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Se termine le 31 déc.( plus que 7 jours )
AT-1015 hydrochloride monohydrate
CAS :AT-1015 hydrochloride monohydrate is a serotonin (5-HT)2 receptor antagonist that blocks vascular and platelet 5-HT2A receptors.Formule :C29H36ClN3O3Couleur et forme :SolidMasse moléculaire :510.08MDK6465
CAS :MDK6465 (PCSK9-IN-8b), CAS#1900686-46-5, is a liver-targeted PCSK9 synthesis inhibitor.Formule :C27H29ClFN9O4Couleur et forme :SolidMasse moléculaire :598.03UNC2025
CAS :<p>UNC2025 (mrx-6313)(IC50 of 0.74 nM and 0.8 nM) is a potent and orally bioavailable dual MER/FLT3 inhibitor.</p>Formule :C28H40N6ODegré de pureté :99.53% - 99.74%Couleur et forme :SolidMasse moléculaire :476.66Cisapride tartrate
CAS :Cisapride tartrate is chemically related to metoclopramide, but unlike metoclopramide, it does not cross the blood-brain barrier or have antidopaminergicFormule :C27H35ClFN3O10Couleur et forme :SolidMasse moléculaire :616.04SLM6031434 (free base)
CAS :SLM6031434 (free base) is an inhibitor of sphingosine kinase type 2 (SphK2). It consists of pedant 1-guanidino-2-phenyloxadiazolylpyrrolidine group.Formule :C22H30F3N5O2Couleur et forme :SolidMasse moléculaire :453.5Aplindore
CAS :<p>Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.</p>Formule :C18H18N2O3Couleur et forme :SolidMasse moléculaire :310.35Fabomotizole dihydrochloride
CAS :<p>Fabomotizole (Afobazole, Obenoxazine, CM346) is a non-sedative anxiolytic with neuroprotective properties, launched in Russia 2000s; exact mechanism unclear.</p>Formule :C15H23Cl2N3O2SCouleur et forme :SolidMasse moléculaire :380.33SB1-F-21
CAS :SB1-F-21 is an UCHL1 inhibitor.Formule :C15H14N4OSCouleur et forme :SolidMasse moléculaire :298.36KDS2010 mesylate
CAS :<p>KDS2010: potent, reversible MAO-B inhibitor with 12,500x selectivity vs. MAO-A; enhances memory in APP/PS1 mice.</p>Formule :C18H21F3N2O4SCouleur et forme :SolidMasse moléculaire :418.43NOSO-95C
CAS :<p>NOSO-95C, an antibacterial, targets bacterial ribosomes, halting translation, and is effective against Enterobacteriaceae in vitro/in vivo.</p>Formule :C54H101N23O12Couleur et forme :SolidMasse moléculaire :1264.53Fadolmidine HCl
CAS :<p>Fadolmidine (MPV-2426) is a potent alpha2-adrenoceptor agonist for spinal analgesia with high affinity across human subtypes and efficacy in vivo.</p>Formule :C13H15ClN2OCouleur et forme :SolidMasse moléculaire :250.72Fadolmidine
CAS :Fadolmidine is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia.Formule :C13H14N2OCouleur et forme :SolidMasse moléculaire :214.26MPV-1306
CAS :MPV-1306 is a metabolite of Dexmedetomidine -- a novel alpha 2-adrenergic receptor agonist.Formule :C13H14N2O2Couleur et forme :SolidMasse moléculaire :230.26Vacquinol-1
CAS :Vacquinol-1 is an MKK4 activator, which rapidly and selectively induces glioma cell death.Formule :C21H21ClN2ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :352.86Methasquin
CAS :<p>Methasquin is a folic acid antagonist that has been used in the treatment of experimental leukemia; acts by inhibiting the dihydrofolate reductase in the cell.</p>Formule :C21H22N6O5Couleur et forme :SolidMasse moléculaire :438.44Pd 158771
CAS :Pd 158771 is a D2 and 5-HT1A agonist.Formule :C22H31N5Couleur et forme :SolidMasse moléculaire :365.52Pyrithione cadmium
CAS :Pyrithione cadmium suppresses tumor growth in vitro and in vivo through inhibition of proteasomal deubiquitinaseFormule :C10H8CdN2O2S2Couleur et forme :SolidMasse moléculaire :364.73Cilengitide hydrochloride
CAS :Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.Formule :C27H41ClN8O7Couleur et forme :SolidMasse moléculaire :625.12Dersalazine
CAS :<p>Dersalazine, a PAF inhibitor, reduces IL-17 to treat colitis in rodents, potentially aiding ulcerative colitis patients.</p>Formule :C35H32N6O4Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :600.67IND 1316
CAS :IND 1316 is an activator of AMP-activated protein kinase (AMPK).Formule :C22H17NO3Couleur et forme :SolidMasse moléculaire :343.38EPZ033294
CAS :EPZ033294 has potential anticancer and antiproliferative activity.Formule :C20H22ClN7ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :411.89EPZ032597
CAS :EPZ032597 is a novel selective inhibitor of SMYD2 with an IC50 of 16 nM. EPZ032597 has anticancer activity and prevent and treat pancreatic cancerFormule :C20H23N7ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :377.44Grp94-IN-2
CAS :Grp94-IN-2 is a inhibitor of Grp94.Formule :C22H23ClN2O5Couleur et forme :SolidMasse moléculaire :430.88Colterol (free base)
CAS :Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Formule :C12H19NO3Couleur et forme :SolidMasse moléculaire :225.28Soyacerebroside II
CAS :Soyacerebroside II is a Ca2+ ionophore; both I and II inhibit IL-18 in PBMCs and modulate immune responses.Formule :C40H75NO9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :714.02Nizatidine amide
CAS :Nizatidine amide blocks H2 receptors, reducing stomach acid to treat ulcers and GERD.Formule :C11H18N4O3S2Couleur et forme :SolidMasse moléculaire :318.42IACS-4759
CAS :IACS-4759 is a novel potent and selective MTH1 inhibitor with excellent cell permeability and good metabolic stability in microsomes.Formule :C10H17N3O2Couleur et forme :SolidMasse moléculaire :211.26ent-Entecavir
CAS :Ent-Entecavir, an enantiomeric impurity of Entecavir (an oral HBV drug), inhibits HBV replication as a reverse transcriptase inhibitor.Formule :C12H15N5O3Couleur et forme :SolidMasse moléculaire :277.28JTP 103237
CAS :<p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>Formule :C24H29F3N6OCouleur et forme :SolidMasse moléculaire :474.52MS-049 oxalate salt
CAS :MS-049 oxalate salt is a potent and selective inhibitor of protein arginine methyltransferases (PRMTs) PRMT 4 and PRMT6.Formule :C17H26N2O5Couleur et forme :SolidMasse moléculaire :338.4Mps1-IN-1 dihydrochloride
CAS :Mps1-IN-1 dihydrochloride, a potent ATP-competitive inhibitor of Mps1 kinase, exhibits an IC50 of 367 nM.Formule :C28H35Cl2N5O4SCouleur et forme :SolidMasse moléculaire :608.58AEG40730 HCl
CAS :<p>AEG40730: A potent, selective IAP inhibitor, induces cIAP1/2 degradation, reduces RIP1 ubiquitination, and depletes XIAP, c-IAP1.</p>Formule :C52H70Cl2F6N8O8Couleur et forme :SolidMasse moléculaire :1120.0704Acefylline piperazine
CAS :Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.Formule :C9H10N4O4·xC4H10N2Couleur et forme :SolidMasse moléculaire :562.54CDK8-IN-18
CAS :CDK8-IN-18, also known as ZINC584617986, is a potent and selective inhibitor of CDK8, also modulating CDK19.Formule :C18H17N5OCouleur et forme :SolidMasse moléculaire :319.36Methylsilanol ascorbate
CAS :Methylsilanol ascorbate is a silanol analogue and inhibitor of angiotensin-converting enzyme.Formule :C7H12O8SiCouleur et forme :SolidMasse moléculaire :252.25VER-155008
CAS :<p>VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively.</p>Formule :C25H23Cl2N7O4Degré de pureté :97.03% - 99.55%Couleur et forme :SolidMasse moléculaire :556.4SG3-179
CAS :SG3-179 is a BET inhibitor.Formule :C28H35ClFN7O3SCouleur et forme :SolidMasse moléculaire :604.14EMD-66684
CAS :EMD-66684 is a non-peptide angiotensin II receptor antagonist.Formule :C28H31ClN8O2Couleur et forme :SolidMasse moléculaire :547.06KFP-H008
CAS :KFP-H008 is a potassium-competitive acid blocker.Formule :C19H18N4O2SCouleur et forme :SolidMasse moléculaire :366.44KSK213
CAS :KSK213: Strongly inhibits C. trachomatis (EC50=60 nM); non-toxic to commensals/host cells at 25 μM.Formule :C28H25N3O2SCouleur et forme :SolidMasse moléculaire :467.58Verubecestat tosylate
CAS :Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.Formule :C25H26N4O4S2Couleur et forme :SolidMasse moléculaire :510.627Chlorpromazine Sulfone Hydrochloride
CAS :Chlorpromazine Sulfone Hydrochloride: metabolite of anti-psychotic, may inhibit N-methyltransferase.Formule :C17H20Cl2N2O2SCouleur et forme :SolidMasse moléculaire :387.32F-050
CAS :F-050 inhibits platelet aggregation, potentially treating thrombosis in guinea pigs, rabbits, and rats.Formule :C21H20OCouleur et forme :SolidMasse moléculaire :288.38Olcorolimus
CAS :Olcorolimus blocks specific allergen-induced inflammation, reducing eosinophil, lymphocyte infiltration, and IL-4/IL-5 mRNA expression.Formule :C51H81NO12Couleur et forme :SolidMasse moléculaire :900.19Fasudil hydrochloride hydrate
CAS :Fasudil HCl hydrate is a ROCK inhibitor that hinders mature CCM development and lowers portal pressure in cirrhotic rats.Formule :C28H38Cl2N6O5S2Couleur et forme :SolidMasse moléculaire :673.67Delucemine Free Base
CAS :Delucemine Free Base is an NMDA Receptor AntagonistFormule :C16H17F2NCouleur et forme :SolidMasse moléculaire :261.31Verubecestat
CAS :<p>Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.</p>Formule :C17H17F2N5O3SDegré de pureté :92.24% - 99.55%Couleur et forme :SolidMasse moléculaire :409.41CVS-1578
CAS :CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.Formule :C20H30N6O5SCouleur et forme :SolidMasse moléculaire :466.55GT-2394
CAS :GT-2394 is a histamine H3 receptor agonist.Formule :C14H21N3O2Couleur et forme :SolidMasse moléculaire :263.34GT-2227
CAS :<p>GT-2227 is a histamine H3 receptor antagonist.</p>Formule :C15H24N2Couleur et forme :SolidMasse moléculaire :232.36
