Endocrinologia/Ormoni
Gli inibitori dell'endocrinologia/oromone sono composti che bloccano l'azione degli ormoni o interferiscono con le vie di segnalazione ormonale. Questi inibitori sono fondamentali per studiare la regolazione dei sistemi endocrini e per sviluppare trattamenti per malattie correlate agli ormoni, come il diabete, i disturbi della tiroide e i tumori ormono-dipendenti. Modulando l'attività ormonale, questi inibitori possono aiutare a chiarire le complesse interazioni all'interno del sistema endocrino. Presso CymitQuimica, offriamo un'ampia gamma di inibitori di alta qualità per endocrinologia/oromone per supportare le tue ricerche in endocrinologia, farmacologia e scienze mediche.
Sottocategorie di "Endocrinologia/Ormoni"
- Recettore degli androgeni(229 prodotti)
- Annessina A(16 prodotti)
- Aromatasi(22 prodotti)
- Recettore degli estrogeni/progestogeni(64 prodotti)
- GPR(1 prodotti)
- Recettore dei glucocorticoidi(165 prodotti)
- LHRH(2 prodotti)
- Recettore degli oppioidi(325 prodotti)
- Recettore della prostaglandina(122 prodotti)
- RAAS(86 prodotti)
- Riduttasi(51 prodotti)
- Somatostatina(57 prodotti)
- Recettore dell'ormone tiroideo (THR)(33 prodotti)
- Recettore della vasopressina(48 prodotti)
Mostrare 6 più sottocategorie
Trovati 3369 prodotti di "Endocrinologia/Ormoni"
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Renin FRET Substrate I
CAS:Renin FRET Substrate I, designed for human renin, contains angiotensinogen's N-terminal cleavage site.Formula:C90H120N22O16SColore e forma:SolidPeso molecolare:1798.1515,26-Dihydroxylanosta-7,9(11),24-trien-3-one
CAS:15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is a natural product that can be used as a reference standard. The CAS number of 15,26-Dihydroxylanosta-7,9(11),24-trien-3-one is 420781-85-7.Formula:C30H46O3Colore e forma:SolidPeso molecolare:454.7RLA-5331
RLA-5331: iron activator with anti-androgen properties; inhibits mCRPC cell proliferation.Formula:C40H43F3N6O7SColore e forma:SolidPeso molecolare:808.87PD 123177
CAS:PD 123177 is an inhibitor of Nonpeptide angiotensin AII-2.Formula:C29H28N4O3Purezza:98%Colore e forma:SolidPeso molecolare:480.56AKR1Cs-IN-1
AKR1Cs-IN-1 (Compound 29) is an effective and broad-spectrum inhibitor of the Aldo-Keto Reductase 1C family (AKR1C1-1C4). It achieves subtype inhibition by simultaneously binding to the SP2 and SP3 pockets, thereby blocking metabolic pathways related to drug resistance. In enzyme assays, AKR1Cs-IN-1 exhibits significant inhibitory activity with IC50 values of 0.09, 0.28, 0.05, and 0.51 µM for AKR1C1, AKR1C2, AKR1C3, and AKR1C4, respectively. The compound shows excellent resensitizing effects in doxorubicin (DOX)-resistant breast cancer cell line MCF-7/ADR, effectively enhancing the cytotoxicity of DOX. AKR1Cs-IN-1 holds promise for research on breast cancer resistance.Colore e forma:Odour SolidAH 8529
CAS:AH 8529 is an orally active opioid compound with analgesic properties.Formula:C16H23ClN2OColore e forma:SolidPeso molecolare:294.82Deltorphin
CAS:Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.Formula:C44H62N10O10S2Purezza:98.96%Colore e forma:SolidPeso molecolare:955.15Saprisartan
CAS:Saprisartan (GR-138950, GR-138950X) is an AT1 receptor antagonist used for the treatment of heart failure and blood pressure.Formula:C25H22BrF3N4O4SColore e forma:SolidPeso molecolare:611.43Rofleponide
CAS:Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.Formula:C25H34F2O6Purezza:99.98%Colore e forma:SolidPeso molecolare:468.53ICI 174,864
CAS:Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.Formula:C38H53N5O7Purezza:98%Colore e forma:White SolidPeso molecolare:691.87N-Phenethylnoroxymorphone
CAS:N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.Formula:C24H25NO4Colore e forma:SolidPeso molecolare:391.46SNC 80
CAS:SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.Formula:C28H39N3O2Purezza:99.65%Colore e forma:SolidPeso molecolare:449.63KOR agonist 3
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.Formula:C24H24N2O3Colore e forma:SolidPeso molecolare:388.46Pro8-Oxytocin
CAS:Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects comparedFormula:C42H62N12O12S2Purezza:98%Colore e forma:SolidPeso molecolare:991.14Hemorphin-7
CAS:Hemorphin-7, an atypical opioid peptide from hemoglobin, may enhance memory, promote cell growth, and is a potential breast cancer biomarker.Formula:C49H64N12O11Purezza:98%Colore e forma:SolidPeso molecolare:997.11Corynantheidine
CAS:Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.Formula:C22H28N2O3Colore e forma:SolidPeso molecolare:368.47BAY 1003803
CAS:BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.Formula:C21H18ClF5N2O4Colore e forma:SolidPeso molecolare:492.83PROTAC ERα Degrader-2
CAS:PROTAC ERα Degrader-2 is composed of a cIAP1 ligand binding group, a linker, and an estrogen receptor α (ERα) binding group, serving as an ERα degrader.Formula:C42H61N5O8Purezza:98%Colore e forma:SolidPeso molecolare:763.96Neuropeptide EI, rat
CAS:Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Formula:C63H98N16O23Purezza:98%Colore e forma:SolidPeso molecolare:1447.556α-Methylprednisolone 21-hemisuccinate sodium salt
CAS:6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.Formula:C26H33NaO8Purezza:99.65%Colore e forma:Lyophilized PowderPeso molecolare:496.53
