
Alpha-bloquants
Les alpha-bloquants sont des composés pharmaceutiques qui agissent en inhibant l'activité des récepteurs alpha-adrénergiques, responsables de la contraction des muscles lisses. Ces médicaments sont couramment utilisés pour traiter des affections telles que l'hypertension artérielle et l'hyperplasie bénigne de la prostate, en provoquant la relaxation et la dilatation des vaisseaux sanguins. Chez CymitQuimica, nous proposons une gamme d'alpha-bloquants adaptés à la recherche en pharmacologie et en santé cardiovasculaire.
658 produits trouvés pour "Alpha-bloquants"
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S-Mirtazapine
CAS :Produit contrôlé<p>Applications S-Mirtazapine is an enantiomer of Mirtazapine (M365000); an antidepressant. R-Mirtazapine showed antinociceptive effects in acute thermal nociception, whereas S-Mirtazapine showed pronociceptive effects.<br>References Muth-Selbach, Uta., et al.: Brain Res. Bull., 79(1), 63-68 (2009); Smith, Donald F., et al.: Psychopharmacology, 200(2), 273-279 (2008); Freynhagen, Rainer., et al.: Brain Res. Bull., 69(2), 168-173 (2006)<br></p>Formule :C17H19N3Couleur et forme :NeatMasse moléculaire :265.356,7,8,9-Tetrahydro Carvedilol
CAS :Produit contrôlé<p>Applications Carvedilol (C184625) derivative.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Formule :C24H30N2O4Couleur et forme :NeatMasse moléculaire :410.51Carvedilol
CAS :Produit contrôlé<p>Applications Carvedilol is a nonselective β-adrenergic blocker with α1-blocking activity. Carvedilol is an antihypertensive used in the treatment of congestive heart failure.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990); Packer, M., et al.: N. Engl. J. Med., 334, 1349 (1996);<br></p>Formule :C24H26N2O4Couleur et forme :WhiteMasse moléculaire :406.47(R)-(+)-Carvedilol
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications The optically active isomer of Carvedilol (C184625), a nonselective ß-adrenergic blocker with a1-blocking activity. An antihypertensive used in the treatment of congestive heart failure.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990),<br></p>Formule :C24H26N2O4Couleur et forme :Off White SolidMasse moléculaire :406.47Tamsulosin
CAS :<p>Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.</p>Formule :C20H28N2O5SDegré de pureté :99.93%Couleur et forme :White CrystalsMasse moléculaire :408.514-(2,3-Epoxypropoxy)carbazole
CAS :Produit contrôlé<p>Impurity Carvedilol EP Impurity D; Carvedilol USP-D<br>Applications 4-(2,3-Epoxypropoxy)carbazole (Carvedilol EP Impurity D; Carvedilol USP-D) is an intermediate in the synthesis of Carvedilol (C184625).<br></p>Formule :C15H13NO2Couleur et forme :Beige SolidMasse moléculaire :239.272-(2-Ethoxyphenoxy)ethanamine
CAS :Produit contrôlé<p>Impurity Tamsulosin EP Impurity F<br>Applications 2-(2-Ethoxyphenoxy)ethanamine (Tamsulosin EP Impurity F) is an impurity of Tamsulosin (T006350), a specific α1-adrenoceptor antagonist (1,2). It is used in the treatment of benign prostatic hypertrophy.<br>References 1. Kawabe, K. et al.: J. Urol. 1990 Oct;144(4):908-11;2. Abrams, P. et al.: Br. J. Urol. 1995 Sep;76(3):325-36.<br></p>Formule :C10H15NO2Couleur et forme :NeatMasse moléculaire :181.23Carvedilol-d3
CAS :Produit contrôléFormule :C242H3H23N2O4Couleur et forme :Off WhiteMasse moléculaire :409.498-Hydroxy Mirtazapine β-D-Glucuronide 90%
CAS :<p>Applications A metabolite of Mirtazapine (M365000). This compounds contains some of the alpha anomer.<br>References Sandker, G., et al.: Xenobiotica, 24, 143 (1994), Dahl, M., et al.: Clin. Drug Invest., 13, 37 (1997),<br></p>Formule :C23H27N3O7Degré de pureté :90%Couleur et forme :NeatMasse moléculaire :457.485-Formyl-2-methoxy-benzenesulfonamide
CAS :Produit contrôlé<p>Impurity Tamsulosin EP Impurity E<br>Applications 5-Formyl-2-methoxy-benzenesulfonamide (Tamsulosin EP Impurity E) is an impurity of Tamsulosin (T006350), a specific α1-adrenoceptor antagonist used in the treatment of benign prostatic hypertrophy.<br>References Kawabe, K., et al.: J. Urol., 144, 908 (1990), Abrams, P., et al.: Br. J. Urol., 76, 325 (1995), Michel, M.C., Expert Opin. Pharmacother., 5, 151 (2004),<br></p>Formule :C8H9NO4SCouleur et forme :NeatMasse moléculaire :215.231-(3-Carboxy-2-pyridyl)-4-methyl-2-phenylpiperazine
CAS :Produit contrôlé<p>Applications Mirtazapine (M365000) impurity.<br>References Reddy, T. et al.; J. Liq. Chromatogr. R. T. 31, 1204 (2008)<br></p>Formule :C17H19N3O2Couleur et forme :NeatMasse moléculaire :297.353-Hydroxy Carvedilol
CAS :Produit contrôlé<p>Applications A vascularly inactive metabolite of Carvedilol (C184625). A novel antihypertensive agent, is a potent antioxidant.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Rapola, J., et al.: Lancet, 349, 1715 (1997), Gao, F., et al.: Eur. J. Pharmacol., 406, 109 (2000),<br></p>Formule :C24H26N2O5Couleur et forme :NeatMasse moléculaire :422.472-(2-Methoxyphenoxy)ethylamine Hydrochloride
CAS :<p>Impurity Carvedilol EP Impurity E; Carvedilol Impurity E; Carvedilol USP E<br>Applications 2-(2-Methoxyphenoxy)ethylamine Hydrochloride (Carvedilol EP Impurity E; Carvedilol Impurity E; Carvedilol USP E) is an impurity of Carvedilol synthesis.<br>References Smith, L., et al.: J. Med. Chem., 20, 1653 (1977),<br></p>Formule :C9H13NO2·ClHCouleur et forme :NeatMasse moléculaire :203.67Carvedilol-d5
CAS :Produit contrôlé<p>Applications Carvedilol-d5 is the labelled analog of Carvedilol, a nonselective β-adrenergic blocker with α1-blocking activity. Carvedilol is an antihypertensive used in the treatment of congestive heart failure.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hirohashi, M., et al.: Arzneim.-Forsch., 40, 735 (1990), Packer, M., et al.: N. Engl. J. Med., 334, 1349 (1996),<br></p>Formule :C24H21D5N2O4Couleur et forme :NeatMasse moléculaire :411.51Silodosin
CAS :<p>Applications Silodosin is an α1a-adrenoceptor antagonist. It is used in treatment of benign prostatic hypertrophy.<br>References (1) Shibata, K., et al.: Mol. Pharmacol., 48, 250 (1995) (2) Murata, S., et al.: J. Urol., 164, 578 (2000)<br></p>Formule :C25H32F3N3O4Couleur et forme :NeatMasse moléculaire :495.53Carvedilol Bis-carbazole
CAS :Produit contrôlé<p>Impurity Carvedilol EP Impurity B; Carvedilol Impurity B; Carvedilol USP B<br>Applications Carvedilol Bis-carbazole (Carvedilol EP Impurity B; Carvedilol Impurity B; Carvedilol USP B) is an impurity from the process of Carvedilol (C184625).<br></p>Formule :C39H39N3O6Couleur et forme :Off-White To Light BeigeMasse moléculaire :645.74O-Desmethyl Carvedilol
CAS :Produit contrôlé<p>Applications A metabolite of Carvedilol (C184625), a nonselective β-adrenergic blocker with α1-blocking activity.<br>References Sponer, G., et al.: J. Cardiovasc. Pharmacol., 9, 317 (1987), Fujimaki, M., et al.: Xenobiotica, 20, 1025 (1990), Ruffolo, R., et al.: Eur. J. Clin. Pharmacol., 38, S82 (1990), Clohs, L., et al.: J. Pharm. Biomed. Anal., 31, 407 (2003),<br></p>Formule :C23H24N2O4Couleur et forme :NeatMasse moléculaire :392.45Carvedilol N’-2-Hydroxy-3-[[2-(methoxyphenoxy)ethyl]amine
CAS :Produit contrôlé<p>Impurity Carvedilol Impurity A; Carvedilol USP A<br>Applications An impurity from the process of Carvedilol (C184625). Carvedilol impurity A. Carvedilol USP A.<br></p>Formule :C36H43N3O7Couleur et forme :NeatMasse moléculaire :629.74Mirtazapine-d3
CAS :Produit contrôlé<p>Applications An α2-Adrenergic blocker; analogue of Mianserin. Antidepressant.<br>References De Boer, T., et al.: Neuropharmacology, 27, 399 (1988), Smith, W.T., et al.: Psychopharmacol. Bull., 26, 191 (1990)<br></p>Formule :C172H3H16N3Couleur et forme :White To BeigeMasse moléculaire :268.37


