Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Camostat mesylate - Bio-X ™
CAS :Camostat is a serine protease inhibitor that is used for the treatment of chronic pancreatitis. This drug has shown to reduce inflammation and pain. Studies have shown that Camostat has also inhibited the entry of SARS-CoV-2 in lung cells by inhibiting the priming process of S-protein, necessary for the viral entry into host cells.Formule :C20H22N4O5•CH4O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :494.52 g/molTivozanib
CAS :Inhibitor of VEGF receptorsFormule :C22H19ClN4O5Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :454.86 g/molGefitinib - Bio-X ™
CAS :Gefitinib is an inhibitor of the epidermal growth factor receptor (EGFR) protein. This inhibition is on the EGFR tyrosine kinase domain, where Gefitinib bindings to the ATP-binding site. As a a tyrosine kinase inhibitor, Gefitinib blocks tumor growth and has led to its use in slowing the progression of non-small cell lung cancer. Gefitinib also inhibits invasion and metastasis through inhibition of macrophage receptor interacting protein kinase 2 (RIPK2), rather than EGFR.Formule :C22H24ClFN4O3Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :446.9 g/molPentoxifylline
CAS :Produit contrôléPhosphodiesterase inhibitorFormule :C13H18N4O3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :278.31 g/molO6-Benzylguanine - Bio-X ™
CAS :O6-Benzylguanine is a guanine analog that is an antineoplastic agent. It works by acting as a suicide inhibitor of the enzyme O6-alkylguanine-DNA alkyltransferase. This results to an interruption of DNA repair so that damage can occur to local tumor targets.Formule :C12H11N5ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :241.25 g/mol3-(4-Phenylbutyl)-4-propyloxetan-2-one
CAS :Cis/trans-form of GK 563 [2351820-19-2]Formule :C16H22O2Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :246.34 g/molTrilostane
CAS :Produit contrôléInhibitor of 3β-hydroxysteroid dehydrogenase in steroid biosynthesis
Formule :C20H27NO3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :329.43 g/molMK 4827
CAS :Inhibitor of PARP1 and PARP2 enzymes
Formule :C19H20N4ODegré de pureté :Min. 96 Area-%Couleur et forme :White PowderMasse moléculaire :320.39 g/molRucaparib camsylate
CAS :Inhibitor of poly (ADP-ribose) polymerase enzyme; antineoplasticFormule :C19H18FN3O•C10H16O4SDegré de pureté :Min. 95%Couleur et forme :Off-White To Yellow SolidMasse moléculaire :555.66 g/molAbiraterone acetate - Bio-X ™
CAS :Produit contrôléAbiraterone is an antiandrogen drug used in the treatment of metastatic prostate cancer. It is a derivative of steroidal progesterone. This drug inhibits the enzyme CYP17 irreversibly, thus inhibiting the synthesis of androgen. It specifically inhibits the conversion of 17-hydroxyprognenolone to dehydroepiandrosterone to decrease serum levels of testosterone and other androgens.Formule :C26H33NO2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :391.55 g/molEtoposide phosphate
CAS :Topoisomerase II inhibitor; chemotherapeutic drugFormule :C29H33O16PDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :668.54 g/molDiacerein - Bio-X ™
CAS :Diacerein is a slow-onset anthraquinone IL-1 inhibitor that is used in the treatment of joint diseases such as osteoarthritis. This drug is also being studied for the treatment of insulin resistance and diabetes mellitus. Diacerein works to decrease inflammation and cartilage destruction by reducing the level of interleukin-1.Formule :C19H12O8Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :368.29 g/molFlurbiprofen
CAS :Inhibitor of cytochrome P450; inhibitor of prostaglandin synthesis
Formule :C15H13FO2Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :244.26 g/molImiquimod - Bio-X ™
CAS :Imiquimod is a toll-like receptor 7 agonist drug that is used for the treatment of genital warts, basal cell carcinoma and condyloma acuminata. This drug works by relieving and controlling wart production. Studies in mice have shown that this drug may induce cytokines such as interleukins. Imiquimod helps to increase apoptosis of diseased tissues and an infiltration of lymphocytes into tumor lesions.Formule :C14H16N4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :240.3 g/molBrivanib alaninate
CAS :VEGFR2 a tyrosine kinase receptor inhibitor; antineoplasticFormule :C22H24FN5O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :441.18123Lenalidomide - Bio-X ™
CAS :Produit contrôléLenalidomide is a thalidomide derivative that is used to treat multiple myeloma and anemia. This drug exerts immunomodulatory effects by altering cytokine production. Lenalidomide also directly inhibits the cullin ring E3 ubiquitin ligase complex.Formule :C13H13N3O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :259.26 g/molLeflunomide - Bio-X ™
CAS :Produit contrôléLeflunomide is a pyrimidine synthesis inhibitor drug that is used to treat rheumatoid arthritis. Although its mechanism of action is not fully determined, this drug has shown to interfere with cell cycle progression by inhibiting dihydroorotate dehydrogenase and has shown antiproliferative activity. As a result of this, it interferes with the expansion of activated autoimmune lymphocytes. Additionally, Leflunomide is a tyrosine kinase inhibitor.Formule :C12H9F3N2O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :270.21 g/molSU 0268
CAS :Inhibitor of 8-oxoguanine DNA glycosylase OGG1 with IC50 of 0.059 μM and excellent specificity over other DNA repair enzymes. OGG1 and its substrate 8-oxoguanine are involved in mutagenesis, genotoxicity, inflammation and cancer. The compound can cause accumulation of 8-oxoguanine in DNA in vitro and is a potent tool for the study of OGG1 biology.Formule :C26H25N3O4SDegré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :475.56 g/molGboxin
CAS :Inhibitor of oxidative phosphorylation which acts on the F0F1 ATP synthase in the inner mitochondrial membrane and causes acute increase in mitochondrial membrane potential. Gboxin was shown to accumulate in mitochondria of cancer cells, to cause cellular toxicity and cell growth inhibition in mouse glioblastoma. However, Gboxin did not inhibit growth of mouse embryonic fibroblasts or neonatal astrocytes.Formule :C22H33N2O2•ClDegré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :392.96 g/molMLN120B
CAS :Inhibitor of IKKβ serine kinaseFormule :C19H15ClN4O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :366.8 g/mol
