et forme :White To Off-White SolidMasse moléculaire :525.59(Rac)-MGV354
CAS :<p>(Rac)-MGV354: a racemic sGC activator; EC50s <0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>Formule :C35H37N5O3Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :575.7PF-06882961
CAS :<p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Formule :C31H30FN5O4Degré de pureté :98.06% - 99.54%Couleur et forme :SolidMasse moléculaire :555.6Rimonabant hydrochloride
CAS :<p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>Formule :C22H22Cl4N4ODegré de pureté :98.24% - 99.5%Couleur et forme :Off-White To White Crystalline PowderMasse moléculaire :500.25Atomoxetine hydrochloride
CAS :<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Formule :C17H22ClNODegré de pureté :99.86%Couleur et forme :White SolidMasse moléculaire :291.82Cloroperone
CAS :<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Formule :C22H23ClFNO2Degré de pureté :98.40%Couleur et forme :SoildMasse moléculaire :387.88Dexchlorpheniramine Maleate
CAS :<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Formule :C24H26F3N3O4Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :477.48Brefonalol HCl
<p>Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.</p>Formule :C22H29ClN2O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :388.93Apelin-13
CAS :<p>Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptor</p>Formule :C69H111N23O16SDegré de pureté :96.81%Couleur et forme :SolidMasse moléculaire :1550.83Bromopride
CAS :<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formule :C14H22BrN3O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :344.25Flopropione
CAS :<p>Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.</p>Formule :C9H10O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :182.17Metoclopramide hydrochloride
CAS :<p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>Formule :C14H22ClN3O2·HClDegré de pureté :99.99%Couleur et forme :White To Off-White PowderMasse moléculaire :336.26DREADD agonist 21
CAS :<p>DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).</p>Formule :C17H18N4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :278.35Hydroxyzine Pamoate
CAS :<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Formule :C44H43ClN2O8Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :763.27Famotidine
CAS :<p>Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.</p>Formule :C8H15N7O2S3Degré de pureté :98.93% - 99.91%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :337.45Evatanepag
CAS :<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formule :C25H28N2O5SDegré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :468.57(R)-Elagolix
CAS :<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Formule :C32H30F5N3O5Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :631.59Terazosin hydrochloride
CAS :<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Formule :C19H26ClN5O4Degré de pureté :99.69% - 99.91%Couleur et forme :SolidMasse moléculaire :423.89RS102895 hydrochloride
CAS :<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Formule :C21H22ClF3N2O2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :426.86(-)-GSK598809 hydrochloride
CAS :<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Formule :C22H24ClF4N5OSDegré de pureté :98.36%Couleur et forme :SoildMasse moléculaire :517.97Benserazide hydrochloride
CAS :<p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>Formule :C10H15N3O5·HClDegré de pureté :98.63% - 99.74%Couleur et forme :White Crystalline SolidMasse moléculaire :293.7Glycerol phenylbutyrate
CAS :<p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>Formule :C33H38O6Degré de pureté :98.54% - 99.74%Couleur et forme :SolidMasse moléculaire :530.65EMPA
CAS :<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Formule :C23H26N4O4SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :454.54Chlorprothixene hydrochloride
CAS :<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Formule :C18H18ClNS·HClDegré de pureté :99.76%Couleur et forme :White PowderMasse moléculaire :352.32Aniracetam
CAS :<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Formule :C12H13NO3Degré de pureté :99.88% - 99.89%Couleur et forme :White Crystalline Or Crystalline PowdeMasse moléculaire :219.24Carvedilol EP IMpurity E
CAS :<p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>Formule :C9H14ClNO2Degré de pureté :99.53%Couleur et forme :White To Almost White Solid CrystallineMasse moléculaire :203.666Acetophenazine dimaleate
CAS :<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Formule :C31H37N3O10SDegré de pureté :99.39% - 99.48%Couleur et forme :SolidMasse moléculaire :643.71Isoxsuprine hydrochloride
CAS :<p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>Formule :C18H24ClNO3Degré de pureté :99.38%Couleur et forme :Crystals From Water SolidMasse moléculaire :337.84Astressin acetate
<p>Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned</p>Formule :C163H273N49O44Degré de pureté :96.87%Couleur et forme :SolidMasse moléculaire :3623.21Phentolamine mesylate
CAS :<p>Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.</p>Formule :C17H19N3O·CH4O3SDegré de pureté :99.77% - >99.99%Couleur et forme :By The Metabolic Processes Of Bacillus Subtilis And LicheniformisMasse moléculaire :377.46Vabicaserin hydrochloride
CAS :<p>Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).</p>Formule :C15H21ClN2Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :264.79Moxisylyte hydrochloride
CAS :<p>Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.</p>Formule :C16H26ClNO3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :315.84Amiselimod hydrochloride
CAS :<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Formule :C19H31ClF3NO3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :413.9CYM 50769
CAS :<p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>Formule :C24H17ClN2O3Degré de pureté :98% - 99.08%Couleur et forme :SolidMasse moléculaire :416.86Indacaterol maleate
CAS :<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Formule :C28H32N2O7Degré de pureté :99.03% - 99.67%Couleur et forme :SolidMasse moléculaire :508.56Carteolol hydrochloride
CAS :<p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>Formule :C16H24N2O3·HClDegré de pureté :99.84% - 99.91%Couleur et forme :SolidMasse moléculaire :328.83Ro 10-5824 dihydrochloride
CAS :<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Formule :C17H22Cl2N4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :353.29AH 6809
CAS :<p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>Formule :C17H14O5Degré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :298.29Ramelteon
CAS :<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Formule :C16H21NO2Degré de pureté :97.21% - 99.92%Couleur et forme :Crystalline SolidMasse moléculaire :259.34Protriptyline hydrochloride
CAS :<p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>Formule :C19H21N·HClDegré de pureté :98.54% - 99.98%Couleur et forme :SolidMasse moléculaire :299.84Erenumab
CAS :<p>Erenumab: human antibody blocking CGRP receptors to prevent migraines.</p>Degré de pureté :99.43% (SEC-HPLC) - > 95%Couleur et forme :LiquidMasse moléculaire :146.2 kDaTiclopidine hydrochloride
CAS :<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formule :C14H15Cl2NSDegré de pureté :99.85% - >99.99%Couleur et forme :White PowderMasse moléculaire :300.25Adrenalone hydrochloride
CAS :<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Formule :C9H11NO3·HClDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :217.65Indusatumab
CAS :<p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145.18 kDaAnatibant 2HCl
CAS :<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formule :C34H36Cl2N6O5S·2ClHDegré de pureté :99.17% - 99.58%Couleur et forme :SoildMasse moléculaire :784.58Sonepcizumab
CAS :<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.90%Couleur et forme :LiquidMasse moléculaire :146.43 kDaBenztropine mesylate
CAS :<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Formule :C21H25NO·CH4SO3Degré de pureté :98.41% - 99.96%Couleur et forme :White Crystalline Powder; Odourless Or Almost OdourlessMasse moléculaire :403.53Nylidrin hydrochloride
CAS :<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Formule :C19H26ClNO2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :335.87Filorexant
CAS :<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Formule :C24H25FN4O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :420.48Roxatidine Acetate hydrochloride
CAS :<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Formule :C19H29ClN2O4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :384.9Labetalol hydrochloride
CAS :<p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>Formule :C19H25ClN2O3Degré de pureté :99.54% - 99.85%Couleur et forme :SolidMasse moléculaire :364.87Gevotroline
CAS :<p>Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.</p>Formule :C19H20FN3Degré de pureté :98.65%Couleur et forme :SolidMasse moléculaire :309.38Sergliflozin A
CAS :<p>Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.</p>Formule :C20H24O7Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :376.4Fezolinetant
CAS :<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Formule :C16H15FN6OSDegré de pureté :98.62% - 99.7%Couleur et forme :SolidMasse moléculaire :358.39Promethazine hydrochloride
CAS :<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formule :C17H20N2S·HClDegré de pureté :99.85%Couleur et forme :Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Masse moléculaire :320.88Rimonabant
CAS :<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formule :C22H21Cl3N4ODegré de pureté :98% - 99.91%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :463.79Ezlopitant
CAS :<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Formule :C31H38N2ODegré de pureté :97.49%Couleur et forme :SolidMasse moléculaire :454.65Blonanserin
CAS :<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.5Fluvoxamine maleate
CAS :<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Formule :C19H25F3N2O6Degré de pureté :99.92% - 99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :434.41ML-180
CAS :<p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>Formule :C20H25ClN4O2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :388.89Tetrahydrozoline
CAS :<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Formule :C13H16N2Degré de pureté :97.85% - 99.77%Couleur et forme :SolidMasse moléculaire :200.28Aripiprazole
CAS :<p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>Formule :C23H27Cl2N3O2Degré de pureté :99.43% - 99.62%Couleur et forme :Colourless Flake Crystalline SolidMasse moléculaire :448.39hGPR91 antagonist 1
CAS :<p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>Formule :C31H23F4N3ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :529.53Mizolastine
CAS :<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Formule :C24H25FN6ODegré de pureté :98% - 99.75%Couleur et forme :SolidMasse moléculaire :432.49Quetiapine hemifumarate
CAS :Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formule :C46H54N6O8S2Degré de pureté :99.32% - >99.99%Couleur et forme :White Crystalline SolidMasse moléculaire :883.09Dimenhydrinate
CAS :<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Formule :C24H28ClN5O3Degré de pureté :99.57% - 99.77%Couleur et forme :Crystals Physical Description Crystalline White Powder (Ntp 1992)Masse moléculaire :469.96Cefaclor monohydrate
CAS :<p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>Formule :C15H16ClN3O5SDegré de pureté :97.36% - 99.9%Couleur et forme :White Crystaling PowderMasse moléculaire :385.82Acebutolol hydrochloride
CAS :<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Formule :C18H29ClN2O4Degré de pureté :99.92% - >99.99%Couleur et forme :White Or Slightly Off-White Crystalline Powder SolidMasse moléculaire :372.89Fenspiride hydrochloride
CAS :<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formule :C15H20N2O2·HClDegré de pureté :99.64% - 99.92%Couleur et forme :SolidMasse moléculaire :296.79Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Degré de pureté :97.76%Couleur et forme :SoildCarbinoxamine Maleate Salt
CAS :<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Formule :C20H23ClN2O5Degré de pureté :99.97%Couleur et forme :Off-White SolidMasse moléculaire :406.86Deoxycholic acid
CAS :<p>Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.</p>Formule :C24H40O4Degré de pureté :99.91% - 99.91%Couleur et forme :Crystals From Alc SolidMasse moléculaire :392.57Prochlorperazine Maleate
CAS :<p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>Formule :C28H32ClN3O8SDegré de pureté :99.78%Couleur et forme :Off-White PowderMasse moléculaire :606.09Talastine
CAS :<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Formule :C19H21N3ODegré de pureté :98.50% - 99.44%Couleur et forme :SolidMasse moléculaire :307.39Dopexamine hydrochloride
CAS :<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Formule :C22H34Cl2N2O2Degré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :429.42Clonidine hydrochloride
CAS :<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Formule :C9H10Cl3N3Degré de pureté :99.16% - 99.86%Couleur et forme :SolidMasse moléculaire :266.55Levocetirizine
CAS :<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Formule :C21H25ClN2O3Degré de pureté :98% - 99.9%Couleur et forme :White PowderMasse moléculaire :388.89NF-56-EJ40 hydrochloride
CAS :<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Formule :C27H31Cl2N3O3Degré de pureté :99.33%Couleur et forme :SoildMasse moléculaire :516.46Anamorelin
CAS :<p>Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).</p>Formule :C31H42N6O3Degré de pureté :99.35% - 99.94%Couleur et forme :SolidMasse moléculaire :546.7SR59230A
CAS :<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Formule :C23H29NO6Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :415.48Tripelennamine hydrochloride
CAS :<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Formule :C16H21N3·HClDegré de pureté :99.54% - 99.81%Couleur et forme :White SolidMasse moléculaire :291.82Fluparoxan hydrochloride
CAS :<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formule :C10H11ClFNO2Degré de pureté :99.98%Couleur et forme :SoildMasse moléculaire :231.65Terlipressin Acetate
CAS :<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Formule :C56H82N16O19S2Degré de pureté :98.50% - 99.69%Couleur et forme :SolidMasse moléculaire :1347.5Silodosin
CAS :<p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>Formule :C25H32F3N3O4Degré de pureté :99.282% - 99.76%Couleur et forme :Colorless To Pink SolidMasse moléculaire :495.53Metaproterenol hemisulfate
CAS :<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Formule :C11H17NO3·5H2O4SDegré de pureté :98.53% - 99.74%Couleur et forme :SolidMasse moléculaire :260.3Oxeladin citrate
CAS :<p>Oxeladin citrate: potent, non-addictive cough suppressant safe for all ages and heart patients; no common antitussive side effects.</p>Formule :C26H41NO10Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :527.6Desipramine hydrochloride
CAS :<p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>Formule :C18H23ClN2Degré de pureté :99.58% - 99.94%Couleur et forme :White To Off-White PowderMasse moléculaire :302.842Evocalcet
CAS :<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Formule :C24H26N2O2Degré de pureté :98.88% - 99.68%Couleur et forme :SolidMasse moléculaire :374.48Zolmitriptan
CAS :<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36Azatadine dimaleate
CAS :<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Formule :C28H30N2O8Degré de pureté :99.7% - >99.99%Couleur et forme :PowderMasse moléculaire :522.55LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Formule :C30H58ClN7O8SDegré de pureté :98.02% - 99.31%Couleur et forme :SolidMasse moléculaire :712.34Doxylamine succinate
CAS :<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formule :C21H28N2O5Degré de pureté :99.61%Couleur et forme :5 1 (Ntp 1992)Masse moléculaire :388.46Noradrenaline bitartrate
CAS :<p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>Formule :C12H19NO10Degré de pureté :99.53% - >99.99%Couleur et forme :SolidMasse moléculaire :337.28(3aR,9aR)-Fluparoxan
CAS :<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formule :C10H10FNO2Degré de pureté :97.82%Couleur et forme :SoildMasse moléculaire :195.19Frovatriptan succinate hydrate
CAS :<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Formule :C18H25N3O6Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :379.41Alarelin Acetate
CAS :<p>Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.</p>Formule :C56H78N16O12Degré de pureté :99.81% - >99.99%Couleur et forme :White PowderMasse moléculaire :1167.34Bambuterol hydrochloride
CAS :<p>Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.</p>Formule :C18H30ClN3O5Degré de pureté :99.53% - 99.61%Couleur et forme :White SolidMasse moléculaire :403.91Methoxamine hydrochloride
CAS :<p>Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.</p>Formule :C11H18ClNO3Degré de pureté :99.84% - >99.99%Couleur et forme :Colorless Or White Plate-Like Crystals Or White Crystalline Powder SolidMasse moléculaire :247.719Tiapride hydrochloride
CAS :<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Formule :C15H24N2O4S·HClDegré de pureté :99.4% - 99.77%Couleur et forme :SolidMasse moléculaire :364.89Degarelix acetate(214766-78-6 free base)
CAS :<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formule :C84H107ClN18O18Degré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :1692.34Olinciguat
CAS :<p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>Formule :C21H16F5N7O3Degré de pureté :99.33% - 99.71%Couleur et forme :SolidMasse moléculaire :509.39Ziprasidone
CAS :<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formule :C21H21ClN4OSDegré de pureté :99.55%Couleur et forme :Tan SolidMasse moléculaire :412.94JP1302 dihydrochloride
CAS :<p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>Formule :C24H26Cl2N4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :441.4Sulpiride
CAS :<p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>Formule :C15H23N3O4SDegré de pureté :99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Loxapine succinate
CAS :<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.9BIBO3304 TFA
CAS :<p>BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).</p>Formule :C31H36F3N7O5Degré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :643.66CD80-IN-3
CAS :<p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>Formule :C17H10FN3O3Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :323.28Fosopamine(HCl)
CAS :<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Formule :C9H15ClNO5PDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :283.65Methyldopa
CAS :<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Formule :C10H13NO4Degré de pureté :98.95% - 99.86%Couleur et forme :Less Or Almost Colorless Crystals Or White To Yellowish-White FineMasse moléculaire :211.21(±) Clopidogrel hydrogen sulfate
CAS :<p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>Formule :C16H16ClNO2S·H2SO4Degré de pureté :98.67% - 99.04%Couleur et forme :Colorless To Light Yellow LiquidMasse moléculaire :419.9YNT-185
CAS :<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Formule :C33H37N5O5SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :615.74Desvenlafaxine
CAS :<p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>Formule :C16H25NO2Degré de pureté :99.46% - 99.81%Couleur et forme :White Crystalline PowderMasse moléculaire :263.38Ziprasidone hydrochloride monohydrate
CAS :<p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>Formule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12Trimipramine maleate
CAS :<p>Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.</p>Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51TSHR antagonist S37
CAS :<p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>Formule :C25H20N2O3S2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :460.57KGA-2727
CAS :<p>KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.</p>Formule :C26H40N4O8Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :536.62Phenothiazine
CAS :<p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>Formule :C12H9NSDegré de pureté :99.95%Couleur et forme :Yellow Solid PelletsMasse moléculaire :199.27Antazoline hydrochloride
CAS :<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Formule :C17H19N3·HClDegré de pureté :98% - 99.53%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :301.82Fexofenadine hydrochloride
CAS :<p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>Formule :C32H40ClNO4Degré de pureté :>99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :538.12Proglumide
CAS :<p>Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.</p>Formule :C18H26N2O4Degré de pureté :99.4% - 99.45%Couleur et forme :White Crystalline PowderMasse moléculaire :334.41Pericyazine
CAS :<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formule :C21H23N3OSDegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :365.49Levosulpiride
CAS :<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Formule :C15H23N3O4SDegré de pureté :98.20% - 99.88%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Xylometazoline hydrochloride
CAS :<p>Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.</p>Formule :C16H24N2·HClDegré de pureté :99.77% - 99.87%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :280.84Agomelatine
CAS :<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formule :C15H17NO2Degré de pureté :99.92%Couleur et forme :White SolidMasse moléculaire :243.3Mefexamide hydrochloride
CAS :<p>Mefexamide hydrochloride is a central stimulant.</p>Formule :C15H25ClN2O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :316.83Trazodone hydrochloride
CAS :<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Formule :C19H23Cl2N5ODegré de pureté :99.5% - 99.52%Couleur et forme :SolidMasse moléculaire :408.33Granisetron hydrochloride
CAS :<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Formule :C18H25ClN4ODegré de pureté :99.88% - 99.93%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :348.87Levodropropizine
CAS :<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Formule :C13H20N2O2Degré de pureté :99.87% - 99.93%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.312-(1-Piperazinyl)pyrimidine
CAS :<p>2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.</p>Formule :C8H12N4Degré de pureté :98.46%Couleur et forme :Liquid - Crystal - LumpMasse moléculaire :164.21Salmeterol
CAS :<p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>Formule :C25H37NO4Degré de pureté :99.2% - 99.9%Couleur et forme :SolidMasse moléculaire :415.57Tolnaftate
CAS :<p>Tolnaftate (NP-27) is a synthetic antifungal agent.</p>Formule :C19H17NOSDegré de pureté :98.85%Couleur et forme :White PowderMasse moléculaire :307.41

