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Recettore dei glucocorticoidi

Recettore dei glucocorticoidi

Il recettore dei glucocorticoidi (GR) è un recettore ormonale nucleare che media gli effetti dei glucocorticoidi, una classe di ormoni steroidei coinvolti nella regolazione del metabolismo, della risposta immunitaria e dello stress. Gli agonisti e antagonisti del recettore dei glucocorticoidi sono ampiamente utilizzati nel trattamento delle malattie infiammatorie e autoimmuni, così come nella terapia del cancro. I modulatori del GR sono anche strumenti importanti per studiare i ruoli fisiologici e patologici dei glucocorticoidi. Presso CymitQuimica, offriamo una vasta gamma di modulatori del recettore dei glucocorticoidi di alta qualità per supportare la tua ricerca in endocrinologia, immunologia e regolazione ormonale.

Trovati 167 prodotti di "Recettore dei glucocorticoidi"

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  • Betamethasone acibutate

    CAS:
    Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.
    Formula:C28H37FO7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:504.59
  • BI 653048 phosphate

    CAS:
    BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).
    Formula:C23H28F4N3O8PS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:613.52
  • Flucloronide

    CAS:
    Flucloronide is a corticosteroid for topical use on the skin. It has anti-inflammatory properties.
    Formula:C24H29Cl2FO5
    Colore e forma:Solid
    Peso molecolare:487.39
  • β-S-ARCA triammonium


    β-S-ARCA (triammonium) is an analog of the mRNA7-methylguanosine (m7G) cap structure, featuring a thio-phosphorylated segment. When bound to mRNA, β-S-ARCA (triammonium) extends the cellular half-life and enhances protein expression. This compound is utilized in research for mRNA-based cancer vaccines.
    Formula:C22H40N13O17P3S
    Colore e forma:Solid
    Peso molecolare:883.62
  • BI 653048

    CAS:
    BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.
    Formula:C23H25F4N3O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:515.52
  • Dexamethasone cipecilate

    CAS:
    Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.
    Formula:C33H43FO7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:570.69
  • RU26988

    CAS:
    RU26988 is a bioactive chemical.
    Formula:C22H26O3
    Colore e forma:Solid
    Peso molecolare:338.44
  • Paramethasone

    CAS:
    Parametasone is a glucocorticoid with the general properties of corticosteroids.
    Formula:C22H29FO5
    Colore e forma:Solid
    Peso molecolare:392.46
  • BAY 1003803

    CAS:
    BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.
    Formula:C21H18ClF5N2O4
    Colore e forma:Solid
    Peso molecolare:492.83
  • OP-3633

    CAS:
    OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.
    Formula:C30H39NO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:445.64
  • ACTH (6-24) (human)

    CAS:
    Adrenocorticotropic hormone (6-24) (ACTH (6-24) (human)) is a fragment of ACTH that acts as a competitive inhibitor of steroidogenesis prompted by full-length
    Formula:C111H175N35O21
    Peso molecolare:2335.8
  • Desoxycorticosterone pivalate

    CAS:
    DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.
    Formula:C26H38O4
    Colore e forma:Solid
    Peso molecolare:414.58
  • Fluocinolone (Acetonide) (Standard)

    CAS:
    Fluocinolone (Acetonide) (Standard) is the standard substance of Fluocinolone (Acetonide), and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, or ointment. It has also been used topically in the treatment of inflammatory eye, ear, and nose disorders.
    Formula:C24H30F2O6
    Peso molecolare:452.49
  • Diflorasone Diacetate

    CAS:
    Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.
    Formula:C26H32F2O7
    Colore e forma:Crystals
    Peso molecolare:494.53
  • Anti-NR3C1 Antibody (9X89)


    <p>Anti-NR3C1 Antibody (9X89) is an antibody targeting NR3C1. Anti-NR3C1 Antibody (9X89) can be used in ELISA, WB, FCM.</p>
    Colore e forma:Odour Liquid
  • Flurandrenolide

    CAS:
    Fludroxycortide, a synthetic topical steroid, serves as an anti-inflammatory treatment for skin irritations.
    Formula:C24H33FO6
    Colore e forma:Crystals From Acetone + Hexane Solid
    Peso molecolare:436.51
  • Hydrocortisone buteprate

    CAS:
    Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.
    Formula:C28H40O7
    Purezza:99.19%
    Colore e forma:Solid
    Peso molecolare:488.61
  • Prednisolone valerate acetate

    CAS:
    <p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>
    Formula:C28H38O7
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:486.6
  • ZK 216348

    CAS:
    ZK 216348 is a selective glucocorticoid receptor agonist with an IC50 of 20.3 nM. also binds to progesterone receptors and mineralocorticoid receptors.
    Formula:C24H23F3N2O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:476.45
  • Hydrocortisone hemisuccinate (Standard)

    CAS:
    Hydrocortisone hemisuccinate (Standard) is the standard substance of Hydrocortisone hemisuccinate, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
    Formula:C25H34O8
    Peso molecolare:462.53