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Syk

Syk

Gli inibitori della chinasi splenica (Syk) sono composti che prendono di mira Syk, una chinasi coinvolta nella segnalazione delle cellule immunitarie e nella regolazione dell'angiogenesi. Syk svolge un ruolo nelle risposte infiammatorie che possono contribuire all'angiogenesi tumorale. L'inibizione di Syk può ridurre la formazione di vasi sanguigni indotta dall'infiammazione nei tumori, rendendo questi inibitori preziosi nella terapia del cancro e nella ricerca sull'infiammazione. Presso CymitQuimica, offriamo una gamma diversificata di inibitori di Syk di alta qualità per supportare la tua ricerca in immunologia, oncologia e angiogenesi.

Trovati 37 prodotti di "Syk"

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  • Piceatannol

    CAS:
    Formula:C14H12O4
    Purezza:>98.0%(HPLC)
    Colore e forma:White to Light yellow to Light red powder to crystal
    Peso molecolare:244.25

    Ref: 3B-P1928

    1g
    478,00€
    100mg
    77,00€
  • Gusacitinib

    CAS:
    <p>Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).</p>
    Formula:C24H28N8O2
    Purezza:98.06% - 99.94%
    Colore e forma:Solid
    Peso molecolare:460.53
  • Adrenalone hydrochloride

    CAS:
    <p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>
    Formula:C9H11NO3·HCl
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:217.65
  • 1,3-Benzodioxole, 5-(2-nitroethenyl)-

    CAS:
    Formula:C9H7NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:193.1562

    Ref: IN-DA001KYU

    1g
    44,00€
    5g
    66,00€
    10g
    73,00€
    25g
    114,00€
    50g
    203,00€
    100g
    240,00€
    250g
    632,00€
    250mg
    28,00€
  • Piceatannol

    CAS:
    <p>Piceatannol (Astringenin) is a synthetic anti-inflammatory that blocks p56lck, syk kinases, and NF-κB, made from resveratrol.</p>
    Formula:C14H12O4
    Purezza:98.66% - 99.73%
    Colore e forma:Light Tan To Yellow Powder
    Peso molecolare:244.24
  • Lanraplenib

    CAS:
    <p>Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.</p>
    Formula:C23H25N9O
    Purezza:98.35%
    Colore e forma:Solid
    Peso molecolare:443.5
  • 1,2-Benzenediol, 4-[(1E)-2-(3,5-dihydroxyphenyl)ethenyl]-

    CAS:
    Formula:C14H12O4
    Purezza:97%
    Colore e forma:Solid
    Peso molecolare:244.2427

    Ref: IN-DA0002ZH

    1g
    26,00€
    5g
    68,00€
    10g
    105,00€
    25g
    198,00€
    100mg
    25,00€
    250mg
    29,00€
  • Tyrosine Kinase Inhibitor Library


    <p>A unique collection of 1016 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related</p>
    Colore e forma:Odour Solid
  • Syk Kinase Peptide Substrate, Biotin labeled


    <p>The compound, Biotin-labeled Syk Kinase Peptide Substrate, is a peptide substrate of Syk kinase that is labeled with biotin.</p>
    Formula:C76H108N18O24S1
    Colore e forma:Solid
    Peso molecolare:1689.9
  • Cevidoplenib dimesylate

    CAS:
    <p>Cevidoplenib dimesylate is an inhibitor of spleen tyrosine kinase (Syk), possessing anti-inflammatory and immunomodulating properties.</p>
    Formula:C27H35N7O9S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:665.74
  • Syk-IN-7


    <p>Syk-IN-7 (compound 17) acts as an inhibitor of spleen tyrosine kinase (SYK) [1].</p>
    Formula:C26H31N9O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:533.58
  • Lanraplenib succinate

    CAS:
    <p>Lanraplenib succinate is an oral SYK inhibitor (IC50=9.5 nM) that doesn't extend BT, targeting GPVI in platelets for inflammation treatment.</p>
    Formula:C58H68N18O14
    Colore e forma:Solid
    Peso molecolare:1241.294
  • MNS

    CAS:
    Formula:C9H7NO4
    Purezza:>98.0%(GC)
    Colore e forma:Light yellow to Yellow to Green powder to crystal
    Peso molecolare:193.16

    Ref: 3B-M3390

    100mg
    58,00€
    500mg
    174,00€
  • BAY 61-3606 dihydrochloride

    CAS:
    <p>BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).</p>
    Formula:C20H18N6O3·2HCl
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:463.32
  • Fostamatinib

    CAS:
    <p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>
    Formula:C23H26FN6O9P
    Purezza:93.08% - 99.38%
    Colore e forma:Solid
    Peso molecolare:580.46
  • TAK-659 hydrochloride

    CAS:
    <p>TAK-659 hydrochloride (TAK-659) is a potent and selective inhibitor of spleen tyrosine kinase (SYK) with an IC50 value of 3.2 nM.</p>
    Formula:C17H22ClFN6O
    Purezza:99.28% - 99.82%
    Colore e forma:Solid
    Peso molecolare:380.85
  • Flavanomarein

    CAS:
    <p>Flavanomarein: Antioxidant with radical scavenging, lipid peroxidation inhibition, and lipid-lowering in HepG2 cells.</p>
    Formula:C21H22O11
    Purezza:98.63% - 99.54%
    Colore e forma:Solid
    Peso molecolare:450.39
  • PRT-060318

    CAS:
    <p>PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach to HIT treatment.</p>
    Formula:C18H24N6O
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:340.42
  • PRT062607 hydrochloride

    CAS:
    <p>PRT062607 hydrochloride (P505-15 Hydrochloride) is a selective inhibitor of Syk. PRT062607 displays at least 80-fold selectivity for Syk over other kinases.</p>
    Formula:C19H23N9O·HCl
    Purezza:97.7% - 99.81%
    Colore e forma:Solid
    Peso molecolare:429.91
  • BAY 61-3606

    CAS:
    <p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>
    Formula:C20H18N6O3
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:390.4