Recettore degli estrogeni/progestogeni

Ethinyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic …

(+)-Medicarpin potently inhibits osteoclastogenesis and promotes bone healing and increases bone mass by osteoblast differentiation …

Fulvestrant is a potent Estrogen Receptor antagonist (IC50: 9.4 nM).

AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.

(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective …

PHTPP is a selective ERβ antagonist.

Synthetic pentapeptide corresponding to the amino acids 32-36 of thymopoietin and exhibiting the full biological …

PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 …

Norgestrel is a synthetic progestin commonly used alone or in combination with an estrogen for …

Gestrinone is a synthetic androgen receptor agonist and ER and progesterone receptor antagonist used to …

DY131 is a novel selective agonist of ERRβ and ERRγ.

NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 …

Allylestrenol is a synthetic steroid with progestational activity.

Estropipate is a natural estrogenic substance composed of estrone sulfate and piperazine.

Dienogest is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic …

Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.

Lasofoxifene Tartrate is a third-generation, non-steroidal selective estrogen receptor modulator.

Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated …

Altrenogest(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.

Astragaloside IV, an active component isolated from Astragalus membranaceus, suppresses the activation of ERK1/2 and …

Ulipristal Acetate is an orally bioavailable, acetate salt of ulipristal, a selective progesterone receptor modulator …

Nestoron, a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).

Chlorotrianisene is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor …

Ethynodiol diacetate is a synthetic progestational hormone used alone or in combination with estrogens as …

Etonogestrel is a steroidal progestin used as hormonal contraceptives.

Ethisterone is a progestogen hormone.

(R)-Zanubrutinib is the R enantiomer of Zanubrutinib. Zanubrutinib is a selective inhibitor of Bruton tyrosine …

(20S)-Protopanaxatriol(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and …

GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with …

Estradiol Benzoate is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to …

CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor …

Toremifene citrate is a selective estrogen receptor modulator (SERM). It is an estrogen agonist for …

Butoconazole Nitrate is the nitrate salt form of butoconazole, a synthetic imidazole derivative with fungistatic …

GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)

PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 …

Dienestrol is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can …

Tamoxifen is an antagonist of the estrogen receptor in breast tissue.

Estradiol is an Estrogen. The mechanism of action of estradiol is as an Estrogen Receptor …

Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by …

Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator …

Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone …

Promestriene (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. …

Lynestrenol is a synthetic progestational hormone, is the progesterone receptor agonist

Gestodene is a progestogen hormonal contraceptive.

Giredestrant potently competes with estradiol for binding and induces a conformational change within the ER …

Bazedoxifene acetate is a novel selective estrogen receptor modulator (SERM).

Mifepristone is a Progestin Antagonist. The mechanism of action of mifepristone is as a Progestational …

Ferrous Bisglycinate is used in the fortification of infant formulations and foods.

ERRα antagonist-1 does not inhibit the interaction of either ERRβ or ERRγ with PGC-1α and …

4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM).

SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding …

Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).

Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.

Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.

Quinestrol is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in …

Bavachin is a phytoestrogen that activates the estrogen receptors ERα and ERβ.

Medroxyprogesterone acetate is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting …

Toremifene is a selective estrogen-receptor modulator (SERM).