PKC
Gli inibitori della proteina chinasi C (PKC) prendono di mira la famiglia delle chinasi PKC, coinvolte in una vasta gamma di processi cellulari, tra cui la regolazione del ciclo cellulare, l'apoptosi e la differenziazione. La PKC svolge un ruolo chiave nelle vie di trasduzione del segnale che influenzano la proliferazione e la sopravvivenza cellulare. L'inibizione della PKC può portare a cambiamenti nella progressione del ciclo cellulare, rendendo questi inibitori strumenti preziosi nella ricerca sul cancro, la neurobiologia e le malattie cardiovascolari. Presso CymitQuimica, offriamo una selezione diversificata di inibitori della PKC di alta qualità per supportare la tua ricerca sulla trasduzione del segnale, la regolazione del ciclo cellulare e lo sviluppo terapeutico.
Trovati 130 prodotti per "PKC".
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PKCα (C2-4) inhibitor peptide
PKCα (C2-4) inhibitor peptide is a specific antagonist to PKCα that impedes the α1A-adrenoreceptor agonist A-61603 [1] from inhibiting I_Kr.Formula:C47H74N14O17Purezza:98%Colore e forma:SolidPeso molecolare:1107.17[Ala113]MBP(104-118)
CAS:Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 28 - 62 mM).Formula:C67H104N20O19Purezza:98%Colore e forma:SolidPeso molecolare:1493.68TAT-P4-(DATC5)2 TFA
TAT-P4-(DATC5)2 TFA, a high-affinity peptide inhibitor targeting the PDZ domain of protein interacting with C kinase-1 (PICK1), exhibits a K i of 1.7 nM andColore e forma:Odour Solid[Ala107]MBP(104-118)
CAS:Synthetic peptide analog of bovine myelin basic protein (MBP). Non-competitive inhibitor of PKC (IC50 = 46 - 145 mM).Formula:C67H104N20O19Purezza:98%Colore e forma:SolidPeso molecolare:1493.68Neuropeptide DF2
CAS:Neuropeptide DF2 is an FMRFamide-related neuropeptide from crayfish.Formula:C44H67N15O10Purezza:98%Colore e forma:SolidPeso molecolare:966.1PKC-ε translocation inhibitor peptide
PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαRPurezza:98%Colore e forma:Odour SolidLys-arg-ala-lys-ala-lys-thr-thr-lys-lys-arg
CAS:Lys-arg-ala-lys-ala-lys-thr-thr-lys-lys-arg is a protein kinase C substrate.Formula:C56H110N22O14Purezza:98%Colore e forma:SolidPeso molecolare:1315.61PKCiota-IN-2
CAS:PKCiota-IN-2 selectively inhibits PKC-ι (IC50=2.8nM) and also blocks PKC-α, ε (IC50s=71nM, 350nM).Formula:C24H21N5OPurezza:98.86%Colore e forma:SolidPeso molecolare:395.46Ref: TM-T9863
1mg109,00€2mg163,00€5mg243,00€1mL*10mM (DMSO)264,00€10mg355,00€25mg532,00€50mg750,00€100mg1.009,00€Delcasertib acetate
Delcasertib acetate is a selective δ protein kinase C (δPKC) inhibitor for the study of acute myocardial infarction and pain.Formula:C122H203N45O36S2Purezza:98.92%Colore e forma:SolidPeso molecolare:2940.33Ref: TM-T11740L
1mg166,00€2mg213,00€5mg313,00€10mg442,00€25mg642,00€50mg880,00€100mg1.179,00€200mg1.594,00€Mitoxantrone-D8
CAS:Mitoxantrone-D8 is the deuterated form of Mitoxantrone. Mitoxantrone (T6588) acts as a topoisomerase II (topoisomeraseII) inhibitor and also inhibits protein kinase C (PKC) with an IC50 value of 8.5 μM.Formula:C22H28N4O6Colore e forma:SolidPeso molecolare:452.53PKCδ Peptide Substrate
CAS:PKCδ Peptide Substrate is a highly specific substrate for the δ-type of Protein kinase C, composed of a sequence that mirrors murine eEF-1α (422-443) andFormula:C109H191N35O29SColore e forma:SolidPeso molecolare:2487.97Protein kinase C α peptide TFA
CAS:Protein Kinase C (alpha) Peptide (TFA) is a PKC-α-associated peptide functioning as a lipid-dependent serine/threonine protein kinase.Formula:C68H115F3N24O26SColore e forma:SolidPeso molecolare:1773.85NPC-15437 dihydrochloride
CAS:NPC-15437 dihydrochloride is a PKC inhibitor blocking enzyme activity and phorbol ester binding, selective over other kinases, in cellular signaling research.Formula:C25H52Cl2N4O2Colore e forma:White SolidPeso molecolare:511.62Bisindolylmaleimide III
CAS:Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively interacts with PKCα or ribosomal S6Formula:C23H20N4O2Purezza:97.2%Colore e forma:SolidPeso molecolare:384.43pep2-EVKI
CAS:Peptide inhibits GluA2-PICK1 binding, sparing GluA2-GRIP/ABP interaction and LTD, without boosting AMPA current.Formula:C62H95N13O19Purezza:98%Colore e forma:SolidPeso molecolare:1326.51PKCε Inhibitor Peptide acetate
PKCε Inhibitor Peptide acetate is a selective PKCε inhibitor containing the site for its specific receptor for activated C kinase (RACK).Formula:C39H69N9O15Purezza:99.62%Colore e forma:SolidPeso molecolare:904.02Ref: TM-T35827L
1mg62,00€2mg89,00€5mg110,00€10mg177,00€25mg298,00€50mg429,00€100mg587,00€200mg792,00€PKCβII Peptide Inhibitor I
CAS:PKCβII Peptide Inhibitor I, a specific PKCβII inhibitor, exhibits cardioprotective properties in a rat cardiac ischemia/reperfusion injury model and mitigatesFormula:C61H94N12O19Purezza:98%Colore e forma:SolidPeso molecolare:1299.471-Oleoyl-2-acetyl-sn-glycerol
CAS:1-Oleoyl-2-acetyl-sn-glycerol (1-oleoyl-2-acetyl-glycerol) is a PKC activator that induces superoxide production.Formula:C23H42O5Colore e forma:SolidPeso molecolare:398.58Protein kinase inhibitor H-7 dihydrochloride
CAS:Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride) is a potent protein kinase C (PKC) inhibitor.Formula:C14H19Cl2N3O2SPurezza:99.81%Colore e forma:White Crystalline SolidPeso molecolare:364.29PKC-θ inhibitor
CAS:PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.Formula:C20H25F3N6O3Purezza:99.46%Colore e forma:SolidPeso molecolare:454.45Ref: TM-T5423
1mg101,00€5mg236,00€1mL*10mM (DMSO)259,00€10mg313,00€25mg442,00€50mg580,00€100mg893,00€200mg1.198,00€
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