
Recettore della prostaglandina
I recettori delle prostaglandine sono un gruppo di recettori accoppiati alle proteine G che mediano gli effetti delle prostaglandine, composti lipidici coinvolti in una vasta gamma di processi fisiologici, tra cui infiammazione, dolore, febbre e regolazione del flusso sanguigno. I modulatori dei recettori delle prostaglandine sono studiati per il loro ruolo nella gestione delle condizioni infiammatorie, delle malattie cardiovascolari e della salute riproduttiva. Questi recettori sono obiettivi chiave nello sviluppo di farmaci anti-infiammatori e analgesici. Presso CymitQuimica, offriamo una selezione di modulatori dei recettori delle prostaglandine di alta qualità per supportare la tua ricerca in endocrinologia, infiammazione e farmacologia.
Trovati 122 prodotti di "Recettore della prostaglandina"
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ONO-AE3-208
CAS:<p>ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.</p>Formula:C24H21FN2O3Purezza:98.04% - 99.55%Colore e forma:SolidPeso molecolare:404.43Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purezza:98.90%Colore e forma:SolidPeso molecolare:376.41Ref: TM-T9153
1mg40,00€5mg97,00€10mg156,00€25mg255,00€50mg368,00€100mg505,00€200mg692,00€1mL*10mM (DMSO)99,00€MRE-269
CAS:<p>MRE-269 (ACT-333679) is an orally available and long-acting prostacyclin receptor agonist prodrug, used for the treatment of pulmonary arterial hypertension.</p>Formula:C25H29N3O3Purezza:98.25%Colore e forma:SolidPeso molecolare:419.52Fevipiprant
CAS:Fevipiprant (NVP-QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.Formula:C19H17F3N2O4SPurezza:99.32% - 99.59%Colore e forma:SolidPeso molecolare:426.41Taprenepag
CAS:Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).Formula:C24H22N4O5SPurezza:98.89% - 99.15%Colore e forma:SolidPeso molecolare:478.52Ref: TM-T3174
1mg35,00€5mg65,00€10mg97,00€25mg188,00€50mg311,00€100mg449,00€200mg628,00€1mL*10mM (DMSO)70,00€Tranilast
CAS:Tranilast (SB 252218), an antiallergic drug, suppresses lipid mediator and cytokine release from inflammatory cells, therefore utilized in the treatment ofFormula:C18H17NO5Purezza:99.67% - >99.99%Colore e forma:White With Light Yellow Crystalline PowderPeso molecolare:327.33Ref: TM-T2690
5mg43,00€10mg55,00€25mg66,00€50mg93,00€100mg119,00€200mg175,00€500mg298,00€1mL*10mM (DMSO)55,00€Ozagrel hydrochloride
CAS:Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormula:C13H12N2O2·HClPurezza:99.80%Colore e forma:White Or Off White Crystalline PowderPeso molecolare:264.71Prostaglandin E2
CAS:Prostaglandin E2 (PGE2): Key in muscle function, blood flow regulation, and inflammation control.Formula:C20H32O5Purezza:99.76% - 99.95%Colore e forma:LiquidPeso molecolare:352.47Ref: TM-T5014
1mg35,00€2mg49,00€5mg71,00€10mg87,00€25mg170,00€50mg244,00€100mg351,00€200mg515,00€1mL*10mM (DMSO)55,00€TG6-10-1
CAS:TG6-10-1 is an EP2 antagonist.Formula:C23H23F3N2O4Purezza:99.66% - ≥95%Colore e forma:SolidPeso molecolare:448.43Ginsenoside Ro
CAS:Ginsenoside Ro (Chikusetsusaponin V) can reduce TXA2 production, weakly reduce COX-1 and TXAS activities, and has antiplatelet effects as a Ca2+ antagonist withFormula:C48H76O19Purezza:98% - 99.66%Colore e forma:SolidPeso molecolare:957.11Asapiprant
CAS:Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited high affinity and selectivity for the DP1 receptor.Formula:C24H27N3O7SPurezza:99.64%Colore e forma:SolidPeso molecolare:501.55Ref: TM-T5386
1mg40,00€5mg97,00€10mg156,00€25mg284,00€50mg449,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)105,00€ONO-8130
CAS:ONO-8130 is an orally available antagonist of EP1 receptor.Formula:C25H28N2O5S2Purezza:97.82%Colore e forma:SolidPeso molecolare:500.63Pectolinarin
CAS:Pectolinarin is a Cirsium isolate with anti-inflammatory activity.Formula:C29H34O15Purezza:98% - 99.79%Colore e forma:SolidPeso molecolare:622.57p-Hydroxycinnamic acid
CAS:p-Hydroxycinnamic acid (NSC-59260) can inhibit platelet activity, with IC50s of 371 μM, 126 μM for thromboxane B2 production and lipopolysaccharide-inducedFormula:C9H8O3Purezza:99.67% - 99.83%Colore e forma:SolidPeso molecolare:164.16E7046
CAS:E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.Formula:C22H18F5N3O4Purezza:99.86%Colore e forma:SolidPeso molecolare:483.4Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purezza:99.62%Colore e forma:SolidPeso molecolare:508.61Cloprostenol sodium salt
CAS:Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.Formula:C22H28ClNaO6Purezza:97.17% - 98.47%Colore e forma:White To Almost White Hygroscopic PowderPeso molecolare:446.9Benorilate
CAS:Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formula:C17H15NO5Purezza:98.39% - 99.85%Colore e forma:SolidPeso molecolare:313.3CAY10471 Racemate
CAS:CAY10471 Racemate is a potent CRTH2/DP2 antagonist with Ki of 0.6 nM; less active on DP1 and TP.Formula:C21H21FN2O4SPurezza:99.08%Colore e forma:SolidPeso molecolare:416.47Agnuside
CAS:<p>Agnuside (chasteberry oil) inhibits COX-2 (IC50: 0.026 mg/ml) but exhibits less than 10% inhibition of COX-1 at this concentration.</p>Formula:C22H26O11Purezza:99.08% - 99.81%Colore e forma:Orangish-Yellow To Light Yellow LiquidPeso molecolare:466.44
