Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Gabexate mesylate
CAS :Serine protease inhibitorFormule :C17H27N3O7SDegré de pureté :Min. 95%Masse moléculaire :417.15697Ro492097
CAS :Inhibitor of γ-secretase and Notch signallingFormule :C22H20F5N3O3Degré de pureté :Min. 95%Masse moléculaire :469.4 g/molZofenopril calcium
CAS :Angiotensin-converting enzyme inhibitor; antioxidantFormule :C44H46N2O8S4•CaDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :899.17 g/molTiludronic acid disodium
CAS :Farnesyltransferase inhibitorFormule :C7H9ClO6P2S•Na2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :364.59 g/molNVP-TAE684
CAS :Inhibitor of NPM-ALK kinaseFormule :C30H40ClN7O3SDegré de pureté :Min. 95%Masse moléculaire :614.2 g/molGinkgolic acid (C13:0)
CAS :Sumoylation inhibitor; reported to inhibit histone acetylation transferaseFormule :C20H32O3Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :320.47 g/molMG 132
CAS :MG 132 is a modified tripeptide that acts as proteasomal inhibitor. In 2006, MG 132 has been experimentally tested in in vitro cell-based and in vivo models for to assess its use in the medical treatment of Parkinson's disease.Formule :C26H41N3O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :475.30462SU 3327
CAS :SU 3327, originally introduced as a thiadiazole JNK inhibitor (De et al. 2009) has recently been identified as having antibiotic activity against a broad range of bacteria including drug-resistant gram positive and negative strains (Strokes et al. 2020). This molecule has been given the fictional name ‘Halicin’ inspired by the AI approach used to discover its novel biological activity.Formule :C5H3N5O2S3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :261.31 g/molRapamycin-13C,d3 (contains d0) - Technical Grade
CAS :Produit contrôléBinds to FK506 binding proteins (FKBPs) to form a complex that inhibits mammalian targets of rapamycin (mTOR). Blocks p70 S6 kinase activation by interleukin-2 and thereby inhibits proliferation of T cells. Induces differentiation of human pluripotent stem cells (hPSCs) to mesendoderm and blood progenitor cells.Formule :C50CH76D3NO13Degré de pureté :Min. 95%Masse moléculaire :918.18 g/molSurfen
CAS :Small molecule antagonist of heparan sulfate that binds to glycosaminoglycans electrostatically. Surfen neutralised anti-coagulant activity of unfractionated and low molecular weight heparins, inhibited enzymatic sulfation and degradation reactions. Surfen also blocked signalling and cell adhesion to fibronectin that was triggered by heparan sulphate.Formule :C21H22Cl2N6ODegré de pureté :Min. 95%Masse moléculaire :445.34 g/molZanubrutinib
CAS :Inhibitor of Bruton's tyrosine kinase (BTK)Formule :C27H29N5O3Degré de pureté :Min. 95%Masse moléculaire :471.55 g/molYM 60828
CAS :Inhibits factor Xa; anti-thrombotic
Formule :C27H33Cl2N5O5SDegré de pureté :Min. 95%Masse moléculaire :610.55 g/molSpirapril hydrochloride
CAS :Spirapril hydrochloride is an antihypertensive agent, which is a synthetic pharmaceutical compound designed to treat high blood pressure. The compound is derived from laboratory synthesis aimed at modulating the renin-angiotensin-aldosterone system. Its mode of action involves the inhibition of angiotensin-converting enzyme (ACE), which is crucial for the conversion of angiotensin I to the vasoconstrictor peptide angiotensin II. Angiotensin II is responsible for the constriction of blood vessels and an increase in blood pressure. By inhibiting this enzyme, Spirapril hydrochloride effectively reduces vascular resistance and lowers blood pressure.Formule :C22H30N2O5S2•HClDegré de pureté :Min. 95%Masse moléculaire :503.08 g/molSorafenib
CAS :Sorafenib is a drug that belongs to the class of multikinase inhibitors. It inhibits a number of kinases, including the Mcl-1 protein, which is involved in apoptosis along with blocking picolinic acid (PA), an endogenous metabolite involved in apoptosis signal transduction. Sorafenib also binds to epidermal growth factor receptor (EGFR) on the surface of cancer cells, inhibiting the production of proteins that are required for angiogenesis, thus blocking the formation of new blood vessels. Sorafenib may also inhibit P-glycoprotein (Pgp) activity. Overall, these cytotoxic effects give Sorafenib anti-tumor properties, inhibiting angiogenesis and cellular transformation, which are the two main processes of tumor growth and metastasis. Sorafenib has been shown to be effective against a range of solid tumors such as breast, prostate and lung cancers and is also used for the treatment of metastatic colorectal cancer and renal cell carcinoma. A combination therapy group found that sorafenib was more effective when used with interferon alfa-2b for the treatment of advanced renal cell carcinoma. Sorafenib also has the potential for drug interactions with other drugs that are metabolized by cytochrome P450 enzymes.
Formule :C21H16ClF3N4O3Degré de pureté :Min. 98.0 Area-%Couleur et forme :White PowderMasse moléculaire :464.82 g/molSB 505124
CAS :Inhibitor of ALK4, ALK5, and ALK7 receptorsFormule :C20H21N3O2Degré de pureté :Min. 95%Masse moléculaire :335.4 g/molForetinib
CAS :Inhibits MET, VEGFR2, Ron, AXL, Tie-2, Flt-1, Flt-3 and Flt-4 tyrosine kinases
Formule :C34H34F2N4O6Degré de pureté :Min. 95%Couleur et forme :White To Off-White SolidMasse moléculaire :632.24464Regorafenib monohydrate
CAS :Multi-kinase inhibitor; inhibits epoxide hydrolase; antineoplasticFormule :C21H15ClF4N4O3•H2ODegré de pureté :Min. 95%Masse moléculaire :500.83 g/molMLN 0905
CAS :Inhibitor of Polo-like kinase 1Formule :C24H25F3N6SDegré de pureté :Min. 95%Masse moléculaire :486.56 g/molErlotinib base
CAS :Tyrosine kinase inhibitor; affects EGFR receptor; pancreatic cancer treatmentFormule :C22H23N3O4Degré de pureté :Min. 99 Area-%Couleur et forme :PowderMasse moléculaire :393.44 g/molIWP-2
CAS :Antagonist of Wnt signalling pathway by inhibiting the activity of Porcn, a member of the membrane-bound O-acyltransferase (MBOAT) family. Porcn is required for the palmitoylation of Wnt, mediating its secretion and signalling. Inhibits self-renewal in embryonic stem cells, whilst promoting differentiation to epiblast stem cells.Formule :C22H18N4O2S3Degré de pureté :Min. 95%Couleur et forme :White To Off-White SolidMasse moléculaire :466.05919
