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Syk

Syk

Gli inibitori della chinasi splenica (Syk) sono composti che prendono di mira Syk, una chinasi coinvolta nella segnalazione delle cellule immunitarie e nella regolazione dell'angiogenesi. Syk svolge un ruolo nelle risposte infiammatorie che possono contribuire all'angiogenesi tumorale. L'inibizione di Syk può ridurre la formazione di vasi sanguigni indotta dall'infiammazione nei tumori, rendendo questi inibitori preziosi nella terapia del cancro e nella ricerca sull'infiammazione. Presso CymitQuimica, offriamo una gamma diversificata di inibitori di Syk di alta qualità per supportare la tua ricerca in immunologia, oncologia e angiogenesi.

Trovati 37 prodotti di "Syk"

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  • Piceatannol

    CAS:
    Formula:C14H12O4
    Purezza:>98.0%(HPLC)
    Colore e forma:White to Light yellow to Light red powder to crystal
    Peso molecolare:244.25

    Ref: 3B-P1928

    1g
    478,00€
    100mg
    77,00€
  • Gusacitinib

    CAS:
    <p>Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).</p>
    Formula:C24H28N8O2
    Purezza:98.06% - 99.94%
    Colore e forma:Solid
    Peso molecolare:460.53

    Ref: TM-T14331

    1mg
    42,00€
    5mg
    88,00€
    10mg
    123,00€
    25mg
    188,00€
    50mg
    350,00€
    100mg
    522,00€
    200mg
    750,00€
  • Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Formula:C9H11NO3·HCl
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:217.65

    Ref: TM-T0948

    1g
    145,00€
    50mg
    35,00€
    100mg
    50,00€
    500mg
    97,00€
  • 1,3-Benzodioxole, 5-(2-nitroethenyl)-

    CAS:
    Formula:C9H7NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:193.1562

    Ref: IN-DA001KYU

    1g
    44,00€
    5g
    66,00€
    10g
    73,00€
    25g
    114,00€
    50g
    203,00€
    100g
    240,00€
    250g
    632,00€
    250mg
    28,00€
  • Piceatannol

    CAS:
    Piceatannol (Astringenin) is a synthetic anti-inflammatory that blocks p56lck, syk kinases, and NF-κB, made from resveratrol.
    Formula:C14H12O4
    Purezza:98.66% - 99.73%
    Colore e forma:Light Tan To Yellow Powder
    Peso molecolare:244.24

    Ref: TM-T0610

    5mg
    42,00€
    10mg
    60,00€
    25mg
    103,00€
    50mg
    150,00€
    100mg
    207,00€
    1mL*10mM (DMSO)
    50,00€
  • Lanraplenib

    CAS:
    Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.
    Formula:C23H25N9O
    Purezza:98.35%
    Colore e forma:Solid
    Peso molecolare:443.5

    Ref: TM-T11824LL

    1mg
    51,00€
    2mg
    74,00€
    5mg
    99,00€
    10mg
    167,00€
    25mg
    290,00€
    50mg
    430,00€
    100mg
    633,00€
    1mL*10mM (DMSO)
    115,00€
  • 1,2-Benzenediol, 4-[(1E)-2-(3,5-dihydroxyphenyl)ethenyl]-

    CAS:
    Formula:C14H12O4
    Purezza:97%
    Colore e forma:Solid
    Peso molecolare:244.2427

    Ref: IN-DA0002ZH

    1g
    26,00€
    5g
    68,00€
    25g
    198,00€
    100mg
    25,00€
    250mg
    29,00€
  • Tyrosine Kinase Inhibitor Library


    A unique collection of 1016 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related
    Colore e forma:Odour Solid

    Ref: TM-L2200

    1mg
    Prezzo su richiesta
    30μL*10mM (DMSO)
    Prezzo su richiesta
    50μL*10mM (DMSO)
    Prezzo su richiesta
    100μL*10mM (DMSO)
    Prezzo su richiesta
    250μL*10mM (DMSO)
    Prezzo su richiesta
  • Syk Kinase Peptide Substrate, Biotin labeled


    The compound, Biotin-labeled Syk Kinase Peptide Substrate, is a peptide substrate of Syk kinase that is labeled with biotin.
    Formula:C76H108N18O24S1
    Colore e forma:Solid
    Peso molecolare:1689.9

    Ref: TM-T76083

    5mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • Cevidoplenib dimesylate

    CAS:
    <p>Cevidoplenib dimesylate is an inhibitor of spleen tyrosine kinase (Syk), possessing anti-inflammatory and immunomodulating properties.</p>
    Formula:C27H35N7O9S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:665.74

    Ref: TM-T39437

    1mg
    65,00€
    5mg
    140,00€
    10mg
    188,00€
    25mg
    374,00€
    50mg
    560,00€
  • Syk-IN-7


    <p>Syk-IN-7 (compound 17) acts as an inhibitor of spleen tyrosine kinase (SYK) [1].</p>
    Formula:C26H31N9O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:533.58

    Ref: TM-T78943

    5mg
    Prezzo su richiesta
    50mg
    Prezzo su richiesta
  • Lanraplenib succinate

    CAS:
    Lanraplenib succinate is an oral SYK inhibitor (IC50=9.5 nM) that doesn't extend BT, targeting GPVI in platelets for inflammation treatment.
    Formula:C58H68N18O14
    Colore e forma:Solid
    Peso molecolare:1241.294

    Ref: TM-T11824

    2mg
    65,00€
  • MNS

    CAS:
    Formula:C9H7NO4
    Purezza:>98.0%(GC)
    Colore e forma:Light yellow to Yellow to Green powder to crystal
    Peso molecolare:193.16

    Ref: 3B-M3390

    100mg
    58,00€
    500mg
    174,00€
  • BAY 61-3606 dihydrochloride

    CAS:
    BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).
    Formula:C20H18N6O3·2HCl
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:463.32

    Ref: TM-T6776

    1mg
    38,00€
    5mg
    84,00€
    10mg
    116,00€
    25mg
    187,00€
    50mg
    279,00€
    100mg
    406,00€
    200mg
    565,00€
    1mL*10mM (DMSO)
    87,00€
  • Fostamatinib

    CAS:
    <p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>
    Formula:C23H26FN6O9P
    Purezza:93.08% - 99.38%
    Colore e forma:Solid
    Peso molecolare:580.46

    Ref: TM-T6115

    1mg
    43,00€
    2mg
    57,00€
    5mg
    88,00€
    10mg
    118,00€
    25mg
    210,00€
    50mg
    335,00€
    100mg
    548,00€
    500mg
    1.198,00€
  • TAK-659 hydrochloride

    CAS:
    TAK-659 hydrochloride (TAK-659) is a potent and selective inhibitor of spleen tyrosine kinase (SYK) with an IC50 value of 3.2 nM.
    Formula:C17H22ClFN6O
    Purezza:99.28% - 99.82%
    Colore e forma:Solid
    Peso molecolare:380.85

    Ref: TM-T4209

    1mg
    39,00€
    5mg
    84,00€
    10mg
    111,00€
    25mg
    216,00€
    50mg
    329,00€
    100mg
    512,00€
  • Flavanomarein

    CAS:
    Flavanomarein: Antioxidant with radical scavenging, lipid peroxidation inhibition, and lipid-lowering in HepG2 cells.
    Formula:C21H22O11
    Purezza:98.63% - 99.54%
    Colore e forma:Solid
    Peso molecolare:450.39

    Ref: TM-TN1644

    1mg
    35,00€
    5mg
    64,00€
    10mg
    95,00€
    25mg
    157,00€
    50mg
    221,00€
    1mL*10mM (DMSO)
    81,00€
  • PRT-060318

    CAS:
    PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach to HIT treatment.
    Formula:C18H24N6O
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:340.42

    Ref: TM-T6957

    1mg
    42,00€
    2mg
    52,00€
    5mg
    94,00€
    10mg
    135,00€
    25mg
    274,00€
    50mg
    465,00€
    100mg
    680,00€
  • PRT062607 hydrochloride

    CAS:
    PRT062607 hydrochloride (P505-15 Hydrochloride) is a selective inhibitor of Syk. PRT062607 displays at least 80-fold selectivity for Syk over other kinases.
    Formula:C19H23N9O·HCl
    Purezza:97.7% - 99.81%
    Colore e forma:Solid
    Peso molecolare:429.91

    Ref: TM-T2696

    1mg
    60,00€
    2mg
    86,00€
    5mg
    127,00€
    10mg
    187,00€
    25mg
    326,00€
    50mg
    500,00€
    200mg
    948,00€
    1mL*10mM (DMSO)
    139,00€
  • BAY 61-3606

    CAS:
    <p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>
    Formula:C20H18N6O3
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:390.4

    Ref: TM-T4263

    1mg
    56,00€
    2mg
    79,00€
    5mg
    140,00€
    10mg
    230,00€
    25mg
    378,00€
    50mg
    563,00€