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Caspasi

Caspasi

Gli inibitori delle caspasi sono composti che bloccano l'attività delle caspasi, una famiglia di proteasi che sono esecutori centrali dell'apoptosi. Le caspasi clivano substrati specifici all'interno della cellula per innescare il processo apoptotico, portando alla morte cellulare programmata. Gli inibitori delle caspasi sono utilizzati per studiare i meccanismi dell'apoptosi, nonché per prevenire la morte cellulare indesiderata in vari modelli di ricerca. Questi inibitori sono anche esplorati in contesti terapeutici per proteggere le cellule dall'apoptosi in malattie come la neurodegenerazione. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle caspasi di alta qualità per supportare la tua ricerca in apoptosi, morte cellulare e campi correlati.

Trovati 143 prodotti di "Caspasi"

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  • PAC-1

    CAS:
    <p>PAC-1 (Procaspase activating compound 1) has been used in trials studying the treatment of Lymphoma, Melanoma, Solid Tumors, Breast Cancer and Thoracic Cancers.</p>
    Formula:C23H28N4O2
    Purezza:96.78% - 99.77%
    Colore e forma:Solid
    Peso molecolare:392.49
  • Ivachtin

    CAS:
    <p>Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining</p>
    Formula:C20H21N3O7S
    Purezza:99.74%
    Colore e forma:Solid
    Peso molecolare:447.46
  • Penicillic acid

    CAS:
    <p>Penicillic acid, a mycotoxin from Aspergillus/Penicillium, blocks Fas ligand apoptosis and is cytotoxic to rat lung macrophages.</p>
    Formula:C8H10O4
    Purezza:98%
    Colore e forma:Needles From Petroleum Ether Slight Yellow Powder
    Peso molecolare:170.16
  • Ginsenoside Rh2

    CAS:
    <p>Ginsenoside Rh2 (20(S)-Ginsenoside Rh2), an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug.</p>
    Formula:C36H62O8
    Purezza:99.20% - 99.76%
    Colore e forma:White Powder
    Peso molecolare:622.87
  • Guggulsterone

    CAS:
    <p>Guggulsterone (Guggulsterone E&amp;Z) E&amp;Z is a 3-hydroxy steroid. It has a role as an androgen.</p>
    Formula:C21H28O2
    Purezza:99.4% - 99.8%
    Colore e forma:Light Yellow Powder
    Peso molecolare:312.45
  • AVN-944

    CAS:
    <p>AVN-944 (VX-944)(VX-944) is a selective, noncompetitive inhibitor of human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.</p>
    Formula:C25H27N5O5
    Purezza:99.07% - ≥95%
    Colore e forma:Solid
    Peso molecolare:477.51
  • Z-IETD-FMK

    CAS:
    <p>Z-IETD-FMK (Z-IE(OMe)TD(OMe)-FMK) is a selective caspase 8 inhibitor, which has cell permeable.</p>
    Formula:C30H43FN4O11
    Purezza:95% - 99.81%
    Colore e forma:Solid
    Peso molecolare:654.68
  • Z-VAD-FMK

    CAS:
    <p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>
    Formula:C21H28FN3O7
    Purezza:98.24% - 99.79%
    Colore e forma:Solid
    Peso molecolare:453.46
  • PHYTOSPHINGOSINE

    CAS:
    <p>Phytosphingosine: anticancer phospholipid; triggers apoptosis in cancer cells via caspase 8 activation and Bax translocation.</p>
    Formula:C18H39NO3
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:317.51
  • TC11

    CAS:
    <p>TC11 (1H-Isoindole-1,3(2H)-dione, 5-amino-2-[2,6-bis(1-methylethyl)phenyl]-TC11) is a potent inhibitor of tumor cell proliferation and an inducer of apoptosis</p>
    Formula:C20H22N2O2
    Purezza:97.86%
    Colore e forma:Solid
    Peso molecolare:322.4
  • Z-VAD(OMe)-FMK

    CAS:
    <p>View and buy Z-VAD(OMe)-FMK from TargetMol.Z-VAD(OMe)-FMK is a cell-permeable and irreversible pan-caspase inhibitor.Cited in 10 publications.</p>
    Formula:C22H30FN3O7
    Purezza:95.92% - 99.71%
    Colore e forma:Solid
    Peso molecolare:467.49
  • Belnacasan

    CAS:
    Belnacasan (VX-765) is an orally active IL-converting enzyme/caspase-1 inhibitor.
    Formula:C24H33ClN4O6
    Purezza:96.53% - 99.5%
    Colore e forma:Solid
    Peso molecolare:508.99
  • Paris saponin VII

    CAS:
    <p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>
    Formula:C51H82O21
    Purezza:99.51% - 99.63%
    Colore e forma:Solid
    Peso molecolare:1031.18
  • Tauroursodeoxycholate sodium

    CAS:
    Tauroursodeoxycholate sodium (TUDC) is an endoplasmic reticulum (ER) stress inhibitor, used for the treatment of gallstones and liver cirrhosis.
    Formula:C26H44NNaO6S
    Purezza:97.90%
    Colore e forma:Solid
    Peso molecolare:521.69
  • Daphnetin

    CAS:
    <p>Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),</p>
    Formula:C9H6O4
    Purezza:97.47% - 99.8%
    Colore e forma:Solid
    Peso molecolare:178.14
  • Ac-DEVD-pNA

    CAS:
    Ac-DEVD-pNA is the preferred peptidic substrate for caspase-3.
    Formula:C26H34N6O13
    Purezza:>99.99%
    Colore e forma:White
    Peso molecolare:638.58
  • Senkyunolide I

    CAS:
    1. Senkyunolide I has neuroprotective effect, associated with its anti-oxidation and anti-apoptosis properties.
    Formula:C12H16O4
    Purezza:99.73% - 99.88%
    Colore e forma:Solid
    Peso molecolare:224.25
  • Z-YVAD-FMK

    CAS:
    AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.
    Formula:C31H39FN4O9
    Purezza:98.00%
    Colore e forma:Solid
    Peso molecolare:630.66
  • Dihydrocapsaicin

    CAS:
    Dihydrocapsaicin, similar to capsaicin, is an irritant found in Capsicum, used in "pure" capsaicin products at about 10%, activates VR1, and is an antioxidant.
    Formula:C18H29NO3
    Purezza:99.8% - ≥95%
    Colore e forma:White Crystal
    Peso molecolare:307.43
  • BC-1471

    CAS:
    BC-1471 is a STAMBP deubiquitinase inhibitor that blocks NALP7 inflammasome activity.
    Formula:C27H32N4O4S
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:508.63