Dérivés de Quinazoline et de Quinoléine
Les quinazolines et les quinoléines sont des composés hétérocycliques azotés à structure aromatique qui jouent un rôle clé dans la synthèse de médicaments à activité anticancéreuse, antimicrobienne et anti-inflammatoire. Leurs dérivés présentent des modifications structurelles qui optimisent leur biodisponibilité et leur sélectivité, permettant ainsi le développement de nouveaux principes actifs pour diverses applications thérapeutiques. Ces composés sont utilisés dans la fabrication d’API destinés au traitement du cancer, des infections, des maladies neurodégénératives et cardiovasculaires. De plus, les dérivés de quinazoline et de quinoléine sont essentiels dans la recherche d’inhibiteurs enzymatiques et dans la conception de molécules bioactives innovantes.
Chez CymitQuimica, nous proposons des dérivés de quinazoline et de quinoléine de haute pureté pour des applications en synthèse chimique, développement pharmaceutique et biotechnologie.
65576 produits trouvés pour "Dérivés de Quinazoline et de Quinoléine"
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Selatinib
CAS :<p>Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer activity that inhibits the growth of NCI-N87 tumor cells.</p>Formule :C29H26ClFN4O3SDegré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :565.06Vasicinone
CAS :<p>Vasicinone may act as a hepatoprotective agent.</p>Formule :C11H10N2O2Degré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :202.21Hemustine
CAS :<p>Hemustine is an inhibitor of human glutathione reductase and widely used as an anti-tumor agent.</p>Formule :C5H10ClN3O3Couleur et forme :SolidMasse moléculaire :195.6Blonanserin HCl
CAS :<p>Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.</p>Formule :C23H32Cl2FN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.42Gilteritinib hemifumarate
CAS :<p>Gilteritinib hemifumarate (ASP2215 hemifumarate) is a potent ATP-competitive dual FLT3 (IC50: 0.29 nM) and AXL (IC50: 0.73 nM) inhibitor for the treatment of</p>Formule :C29H44N8O3C4H4O4Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :610.75Thiochrome
CAS :<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Formule :C12H14N4OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.33(S)-Hydroxychloroquine
CAS :<p>(S)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine shows efficiently inhibits SARS-CoV-2 infection in vitro.</p>Formule :C18H26ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :335.87cis-Tadalafil
CAS :<p>Cis-Tadalafil is a potent inhibitor of phosphodiesterase 5, which is used to treat erectile dysfunction (ED) and primary pulmonary hypertension (PPH). It works by increasing blood flow to the penis, allowing men with ED to achieve and maintain an erection. Cis-Tadalafil is also used to treat symptoms of prostatic hyperplasia (enlarged prostate) in men. This drug has been shown to be effective in treating PPH by reducing pulmonary arterial pressure and improving exercise capacity. Cis-Tadalafil belongs to the carboline class of drugs and is a phosphodiesterase 5 inhibitor that selectively inhibits cGMP-specific phosphodiesterase type 5 (PDE5). This drug has been shown to be highly effective in treating both ED and PPH with minimal side effects.</p>Formule :C22H19N3O4Degré de pureté :Min. 95%Couleur et forme :White/Off-White SolidMasse moléculaire :389.4 g/molCarisbamate
CAS :<p>CarisbAMate (JNJ-10234094, RWJ 333369, YKP-509) is an antiepileptic drug candidate.</p>Formule :C9H10ClNO3Couleur et forme :SolidMasse moléculaire :215.63Palonosetron
CAS :<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Formule :C19H24N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.41Clofedanol
CAS :<p>Clofedanol, also known as chlophedianol or antitussin, is used in the treatment of pediatric pertussis.</p>Formule :C17H20ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :289.8(R)-ND-336
CAS :<p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>Formule :C16H18ClNO3S2Couleur et forme :SolidMasse moléculaire :371.89BR351
CAS :<p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Formule :C20H25FN2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.49Rufloxacin hydrochloride
CAS :<p>Rufloxacin HCl (MF-934 HCl): a fluoroquinolone that inhibits topoisomerase and B-cell differentiation.</p>Formule :C17H19ClFN3O3SDegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :399.867Alimemazine
CAS :<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Formule :C18H22N2SDegré de pureté :98%Couleur et forme :Crystals SolidMasse moléculaire :298.45Bifeprunox Mesylate
CAS :<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Formule :C25H27N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.56(S)-Azelastine
CAS :<p>(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.</p>Formule :C22H24ClN3OCouleur et forme :SolidMasse moléculaire :381.9PTIQ
CAS :<p>MMP-3 expression inhibitor</p>Formule :C13H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :235.28RS-104966
CAS :<p>RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.</p>Formule :C19H21NO6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.44U 27391
CAS :<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Formule :C23H36N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.56PF-00356231 hydrochloride
CAS :<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Formule :C25H21ClN2O3SDegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :464.96Enadoline (Free Base)
CAS :<p>Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.</p>Formule :C24H32N2O3Couleur et forme :SolidMasse moléculaire :396.52Otamixaban
CAS :<p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>Formule :C25H26N4O4Degré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :446.5(R,R)-Glycopyrrolate
CAS :<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Formule :C19H28BrNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :398.34Midodrine (R-isomer HCl)
CAS :<p>Midodrine is a vasopressor/antihypertensive agent for the treatment of symptomatic postural hypotension.</p>Formule :C12H19ClN2O4Couleur et forme :SolidMasse moléculaire :290.74BP-5-087
CAS :<p>BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.</p>Formule :C36H30F8N2O6SCouleur et forme :SolidMasse moléculaire :770.69Pridinol
CAS :<p>Pridinol is an antispasmodic and muscle relaxant.</p>Formule :C20H25NODegré de pureté :98%Couleur et forme :Crystals SolidMasse moléculaire :295.42Esreboxetine
CAS :<p>Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.</p>Formule :C19H23NO3Couleur et forme :SolidMasse moléculaire :313.39Zuclopenthixol decanoate
CAS :<p>Zuclopenthixol decanoate is an anti-schizophrenia drug.</p>Formule :C32H43ClN2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :555.21Indisetron Dihydrochloride
CAS :<p>Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.</p>Formule :C17H24ClN5OCouleur et forme :SolidMasse moléculaire :349.86Propoxur
CAS :<p>Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; carcinogenicity unclassified by EPA.</p>Formule :C11H15NO3Degré de pureté :99.84% - 99.87%Couleur et forme :Minute Crystals (Niosh 2016)Masse moléculaire :209.24GW-3333
CAS :<p>GW-3333 inhibits matrix metalloproteinases and TNF-Converting Enzyme, showing potential as an antiarthritic therapy.</p>Formule :C22H36N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.55Camylofine
CAS :<p>Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.</p>Formule :C19H32N2O2·2HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.4ABT-770
CAS :<p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>Formule :C22H22F3N3O6Couleur et forme :SolidMasse moléculaire :481.42MMP-1-IN-1
<p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>Formule :C14H17ClN2O3Couleur et forme :SolidMasse moléculaire :296.75NNGH
CAS :<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Formule :C13H20N2O5SDegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :316.37Enflicoxib
CAS :<p>Enflicoxib is an effective treatment for canine osteoarthritis pain and inflammation, with faster onset than mavacoxib, improving veterinary outcomes.</p>Formule :C16H12F5N3O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :405.34Ketotifen
CAS :<p>Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.</p>Formule :C19H19NOSCouleur et forme :SolidMasse moléculaire :309.43Phenindamine Tartrate
CAS :<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Formule :C23H25NO6Couleur et forme :SolidMasse moléculaire :411.454Hexazinone
CAS :<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Formule :C12H20N4O2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :252.31Lanicemine
CAS :<p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>Formule :C13H14N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :198.26(Rac)-Tanomastat
CAS :<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Formule :C23H19ClO3SCouleur et forme :SolidMasse moléculaire :410.91Ingavirin
CAS :<p>Ingavirin, a novel inhibitor of the influenza virus reproduction, inhubits the formation of the virus specific hemagglutinin.</p>Formule :C10H15N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :225.24Mesopram
CAS :<p>PDE4 inhibitor, orally active</p>Formule :C14H19NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.3AZD5248
CAS :<p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>Formule :C22H22N4O2Couleur et forme :SolidMasse moléculaire :374.44TAPI-1
CAS :<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Formule :C26H37N5O5Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :499.6Benzatropine
CAS :<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Formule :C21H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.43Nifekalant hydrochloride
CAS :<p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>Formule :C19H28ClN5O5Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :441.91Gallopamil hydrochloride
CAS :<p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>Formule :C28H41ClN2O5Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :521.09Levobetaxolol
CAS :<p>Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.</p>Formule :C18H29NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.43Tanomastat
CAS :<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Formule :C23H19ClO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.91Robenidine
CAS :<p>Robenidine, an anticoccidial guanidine, is used as an additive in rabbit fodder.</p>Formule :C15H13Cl2N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :334.2Metaproterenol
CAS :<p>Metaproterenol also has anti-inflammatory activity. Metaproterenol is a direct-acting sympathomimetic and a β2-adrenergic receptor (β2AR) agonist (IC50: 68 nM).</p>Formule :C11H17NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :211.26ND-322 HCl
CAS :<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Formule :C15H16ClNO3S2Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :357.88TAPI-0
CAS :<p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>Formule :C24H32N4O5Couleur et forme :SolidMasse moléculaire :456.53Amorolfine
CAS :<p>Amorolfine is available in the nail lacquer and can be used to treat fungal nail infections.</p>Formule :C21H35NOCouleur et forme :White To Off-White Crystalline PowderMasse moléculaire :317.517WAY-151693
CAS :<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Formule :C21H22ClN3O5SCouleur et forme :SolidMasse moléculaire :463.93(S)-Terazosin
CAS :<p>(S)-Terazosin is an active S-enantiomer of Terazosin.</p>Formule :C19H25N5O4Couleur et forme :SolidMasse moléculaire :387.43Chlophedianol Hydrochloride
CAS :<p>Chlophedianol hydrochloride: a cough suppressant for dry cough with antihistamine and local anesthetic traits; possibly anticholinergic at high doses.</p>Formule :C17H21Cl2NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.26Protriptyline
CAS :<p>Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.</p>Formule :C19H21NCouleur et forme :SolidMasse moléculaire :263.38Diethyl pyimDC
CAS :<p>Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).</p>Formule :C14H15N3O4Couleur et forme :SolidMasse moléculaire :289.29Guanfacine
CAS :<p>Guanfacine is a selective agonist of the α2A receptor.</p>Formule :C9H9Cl2N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :246.09BR351 precursor
CAS :<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Formule :C27H32N2O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :576.68NBI-42902
CAS :<p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>Formule :C27H24F3N3O3Couleur et forme :SolidMasse moléculaire :495.49RH01617
CAS :<p>RH01617 possesses potent inhibitory activities against Kv1.5.</p>Formule :C22H26N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :430.52CP 93129 dihydrochloride
CAS :<p>5-HT1B agonist, potent and highly selective</p>Formule :C12H14ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :251.71Vapendavir
CAS :<p>Vapendavir binds enterovirus capsids; effective against EV71 with EC50 of 0.5-1.4 μM.</p>Formule :C21H26N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.46Moricizine
CAS :<p>Moricizine is an antiarrhythmia agent which is used primarily for ventricular rhythm disturbances.</p>Formule :C22H25N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.52Landiolol
CAS :<p>Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.</p>Formule :C25H39N3O8Degré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :509.59Ivaltinostat
CAS :<p>CG-200745 is a potent inhibitor of HDAC. CG200745 induces apoptosis and also inhibits the deacetylation of histone H3 and tubulin.</p>Formule :C24H33N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.54Fidarestat
CAS :<p>Fidarestat (SNK 860),Aldose reductase inhibitor (IC50=26 nM). Targets AKR1B10 (33 μM) and V301L AKR1B10 (1.8 μM). Potential diabetes treatment.</p>Formule :C12H10FN3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.22Benproperine
CAS :<p>Benproperine is a bioactive molecule with antineoplastic properties.</p>Formule :C21H27NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :309.45(S)-Carvedilol
CAS :<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Formule :C24H26N2O4Degré de pureté :98%Couleur et forme :Less Crystalline Solid Colourless Crystalline SolidMasse moléculaire :406.47Levomepromazine Maleate
CAS :<p>Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.</p>Formule :C23H28N2O5SCouleur et forme :SolidMasse moléculaire :444.546(R)-Carvedilol
CAS :<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Formule :C24H26N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :406.47Ivabradine
CAS :<p>Ivabradine: oral HCN blocker, lowers heart rate without affecting blood pressure, has anticonvulsant and anti-anginal properties.</p>Formule :C27H36N2O5Couleur et forme :SolidMasse moléculaire :468.59Levobunolol
CAS :<p>Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.</p>Formule :C17H25NO3Couleur et forme :White To Pink PowderMasse moléculaire :291.39LPA2 antagonist 1
CAS :<p>LPA2 antagonist 1 is a potent LPA2 antagonist.</p>Formule :C20H23Cl2N5O2S2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :500.47Sarafloxacin
CAS :<p>Sarafloxacin (A56620) has antibacterial activities against Gram-positive and Gram-negative bacteria.</p>Formule :C20H17F2N3O3Degré de pureté :98.07% - 98.94%Couleur et forme :SolidMasse moléculaire :385.36Indenolol
CAS :<p>Indenolol is a blocker of beta-adrenergic.</p>Formule :C15H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.33Tropatepine
CAS :<p>Tropatepine: oral anticholinergic, treats extrapyramidal symptoms, anti-Parkinson's.</p>Formule :C22H23NSCouleur et forme :SolidMasse moléculaire :333.49Licogliflozin
CAS :<p>Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).</p>Formule :C23H28O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.46PPNDS
CAS :<p>P2X1 receptor antagonist</p>Formule :C18H15N4NaO14PS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :629.42Laropiprant
CAS :<p>Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki</p>Formule :C21H19ClFNO4SDegré de pureté :98.24% - 99.89%Couleur et forme :SolidMasse moléculaire :435.9Niclosamide monohydrate
CAS :<p>Niclosamide Monohydrate is used for the treatment of most tapeworm infections by inhibiting DNA replication.</p>Formule :C13H10Cl2N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.14Adrafinil, (R)-
CAS :<p>Adrafinil (R)-isomer, former eugeroic for enhancing alertness, attention, and mood in elderly.</p>Formule :C15H15NO3SCouleur et forme :SolidMasse moléculaire :289.35(R)-Azelastine
CAS :<p>(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.</p>Formule :C22H24ClN3OCouleur et forme :SolidMasse moléculaire :381.9Afacifenacin
CAS :<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Formule :C27H26F3N3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :481.51Distigmine Bromide
CAS :<p>Distigmine Bromide is an acetylcholinesterase inhibitor. It is used for the treatment of underactive neurogenic bladder and myasthenia gravis.</p>Formule :C22H32BrN4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :496.42Cibenzoline
CAS :<p>Cibenzoline: antiarrhythmic, blocks KATP channels, minimizes LVPG, useful in hypertrophic cardiomyopathy studies.</p>Formule :C18H18N2Couleur et forme :SolidMasse moléculaire :262.35Arasertaconazole
CAS :<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Formule :C20H15Cl3N2OSCouleur et forme :SolidMasse moléculaire :437.77Oxolamine
CAS :<p>Oxolamine is an agent of a cough suppressant.</p>Formule :C14H19N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :245.32Tiropramide
CAS :<p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>Formule :C28H41N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :467.64Piribedil dihydrochloride
CAS :<p>dopamine agonist</p>Formule :C16H20Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :371.26TAK-875 Hemihydrate
CAS :<p>TAK-875 Hemihydrate (Fasiglifam) is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than oleic acid.</p>Formule :C29H32O7SH2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :533.63Phenindamine
CAS :<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Formule :C19H19NCouleur et forme :SolidMasse moléculaire :261.36Omeprazole Sodium
CAS :<p>Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.</p>Formule :C17H18N3NaO3SDegré de pureté :99.84%Couleur et forme :Clear In WaterMasse moléculaire :367.4Vandetanib Fumarate
CAS :<p>Oral tyrosine kinase inhibitor Vandetanib Fumarate targets RET, VEGFRs, EGFR in thyroid cancer.</p>Formule :C26H28BrFN4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :591.43Evogliptin HCl
CAS :<p>Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.</p>Formule :C19H27ClF3N3O3Couleur et forme :SolidMasse moléculaire :437.88Atomoxetine
CAS :<p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>Formule :C17H21NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :255.35Azelastine
CAS :<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formule :C22H24ClN3ODegré de pureté :99.35%Couleur et forme :White Crystal PowderMasse moléculaire :381.90Vernakalant
CAS :<p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>Formule :C20H31NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.46Batimastat sodium salt
CAS :<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Formule :C23H31N3NaO4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :500.63Givinostat hydrochloride monohydrate
CAS :<p>Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.</p>Formule :C24H27N3O4·HCl·H2ODegré de pureté :97.97% - 99.51%Couleur et forme :SolidMasse moléculaire :475.97Famotidine disulfide
CAS :<p>Famotidine disulfide blocks histamine, reduces acid, treats ulcers and GERD.</p>Formule :C10H14N8S4Couleur et forme :SolidMasse moléculaire :374.53Propentofylline
CAS :<p>Propentofylline (Hextol) has neuroprotective, antiproliferative and anti-inflammatory activities and can be used in the study of Alzheimer's disease.</p>Formule :C15H22N4O3Degré de pureté :99.76% - 99.86%Couleur et forme :Off-White SolidMasse moléculaire :306.36(S)-Propafenone
CAS :<p>(S)-Propafenone, or (S)-SA-79, is an S-enantiomer with beta-blocking effects and sodium channel blocking class 1 antiarrhythmic properties.</p>Formule :C21H27NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :341.44Repirinast
CAS :<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Formule :C20H21NO5Couleur et forme :SolidMasse moléculaire :355.38Thiorphan disulfide
CAS :<p>Thiorphan disulfide: Racecadotril impurity; antidiarrheal; limits water/electrolyte intestinal absorption.</p>Formule :C24H28N2O6S2Couleur et forme :SolidMasse moléculaire :504.62CP-471474
CAS :<p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>Formule :C16H17FN2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.38Propiomazine
CAS :<p>Propiomazine is an orally active antihistamine compound with sedative properties, useful for controlling insomnia in neurological disorders.</p>Formule :C20H24N2OSDegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :340.48ND-336
CAS :<p>ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.</p>Formule :C16H18ClNO3S2Couleur et forme :SolidMasse moléculaire :371.9Anitrazafen
CAS :<p>Anitrazafen is a locally effective anti-inflammatory agent that has been shown to have COX-2 inhibitor activity.</p>Formule :C18H17N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.35Mianserin
CAS :<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Formule :C18H20N2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :264.36Riodoxol
CAS :<p>Riodoxol is an antiviral agent that effectively affects the reproduction and maturation of viruses.</p>Formule :C6H3I3O2Couleur et forme :SolidMasse moléculaire :487.8Trifluperidol HCl
CAS :Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Formule :C22H24ClF4NO2Couleur et forme :SolidMasse moléculaire :445.88Clencyclohexerol
CAS :<p>Clencyclohexerol, like clenbuterol, is a β-adrenoceptor agonist with potential in muscle disorders but poses cardiovascular risks at high doses.</p>Formule :C14H20Cl2N2O2Couleur et forme :SolidMasse moléculaire :319.23Pipotiazine
CAS :<p>Pipotiazine treats chronic schizophrenia with less sedation, low hypotension risk, but high extrapyramidal side effects.</p>Formule :C24H33N3O3S2Couleur et forme :SolidMasse moléculaire :475.67Bromhexine
CAS :<p>Bromhexine is an expectorant/mucolytic agent which can be used in the treatment of respiratory disorders associated with excessive mucus or viscid.</p>Formule :C14H20Br2N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.13MMP-2/9-IN-1
CAS :<p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>Formule :C14H16IN7SCouleur et forme :SolidMasse moléculaire :441.29(R)-Praziquantel
CAS :<p>(R)-Praziquantel is an active enantiomer of praziquantel.</p>Formule :C19H24N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :312.41Procarbazine free base
CAS :<p>Procarbazine: chemo drug for Hodgkin's, brain cancer; liver-activated; MAO inhibitor.</p>Formule :C12H19N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :221.3Safironil
CAS :<p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>Formule :C15H23N3O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :309.36Rolapitant
CAS :<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Formule :C25H26F6N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :500.48Isothipendyl
CAS :<p>Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.</p>Formule :C16H19N3SCouleur et forme :SolidMasse moléculaire :285.41Evogliptin
CAS :<p>Evogliptin (DA-1229) is an oral DPP4 inhibitor effective in reducing blood sugar and liver inflammation.</p>Formule :C19H26F3N3O3Couleur et forme :SolidMasse moléculaire :401.42Linagliptin impurity G
CAS :<p>Linagliptin impurity G is an impurity in the drug product Linagliptin. It is a natural substance and its CAS number is 668270-11-9. Impurity G can be synthesized from L-phenylalanine and cyclohexane carboxaldehyde in a two step process. The first step involves the reaction of L-phenylalanine with cyclohexane carboxaldehyde to yield methylcyclohexanecarboxylate, which then undergoes hydrolysis to give phenylcyclohexanol. In the second step, phenylcyclohexanol reacts with hydrochloric acid to produce phenylcyclohexanone, which is then oxidized with hydrogen peroxide to yield impurity G. Impurity G can also be found in the pharmacopoeia as a high purity HPLC standard for linagliptin.</p>Formule :C25H28N8O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :472.54 g/molEmpagliflozin S-furanose
CAS :<p>Empagliflozin S-furanose is a Custom synthesis drug product. It is an analytical standard with CAS No. 1620758-32-8, and it is used in research and development of new drugs. Empagliflozin S-furanose has been found to be a metabolite of empagliflozin, a drug that is used to treat type 2 diabetes mellitus. It is also used as an impurity standard for HPLC analysis of empagliflozin because it does not have any biological activity.</p>Formule :C23H27ClO7Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :450.91 g/molN-De[2-(methylsulfonyl)ethyl] lapatinib
CAS :<p>Lapatinib is a tyrosine kinase inhibitor that blocks the epidermal growth factor receptor (EGFR) and other tyrosine kinases. It is used in cancer treatment to inhibit tumor growth, with a high success rate. Lapatinib is also used to treat lung cancer and other types of cancer. The drug has been shown to inhibit EGFR phosphorylation in vitro, which leads to inhibition of cell proliferation and induction of apoptosis. Lapatinib also inhibits the expression of EGFR downstream target genes such as b-raf, serine/threonine-protein kinase, and cyp3a5.</p>Formule :C26H20ClFN4O2Degré de pureté :Min. 95%Masse moléculaire :474.91 g/molVildagliptin related compound F
CAS :<p>Vildagliptin related compound F (VRCF) is a drug product that has been custom synthesized. VRCF is a high purity, analytical standard. It is metabolized in the body and can be used as a research and development standard to study the metabolism of vildagliptin. VRCF is a natural metabolite that has been identified as an impurity in the drug product Vildagliptin. VRCF has not been recognized by the USP or EP for use as an impurity standard. CAS no: 1789703-36-1</p>Formule :C17H24N2O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :304.4 g/molViloxazine
CAS :<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Formule :C13H19NO3Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :237.29Vildagliptin carboxylic acid methyl ester
CAS :<p>Please enquire for more information about Vildagliptin carboxylic acid methyl ester including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C18H28N2O4Degré de pureté :Min. 95%Masse moléculaire :336.43 g/molGallopamil
CAS :<p>Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.</p>Formule :C28H40N2O5Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :484.63Amlodipine EP Impurity F maleate
CAS :<p>Amlodipine EP Impurity F maleate is an impurity of amlodipine, a drug product. It is a natural substance that has been classified as an API impurity in the United States Pharmacopeia (USP). The chemical name for this drug is 3-(2-chlorophenyl)-1-methyl-5-(o-tolyloxy)-2,4-dihydro-6H-[1,3]thiazolo[3,2-a]pyrimidin-7-one. Amlodipine EP Impurity F maleate has the following properties: C12H9ClNO2S and a melting point of 210°C with a purity of 99.5%. This compound was synthesized by custom synthesis and is used as an analytical standard for HPLC. This compound was also used during the development of amlodipine to determine its metabolism studies.</p>Formule :C19H23ClN2O5•C4H4O4Degré de pureté :Min. 95%Masse moléculaire :510.92 g/mol(Z)-Thiothixene
CAS :<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Formule :C23H29N3O2S2Degré de pureté :99.21%Couleur et forme :Yellow To Yellow With A Tan Cast PowderMasse moléculaire :443.63MMP-2/MMP-9 Inhibitor I
CAS :<p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>Formule :C21H19NO4SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :381.44Sovaprevir
CAS :<p>Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.</p>Formule :C43H53N5O8SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :799.97Vildagliptin Related Compound 2
CAS :<p>Vildagliptin Related Compound 2 is a synthetic compound that has been shown to be an inhibitor of DPP-4. It is a white solid that can be synthesized by condensation of vildagliptin with chloroacetyl chloride in the presence of an alkali. The compound was found to have impurities, including 1-(2-chlorophenyl)ethanol and 3-chlorobenzaldehyde.</p>Formule :C17H25N3O2Degré de pureté :Min. 95%Masse moléculaire :303.4 g/molGivinostat hydrochloride
CAS :<p>Givinostat HCl (ITF2357 HCl) inhibits HDAC1/3 (IC50: 198/157 nM) with anti-inflammatory, anti-angiogenic, and antineoplastic properties.</p>Formule :C24H28ClN3O4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :457.95PG-116800
CAS :<p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>Formule :C24H27N3O7SDegré de pureté :98.03% - 99.66%Couleur et forme :SolidMasse moléculaire :501.55Moveltipril
CAS :<p>Moveltipril (Moveltipril calcium) is a potent angiotensin-converting enzyme (ACE) inhibitor.Moveltipril is converted to captopril in the body for action.</p>Formule :C19H30N2O5SDegré de pureté :97.55% - 98.28%Couleur et forme :SolidMasse moléculaire :398.52Laduviglusib trihydrochloride
CAS :<p>Laduviglusib trihydrochloride, a GSK-3α/β inhibitor (IC50: 10/6.7 nM), activates Wnt/β-catenin signaling and induces autophagy.</p>Formule :C22H20Cl5N8Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :573.71CP-544439
CAS :<p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>Formule :C18H19FN2O6SDegré de pureté :95.02% - 98.66%Couleur et forme :SolidMasse moléculaire :410.42Cyamemazine
CAS :<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Formule :C19H21N3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :323.46Fenoverine
CAS :<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Formule :C26H25N3O3SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :459.562,3,4,5-Tetradehydro alfuzosin hydrochloride
CAS :<p>Alfuzosin is a potent, selective, and long-acting α1A-adrenergic receptor antagonist. It is used to treat benign prostatic hyperplasia (BPH) in males. Alfuzosin is also used as an antihypertensive agent, for the treatment of pheochromocytoma, and for the treatment of benign prostatic hyperplasia in males. The hydrogenation of 2,3,4,5-tetradehydroalfuzosin to alfuzosin hydrochloride is performed by liquid hydrogenation or by hydrogenation on a palladium catalyst in a mixture of dimethylformamide and hexamethylphosphoramide. This process minimizes the formation of impurities such as 2,3,4-trimethoxy alfuzosin.</p>Formule :C19H24ClN5O4Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :421.88 g/molDesfluoro ezetimibe
CAS :<p>Desfluoro ezetimibe is a synthetic cholesterol-lowering drug that inhibits intestinal cholesterol absorption. It is chemically synthesized, and the process includes the introduction of fluorine at the 3-position of the C-ring. Desfluoro ezetimibe is not metabolized in humans, but it may be subject to oxidative degradation. The product is also subject to oxidation by light and air, which may result in formation of impurities. The drug substance has been validated as well as its isomers and efficiencies in mass spectrometry detection.</p>Formule :C24H22FNO3Degré de pureté :Min. 95%Couleur et forme :White To Off-White SolidMasse moléculaire :391.43 g/mol(R,R)-Montelukast bis-sulfide
CAS :<p>(R,R)-Montelukast bis-sulfide is a drug product that is used in the analytical and research and development of drugs. It is also used as an impurity standard for HPLC. (R,R)-Montelukast bis-sulfide has been shown to have niche applications in drug development and research, as well as being a high purity API.</p>Formule :C41H46ClNO5S2Degré de pureté :90%MinMasse moléculaire :732.39 g/molEltenac
CAS :<p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>Formule :C12H9Cl2NO2SDegré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :302.18(R)-Zanubrutinib
CAS :<p>(R)-Zanubrutinib ((R)-BGB-3111) is a selective inhibitor of Bruton tyrosine kinase (BTK).</p>Formule :C27H29N5O3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :471.55Pantoprazole sulphide
CAS :<p>Pantoprazole sulphide is a benzimidazole derivative that has been synthesized in an asymmetric synthesis. The purified compound was characterized by its nmr spectra, which showed the presence of the carboethoxy group and the chromatographic method. The compound belongs to a family of inhibitors known as benzimidazole derivatives and has shown inhibitory activity against a number of bacterial species including Staphylococcus aureus, Clostridium perfringens, and Mycobacterium tuberculosis. Pantoprazole sulphide has been used as an inhibitor to treat gastric acid pump disorders such as Zollinger-Ellison syndrome. It is also used for treating pathological conditions such as duodenal ulcers or gastroesophageal reflux disease.</p>Formule :C16H15F2N3O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :367.37 g/molUNC0321
CAS :<p>UNC0321 is an effective inhibitor of histone methyltransferase G9a with a Ki of 63 pM and with IC50s 9 nM and 6 nM in ECSD and CLOT assays.</p>Formule :C27H45N7O3Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :515.69MMP2-IN-3
CAS :<p>MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).</p>Formule :C23H21N3ODegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :355.43Pitolisant
CAS :<p>Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Formule :C17H26ClNODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :295.85Edoxaban
CAS :<p>Edoxaban: potent, selective FXa inhibitor; Ki 0.561 nM. Used as an oral anticoagulant for stroke prevention, also inhibits thrombin and FIXa.</p>Formule :C24H30ClN7O4SDegré de pureté :97.67% - 99.71%Couleur et forme :SolidMasse moléculaire :548.061-Oxo mirtazapine
CAS :<p>1-Oxo mirtazapine is a metabolite of mirtazapine. It is a synthetic compound and is not found in nature. This product is a research and development impurity standard for the preparation of drug product, which has been synthesized to be highly pure. The material is used for drug development, including pharmacopoeia requirements for analytical studies and metabolism studies. 1-Oxo mirtazapine has been shown to have niche applications in pharmacopoeia and as an HPLC standard.</p>Formule :C17H17N3ODegré de pureté :Min. 95%Masse moléculaire :279.34 g/molDimethindene
CAS :<p>Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.</p>Formule :C20H24N2Degré de pureté :98.3% - 98.99%Couleur et forme :SolidMasse moléculaire :292.42(S)-Rabeprazole sodium
CAS :<p>(S)-Rabeprazole sodium is an anticancer drug that acts as a kinase inhibitor. It is an analog of Rabeprazole and has been shown to inhibit the growth of cancer cells in vitro and in vivo. (S)-Rabeprazole sodium inhibits the activity of kinases, which are enzymes that play a key role in cell signaling pathways. This inhibition leads to apoptosis, or programmed cell death, in cancer cells. (S)-Rabeprazole sodium has been tested against various types of cancer, including Chinese hamster ovary cells and tumor xenografts in mice. It has also been shown to inhibit elastin degradation, which is important for preventing metastasis of cancer cells. (S)-Rabeprazole sodium may be a promising candidate for the development of new anticancer drugs that target specific kinases and proteins involved in cancer cell growth and survival.</p>Formule :C18H21N3O3S•NaDegré de pureté :Min. 95%Masse moléculaire :382.43 g/mol3-Trifluoroacetylamino linagliptin
CAS :<p>Please enquire for more information about 3-Trifluoroacetylamino linagliptin including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C27H27F3N8O3Degré de pureté :Min. 95%Masse moléculaire :568.55 g/molAmlodipine EP Impurity E maleate
CAS :<p>Amlodipine EP Impurity E maleate is a high purity and analytical grade chemical. It is a metabolite of Amlodipine, which is used in the treatment of hypertension. This chemical has been shown to be a natural product that is produced by the human body. It also has been shown to have pharmacological properties, such as anti-inflammatory and vasodilatory effects. The impurity standard for this compound is available from Sigma-Aldrich.br>br></p>Formule :C21H27ClN2O5•C4H4O4Degré de pureté :Min. 95%Masse moléculaire :538.98 g/molethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
CAS :<p>Please enquire for more information about ethyl 6-(4-aMinophenyl)-1-(4-Methoxyphenyl)-7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C22H22N4O4Degré de pureté :Min. 95%Masse moléculaire :406.43 g/molImipramine
CAS :<p>Imipramine (Dimipressin) is a Fascin1 inhibitor with antitumor activity and induces apoptosis.</p>Formule :C19H24N2Degré de pureté :99.4%Couleur et forme :White To Off-White /Hydrochloride/ SolidMasse moléculaire :280.41Roflumilast Impurity A
CAS :<p>Roflumilast impurity A is a metabolite of roflumilast. It is a drug product that is used as an analytical standard for the determination of roflumilast in HPLC analysis. Roflumilast impurity A is not natural and is synthetic. It has been shown to be a substrate for CYP1A2, CYP2C8, CYP2C9, and CYP3A4 enzymes. Studies have shown that it may be involved in the metabolism of roflumilast through hydroxylation and deamination.</p>Formule :C16H14Cl2N2O3Degré de pureté :Min. 95%Masse moléculaire :353.2 g/molEzetimibe ketone
CAS :<p>Ezetimibe ketone is a lipid-lowering agent that inhibits cholesterol absorption through the inhibition of Niemann-Pick C1-like 1 (NPC1L1). Ezetimibe ketone is used to reduce the levels of low-density lipoprotein cholesterol (LDL-C) in patients with primary hypercholesterolemia, sitosterolemia, and familial combined hyperlipidemia. Ezetimibe ketone has been shown to be bioequivalent to ezetimibe, which is an oral drug that inhibits cholesterol absorption by blocking NPC1L1. The drug binds to the NPC1L1 receptor in the brush border membrane of enterocytes and prevents cholesterol uptake. Ezetimibe ketone has a high solubility in organic solvents such as dichloromethane or chloroform. It also has a high melting point, which makes it suitable for use on chromatographic columns.</p>Formule :C24H19F2NO3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :407.41 g/molAGPS-IN-2i
CAS :<p>AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.</p>Formule :C18H17F2N3O2Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :345.34Ecopipam
CAS :<p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>Formule :C19H20ClNODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :313.82Pramipexole EP Impurity C
CAS :<p>Pramipexole EP Impurity C is a synthetic impurity that is used as an impurity standard in the manufacture of Pramipexole EP. It is also used as a research and development tool for drug product, custom synthesis, CAS No. 1973461-14-1, and analytical studies. This compound has been shown to be a metabolite of Pramipexole EP and may have pharmacological properties. Pramipexole EP Impurity C has been found to inhibit the growth of certain bacteria, such as methicillin-resistant Staphylococcus aureus (MRSA) isolates.</p>Formule :C20H32N6S2Degré de pureté :Min. 95%1-Fluoronaphthalene
CAS :<p>1-Fluoronaphthalene is a polyunsaturated compound that is used in analytical chemistry for the determination of test samples. It is an inhibitor of the enzyme IDO1, which plays an important role in the regulation of immune function, and has been shown to have anti-inflammatory properties. 1-Fluoronaphthalene can be synthesized by reacting n-dimethyl formamide with hydrogen fluoride and then adding a diazonium salt and hydrochloric acid. The UV absorption spectrum of 1-fluoronaphthalene displays a maximum at 248 nm. This compound binds to cation channels on cells, causing hyperpolarization.</p>Formule :C10H7FDegré de pureté :Min. 95%Masse moléculaire :146.16 g/molGemigliptin
CAS :<p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>Formule :C18H19F8N5O2Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :489.36N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methyloxirane-2-carboxamide
CAS :<p>N-[4-Cyano-3-(trifluoromethyl)phenyl]-2-methyloxirane-2-carboxamide (NUOX) is a potential anticancer agent that has been shown to have an acidic pKa of 5.8 and to be active against cancer cells in the same way as bicalutamide, which is a known antiandrogen. NUOX has been shown to increase the number of cavities in polybenzimidazole (PBI) films by enhancing the rate of oxidation. NUOX also inhibits the growth of human cancer cells by binding sulfide groups on proteins and DNA, inhibiting cellular respiration. NUOX is not water soluble, so it must be dissolved in solvents such as acetonitrile or chloroform before administration.</p>Formule :C12H9F3N2O2Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :270.21 g/molDB04760
CAS :<p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>Formule :C22H20F2N4O2Degré de pureté :99.93% - 99.99%Couleur et forme :SolidMasse moléculaire :410.42Ephedrine Hydrochloride
CAS :Produit contrôléEphedrine and its saltsFormule :C10H15NO·HClCouleur et forme :White Off-White PowderMasse moléculaire :201.09204Stepronin
CAS :<p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>Formule :C10H11NO4S2Degré de pureté :99.59%Couleur et forme :White Or Off White CrystallineMasse moléculaire :273.33Benperidol
CAS :<p>Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.</p>Formule :C22H24FN3O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :381.44Brivaracetam CV
CAS :Produit contrôléLactams, nesoiFormule :C11H20N2O2Couleur et forme :White Off-White SolidMasse moléculaire :212.15248Pitavastatin N-oxide
CAS :<p>Pitavastatin N-oxide is a drug product that is an analytical standard and natural API impurity. It is used in the synthesis of other drugs, such as pitavastatin, which is a statin drug used to lower cholesterol levels. Pitavastatin N-oxide has been shown to be a potent inhibitor of HMG-CoA reductase, the enzyme that catalyzes the conversion of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) to mevalonate. This inhibits cholesterol production and lowers levels of low density lipoprotein (LDL) cholesterol in the blood.</p>Formule :C25H24FNO5Degré de pureté :Min. 95%Masse moléculaire :437.46 g/molArimoclomol
CAS :<p>Arimoclomol (BRX-220 free base) is a co-inducer of heat shock proteins (HSP) and can be used in studies about the treatment of amyotrophic lateral sclerosis (</p>Formule :C14H20ClN3O3Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :313.78Apixaban Impurity 6
CAS :<p>Please enquire for more information about Apixaban Impurity 6 including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Formule :C26H26N4O5Degré de pureté :Min. 95%Masse moléculaire :474.51 g/molAmiodarone impurity E
CAS :<p>Amiodarone impurity E is a nucleophilic compound that is synthesized by the acylation of a diazonium salt with an amine. It has been shown to be active against staphylococci, but not against subtilis. The reaction may be catalyzed by acid or chloride. Amiodarone impurity E is also demethylated and dehydrated to form the final product, amiodarone.</p>Formule :C19H18O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :294.34 g/molApixaban Impurity 1
CAS :<p>Apixaban Impurity 1 is an impurity found in Apixaban, a drug used for the prevention of stroke. It is produced by condensation of 2-aminopyridine and 3-hydroxybenzaldehyde in ethanol with sodium hydroxide as a catalyst. The reaction proceeds via amination of the pyridine ring followed by transesterification. The yield of this impurity is low at about 4%.</p>Degré de pureté :Min. 95%ROCK2-IN-7
CAS :<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Formule :C26H28FN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :445.53Ro 31-9790
CAS :<p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>Formule :C15H29N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.41Mefenidil
CAS :<p>Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.</p>Formule :C12H11N3Degré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :197.24Quizalofop
CAS :<p>Quizalofop (Xylafop) is a reagent of biochemical.</p>Formule :C17H13ClN2O4Degré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :344.75Etidocaine Hydrochloride
CAS :<p>Etidocaine Hydrochloride (W19053) is a long-acting anesthetic and a blocker of the voltage-gated sodium channel.</p>Formule :C17H29ClN2ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :312.88LY52
CAS :<p>LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.</p>Formule :C22H24N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.45Brilaroxazine
CAS :<p>Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.</p>Formule :C22H25Cl2N3O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :450.36Dibenamine hydrochloride
CAS :<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Formule :C16H19Cl2NDegré de pureté :96.43%Couleur et forme :Oily Liquid SolidMasse moléculaire :296.23Frovatriptan
CAS :<p>Frovatriptan, potent 5-HT 1B/D agonist, shows high cerebroselectivity and efficacy for migraine with aura.</p>Formule :C14H17N3OCouleur et forme :SolidMasse moléculaire :243.3Yonkenafil
CAS :<p>Yonkenafil, a PDE5 inhibitor, may reduce stroke damage and aid in Alzheimer's treatment.</p>Formule :C24H33N5O4SCouleur et forme :SolidMasse moléculaire :487.61RU 58668
CAS :<p>Pure antiestrogen that downregulates estrogen receptor expression</p>Formule :C34H43F5O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :658.76Ro 32-7315
CAS :<p>Ro 32-7315 is a selective inhibitor of ADAM17.</p>Formule :C22H35N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.6FGIN-1-27
CAS :<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Formule :C28H37FN2ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :436.6Apratastat
CAS :<p>Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs)</p>Formule :C17H22N2O6S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.5ND-378
CAS :<p>ND-378 is a potent and selective inhibitor of MMP-2 with no inhibition on MMP-9 and MMP-14.</p>Formule :C18H19NO4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.48MMP-145
CAS :<p>MMP-145 is used as a protease inhibitor.</p>Formule :C20H20N2O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.45MMP13-IN-3
CAS :<p>MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.</p>Formule :C24H22N4O5Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :446.46XL-784
CAS :<p>XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.</p>Formule :C42H42Cl2F4MgN6O16S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1122.15AZD-1656
CAS :<p>AZD-1656 is a glucokinase activator (GKA) that can cause dose-limiting hypoglycemia in normal animals used in embryofetal development studies and type 2</p>Formule :C24H26N6O5Degré de pureté :97.07% - 99.37%Couleur et forme :SolidMasse moléculaire :478.5ONO 4817
CAS :<p>ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.</p>Formule :C22H28N2O6Couleur et forme :SolidMasse moléculaire :416.47
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