
Syk
Gli inibitori della chinasi splenica (Syk) sono composti che prendono di mira Syk, una chinasi coinvolta nella segnalazione delle cellule immunitarie e nella regolazione dell'angiogenesi. Syk svolge un ruolo nelle risposte infiammatorie che possono contribuire all'angiogenesi tumorale. L'inibizione di Syk può ridurre la formazione di vasi sanguigni indotta dall'infiammazione nei tumori, rendendo questi inibitori preziosi nella terapia del cancro e nella ricerca sull'infiammazione. Presso CymitQuimica, offriamo una gamma diversificata di inibitori di Syk di alta qualità per supportare la tua ricerca in immunologia, oncologia e angiogenesi.
Trovati 37 prodotti di "Syk"
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Piceatannol
CAS:Formula:C14H12O4Purezza:>98.0%(HPLC)Colore e forma:White to Light yellow to Light red powder to crystalPeso molecolare:244.25Gusacitinib
CAS:<p>Gusacitinib (ASN-002) (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).</p>Formula:C24H28N8O2Purezza:98.06% - 99.94%Colore e forma:SolidPeso molecolare:460.53Adrenalone hydrochloride
CAS:<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Formula:C9H11NO3·HClPurezza:99.94%Colore e forma:SolidPeso molecolare:217.651,3-Benzodioxole, 5-(2-nitroethenyl)-
CAS:Formula:C9H7NO4Purezza:98%Colore e forma:SolidPeso molecolare:193.1562Piceatannol
CAS:<p>Piceatannol (Astringenin) is a synthetic anti-inflammatory that blocks p56lck, syk kinases, and NF-κB, made from resveratrol.</p>Formula:C14H12O4Purezza:98.66% - 99.73%Colore e forma:Light Tan To Yellow PowderPeso molecolare:244.24Lanraplenib
CAS:<p>Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.</p>Formula:C23H25N9OPurezza:98.35%Colore e forma:SolidPeso molecolare:443.51,2-Benzenediol, 4-[(1E)-2-(3,5-dihydroxyphenyl)ethenyl]-
CAS:Formula:C14H12O4Purezza:97%Colore e forma:SolidPeso molecolare:244.2427Tyrosine Kinase Inhibitor Library
<p>A unique collection of 1016 tyrosine kinase inhibitors for high throughput screening and high content screening for drug discovery in tyrosine kinase related</p>Colore e forma:Odour SolidSyk Kinase Peptide Substrate, Biotin labeled
<p>The compound, Biotin-labeled Syk Kinase Peptide Substrate, is a peptide substrate of Syk kinase that is labeled with biotin.</p>Formula:C76H108N18O24S1Colore e forma:SolidPeso molecolare:1689.9Cevidoplenib dimesylate
CAS:<p>Cevidoplenib dimesylate is an inhibitor of spleen tyrosine kinase (Syk), possessing anti-inflammatory and immunomodulating properties.</p>Formula:C27H35N7O9S2Purezza:98%Colore e forma:SolidPeso molecolare:665.74Syk-IN-7
<p>Syk-IN-7 (compound 17) acts as an inhibitor of spleen tyrosine kinase (SYK) [1].</p>Formula:C26H31N9O4Purezza:98%Colore e forma:SolidPeso molecolare:533.58Lanraplenib succinate
CAS:<p>Lanraplenib succinate is an oral SYK inhibitor (IC50=9.5 nM) that doesn't extend BT, targeting GPVI in platelets for inflammation treatment.</p>Formula:C58H68N18O14Colore e forma:SolidPeso molecolare:1241.294MNS
CAS:Formula:C9H7NO4Purezza:>98.0%(GC)Colore e forma:Light yellow to Yellow to Green powder to crystalPeso molecolare:193.16BAY 61-3606 dihydrochloride
CAS:<p>BAY 61-3606 dihydrochloride (BAY 61-3606) is a potent and selective inhibitor of Syk kinase (Ki = 7.5 nM).</p>Formula:C20H18N6O3·2HClPurezza:99.46%Colore e forma:SolidPeso molecolare:463.32Fostamatinib
CAS:<p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>Formula:C23H26FN6O9PPurezza:93.08% - 99.38%Colore e forma:SolidPeso molecolare:580.46TAK-659 hydrochloride
CAS:<p>TAK-659 hydrochloride (TAK-659) is a potent and selective inhibitor of spleen tyrosine kinase (SYK) with an IC50 value of 3.2 nM.</p>Formula:C17H22ClFN6OPurezza:99.28% - 99.82%Colore e forma:SolidPeso molecolare:380.85Flavanomarein
CAS:<p>Flavanomarein: Antioxidant with radical scavenging, lipid peroxidation inhibition, and lipid-lowering in HepG2 cells.</p>Formula:C21H22O11Purezza:98.63% - 99.54%Colore e forma:SolidPeso molecolare:450.39PRT-060318
CAS:<p>PRT-060318 (P142-76) is a novel selective inhibitor of the Syk tyrosine kinase, as an approach to HIT treatment.</p>Formula:C18H24N6OPurezza:99.98%Colore e forma:SolidPeso molecolare:340.42PRT062607 hydrochloride
CAS:<p>PRT062607 hydrochloride (P505-15 Hydrochloride) is a selective inhibitor of Syk. PRT062607 displays at least 80-fold selectivity for Syk over other kinases.</p>Formula:C19H23N9O·HClPurezza:97.7% - 99.81%Colore e forma:SolidPeso molecolare:429.91BAY 61-3606
CAS:<p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>Formula:C20H18N6O3Purezza:98.72%Colore e forma:SolidPeso molecolare:390.4



