Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
693 produits trouvés pour "Modulateurs d'enzymes"
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Licofelone
CAS :Dual COX/5-LO inhibitor; anti-inflammatory; analgesic
Formule :C23H22ClNO2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :379.88 g/molGefitinib hydrochloride
CAS :RIPK2 protein kinase inhibitor; EGFR inhibitorFormule :C22H24ClFN4O3·HClDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :483.36 g/molAZD 1152
CAS :AZD 1152 is an Aurora kinase inhibitor, which is a type of small-molecule therapeutic agent. It is derived from the pharmaceutical research conducted by AstraZeneca. Its primary mode of action involves the selective inhibition of Aurora B kinase, an enzyme crucial for the regulation of mitosis. By interfering with this enzyme, AZD 1152 disrupts the normal progression of cell division, leading to the inhibition of proliferation and induction of apoptosis in rapidly dividing cells.Formule :C26H31FN7O6PDegré de pureté :Min. 97 Area-%Couleur et forme :Slightly Yellow PowderMasse moléculaire :587.54 g/molCerivastatin sodium
CAS :An inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase that reduces total cholesterol and low-density lipoprotein (LDL). Cerivastatin is cardioprotective and anti-atherosclerotic. Cerivastatin inhibits the expression of the atherosclerotic genes monocyte chemoattractant protein-1 (MCP-1) and C-C chemokine receptor type 2 (CCR2), whilst inducing the expression of Kruppel-like factor 2 (KLF2).Formule :C26H33FNNaO5Degré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :481.53 g/molSU 11274
CAS :MET tyrosine kinase inhibitor; anti-proliferative; pro-apoptoticFormule :C28H30ClN5O4SDegré de pureté :Min. 95%Couleur et forme :Yellow To Orange SolidMasse moléculaire :568.09 g/molOmeprazole - Bio-X ™
CAS :Omeprazole is a proton pump inhibitor (PPI) that inhibits the production of gastric acid in the stomach. This is due to Omeprazole binding through a stable disulphide bond to the H+/K+ ATPase enzyme found on parietal cells, and preventing hydrogen ion transport. Consequently, gastric acid secretion is supressed. As a PPI, Omerprazole can be used to treat disorders where gastric acid is over-secreted. Examples of these disorders are gastroesophageal reflux disease (GERD) and peptic ulcer disease.Formule :C17H19N3O3SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :345.42 g/molAceclofenac - Bio-X ™
CAS :Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.Formule :C16H13Cl2NO4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :354.18 g/molUNC 4203
CAS :Potent and specific inhibitor of the tyrosine protein kinase Mer precursor (MERTK) with 38-fold selectivity over the FMS-like protein kinase FLT3. UNC 4203 inhibits MERTK with an IC50 value of 2.4 nM and shows favourable pharmacokinetic properties. In vivo experiments in mice showed that UNC 4203 dramatically decreased the phosphorylation of MERTK in bone marrow leukemia cells.Formule :C30H44N6ODegré de pureté :Min. 95%Couleur et forme :Yellow PowderMasse moléculaire :504.71 g/molIrsogladine maleate - Bio-X ™
CAS :Irsogladine is a gastroprotective drug that is used for the treatment of GERD and gastric ulcers. This drug also has antioxidant properties. Irsogladine is a phosphodiesterase-4 inhibitor and increases levels of cAMP. It helps to prevent and heal damage to the stomach lining.Formule :C13H11Cl2N5O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :372.16 g/molChymostatin
CAS :Inhibitor of chymotrypsinFormule :C31H41N7O6Couleur et forme :White To Yellowish SolidMasse moléculaire :607.7 g/molBAY 607550
CAS :A selective and potent inhibitor of phosphodiesterase 2 (PDE2). Raises cAMP and cGMP levels in neurons, improves social recognition and object memory in murine animals. Reverses anxiolytic effects induced by oxidative stress in mice by blocking cGMP-PKG signaling.
Formule :C27H32N4O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :476.24236Zotarolimus
CAS :Inhibitor of immunophilin FKBP12 and mTOR signalling with immunosuppressant activity. Zotarolimus inhibits proliferation of endothelial cells and smooth muscle cells and is employed in vascular interventional therapies.Formule :C52H79N5O12Degré de pureté :Min. 95%Couleur et forme :White PowderMasse moléculaire :966.21 g/molRebamipide - Bio-X ™
CAS :Rebamipide is a gastroprotective agent that is used to treat various gastrointestinal disorders such as gastric ulcers and GERD. This drug’s mechanism of action is not fully understood however, it is thought to exert its effects by promoting the secretion of protective mucus in the stomach and intestine, which helps to create a barrier against stomach acid and other irritants. Additionally, it has antioxidant and anti-inflammatory properties that can help reduce tissue damage.Formule :C19H15ClN2O4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :370.79 g/molThioglycosyl Naphthalimide
CAS :Thioglycosyl Naphthalimide is a highly potent human O-GlcNAcase (hOGA) inhibitor with good selectivity against human β-N-acetylhexosaminidase B (HsHexB).Formule :C30H40N4O7SDegré de pureté :Min. 95%Masse moléculaire :600.73 g/molGilteritinib
CAS :Inhibitor of FLT3 and AXL tyrosine kinasesFormule :C29H44N8O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :552.71 g/mol(-)-Huperzine A
CAS :Acetylcholinesterase inhibitor; therapy for Alzheimer's diseaseFormule :C15H18N2ODegré de pureté :(%) Min. 98%Couleur et forme :PowderMasse moléculaire :242.32 g/molLY 411575
CAS :Potent inhibitor of γ-secretase. LY 411575 inhibited production of amyloid β (Aβ) peptides with IC50 of 0.078 nM in vitro as well as decreased levels of Aβ40 and Aβ42 amyloids in brain of a mouse model for Alzheimer’s disease. In vitro studies confirmed that LY 411575 inhibited cleavage of Notch receptor at S3 site with IC50 of 0.39 nM, which blocked Notch activation and downstream signalling, leading to apoptosis in primary and immortalized Kaposi's sarcoma cells.Formule :C26H23F2N3O4Degré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :479.48 g/molLovastatin - Bio-X ™
CAS :Lovastatin is an HMG-CoA reductase inhibitor that is used to lower LDL cholesterol levels and to aid in the management of cardiovascular diseases. Animal studies have demonstrated that this drug has vasculoprotective properties.Formule :C24H36O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :404.54 g/molMRK 560
CAS :γ-secretase inhibitor; reduces amyloid-β in brainÂ
Formule :C19H17ClF5NO4S2Degré de pureté :Min. 95%Masse moléculaire :517.92 g/molRofecoxib - Bio-X ™
CAS :Produit contrôléRofecoxib is a non-steroidal anti-inflammatory drug that is used to treat osteoarthritis, acute pain and migraine attacks. This drug is also a COX-2 inhibitor. As a result, it reduces inflammation and pain.Formule :C17H14O4SDegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :314.36 g/mol
