Enzima
Gli inibitori enzimatici sono molecole che si legano agli enzimi e ne diminuiscono l'attività. Questi inibitori sono ampiamente utilizzati nella ricerca per studiare la cinetica enzimatica, la regolazione e il ruolo di specifici enzimi nelle vie metaboliche. Gli inibitori enzimatici sono anche fondamentali nello sviluppo di farmaci, poiché molti agenti terapeutici agiscono inibendo enzimi coinvolti in processi patologici. Mirando agli enzimi, questi inibitori possono modulare le vie biochimiche e offrire potenziali trattamenti per varie malattie. Presso CymitQuimica, offriamo una vasta selezione di inibitori enzimatici di alta qualità per supportare le tue ricerche in biochimica, farmacologia e scoperta di farmaci.
Sottocategorie di "Enzima"
- Anidrasi carbonica(189 prodotti)
- Idrossilasi(35 prodotti)
- MPO(2 prodotti)
- Riduttasi(50 prodotti)
- Tirosinasi(72 prodotti)
Trovati 3610 prodotti di "Enzima"
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ACT-678689
CAS:<p>ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].</p>Formula:C23H22ClFN6O4S2Purezza:99.46%Colore e forma:SolidPeso molecolare:565.04Brinzolamide
CAS:<p>Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.</p>Formula:C12H21N3O5S3Purezza:99.84% - >99.99%Colore e forma:Crystalline SolidPeso molecolare:383.51KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Formula:C29H31N5O5SPurezza:99.28%Colore e forma:SolidPeso molecolare:561.65Methazolamide
CAS:Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.Formula:C5H8N4O3S2Purezza:99.31% - 99.77%Colore e forma:Crystals From Water SolidPeso molecolare:236.27Actarit
CAS:Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug.Formula:C10H11NO3Purezza:99.64% - 99.74%Colore e forma:White Or Off-White Crystal Or Crystalline SolidPeso molecolare:193.2pNNP
CAS:pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.Formula:C6H6NO6PPurezza:99.82%Colore e forma:SolidPeso molecolare:219.09Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Formula:C11H15NO5Purezza:99.96%Colore e forma:Crystals From Benzene SolidPeso molecolare:241.24Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formula:C12H21NO8SPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:339.36Benzthiazide
CAS:<p>Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.</p>Formula:C15H14ClN3O4S3Purezza:99.34% - 99.79%Colore e forma:Crystals From Acetone SolidPeso molecolare:431.94p-Ethynylphenylalanine hydrochloride
CAS:p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].Formula:C11H12ClNO2Purezza:99.03%Colore e forma:SolidPeso molecolare:225.67Arbutin
CAS:Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.Formula:C12H16O7Purezza:99.58% - 99.93%Colore e forma:Colorless Elongated Prisms From Moist Ethyl Acetate White PowderPeso molecolare:272.25Telotristat ethyl
CAS:Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.Formula:C27H26ClF3N6O3Purezza:98% - 99.89%Colore e forma:White SolidPeso molecolare:574.98Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Purezza:> 95%Colore e forma:LiquidPeso molecolare:145.42 kDa4-Chlorosalicylic acid
CAS:<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Formula:C7H5ClO3Purezza:98.59%Colore e forma:Off-White To Light Beige PowderPeso molecolare:172.57Acipimox
CAS:<p>Acipimox (K-9321), a niacin derivative, treats hyperlipidemia in type 2 diabetics.</p>Formula:C6H6N2O3Purezza:98.98%Colore e forma:Low Yellow Liquid Or CrystallinePeso molecolare:154.12Fenclonine
CAS:Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.Formula:C9H10ClNO2Purezza:98.81% - >99.99%Colore e forma:Crystals From Methanol White SolidPeso molecolare:199.635-Feruloylquinic acid
CAS:5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.Formula:C17H20O9Purezza:99.03%Colore e forma:SolidPeso molecolare:368.34Zonisamide
CAS:<p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>Formula:C8H8N2O3SPurezza:99.05% - 99.9%Colore e forma:Off-White PowderPeso molecolare:212.23Tioxolone
CAS:Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.Formula:C7H4O3SPurezza:97.79%Colore e forma:Light Yellow To Beige PowderPeso molecolare:168.17Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Colore e forma:Odour SolidCAIX/CAXII-IN-3
CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.Colore e forma:Odour SolidCAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Formula:C23H21N5O3SColore e forma:SolidPeso molecolare:447.51Pyrocatechol
CAS:Pyrocatechol, often known as catechol or benzene-1,2-diol, is a benzenediol, Pyrocatechol was produced at a large scale industrially, mainly as precursors to pesticides, flavors, and fragrances. Its sulfonic acid is often present in the urine of many mammals.Formula:C6H6O2Purezza:99.96%Colore e forma:SolidPeso molecolare:110.11Chlorothiazide
CAS:Chlorothiazide (Diuril) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE.Formula:C7H6ClN3O4S2Purezza:98.46% - 98.91%Colore e forma:Crystals Physical Description Crystals; White Powder (Ntp 1992)Peso molecolare:295.72CAIX Inhibitor S4
CAS:<p>CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.</p>Formula:C15H17N3O4SPurezza:99.07%Colore e forma:SolidPeso molecolare:335.38hCAIX-IN-19
<p>hCAIX-IN-19 is a sulfonamide inhibitor with an inhibition constant (KI) of 6.2 nM for hCAIX, exhibiting significant selectivity towards hCAIX over hCAI (hCA I/</p>Colore e forma:Odour Solid2-Methoxy-4-propylphenol
CAS:<p>2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.</p>Formula:C10H14O2Colore e forma:SolidPeso molecolare:166.22Carbonic anhydrase inhibitor 30
Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].Formula:C23H22FN3O5SColore e forma:SolidPeso molecolare:471.12642Xanthine Oxidase, ammonium sulfate suspension
CAS:Colore e forma:Faint brown to dark brown suspensionAnhydrotetracycline hydrochloride
CAS:Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.Formula:C22H23ClN2O7Purezza:98% - 98.90%Colore e forma:SolidPeso molecolare:462.88Tyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Formula:C19H14BrClN4OColore e forma:SolidPeso molecolare:429.7Tyrosinase-IN-32
<p>Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.</p>Formula:C15H19NO3Colore e forma:SolidPeso molecolare:261.32Calmodulin-dependent Protein Kinase II fragment 290-309
CAS:Formula:C103H185N31O24SPeso molecolare:2273.83(E)-Dehydrodiconiferyl alcohol
CAS:(E)-Dehydrodiconiferyl alcohol inhibits hCA IX/XII enzymes and blocks NF-κB nuclear translocation in healing tissues.Formula:C20H22O6Colore e forma:SolidPeso molecolare:358.395,6-Dihydro-2H-pyran-2-one
CAS:5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.Formula:C5H6O2Colore e forma:SolidPeso molecolare:98.1Peroxidase
CAS:Purezza:≥ 85units/mg (dry basis)Colore e forma:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecolare:-
