
Canale del potassio
I canali del potassio sono un gruppo diversificato di proteine di membrana che facilitano il flusso di ioni potassio (K+) attraverso la membrana cellulare. Questi canali svolgono un ruolo cruciale nel mantenimento del potenziale di membrana a riposo, nella regolazione del volume cellulare e nel controllo dell'eccitabilità dei neuroni e delle cellule muscolari. I canali del potassio sono coinvolti in vari processi fisiologici, tra cui la regolazione del ritmo cardiaco, la secrezione di insulina e il rilascio di neurotrasmettitori. La disfunzione dei canali del potassio è legata a condizioni come aritmie, epilessia e ipertensione. Presso CymitQuimica, offriamo una vasta gamma di modulatori dei canali del potassio per supportare la tua ricerca in elettrofisiologia, salute cardiovascolare e neurobiologia.
Trovati 283 prodotti di "Canale del potassio"
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NS 11021
CAS:NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channelsFormula:C16H9BrF6N6SPurezza:97.26%Colore e forma:SolidPeso molecolare:511.24Ref: TM-T4294
1mg42,00€5mg88,00€10mg128,00€25mg263,00€50mg447,00€100mg760,00€200mg1.018,00€1mL*10mM (DMSO)89,00€Tetraethylammonium bromide
CAS:Tetraethylammonium bromide (TEA bromide) can selectively block potassium channels.
Formula:C8H20BrNPurezza:98%Colore e forma:White SolidPeso molecolare:210.16VU0810464
CAS:VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK, Kir3) activator.Formula:C18H21ClFN3OPurezza:99.62%Colore e forma:SolidPeso molecolare:349.83Ref: TM-T7899
1mg47,00€5mg95,00€10mg150,00€25mg245,00€50mg325,00€100mg434,00€200mg590,00€1mL*10mM (DMSO)104,00€Atpenin A5
CAS:Atpenin A5 is a potent and highly specific complex II inhibitor (IC50 ~10 nM).Formula:C15H21Cl2NO5Purezza:97.33% - 99.91%Colore e forma:SolidPeso molecolare:366.24ML133 hydrochloride
CAS:ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.Formula:C19H19NO·HClPurezza:99.48%Colore e forma:SolidPeso molecolare:313.82Ref: TM-T6592
5mg50,00€10mg66,00€25mg106,00€50mg170,00€100mg274,00€200mg354,00€500mg597,00€1mL*10mM (DMSO)52,00€20(S)-Ginsenoside Rg3
CAS:20(S)-Ginsenoside Rg3 (Rg3) possess an ability to inhibit the lung metastasis of tumor cells via inhibition of the adhesion and invasion of tumor cells.Formula:C42H72O13Purezza:98.11% - 99.93%Colore e forma:SolidPeso molecolare:785.01XE 991 dihydrochloride
CAS:XE 991 dihydrochloride is a Kv7 (KCNQ) channel blocker.Formula:C26H22Cl2N2OPurezza:98.68%Colore e forma:SolidPeso molecolare:449.37SKF-96365 hydrochloride
CAS:SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal YFormula:C22H27ClN2O3Purezza:99.47% - 99.92%Colore e forma:SolidPeso molecolare:402.91Ref: TM-T2170
5mg57,00€10mg86,00€25mg138,00€50mg243,00€100mg470,00€200mg717,00€500mg1.111,00€1mL*10mM (DMSO)63,00€Nigericin sodium salt
CAS:Nigericin sodium salt, an antibiotic and NLRP3 activator from S. hygroscopicus, inhibits Golgi and gram-positive bacteria, blocking viral activation.Formula:C40H67NaO11Purezza:98.2% - 99.52%Colore e forma:SolidPeso molecolare:746.94Senicapoc
CAS:Senicapoc (ICA-17043) blocks Gardos channel, reduces RBC dehydration, IC50: 11 nM for rubidium flux, 30 nM for dehydration. Used in Sickle Cell therapy.Formula:C20H15F2NOPurezza:95.7% - 99.47%Colore e forma:SolidPeso molecolare:323.34Rimtuzalcap
CAS:Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and ET.Formula:C18H24F2N6OPurezza:99.64%Colore e forma:SolidPeso molecolare:378.42Ref: TM-T9522
1mg35,00€5mg78,00€10mg111,00€25mg215,00€50mg320,00€100mg452,00€200mg632,00€1mL*10mM (DMSO)34,00€BMS-191011
CAS:BMS-191011 (BMS-A) is an activator of large-conductance calcium-activated potassium (BKCa) channels ,effective in stroke modelsFormula:C16H10ClF3N2O3Purezza:97.43%Colore e forma:SolidPeso molecolare:370.71VU0071063
CAS:VU0071063 is a Kir6.2/SUR1 activator.Formula:C18H22N4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:326.39Guanosine 5'-diphosphate disodium salt
CAS:5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.
Formula:C10H13N5Na2O11P2Purezza:99.40%Colore e forma:White PowderPeso molecolare:487.16ML365
CAS:ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).Formula:C22H20N2O3Purezza:98.78%Colore e forma:SolidPeso molecolare:360.41PAP-1
CAS:PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).Formula:C21H18O5Purezza:99.35% - 99.75%Colore e forma:White SolidPeso molecolare:350.36Ref: TM-TQ0179
2mg63,00€5mg88,00€10mg136,00€25mg291,00€50mg520,00€100mg550,00€200mg785,00€1mL*10mM (DMSO)90,00€Loureirin B
CAS:Loureirin B suppresses fibrosis by modulating MMPs/TIMPs, hindering fibroblast growth, and targeting TGF-β1/Smad2/3 pathway.Formula:C18H20O5Purezza:99.33% - 99.86%Colore e forma:SolidPeso molecolare:316.35Paederosidic acid methyl ester
CAS:Paederosidic acid methyl ester has antinociception, is possibly related to the pathway of NO-cGMP-ATP sensitive K(+) channels.
Formula:C19H26O12SPurezza:99.67% - 99.91%Colore e forma:SolidPeso molecolare:478.47A2764 dihydrochloride
CAS:A2764 dihydrochloride is a highly selective inhibitor of TRESK.Formula:C15H21Cl3N2OPurezza:99.05%Colore e forma:SolidPeso molecolare:351.7CLP290
CAS:CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatricFormula:C19H21FN4O3SPurezza:99.93% - >99.99%Colore e forma:SolidPeso molecolare:404.46Ref: TM-T5444
1mg34,00€5mg73,00€10mg116,00€25mg190,00€50mg286,00€100mg430,00€200mg628,00€1mL*10mM (DMSO)62,00€
