
Recettore dei glucocorticoidi
Il recettore dei glucocorticoidi (GR) è un recettore ormonale nucleare che media gli effetti dei glucocorticoidi, una classe di ormoni steroidei coinvolti nella regolazione del metabolismo, della risposta immunitaria e dello stress. Gli agonisti e antagonisti del recettore dei glucocorticoidi sono ampiamente utilizzati nel trattamento delle malattie infiammatorie e autoimmuni, così come nella terapia del cancro. I modulatori del GR sono anche strumenti importanti per studiare i ruoli fisiologici e patologici dei glucocorticoidi. Presso CymitQuimica, offriamo una vasta gamma di modulatori del recettore dei glucocorticoidi di alta qualità per supportare la tua ricerca in endocrinologia, immunologia e regolazione ormonale.
Trovati 167 prodotti di "Recettore dei glucocorticoidi"
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Betamethasone acibutate
CAS:Betamethasone acibutate, a glucocorticoid, is derived from Betamethasone.Formula:C28H37FO7Purezza:98%Colore e forma:SolidPeso molecolare:504.59BI 653048 phosphate
CAS:BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : 55 nM).Formula:C23H28F4N3O8PSPurezza:98%Colore e forma:SolidPeso molecolare:613.52Flucloronide
CAS:Flucloronide is a corticosteroid for topical use on the skin. It has anti-inflammatory properties.Formula:C24H29Cl2FO5Colore e forma:SolidPeso molecolare:487.39β-S-ARCA triammonium
β-S-ARCA (triammonium) is an analog of the mRNA7-methylguanosine (m7G) cap structure, featuring a thio-phosphorylated segment. When bound to mRNA, β-S-ARCA (triammonium) extends the cellular half-life and enhances protein expression. This compound is utilized in research for mRNA-based cancer vaccines.Formula:C22H40N13O17P3SColore e forma:SolidPeso molecolare:883.62BI 653048
CAS:BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.Formula:C23H25F4N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:515.52Dexamethasone cipecilate
CAS:Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.Formula:C33H43FO7Purezza:98%Colore e forma:SolidPeso molecolare:570.69RU26988
CAS:RU26988 is a bioactive chemical.Formula:C22H26O3Colore e forma:SolidPeso molecolare:338.44Paramethasone
CAS:Parametasone is a glucocorticoid with the general properties of corticosteroids.Formula:C22H29FO5Colore e forma:SolidPeso molecolare:392.46BAY 1003803
CAS:BAY 1003803 is a glucocorticoid receptor agonist for the topical treatment of psoriasis or severe atopic dermatitis.Formula:C21H18ClF5N2O4Colore e forma:SolidPeso molecolare:492.83OP-3633
CAS:OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.Formula:C30H39NO2Purezza:98%Colore e forma:SolidPeso molecolare:445.64ACTH (6-24) (human)
CAS:Adrenocorticotropic hormone (6-24) (ACTH (6-24) (human)) is a fragment of ACTH that acts as a competitive inhibitor of steroidogenesis prompted by full-lengthFormula:C111H175N35O21Peso molecolare:2335.8Desoxycorticosterone pivalate
CAS:DOCP, a mineralocorticoid, treats dogs with adrenal insufficiency.Formula:C26H38O4Colore e forma:SolidPeso molecolare:414.58Fluocinolone (Acetonide) (Standard)
CAS:Fluocinolone (Acetonide) (Standard) is the standard substance of Fluocinolone (Acetonide), and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion, or ointment. It has also been used topically in the treatment of inflammatory eye, ear, and nose disorders.Formula:C24H30F2O6Peso molecolare:452.49Diflorasone Diacetate
CAS:Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.Formula:C26H32F2O7Colore e forma:CrystalsPeso molecolare:494.53Anti-NR3C1 Antibody (9X89)
<p>Anti-NR3C1 Antibody (9X89) is an antibody targeting NR3C1. Anti-NR3C1 Antibody (9X89) can be used in ELISA, WB, FCM.</p>Colore e forma:Odour LiquidFlurandrenolide
CAS:Fludroxycortide, a synthetic topical steroid, serves as an anti-inflammatory treatment for skin irritations.Formula:C24H33FO6Colore e forma:Crystals From Acetone + Hexane SolidPeso molecolare:436.51Hydrocortisone buteprate
CAS:Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.Formula:C28H40O7Purezza:99.19%Colore e forma:SolidPeso molecolare:488.61Prednisolone valerate acetate
CAS:<p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>Formula:C28H38O7Purezza:99.93%Colore e forma:SolidPeso molecolare:486.6ZK 216348
CAS:ZK 216348 is a selective glucocorticoid receptor agonist with an IC50 of 20.3 nM. also binds to progesterone receptors and mineralocorticoid receptors.Formula:C24H23F3N2O5Purezza:98%Colore e forma:SolidPeso molecolare:476.45Hydrocortisone hemisuccinate (Standard)
CAS:Hydrocortisone hemisuccinate (Standard) is the standard substance of Hydrocortisone hemisuccinate, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.Formula:C25H34O8Peso molecolare:462.53

