Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Teriflunomide
CAS :Produit contrôlé<p>Inhibitor of dihydroorotate dehydrogenase; anti-inflammatory; immunomodulatory</p>Formule :C12H9F3N2O2Degré de pureté :Min. 98 Area-%Couleur et forme :White PowderMasse moléculaire :270.21 g/molCX 4945
CAS :<p>Inhibitor of CK2 protein kinase; anti-proliferative</p>Formule :C19H12ClN3O2Degré de pureté :Min. 98 Area-%Couleur et forme :SolidMasse moléculaire :349.0618BAY 607550
CAS :<p>A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.</p>Formule :C27H32N4O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :476.24236Vildagliptin - Bio-X ™
CAS :<p>Vildagliptin is an antihyperglycemic agent that is used for the management of type 2 diabetes mellitus. This drug is a dipeptidyl peptidase 4 inhibitor and prevents the degradation of glucagon-like peptide 1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP). This leads to improved glycemic control.</p>Formule :C17H25N3O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :303.4 g/molMK 886 - Bio-X ™
CAS :<p>MK 886 is a leukotriene antagonist that has been studied for use in treating atherosclerosis. This drug inhibits the 5-lipoxygenase activating protein thus inhibiting 5-lipoxygenase.</p>Formule :C27H34ClNO2SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :472.08 g/molSCH 772984
CAS :<p>Inhibitor of ERK1 and ERK2 serine/threonine kinases</p>Formule :C33H33N9O2Degré de pureté :Min. 95%Couleur et forme :Light (Or Pale) Yellow To Yellow SolidMasse moléculaire :587.67 g/molSB 431542
CAS :<p>Inhibitor of activin receptor-like kinases (ALK4, ALK5 and ALK7), members of TGFβ type I receptor family. Blocks activin- and TGFβ-mediated signaling and phosphorylation of Smad2 downstream. Suppresses tumor-promoting and tumor-suppressing effects of TGFβ. Promotes differentiation of human embryonic stem cells (hESCs), whilst sustaining mouse ESCs in the undifferentiated state.</p>Formule :C22H16N4O3Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :384.4 g/moleCF506
CAS :<p>Selective inhibitor of the Src kinase family with subnanomolar IC50 values and good selectivity over c-Abl, PDGFRα and c-Kit kinases. The compound is effective in inhibiting growth in drug resistant cancer cell lines. In a recent study, it inhibited the growth of HER2-positive breast cancer cell lines which were resistant to pan-HER family kinase inhibitors such as lapatinib.</p>Formule :C26H38N8O3Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :510.63 g/molBLU 667
CAS :<p>RET receptor tyroine kinase inhibitor</p>Formule :C27H32FN9O2Degré de pureté :Min. 95%Couleur et forme :White/Off-White SolidMasse moléculaire :533.6 g/molRigosertib sodium
CAS :<p>Rigosertib sodium is an experimental chemotherapeutic agent that is a derivative of benzyl styryl sulfone. It is synthesized chemically and functions primarily by inhibiting key signaling pathways involved in cancer cell proliferation. Specifically, Rigosertib targets the RAS signaling pathway along with the phosphatidylinositol-3-kinase/AKT and polo-like kinase 1 (Plk1) pathways, impeding the progression of the cell cycle and inducing apoptosis in malignant cells.</p>Formule :C21H24NNaO8SDegré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :473.47 g/molAbemaciclib
CAS :<p>Inhibitor of cyclin-dependent kinases CDK4 and CDK6</p>Formule :C27H32F2N8Degré de pureté :Min. 95%Masse moléculaire :506.59 g/molLarotrectinib
CAS :<p>A potent ATP-competitive inhibitor of tropomyosin-related kinases (TRK1, TRK2 and TRK3), members of the receptor tyrosine kinase family of neurotrophin receptors. Tumors with oncogenic TRK fusions are sensitive to larotrectinib, leading to reduced proliferation and tumor growth in patients with soft tissue sarcoma, triple-negative breast cancer and lung cancer.</p>Formule :C21H22F2N6O2Degré de pureté :Min. 98 Area-%Couleur et forme :Yellow PowderMasse moléculaire :428.44 g/molSulindac - Bio-X ™
CAS :<p>Sulindac is a non-steroidal anti-inflammatory drug that has anti-inflammatory and analgesic properties. It is used to relieve the pain of osteoarthritis and rheumatoid arthritis by reducing inflammation and inhibiting the production of prostaglandins, which are chemicals that cause inflammation.</p>Formule :C20H17FO3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :356.41 g/molAxitinib
CAS :<p>Inhibits VEGFR1, VEGFR2, VEGFR3, c-kit and PDGFR tyrosine kinases</p>Formule :C22H18N4OSDegré de pureté :Min. 98 Area-%Couleur et forme :White Yellow PowderMasse moléculaire :386.47 g/molCZC 25146
CAS :<p>Inhibitor of leucine-rich repeat kinase LRRK2Â</p>Formule :C22H25FN6O4SDegré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :488.54 g/molMethocarbamol
CAS :<p>Inhibitor of carbonic anhydrase; muscle relaxant</p>Formule :C11H15NO5Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :241.24 g/molLovastatin - Bio-X ™
CAS :<p>Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.</p>Formule :C24H36O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :404.54 g/molPF 06447475
CAS :<p>Inhibitor of LRRK2 kinase</p>Formule :C17H15N5ODegré de pureté :Min. 95%Couleur et forme :White To Off-White To Pink SolidMasse moléculaire :305.33 g/molBetrixaban
CAS :<p>Inhibitor of factor Xa</p>Formule :C23H22ClN5O3Degré de pureté :Min. 95%Couleur et forme :Off-White PowderMasse moléculaire :451.91 g/molIbuprofen - Bio-X ™
CAS :<p>Ibuprofen is a non-steroidal anti-inflammatory drug (NSAID) used to reduce inflammation, relieve pain and reduce fever. The mechanism of action of ibuprofen has not been fully elucidated, but it may be due to inhibiting the enzyme cyclooxygenase and thus decreasing the synthesis of prostaglandins allowing a reduction of pain and inflammation.</p>Formule :C13H18O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :206.28 g/mol
