
Cromatina/Epigenetica
Gli inibitori della cromatina/epigenetica sono composti che modulano la struttura e la funzione della cromatina o interferiscono con le modificazioni epigenetiche, come la metilazione del DNA e la modifica degli istoni. Questi inibitori sono strumenti essenziali per studiare la regolazione dell'espressione genica e il ruolo dell'epigenetica in malattie come il cancro, i disturbi neurologici e le anomalie dello sviluppo. Mirando ai processi epigenetici, questi inibitori possono alterare i modelli di espressione genica e offrire nuove opportunità terapeutiche. Presso CymitQuimica, offriamo un'ampia selezione di inibitori della cromatina/epigenetica di alta qualità per supportare le tue ricerche in biologia molecolare, genetica ed epigenetica.
Sottocategorie di "Cromatina/Epigenetica"
Trovati 2567 prodotti di "Cromatina/Epigenetica"
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Helenalin Acetate
CAS:Helenalin Acetate: anti-inflammatory, anti-cancer, hinders C/EBPß and p300 cooperation.Formula:C17H20O5Purezza:98%Colore e forma:SolidPeso molecolare:304.34DM-01
CAS:DM-01 is a potent and selective inhibitor of EZH2.
Formula:C23H24F3N3O2Colore e forma:SolidPeso molecolare:431.45(1S,2R)-Tranylcypromine hydrochloride
CAS:(1S,2R)-Tranylcypromine hydrochloride ((1S,2R)-SKF 385), a potent antidepressant, functions by inhibiting both MAO and LSD1.Formula:C9H12ClNColore e forma:SolidPeso molecolare:169.651Gue1654
CAS:Gue1654 is an OXE-R inhibitor and cardiomyocyte apoptosis.Gue1654 can be used for the study of cardiovascular diseases.Formula:C23H17N3OS3Purezza:98.02% - 98.04%Colore e forma:SolidPeso molecolare:447.6CID-4785700
CAS:CID-4785700 is a potent pan-GTPase inhibitor that inhibits Rab7 and inhibits the fungal histone acetyltransferase Rtt109 that binds to Asf1 and Vps75Formula:C22H23ClFN3O3Purezza:98.16%Colore e forma:SolidPeso molecolare:431.89Ref: TM-T71740
1mg315,00€5mg873,00€10mg1.080,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.419,00€SMYD2-IN-1
CAS:SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM).Formula:C25H25Cl2F2N7O2Purezza:98%Colore e forma:SolidPeso molecolare:564.41HDAC3-IN-T326
CAS:HDAC3-IN-T326: potent, selective HDAC3 inhibitor, boosts NF-κB acetylation, activates latent HIV gene expression.Formula:C21H18N6O3SPurezza:98%Colore e forma:SolidPeso molecolare:434.47PS432
CAS:PS432 inhibits atypical PKCs, targets PIF-pocket, reduces tumors in mice sans side effects.Formula:C25H19ClN2O5SPurezza:98%Colore e forma:SolidPeso molecolare:494.95Akt Inhibitor X
CAS:Akt Inhibitor X is a cell-permeable and reversible inhibitor of Akt phosphorylation.Formula:C20H25ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:344.88NSC-636819
CAS:NSC-636819 is a novel inhibitor of KDM4A/KDM4B.Formula:C22H12Cl4N2O4Purezza:98%Colore e forma:SolidPeso molecolare:510.15PARP-1/2-IN-1
CAS:PARP-1-/2-IN-1 is a potent inhibitor of PARP-1 (IC50: 0.51 nM) and PARP-2 (IC50: 23.11 nM).Formula:C24H27FN4O3Colore e forma:SolidPeso molecolare:438.49Kgp-IN-1
CAS:Kgp-IN-1 is an arginine-specific gingipain (Rgp) inhibitor.Formula:C19H24F4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:432.41PNZ5
CAS:PNZ5, an isoxazole-based pan-BET inhibitor, demonstrates potent activity and high selectivity comparable to the established (+)-JQ1, exhibiting a dissociationFormula:C20H18N2O2Purezza:99.51% - 99.61%Colore e forma:SolidPeso molecolare:318.37Ref: TM-T12513
1mg109,00€5mg243,00€10mg355,00€25mg532,00€50mg750,00€100mg1.009,00€200mg1.369,00€1mL*10mM (DMSO)240,00€JAK-IN-10
CAS:JAK-IN-10 is a JAK inhibitor. JAK-IN-10 can be used for the research of dry eye disorders.Formula:C20H18FN5O3SPurezza:99.53%Colore e forma:SolidPeso molecolare:427.45Ref: TM-T13571
1mg82,00€5mg167,00€10mg246,00€25mg405,00€50mg572,00€100mg772,00€500mg1.539,00€1mL*10mM (DMSO)178,00€SW155246
CAS:SW155246 is a potent and selective inhibitor of DNMT1 (DNA methyltransferase 1; IC50 of 1.2 μM).Formula:C16H11ClN2O5SPurezza:98.99%Colore e forma:SolidPeso molecolare:378.79SIRT5 inhibitor 5
CAS:SIRT5 inhibitor 5 is a selective and substrate-competitive SIRT5 inhibitor, which does not occupy the NAD+ binding pocket,cancer and metabolism-related disease.Formula:C21H14ClN3O3SPurezza:99.33%Colore e forma:SolidPeso molecolare:423.87Valemetostat tosylate
CAS:Valemetostat tosylate is a dual inhibitor of EZH1/2 and used in the research of relapsed/refractory peripheral T-cell lymphoma.Formula:C33H42ClN3O7SPurezza:98%Colore e forma:SolidPeso molecolare:660.22KP-302
CAS:KP-302 is a selective PAD inhibitor, reversing physical disability in multiple sclerosis (MS) mice and clearing T-cell infiltration in the brain.
Formula:C20H23N5O2Purezza:99.77%Colore e forma:SolidPeso molecolare:365.43Ref: TM-T88080
1mg60,00€5mg127,00€10mg202,00€25mg416,00€50mg677,00€100mg1.074,00€200mg1.454,00€1mL*10mM (DMSO)140,00€GSK360A
CAS:GSK360A is a novel prolyl hydroxylase (PHD) domain-containing enzyme inhibitor.Formula:C17H17FN2O5Purezza:98%Colore e forma:SolidPeso molecolare:348.33ZYJ-34c
CAS:ZYJ-34c is a potent oral antitumor activities histone deacetylase inhibitor (HDACi).Formula:C31H42N4O7Purezza:98%Colore e forma:SolidPeso molecolare:582.69
