CAS 952654-62-5

(3R,4R,5R,6R)-6-[4-[(4-fluorofenil)metilcarbamoil]-1-metil-2-[1-metil-1-[(5-metil-1,3,4-ossadiazolo-2-carbonil)amino]etil]-6-osso-pirimidin-5-il]ossi-3,4,5-triidrossi-tetraidropirano-2-carbossilico acido

Formula: C₂₆H₂₉FN₆O₁₁

InChI: InChI=1/C26H29FN6O11/c1-10-31-32-21(42-10)20(38)30-26(2,3)25-29-13(19(37)28-9-11-5-7-12(27)8-6-11)17(22(39)33(25)4)43-24-16(36)14(34)15(35)18(44-24)23(40)41/h5-8,14-16,18,24,34-36H,9H2,1-4H3,(H,28,37)(H,30,38)(H,40,41)/t14-,15-,16-,18?,24+/m1/s1

Raltegravir Glucuronide

CAS: 952654-62-5

Formula: C₂₆H₂₉FN₆O₁₁

Colore e forma: White To Off-White Solid

Peso molecolare: 620.55

Ref: 4Z-R-243

Raltegravir b-D-glucuronide

CAS: 952654-62-5

Ref: 7W-GC7918

Raltegravir β-D-Glucuronide

CAS: 952654-62-5

Applications A metabolite of Raltegravir.
References Bosma, P., et al.: J. Biol. Chem., 269, 17960 (1994), Richman, D., et al.: Nature, 410, 995 (2001), Williams, J., et al.: Drug Metab. Dispos., 32, 1201 (2004), Miners, J., et al.: Biochem. Pharmacol., 71, 1531 (2006),

Formula: C₂₆H₂₉FN₆O₁₁

Colore e forma: Neat

Peso molecolare: 620.54

Ref: TR-R100310

Raltegravir-d3 b-D-Glucuronide (>90%)

Prodotto controllato

CAS: 952654-62-5

Applications A labelled metabolite of Raltegravir.
References Bosma, P., et al.: J. Biol. Chem., 269, 17960 (1994) , Richman, D., et al.: Nature, 410, 995 (2001), Williams, J., et al.: Drug Metab. Dispos., 32, 1201 (2004), Miners, J., et al.: Biochem. Pharmacol., 71, 1531 (2006),

Formula: C₂₆H₂₆D₃FN₆O₁₁

Purezza: >90%

Colore e forma: Neat

Peso molecolare: 623.56

Ref: TR-R100312

Raltegravir b-D-glucuronide

CAS: 952654-62-5

Raltegravir b-D-glucuronide is a synthetic, fluorinated analog of raltegravir. It is a potent HIV-1 integrase inhibitor that has been shown to be active against the majority of HIV-1 strains. Raltegravir b-D-glucuronide is less potent than the parent compound and exhibits reduced antiviral activity in vitro. Raltegravir b-D-glucuronide is metabolized to raltegravir and eliminated in urine as the glucuronide conjugate.

Formula: C₂₆H₂₉FN₆O₁₁

Purezza: Min. 95%

Colore e forma: White Powder

Peso molecolare: 620.54 g/mol

Ref: 3D-MR09516

Raltegravir β-D-Glucuronide

CAS: 952654-62-5

Formula: C₂₆H₂₉FN₆O₁₁

Peso molecolare: 620.55

Ref: ST-EA-CP-R6020