Modulateurs d'enzymes
Les modulateurs d'enzymes sont des composés qui peuvent augmenter ou inhiber l'activité des enzymes, régulant ainsi la vitesse des réactions biochimiques. Ces modulateurs jouent un rôle essentiel dans le contrôle des voies métaboliques, de la signalisation cellulaire et de divers processus physiologiques. Les modulateurs d'enzymes sont largement utilisés dans la recherche et le développement de médicaments pour étudier les fonctions enzymatiques et développer des agents thérapeutiques. Chez CymitQuimica, nous proposons une gamme complète de modulateurs d'enzymes de haute qualité pour soutenir vos recherches sur la régulation enzymatique et la découverte de médicaments.
Sous-catégories appartenant à la catégorie "Modulateurs d'enzymes"
644 produits trouvés pour "Modulateurs d'enzymes".
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Crenolanib
CAS :Inhibits type III tyrosine kinases (PDGFRα, PDGFRβ, FLT3)Formule :C26H29N5O2Degré de pureté :Min. 95%Couleur et forme :White To Yellow SolidMasse moléculaire :443.54 g/molBMS 754807
CAS :A reversible inhibitor of IGF-1R kinase and insulin receptor. Has anti-growth effects in mesenchymal, epithelial and hematopoietic tumor types. Synergistic with other cytotoxic, hormonal and targeted anti-cancer therapy.
Formule :C23H24FN9ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :461.49 g/molAceclofenac - Bio-X ™
CAS :Acecelofenac is a non-steroidal anti-inflammatory drug that is used in the treatment of osteoarthritis, arthritis, and ankylosing spondylitis. This drug is also a cyclooxygenase inhibitor and works by inhibiting this enzyme so that pain and inflammation is reduced.Formule :C16H13Cl2NO4Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :354.18 g/molSB 239063
CAS :Inhibits p38 MAP kinase; anti-inflammatory; neuroprotectiveFormule :C20H21FN4O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :368.4 g/molMGCD 265
CAS :Inhibits MET, VEGFR1-3, Tie and Ron tyrosine kinases; antineoplasticFormule :C26H20FN5O2S2Degré de pureté :Min. 95%Masse moléculaire :517.60 g/molXMU MP 2
CAS :BRK tyrosine kinase (PTK6) inhibitor; anti-proliferative in breast cancer cells
Formule :C32H33F3N8O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :618.65 g/molSivelestat
CAS :Inhibitor of human neutrophil elastase
Formule :C20H22N2O7SDegré de pureté :Min. 95%Masse moléculaire :434.46 g/molGC376 sodium
CAS :GC 376 is an inhibitor of the main protease Mpro (3CLpro) in coronaviruses as well as picornaviruses. This broad-spectrum antiviral compound has been used as investigational veterinary drug for treatment of feline infectious peritonitis virus (FIPV) infections. Recent studies also showed that GC 376 inhibits the main protease Mpro (3CLpro) from SARS-CoV-2 with IC50 of 0.03 μM and EC50 of 3.37 μM.
Formule :C21H30N3NaO8SDegré de pureté :Min. 95 Area-%Couleur et forme :White PowderMasse moléculaire :507.53 g/molIdelalisib
CAS :Idelalisib is a pharmaceutical drug that functions as a PI3Kδ inhibitor, developed through synthetic chemical processes. Its mode of action involves selectively targeting and inhibiting phosphatidylinositol 3-kinase delta (PI3Kδ), a lipid kinase that plays a crucial role in the signaling pathways responsible for cell proliferation, survival, and differentiation. By inhibiting this enzyme, Idelalisib effectively impedes pathways that are often hyperactivated in certain hematologic malignancies, thereby exerting antitumor effects.Formule :C22H18FN7ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :415.42 g/molSRT1720 hydrochloride
CAS :SIRT1 activatorFormule :C25H23N7OS·xHClDegré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :469.56 g/molAG 221
CAS :Inhibitor of isocitrate dehydrogenase 2Formule :C19H17F6N7ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :473.38 g/molDCC 2036
CAS :Inhibits multiple tyrosine kinases (Abl1, Src family kinases, Tie-2 and VEGFR-2)Formule :C30H28FN7O3Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :553.59 g/molSGC AAK1 1
CAS :Dual inhibitor of the adaptor protein 2-associated kinase 1 (AAK1) and BMP2-inducible kinase (BMP2K) with IC50 values of 270 nM and 1 μM, respectively. In a recent study, SGC AAK1 1 stabilised β-catenin, inhibited phosphorylation of the AP2 complex subunit mu protein (AP2M1) and activated Wnt signalling in in vitro experiments._x000D_Formule :C21H25N5O3SDegré de pureté :Min. 95%Couleur et forme :SolidMasse moléculaire :427.52 g/molEbselen
CAS :Ebselen is a non-toxic organoselenium compound with antioxidant, anti-inflammatory and cytoprotective properties. Ebselen is an inhibitor of lipoxygenases, nitric oxide (NO) synthases, protein kinase C, H+/K+-ATPase, thioredoxin reductase and NADPH oxidase. Recently, ebselen has been identified by several studies as a covalent inhibitor of the main protease Mpro from coronaviruses. For the SARS-CoV-2 main protease Mpro, the IC50 value is 0.67 μM and EC50 is 4.57 μM.Formule :C13H9NOSeDegré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :274.18 g/molPD 169316
CAS :Inhibitor of p38 kinase
Formule :C20H13FN4O2Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :360.34 g/molLY 2886721
CAS :Inhibitor of BACE1 proteaseFormule :C18H16F2N4O2SDegré de pureté :Min. 98 Area-%Couleur et forme :PowderMasse moléculaire :390.41 g/molZileuton- Bio-X ™
CAS :Zileuton is an inhibitor of the 5-lipoxygenase enzyme, thus preventing the leukotrienes LTE4, LDT4, LTB4 and LTC4 from being formed. This in turn reduces inflammation, bronchoconstriction and mucus secretion in the airways. As a result, Zileuton can be used in the treatment and management of asthma and allergic rhinitis. Studies have shown that Zileuton has the potential to reverse dementia-related brain damage.Formule :C11H12N2O2SDegré de pureté :(%) Min. 95%Couleur et forme :PowderMasse moléculaire :236.29 g/molKenpaullone
CAS :Inhibitor of glycogen synthase 3 (GSK-3) and cyclin-dependent kinases CDK1, CDK2 and CDK5. Kenpaullone can substitute transcription factor Klf4 in reprogramming of fibroblast to induced pluripotent stem cells when using the method of ectopic expression of transcriptional factors. In an in vitro model for Alzheimer’s disease, kenpaullone decreased production of amyloid beta peptides Aβ40 and Aβ42.
Formule :C16H11BrN2ODegré de pureté :Min. 95%Couleur et forme :Yellow To Dark Yellow SolidMasse moléculaire :326.00548GSK 2606414
CAS :Inhibitor of EIF2AK3/PERK kinasesFormule :C24H20F3N5ODegré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :451.44 g/molA 485
CAS :Histone acetyltransferase inhibitor of p300/CBP; anti-proliferative
Formule :C25H24F4N4O5Degré de pureté :Min. 95%Couleur et forme :PowderMasse moléculaire :536.48 g/mol
