
Recettore dei glucocorticoidi
Il recettore dei glucocorticoidi (GR) è un recettore ormonale nucleare che media gli effetti dei glucocorticoidi, una classe di ormoni steroidei coinvolti nella regolazione del metabolismo, della risposta immunitaria e dello stress. Gli agonisti e antagonisti del recettore dei glucocorticoidi sono ampiamente utilizzati nel trattamento delle malattie infiammatorie e autoimmuni, così come nella terapia del cancro. I modulatori del GR sono anche strumenti importanti per studiare i ruoli fisiologici e patologici dei glucocorticoidi. Presso CymitQuimica, offriamo una vasta gamma di modulatori del recettore dei glucocorticoidi di alta qualità per supportare la tua ricerca in endocrinologia, immunologia e regolazione ormonale.
Trovati 166 prodotti di "Recettore dei glucocorticoidi"
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Anti-NR3C1 Antibody (9X89)
Anti-NR3C1 Antibody (9X89) is an antibody targeting NR3C1. Anti-NR3C1 Antibody (9X89) can be used in ELISA, WB, FCM.Colore e forma:Odour LiquidHydrocortisone hemisuccinate (Standard)
CAS:Hydrocortisone hemisuccinate (Standard) is the standard substance of Hydrocortisone hemisuccinate, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.Formula:C25H34O8Peso molecolare:462.53Mirodenafil dihydrochloride
CAS:Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.Formula:C26H39Cl2N5O5SPurezza:99.64% - 99.78%Colore e forma:SolidPeso molecolare:604.59Canrenoate potassium
CAS:Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.Formula:C22H29KO4Purezza:99.04% - 99.18%Colore e forma:Light Yellow To Tan PowderPeso molecolare:396.56Osilodrostat
CAS:Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase (CYP11B1) and aldosterone synthase (CYP11B2).Cost-effective and quality-assured.Formula:C13H10FN3Purezza:99.10% - 99.36%Colore e forma:SolidPeso molecolare:227.24Ref: TM-T4277
1mg37,00€5mg74,00€10mg104,00€25mg169,00€50mg246,00€100mg376,00€150mg772,00€1mL*10mM (DMSO)81,00€AZD9977
CAS:AZD9977 is a novel, selective modulator of mineralocorticoid receptor .Formula:C20H18FN3O5Purezza:99.82%Colore e forma:SolidPeso molecolare:399.37Beclometasone dipropionate monohydrate
CAS:Beclometasone dipropionate monohydrate, precursor to oral glucocorticoid for inflammation and asthma research.Formula:C28H39ClO8Colore e forma:SolidPeso molecolare:539.06LY404039
CAS:LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).Formula:C7H9NO6SPurezza:99% - 99.92%Colore e forma:SolidPeso molecolare:235.22AL 082D06
CAS:AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.Formula:C23H24ClN3O2Purezza:99.05% - 99.06%Colore e forma:SolidPeso molecolare:409.91Isoflupredone Acetate
CAS:Isoflupredone Acetate is a corticosteroid with the activity of topical anti-inflammatory.Formula:C23H29FO6Purezza:99.43%Colore e forma:SolidPeso molecolare:420.47Ref: TM-T21193
1mg38,00€5mg80,00€10mg105,00€25mg207,00€50mg311,00€100mg439,00€200mg632,00€1mL*10mM (DMSO)88,00€Osilodrostat phosphate
CAS:Osilodrostat phosphate is a potent oral 11β-hydroxylase inhibitor.Formula:C13H13FN3O4PColore e forma:SolidPeso molecolare:325.23Ref: TM-T28272
1mg35,00€5mg74,00€10mg104,00€25mg169,00€50mg246,00€100mg376,00€150mg602,00€200mg550,00€Cortodoxone
CAS:Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of cortisol in the adrenal gland.Formula:C21H30O4Purezza:99.26% - 99.87%Colore e forma:SolidPeso molecolare:346.46TPI-1
CAS:TPI-1 is a SHP-1 inhibitor.Formula:C12H6Cl2O2Purezza:99.64% - 99.79%Colore e forma:SolidPeso molecolare:253.08Ref: TM-T3962
1mg50,00€2mg73,00€5mg109,00€10mg178,00€25mg349,00€50mg532,00€100mg757,00€1mL*10mM (DMSO)120,00€Velsecorat
CAS:Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).Formula:C32H32F2N4O6Purezza:99.35%Colore e forma:SolidPeso molecolare:606.62Ref: TM-TQ0225
1mg52,00€5mg114,00€10mg158,00€25mg339,00€50mg505,00€100mg722,00€1mL*10mM (DMSO)156,00€Finerenone
CAS:Finerenone (BAY-948862) is a selective and orally nonsteroidal antagonist of the mineralocorticoid receptor (MR). Cost effective and quality assured.Formula:C21H22N4O3Purezza:99.45% - 99.91%Colore e forma:SolidPeso molecolare:378.42Ref: TM-T21395
1mg37,00€5mg81,00€10mg114,00€25mg220,00€50mg355,00€100mg567,00€200mg645,00€500mg945,00€1mL*10mM (DMSO)89,00€Fluorometholone
CAS:Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.Formula:C22H29FO4Purezza:99% - 99.15%Colore e forma:SolidPeso molecolare:376.46Methylprednisolone succinate
CAS:<p>Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory agent.</p>Formula:C26H34O8Purezza:98.41% - 99.82%Colore e forma:White Or Almost-White Solid PowderPeso molecolare:474.54Diflorasone
CAS:Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene expression.Formula:C22H28F2O5Purezza:99.02% - 99.92%Colore e forma:SolidPeso molecolare:410.45(20S)-Protopanaxatriol
CAS:(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoidFormula:C30H52O4Purezza:95% - 99%Colore e forma:SolidPeso molecolare:476.73Ref: TM-T2810
2mg35,00€5mg52,00€10mg70,00€25mg120,00€50mg188,00€100mg311,00€200mg467,00€1mL*10mM (DMSO)58,00€Hydrocortisone hemisuccinate
CAS:Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.Formula:C25H34O8Purezza:98.01% - 98.7%Colore e forma:SolidPeso molecolare:462.53

