
Recettore dei glucocorticoidi
Il recettore dei glucocorticoidi (GR) è un recettore ormonale nucleare che media gli effetti dei glucocorticoidi, una classe di ormoni steroidei coinvolti nella regolazione del metabolismo, della risposta immunitaria e dello stress. Gli agonisti e antagonisti del recettore dei glucocorticoidi sono ampiamente utilizzati nel trattamento delle malattie infiammatorie e autoimmuni, così come nella terapia del cancro. I modulatori del GR sono anche strumenti importanti per studiare i ruoli fisiologici e patologici dei glucocorticoidi. Presso CymitQuimica, offriamo una vasta gamma di modulatori del recettore dei glucocorticoidi di alta qualità per supportare la tua ricerca in endocrinologia, immunologia e regolazione ormonale.
Trovati 167 prodotti di "Recettore dei glucocorticoidi"
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6β-hydroxy Dexamethasone
CAS:6β-hydroxy Dexamethasone is a metabolite of dexamethasone that is more hydrophilic than the parent compound.Formula:C22H29FO6Colore e forma:SolidPeso molecolare:408.46Hydrocortisone sodium succinate
CAS:Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.Formula:C25H34NaO8Colore e forma:SolidPeso molecolare:485.529Deacylcortivazol
CAS:Deacylcortivazol is a potent glucocorticoid that inhibits growth in glucocorticoid-resistant leukemia cells without receptor mediation.Formula:C30H36N2O4Colore e forma:SolidPeso molecolare:488.62PPARγ/GR modulator 1
PPARγ/GR Modulator 1, an orally active dual agonist for the Peroxisome Proliferator-Activated Receptor Gamma (PPARγ) and Glucocorticoid Receptor (GR), exhibitsFormula:C14H10FNO4Colore e forma:SolidPeso molecolare:275.23ACTH (6-24) (human)
CAS:Adrenocorticotropic hormone (6-24) (ACTH (6-24) (human)) is a fragment of ACTH that acts as a competitive inhibitor of steroidogenesis prompted by full-lengthFormula:C111H175N35O21Peso molecolare:2335.8Dexamethasone phosphate
CAS:<p>Dexamethasone phosphate is a synthetic adrenal corticosteroid. It also has potent anti-inflammatory properties.</p>Formula:C22H30FO8PColore e forma:SolidPeso molecolare:472.44RS 21314
CAS:RS 21314 is a thiol ester corticosteroid that is topical.Formula:C24H30F2O5SColore e forma:SolidPeso molecolare:468.55Prednisolone farnesylate
CAS:<p>Prednisolone farnesylate is a novel transdermal corticosteroid with anti-inflammatory activity.</p>Formula:C36H50O6Purezza:98%Colore e forma:SolidPeso molecolare:578.78Rofleponide
CAS:Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.Formula:C25H34F2O6Purezza:99.98%Colore e forma:SolidPeso molecolare:468.53Rimexolone
CAS:Rimexolone is a glucocorticoid steroid used to treat inflammation in the eye.Formula:C24H34O3Colore e forma:SolidPeso molecolare:370.52Nuclear Receptor Compound Library
<p>A unique collection of 531 nuclear receptor signaling targeted compounds for high throughput and high content screening;</p>Colore e forma:Odour SolidBAY 1003803
CAS:BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.Formula:C21H18ClF5N2O4Colore e forma:SolidPeso molecolare:492.83Prednicarbate
CAS:Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.Formula:C27H36O8Purezza:99.88%Colore e forma:SolidPeso molecolare:488.57Glucocorticoids receptor agonist 1
CAS:<p>GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.</p>Formula:C20H23FN2OColore e forma:SolidPeso molecolare:326.41EX-A5386
CAS:<p>EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.</p>Formula:C29H27FN4O2Purezza:99.89%Colore e forma:SoildPeso molecolare:482.55OP-3633
CAS:OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.Formula:C30H39NO2Purezza:98%Colore e forma:SolidPeso molecolare:445.64Glucocorticoids receptor agonist 2
CAS:Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.Formula:C25H25FN2OColore e forma:SolidPeso molecolare:388.48Zavacorilant
CAS:<p>Zavacorilant is capable of modulating glucocorticoid receptor (GR).</p>Formula:C25H26FN7O3S2Colore e forma:SolidPeso molecolare:555.65Methylprednisolone Acetate
Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.Formula:C24H32O6Purezza:99.74%Colore e forma:Off-White SolidPeso molecolare:416.51Betamethasone 17-benzoate
CAS:<p>Betamethasone 17-benzoate is a representative steroid. It also can be used in the treatment of recurrent aphothous ulcers (RAU).</p>Formula:C29H33FO6Purezza:98%Colore e forma:SolidPeso molecolare:496.57

