PKC
Gli inibitori della proteina chinasi C (PKC) prendono di mira la famiglia delle chinasi PKC, coinvolte in una vasta gamma di processi cellulari, tra cui la regolazione del ciclo cellulare, l'apoptosi e la differenziazione. La PKC svolge un ruolo chiave nelle vie di trasduzione del segnale che influenzano la proliferazione e la sopravvivenza cellulare. L'inibizione della PKC può portare a cambiamenti nella progressione del ciclo cellulare, rendendo questi inibitori strumenti preziosi nella ricerca sul cancro, la neurobiologia e le malattie cardiovascolari. Presso CymitQuimica, offriamo una selezione diversificata di inibitori della PKC di alta qualità per supportare la tua ricerca sulla trasduzione del segnale, la regolazione del ciclo cellulare e lo sviluppo terapeutico.
Trovati 111 prodotti di "PKC"
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Protein Kinase C (19-31) (TFA)(121545-65-1,free)
Protein Kinase C (19-31) TFA is a serine-modified PKCa-derived inhibitor for testing PKC activity.Formula:C69H119F3N26O18Purezza:98%Colore e forma:SolidPeso molecolare:1657.84Aurothiomalate tetramer sodium
Aurothiomalate tetramer sodium, a tetrameric form of Aurothiomalate sodium, functions as an anti-arthritis gold agent. It also acts as a potent and selective inhibitor of the oncogenic PKCι signaling pathway.Colore e forma:Odour SolidSAMβA TFA
<p>SAMβA TFA, a selective antagonist of Mfn1-βIIPKC association conjugated to the cell permeable peptide TAT47-57, is a rationally designed inhibitor that improves</p>Formula:C50H73N17O16·xC2HF3O2Purezza:98%Colore e forma:SolidPeso molecolare:1168.22 (free acid)Psychosine
CAS:<p>Psychosine (Galactosylsphingosine) is a PKC inhibitor, and is highly cytotoxic, inducing cell death in a variety of cells.</p>Formula:C24H47NO7Purezza:98%Colore e forma:White PowderPeso molecolare:461.63PKC-θ inhibitor
CAS:PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.Formula:C20H25F3N6O3Purezza:99.46%Colore e forma:SolidPeso molecolare:454.45Protein kinase inhibitor H-7 dihydrochloride
CAS:Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor.Formula:C14H19Cl2N3O2SPurezza:99.81%Colore e forma:White Crystalline SolidPeso molecolare:364.29(±)-1,2-Diolein
CAS:(±)-1,2-Diolein (1,2-Dioleoyl-rac-glycerol) (1,2-Dioleoyl-rac-glycerol) is a PKC activator. (±)-1,2-Diolein could increases myotubes Ca 2+ influx.Formula:C39H72O5Colore e forma:SolidPeso molecolare:620.99R59949
CAS:R59949 is used as a Diacylglycerol kinase (DGK) inhibitor.Formula:C28H25F2N3OSPurezza:97.04%Colore e forma:SolidPeso molecolare:489.58Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formula:C26H44NNaO5SPurezza:99.79% - 99.93%Colore e forma:SolidPeso molecolare:505.69Desmethylglycitein
CAS:Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which hasFormula:C15H10O5Purezza:97.93%Colore e forma:SolidPeso molecolare:270.24Afuresertib
CAS:Afuresertib (GSK2110183) is an orally bioavailable inhibitor of the serine/threonine protein kinase Akt (protein kinase B) with potential antineoplasticFormula:C18H17Cl2FN4OSPurezza:97.51% - 99.51%Colore e forma:SolidPeso molecolare:427.32Bisindolylmaleimide IV
CAS:<p>Bisindolylmaleimide IV is a protein kinase C (PKC) cell permeable inhibitor( IC50 : 0.10 - 0.55 μM)</p>Formula:C20H13N3O2Purezza:98.83%Colore e forma:Dark Red SolidPeso molecolare:327.34Hypocrellin A
CAS:Hypocrellin A is a natural PKC inhibitor with light-induced antitumor, antifungal and antiviral activities.Cost-effective and quality-assured.Formula:C30H26O10Purezza:98% - 99.95%Colore e forma:SolidPeso molecolare:546.52Daphnoretin
CAS:<p>1.</p>Formula:C19H12O7Purezza:98% - 99.85%Colore e forma:SolidPeso molecolare:352.29Bisindolylmaleimide V
CAS:Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.Formula:C21H15N3O2Purezza:90%Colore e forma:Red SolidPeso molecolare:341.36TPPB
CAS:<p>TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).</p>Formula:C27H30F3N3O3Purezza:97.71% - 98.00%Colore e forma:SolidPeso molecolare:501.54Ro 31-8220 Mesylate
CAS:<p>Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor, and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β.</p>Formula:C25H23N5O2S·CH4O3SPurezza:98.79% - 99.02%Colore e forma:SolidPeso molecolare:553.65Staurosporine
CAS:Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6/15/2/3/3000 nM) against PKC, PKA, c-FgrFormula:C28H26N4O3Purezza:99.24% - 99.82%Colore e forma:Off-White PowderPeso molecolare:466.53Procyanidin A1
CAS:Procyanidin A1 (Proanthocyanidin A1) has antiallergic effects, it inhibits degranulation downstream of protein kinase C activation or Ca2+.Formula:C30H24O12Purezza:99.52%Colore e forma:SolidPeso molecolare:576.50Ingenol
CAS:<p>Ingenol mebutate treats actinic keratosis, has anticancer properties, and may reactivate latent HIV.</p>Formula:C20H28O5Purezza:99.78% - 99.87%Colore e forma:SolidPeso molecolare:348.43
