Endocrinologia/Ormoni
Gli inibitori dell'endocrinologia/oromone sono composti che bloccano l'azione degli ormoni o interferiscono con le vie di segnalazione ormonale. Questi inibitori sono fondamentali per studiare la regolazione dei sistemi endocrini e per sviluppare trattamenti per malattie correlate agli ormoni, come il diabete, i disturbi della tiroide e i tumori ormono-dipendenti. Modulando l'attività ormonale, questi inibitori possono aiutare a chiarire le complesse interazioni all'interno del sistema endocrino. Presso CymitQuimica, offriamo un'ampia gamma di inibitori di alta qualità per endocrinologia/oromone per supportare le tue ricerche in endocrinologia, farmacologia e scienze mediche.
Sottocategorie di "Endocrinologia/Ormoni"
- Recettore degli androgeni(229 prodotti)
- Annessina A(16 prodotti)
- Aromatasi(22 prodotti)
- Recettore degli estrogeni/progestogeni(64 prodotti)
- GPR(1 prodotti)
- Recettore dei glucocorticoidi(165 prodotti)
- LHRH(2 prodotti)
- Recettore degli oppioidi(325 prodotti)
- Recettore della prostaglandina(122 prodotti)
- RAAS(86 prodotti)
- Riduttasi(51 prodotti)
- Somatostatina(57 prodotti)
- Recettore dell'ormone tiroideo (THR)(32 prodotti)
- Recettore della vasopressina(48 prodotti)
Mostrare 6 più sottocategorie
Trovati 3368 prodotti di "Endocrinologia/Ormoni"
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2-sec-Butylphenol
CAS:2-sec-Butylphenol is an inhibitor of the androgen receptor and P450 aromatase, and can be used in research and experiments in the field of life sciences.Formula:C10H14OColore e forma:SolidPeso molecolare:150.22[Orn8]-Urotensin II
CAS:[Orn8]-Urotensin II is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.Formula:C63H83N13O18S2Colore e forma:SolidPeso molecolare:1374.55WAY267464 HCl
CAS:WAY267464: nonpeptide OT agonist, anxiolytic, modulates selectivity, improves CNS entry and oral uptake.Formula:C32H37Cl2N7O4Purezza:98%Colore e forma:SolidPeso molecolare:654.59Tibolone
CAS:Tibolone is an estrogen-like compound used for the treatment of the symptoms associated with menopausal transition (i.e., climacteric symptoms) and also for theFormula:C21H28O2Purezza:99.70% - 99.71%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:312.45Dexamethasone phosphate
CAS:Dexamethasone phosphate is a synthetic adrenal corticosteroid. It also has potent anti-inflammatory properties.Formula:C22H30FO8PColore e forma:SolidPeso molecolare:472.44ET receptor antagonist 3
"ET receptor antagonist 3 (compound 17d) is an orally active ET receptor antagonist with an IC50 of 0.26 nM, utilized for pulmonary arterial hypertension (PAH)Formula:C27H28N6O5SPurezza:98%Colore e forma:SolidPeso molecolare:548.61ET receptor antagonist 1
ET Receptor Antagonist 1 (compound 16h), with an IC50 value of 0.18 nM, is an orally active agent that can be utilized for pulmonary arterial hypertension (PAHFormula:C21H25N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:459.52Anticancer agent 135
Anticancer agent 135 (compound 26h) acts as a potent androgen receptor (AR) antagonist, effectively blocking AR nuclear translocation and inhibiting AR/AR-V7
Formula:C23H21F3N4OSPurezza:98%Colore e forma:SolidPeso molecolare:458.5Androgen receptor antagonist 9
CAS:Androgen Receptor Antagonist 9 (compound 28) serves as an antagonist to the androgen receptor [1].Formula:C19H14F3N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:405.39WCA-814
WCA-814, an androgen receptor (AR) antagonist-Hsp90 inhibitor conjugate, induces degradation of both full-length and AR-V7, exhibiting cytotoxic effects inFormula:C46H53ClN10O5Purezza:98%Colore e forma:SolidPeso molecolare:861.43Dynorphin B (1-9)
CAS:Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selectiveFormula:C54H78N16O12Purezza:98%Colore e forma:SolidPeso molecolare:1143.3Vasopressin Dimer (parallel) (TFA)
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four G protein-coupled receptors—namely, V1aR, V1bR, V2R, andFormula:C94H131F3N30O26S4Purezza:98%Colore e forma:SolidPeso molecolare:2282.49Dynorphin A (1-10)
CAS:Dynorphin A (1-10) is an opioid peptide, binds κ-opioid receptor, blocks NMDA current, IC50: 42.0 μM.Formula:C57H91N19O12Purezza:98%Colore e forma:SolidPeso molecolare:1234.4514-3-3σ/ERα stabilizer-1
Compound 181, also known as 14-3-3σ/ERα Stabilizer-1, is a covalent stabilizer targeting the 14-3-3σ/ERα proteins.Formula:C25H35Cl2N3O3Purezza:98%Colore e forma:SolidPeso molecolare:496.47Keap1-IN-1
Keap1-IN-1 (Compound 27) is an inhibitor of Keap1, functioning by covalently modifying the Cys151 residue on the BTB domain of KEAP1, thereby disrupting the interaction between Keap and Nrf. It enhances the mRNA expression of the antioxidant response element (ARE) dependent gene NQO1, with an EC50 of 160 nM, and exhibits cytotoxicity in U2OS cells, with an EC50 of 527 nM.Formula:C17H21Cl2N2O5PS3Colore e forma:SolidPeso molecolare:531.434ERD-3111
CAS:ERD-3111 (Compound 44), an orally active PROTAC ERα degrader (DC50: 0.5 nM), exhibits efficacy in inhibiting tumor growth in both the parental MCF-7 xenograftFormula:C45H46F4N8O5Purezza:98%Colore e forma:SolidPeso molecolare:854.89LY2623091
CAS:LY2623091, a mineralocorticoid receptor antagonist, is utilized in treating refractory hypertension. It demonstrates CYP3A4-dependent clearance and exhibits synergistic effects when combined with CYP3A4 inhibitors.Formula:C30H30FN5O3Colore e forma:SolidPeso molecolare:527.59Angiotensin II 5-valine
CAS:ngiotensin II 5-valine is an angiotensin II analog which is an agonist at angiotensin receptors.Formula:C49H69N13O12Purezza:98%Colore e forma:SolidPeso molecolare:N/AET receptor antagonist 2
ET Receptor Antagonist 2 (Compound 16j) is an orally active ET receptor antagonist with an IC50 of 0.22 nM, suitable for pulmonary arterial hypertension (PAH)Formula:C22H25N5O5SPurezza:98%Colore e forma:SolidPeso molecolare:471.53ERα degrader 6
ERα degrader 6 (Compound 31q) is an ERα degrader with a K I of 75 nM and also inhibits ARO with an IC50 value of 37.7 nM.Formula:C28H23F3N4O4SPurezza:98%Colore e forma:SolidPeso molecolare:568.57
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