
Enzima
Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.
Sottocategorie di "Enzima"
- Anidrasi carbonica(196 prodotti)
- Idrossilasi(36 prodotti)
- MPO(2 prodotti)
- Riduttasi(53 prodotti)
- Tirosinasi(77 prodotti)
Trovati 3669 prodotti per "Enzima".
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Tioxolone
CAS:Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.Formula:C7H4O3SPurezza:97.79%Colore e forma:White SolidPeso molecolare:168.17pNNP
CAS:pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.Formula:C6H6NO6PPurezza:99.82%Colore e forma:White SolidPeso molecolare:219.09Benzthiazide
CAS:Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.Formula:C15H14ClN3O4S3Purezza:98.48% - 99.79%Colore e forma:White SolidPeso molecolare:431.94Methazolamide
CAS:Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.Formula:C5H8N4O3S2Purezza:99.31% - 99.77%Colore e forma:SolidPeso molecolare:236.27CAIX Inhibitor S4
CAS:CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.Formula:C15H17N3O4SPurezza:99.07%Colore e forma:SolidPeso molecolare:335.38Ref: TM-T36758
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg90,00€25mg178,00€50mg334,00€100mg500,00€500mg1.099,00€Brinzolamide
CAS:Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.Formula:C12H21N3O5S3Purezza:99.84% - >99.99%Colore e forma:SolidPeso molecolare:383.51ACT-678689
CAS:ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].Formula:C23H22ClFN6O4S2Purezza:99.46%Colore e forma:SolidPeso molecolare:565.04Ref: TM-T14119
1mg107,00€5mg245,00€1mL*10mM (DMSO)308,00€10mg371,00€25mg620,00€50mg858,00€100mg1.153,00€200mg1.549,00€Topiramate
CAS:Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.Formula:C12H21NO8SPurezza:99.79% - 99.92%Colore e forma:SolidPeso molecolare:339.36KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Formula:C29H31N5O5SPurezza:99.70%Colore e forma:Yellow SolidPeso molecolare:561.655-Feruloylquinic acid
CAS:5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.Formula:C17H20O9Purezza:99.03%Colore e forma:White SolidPeso molecolare:368.34Hydrochlorothiazide
CAS:Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药,可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能,减少纤维化并具有降压作用。Formula:C7H8ClN3O4S2Purezza:99.43% - 99.50%Colore e forma:White SolidPeso molecolare:297.74Zonisamide
CAS:Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.Formula:C8H8N2O3SPurezza:99.05% - 99.9%Colore e forma:SolidPeso molecolare:212.23p-Ethynylphenylalanine hydrochloride
CAS:p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].Formula:C11H12ClNO2Purezza:99.03% - 99.83%Colore e forma:SolidPeso molecolare:225.67Telotristat ethyl
CAS:Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.Formula:C27H26ClF3N6O3Purezza:98% - 99.89%Colore e forma:White SolidPeso molecolare:574.98Fenclonine
CAS:Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.Formula:C9H10ClNO2Purezza:98.81% - >99.99%Colore e forma:Crystals From Methanol White SolidPeso molecolare:199.63Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purezza:99.96%Colore e forma:White SolidPeso molecolare:241.24Arbutin
CAS:Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.Formula:C12H16O7Purezza:99.58% - 99.87%Colore e forma:White SolidPeso molecolare:272.25Actarit
CAS:Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug.Formula:C10H11NO3Purezza:99.64% - 99.74%Colore e forma:White Or Off-White Crystal Or Crystalline SolidPeso molecolare:193.2Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Purezza:> 95%Colore e forma:Transparent LiquidPeso molecolare:145.42 kDaAcipimox
CAS:Acipimox (K-9321), a niacin derivative, treats hyperlipidemia in type 2 diabetics.Formula:C6H6N2O3Purezza:98.98%Colore e forma:SolidPeso molecolare:154.12
