Recettore della vasopressina
I recettori della vasopressina sono una famiglia di recettori accoppiati alle proteine G che mediano gli effetti della vasopressina, un ormone coinvolto nella regolazione dell'equilibrio idrico, della pressione sanguigna e della funzione renale. Gli agonisti e antagonisti dei recettori della vasopressina sono studiati per il loro ruolo nel trattamento di condizioni come il diabete insipido, l'iponatriemia e l'insufficienza cardiaca. Questi recettori sono anche obiettivi importanti nella ricerca sull'equilibrio dei fluidi e sulla salute cardiovascolare. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori della vasopressina di alta qualità per supportare la tua ricerca in endocrinologia, nefrologia e biologia cardiovascolare.
Trovati 46 prodotti di "Recettore della vasopressina"
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Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Formula:C56H82N16O19S2Purezza:98.50% - 99.69%Colore e forma:SolidPeso molecolare:1347.5Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Formula:C30H32ClN3O8SPurezza:98.46% - 99.89%Colore e forma:SolidPeso molecolare:630.11Balovaptan
CAS:Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.Formula:C22H24ClN5OPurezza:99.88%Colore e forma:SolidPeso molecolare:409.91(D-Arg8)-Inotocin
CAS:'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.Formula:C39H68N14O11S2Purezza:98%Colore e forma:SolidPeso molecolare:973.17d[Cha4]-AVP
CAS:Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Formula:C50H71N13O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1094.31(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formula:C52H74N14O12S2Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:1151.38Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFormula:C45H63N15O11S2Colore e forma:SolidPeso molecolare:1054.21[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Colore e forma:SolidPeso molecolare:1033.14(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formula:C44H69N13O13S2Colore e forma:SolidPeso molecolare:1052.23Selepressin acetate
Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.Formula:C48H77N13O13S2Colore e forma:SolidPeso molecolare:1108.33(Phe2,Orn8)-Oxytocin
CAS:(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.Formula:C42H65N13O11S2Colore e forma:SolidPeso molecolare:992.18D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Formula:C49H68F3N11O13S2Colore e forma:SolidPeso molecolare:1140.25(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:<p>Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.</p>Formula:C54H76N14O11Colore e forma:SolidPeso molecolare:1097.27[8-L-arginine] deaminovasopressin
CAS:[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .Formula:C46H64N14O13S2Colore e forma:SolidPeso molecolare:1085.22Endolide F
Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.Formula:C25H32N4O6Peso molecolare:484.23218Velmupressin acetate
CAS:Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).Formula:C44H64ClN11O10S2Purezza:98%Colore e forma:SolidPeso molecolare:1006.63Ornipressin
CAS:Ornipressin is a vasoconstrictor, haemostatic and renal agent.Formula:C45H63N13O12S2Purezza:98%Colore e forma:White PowderPeso molecolare:1042.19c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
CAS:c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm: potent, selective V2R agonist; EC50: 0.25 nM (hV2R), 0.05 nM (rV2R).Formula:C47H69ClN12O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1045.71d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.Formula:C49H71N11O13S2Purezza:98.86%Colore e forma:SolidPeso molecolare:1086.28Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].Formula:C49H70N14O12S2Purezza:98%Colore e forma:SolidPeso molecolare:1111.3Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Formula:C110H161N31O27S2Purezza:98%Colore e forma:SolidPeso molecolare:2413.78[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).Formula:C48H69N13O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1068.27Val9-Oxytocin
CAS:Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.Formula:C46H72N12O12S2Purezza:98%Colore e forma:SolidPeso molecolare:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formula:C52H76N14O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1137.38V1a/V2 antagonist 1
V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.Formula:C25H26ClN5O3Colore e forma:SolidPeso molecolare:479.96d[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formula:C47H67N11O11S2Purezza:98%Colore e forma:SolidPeso molecolare:1026.2d[Cha4]-AVP TFA
d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.Formula:C52H72F3N13O13S2Colore e forma:SolidPeso molecolare:1208.33Atosiban
CAS:Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.Formula:C43H67N11O12S2Purezza:98%Colore e forma:SolidPeso molecolare:994.19Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Formula:C27H34N4O3Purezza:99.33%Colore e forma:SolidPeso molecolare:462.58Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purezza:98%Colore e forma:White PowderPeso molecolare:1084.23Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Formula:C43H77N17O12S2Purezza:99.79%Colore e forma:SolidPeso molecolare:1088.32Desmopressin acetate (16679-58-6 free base)
CAS:Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.Formula:C48H68N14O14S2Purezza:98.84% - >99.99%Colore e forma:SolidPeso molecolare:1129.26Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purezza:98.13% - 99.66%Colore e forma:SolidPeso molecolare:449.54d[Cha4]-AVP acetate(500170-27-4 free base)
'd[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'Formula:C52H75N13O13S2Purezza:99.86%Colore e forma:SolidPeso molecolare:1154.37Atosiban acetate
CAS:Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.Formula:C45H71N11O14S2Purezza:99.84% - 99.92%Colore e forma:SolidPeso molecolare:1054.24Mozavaptan
CAS:Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.Formula:C27H29N3O2Purezza:98.98% - 99.12%Colore e forma:SolidPeso molecolare:427.54LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purezza:98.36%Colore e forma:SolidPeso molecolare:473.93Felypressin
CAS:Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formula:C46H65N13O11S2Purezza:99.65%Colore e forma:SolidPeso molecolare:1040.22Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Formula:C32H26N4O2·HClPurezza:98.33% - 99.86%Colore e forma:SolidPeso molecolare:535.04Tolvaptan
CAS:<p>Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.</p>Formula:C26H25ClN2O3Purezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:448.94RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Formula:C25H28ClN3O2Purezza:99.74%Colore e forma:SolidPeso molecolare:437.96Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Formula:C48H69N13O13S2Purezza:97.06%Colore e forma:SolidPeso molecolare:1100.27TASP0390325
CAS:<p>TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.</p>Formula:C25H30Cl2FN5O4Purezza:98.62%Colore e forma:SolidPeso molecolare:554.44OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formula:C26H32ClN3O2Purezza:98.93% - >99.99%Colore e forma:SolidPeso molecolare:454Elsovaptan
CAS:Elsovaptan is an antagonist of the vasopressin receptor and is applicable for research in Alzheimer's disease.Formula:C19H20ClN5O2Colore e forma:SolidPeso molecolare:385.847RGH-122
CAS:RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 μL/min/mg [1].Formula:C24H25ClN4O3Colore e forma:SolidPeso molecolare:452.93
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