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Caspasi

Caspasi

Gli inibitori delle caspasi sono composti che bloccano l'attività delle caspasi, una famiglia di proteasi che sono esecutori centrali dell'apoptosi. Le caspasi clivano substrati specifici all'interno della cellula per innescare il processo apoptotico, portando alla morte cellulare programmata. Gli inibitori delle caspasi sono utilizzati per studiare i meccanismi dell'apoptosi, nonché per prevenire la morte cellulare indesiderata in vari modelli di ricerca. Questi inibitori sono anche esplorati in contesti terapeutici per proteggere le cellule dall'apoptosi in malattie come la neurodegenerazione. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle caspasi di alta qualità per supportare la tua ricerca in apoptosi, morte cellulare e campi correlati.

Trovati 143 prodotti di "Caspasi"

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  • Biotin-DEVD-CHO TFA


    Biotin-DEVD-CHO (TFA) is the biotin-conjugated form of the caspase-3 and caspase-7 inhibitor Ac-DEVD-CHO. It can be utilized for affinity purification of active caspase-3, -6, -7, and -8 and is also applicable for in vitro detection of active caspase-3.
    Colore e forma:Odour Solid
  • Perfluorodecanoic acid

    CAS:
    Perfluorodecanoic acid is a biochemical.
    Formula:C10HF19O2
    Colore e forma:Physical Description Liquid (Ntp 1992)
    Peso molecolare:514.08
  • Ac-LEVD-CHO

    CAS:
    <p>Ac-LEVD-CHO, a caspase-4 inhibitor, is a peptide with the sequence Ac-Leu-Glu-Val-Asp-al [1].</p>
    Formula:C22H36N4O9
    Colore e forma:Solid
    Peso molecolare:500.54
  • (Iso)-Z-VAD(OMe)-FMK

    CAS:
    (Iso)-Z-VAD(OMe)-FMK is an isomer of Z-VAD(OMe)-FMK, which is a pan-caspase inhibitor with irreversible properties. Z-VAD(OMe)-FMK is also an inhibitor UCHL1.
    Formula:C22H30FN3O7
    Purezza:97.10%
    Colore e forma:Soild
    Peso molecolare:467.49
  • Ac-VDVAD-CHO TFA


    Ac-VDVAD-CHO (TFA) is a caspase-2/3 inhibitor with IC50 values of 46 nM and 15 nM, respectively.
    Colore e forma:Odour Solid
  • Ac-IEPD-AFC

    CAS:
    Ac-IEPD-AFC (IEPD) is a fluorescent substrate for granzyme B and can be used to measure granzyme B activity.
    Formula:C32H38F3N5O11
    Purezza:99.16%
    Colore e forma:Solid
    Peso molecolare:725.67
  • Ac-WEHD-AFC TFA


    Ac-WEHD-AFC TFA: a fluorogenic substrate detecting caspase-1 activity, used in tumor and inflammation research.
    Formula:C40H38F6N8O13
    Colore e forma:Solid
    Peso molecolare:952.77
  • J22352

    CAS:
    J22352, a PROTAC (proteolysis-targeting chimeras)-like and highly selective HDAC6 inhibitor with an IC50 value of 4.7 nM, enhances anticancer effects in
    Formula:C24H21N3O4
    Colore e forma:Solid
    Peso molecolare:415.44
  • Almorexant hydrochloride

    CAS:
    Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.
    Formula:C29H32ClF3N2O3
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:549.02
  • MX1013

    CAS:
    MX1013, a dipeptide pan-caspase inhibitor, inhibits caspase-1, -3, -6, -7, -8, and -9.
    Formula:C18H23FN2O6
    Colore e forma:Solid
    Peso molecolare:382.39
  • Paris saponin VII

    CAS:
    <p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>
    Formula:C51H82O21
    Purezza:99.51% - 99.63%
    Colore e forma:Solid
    Peso molecolare:1031.18
  • Asperosaponin VI

    CAS:
    Asperosaponin VI, from Dipsacus asper rhizome, treats back pain, hematoma, and fractures.
    Formula:C47H76O18
    Purezza:97.15% - 99.79%
    Colore e forma:Solid
    Peso molecolare:929.10
  • 5,​7,​4'-​Trimethoxyflavone

    CAS:
    5,7,4'-Trimethoxyflavone (4',5,7-Trimethoxyflavone) is isolated from Kaempferia parviflora (KP) which is a medicinal plant from Thailand.
    Formula:C18H16O5
    Purezza:97.53%
    Colore e forma:Solid
    Peso molecolare:312.32
  • CASP3 Activator 1541

    CAS:
    CASP3 Activator 1541 is an activator of the proenzyme forms of caspase-3, and induces cell death.
    Formula:C24H17N3O4
    Purezza:98.84%
    Colore e forma:Solid
    Peso molecolare:411.41
  • KEA1-97

    CAS:
    <p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>
    Formula:C15H9Cl2FN4
    Purezza:97.07%
    Colore e forma:Solid
    Peso molecolare:335.16
  • Taurodeoxycholic acid sodium hydrate

    CAS:
    <p>Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate), a hydrophilic bile salt, on bile salt and biliary lipid secretion in the rat.</p>
    Formula:C26H46NNaO7S
    Purezza:99.95%
    Colore e forma:Solid
    Peso molecolare:539.70
  • L67

    CAS:
    <p>L67 (DNA Ligase Inhibitor) is a competitive human DNA ligase inhibitor, inhibits DNA ligases I and III (IC50: 10 μM).</p>
    Formula:C16H14Br2N4O4
    Purezza:98.34% - 99.56%
    Colore e forma:Solid
    Peso molecolare:486.11
  • Diclofenac Potassium

    CAS:
    Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.
    Formula:C14H10Cl2KNO2
    Purezza:99.51%
    Colore e forma:White To Yellowish Crystalline Powder
    Peso molecolare:334.24
  • Chelidonic acid

    CAS:
    Chelidonic acid, in Chelidonium majus, acts as an analgesic, antimicrobial, CNS sedative, and has anti-inflammatory properties.
    Formula:C7H4O6
    Purezza:99.03%
    Colore e forma:Solid
    Peso molecolare:184.10
  • AVN-944

    CAS:
    <p>AVN-944 (VX-944)(VX-944) is a selective, noncompetitive inhibitor of human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.</p>
    Formula:C25H27N5O5
    Purezza:99.07% - ≥95%
    Colore e forma:Solid
    Peso molecolare:477.51