Idrossilasi
Le idrossilasi sono una classe di enzimi che catalizzano l'idrossilazione dei substrati, spesso aggiungendo gruppi idrossilici (-OH) a posizioni specifiche all'interno delle molecole. Questi enzimi sono coinvolti in una vasta gamma di percorsi biochimici, inclusa la sintesi di ormoni, i processi di detossificazione e il metabolismo dei farmaci. Gli inibitori e gli attivatori delle idrossilasi sono strumenti preziosi nella ricerca sui disturbi metabolici, sul metabolismo dei farmaci e sulla regolazione ormonale. Presso CymitQuimica, offriamo una selezione di reagenti per idrossilasi di alta qualità per supportare la tua ricerca in biochimica, farmacologia e regolazione metabolica.
Trovati 36 prodotti di "Idrossilasi"
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Fenclonine
CAS:Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.Formula:C9H10ClNO2Purezza:98.81% - >99.99%Colore e forma:Crystals From Methanol White SolidPeso molecolare:199.63ACT-678689
CAS:ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].Formula:C23H22ClFN6O4S2Purezza:99.46%Colore e forma:SolidPeso molecolare:565.04Ref: TM-T14119
1mg107,00€5mg245,00€10mg371,00€25mg620,00€50mg858,00€100mg1.153,00€200mg1.549,00€1mL*10mM (DMSO)308,00€Telotristat ethyl
CAS:Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.Formula:C27H26ClF3N6O3Purezza:98% - 99.89%Colore e forma:White SolidPeso molecolare:574.98p-Ethynylphenylalanine hydrochloride
CAS:p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].Formula:C11H12ClNO2Purezza:99.03%Colore e forma:SolidPeso molecolare:225.67Butobendine
CAS:Butobendine is a compound derived from gallic acid and exhibits significant antiarrhythmic activity.Formula:C32H48N2O10Colore e forma:SolidPeso molecolare:620.73IOX2-NH2-1
CAS:IOX2-NH2-1 inhibits E. coli EGLN-3 (prolyl hydroxylase) with an IC50 of 0.02–1 μM.Formula:C19H17N3O5Purezza:98.77% - 99.91%Colore e forma:SoildPeso molecolare:367.36TPH1-IN-1
TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.Formula:C21H18N6O4SColore e forma:SolidPeso molecolare:450.47TPT-004
TPT-004, a TPH inhibitor, exhibits superior pharmacokinetic and pharmacodynamic properties, and demonstrates efficacy in preclinical models for attenuatingColore e forma:Odour SolidGSK180
CAS:GSK180 is a selective competitive inhibitor of kynurenine 3-monooxygenase (KMO; IC50: ~6 nM), an enzyme involved in tryptophan metabolism.Formula:C10H7Cl2NO4Colore e forma:SolidPeso molecolare:276.07Cuprizone
CAS:Cuprizone is a copper chelator.Cuprizone is used to induce schizophrenia in mice.Cuprizone induces oligodendrocyte death and induces a demyelination response.Formula:C14H22N4O2Purezza:≥98%Colore e forma:SolidPeso molecolare:278.35FG-2216
CAS:FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.Formula:C12H9ClN2O4Purezza:97.1% - >99.99%Colore e forma:SolidPeso molecolare:280.66Ro 61-8048
CAS:Ro 61-8048 is a potent and selective inhibitor of kynurenine hydroxylase with an IC50 value of 37 nM.Formula:C17H15N3O6S2Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:421.45Ref: TM-T1896
2mg37,00€5mg54,00€10mg73,00€25mg114,00€50mg178,00€100mg284,00€200mg512,00€500mg822,00€1mL*10mM (DMSO)60,00€Telotristat
CAS:Telotristat, active metabolite of LX1606, is an oral tryptophan hydroxylase inhibitor with potential antiserotonergic effects.Formula:C25H22ClF3N6O3Purezza:99.70%Colore e forma:SolidPeso molecolare:546.93Ref: TM-T21506
5mg46,00€10mg62,00€25mg119,00€50mg187,00€100mg304,00€200mg424,00€1mL*10mM (DMSO)52,00€p-Fluoro-L-phenylalanine
CAS:p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.Formula:C9H10FNO2Purezza:99.63%Colore e forma:White To Off-White PowderPeso molecolare:183.18Fenclonine hydrochloride
CAS:Fenclonine hydrochloride is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.Formula:C9H11Cl2NO2Colore e forma:SolidPeso molecolare:236.095Telotristat Etiprate
CAS:Telotristat Etiprate (LX 1606 Hippurate) is an orally bioavailable, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.Formula:C27H26ClF3N6O3·C9H9NO3Purezza:99.21% - 99.83%Colore e forma:White SolidPeso molecolare:754.15Ref: TM-T6044
2mg46,00€5mg66,00€10mg92,00€25mg150,00€50mg183,00€100mg325,00€500mg780,00€1mL*10mM (DMSO)85,00€Tetrahydropapaverine hydrochloride
CAS:Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) , an analogue of salsolinol and tetrahydropapaveroline, has neurotoxicity on dopamine neurons.Formula:C20H26ClNO4Purezza:99.08%Colore e forma:White Crystal PowderPeso molecolare:379.878Mildronate
CAS:Mildronate (Meldonium) is an inhibitor of biosynthesis of L-carnitine by gamma-butyrobetaine (GBB) hydroxylase and as a competitive inhibitor of renal carnitineFormula:C6H14N2O2Purezza:99.94%Colore e forma:White Crystalline PowderPeso molecolare:146.19TETRAHYDROPIPERINE
CAS:Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects.Formula:C17H23NO3Purezza:98.04% - 99.61%Colore e forma:Off-White Low Melting Solid With Characteristic OdourPeso molecolare:289.37Nepicastat
CAS:Nepicastat (SYN117) is a potent, BBB-permeable, selective DBH inhibitor with IC50s of 8.5/9 nM in bovine/human.Formula:C14H15F2N3SColore e forma:SolidPeso molecolare:295.35
