Canale del calcio
I canali del calcio sono proteine di membrana che regolano il flusso di ioni calcio dentro e fuori dalle cellule, essenziale per varie funzioni cellulari, tra cui la contrazione muscolare, il rilascio di neurotrasmettitori e l'espressione genica. La disfunzione dell'attività dei canali del calcio è associata a condizioni come ipertensione, aritmie cardiache e disturbi neurologici. Presso CymitQuimica, offriamo un'ampia selezione di modulatori dei canali del calcio per supportare la tua ricerca in salute cardiovascolare, neurobiologia e trasduzione del segnale.
Trovati 493 prodotti di "Canale del calcio"
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Yangambin
CAS:<p>Yangambin: selective PAF antagonist, hypotensive, inhibits Ca2+ influx, induces peripheral vasodilation, affects CNS.</p>Formula:C24H30O8Purezza:98.02%Colore e forma:SolidPeso molecolare:446.49Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formula:C26H44NNaO5SPurezza:99.79% - 99.93%Colore e forma:SolidPeso molecolare:505.692,5-Di-tert-butylhydroquinone
CAS:<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formula:C14H22O2Purezza:97.11%Colore e forma:PelletslargecrystalsPeso molecolare:222.32CDN1163
CAS:<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Formula:C20H20N2O2Purezza:99.83% - ≥95%Colore e forma:SolidPeso molecolare:320.39MDK-4025
CAS:<p>MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.</p>Formula:C19H15ClOPurezza:98.65%Colore e forma:SolidPeso molecolare:294.77Bevantolol hydrochloride
CAS:<p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>Formula:C20H28ClNO4Purezza:99.49%Colore e forma:SolidPeso molecolare:381.9L-Ascorbic acid sodium salt
CAS:<p>L-Ascorbic acid sodium salt (Vitamin C sodium salt) is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.</p>Formula:C6H7NaO6Purezza:98.73% - 99.75%Colore e forma:Less Solid PowderPeso molecolare:198.11JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formula:C9H10N2O2S2Purezza:97.37%Colore e forma:SolidPeso molecolare:242.32Tetrandrine
CAS:<p>Tetrandrine (Sinomenine A) is a naturally occurring biphenylisoquinoline alkaloid, a calcium channel inhibitor. Cost-effective and quality-assured.</p>Formula:C38H42N2O6Purezza:99.61% - 99.94%Colore e forma:White SolidPeso molecolare:622.75Bay K 8644
CAS:<p>Bay K 8644 (SQ 28,873) is a potent, selective activator of L-type Ca2+ channel with IC50 of 17.3 nM.</p>Formula:C16H15F3N2O4Purezza:99.41%Colore e forma:Yellow PowderPeso molecolare:356.3SEA0400
CAS:<p>SEA0400 is a selective inhibitor of the Na+/Ca2+ exchanger.</p>Formula:C21H19F2NO3Purezza:98.88% - 99.55%Colore e forma:SolidPeso molecolare:371.38SN 6
CAS:<p>SN 6 (SN6) is a selective Na+/Ca2+ exchanger (NCX) inhibitor (IC50s of NCX1: 2.9 μM , NCX2: 16 μM ,NCX3: 8.6 μM)</p>Formula:C20H22N2O5SPurezza:97.28%Colore e forma:SolidPeso molecolare:402.46Pyridaben
CAS:<p>Pyridaben is a METI acaricide that inhibits mitochondrial electron transport at complex I (METI; Ki = 0.36 nmol/mg protein in rat brain mitochondria).</p>Formula:C19H25ClN2OSPurezza:97.11% - 99.75%Colore e forma:SolidPeso molecolare:364.93Bupivacaine
CAS:<p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>Formula:C18H28N2OPurezza:99.83%Colore e forma:SolidPeso molecolare:288.43Diltiazem
CAS:<p>Diltiazem (CRD 401 free base) is an orally available L-type Ca2+ channel blocker with antihypertensive, antiarrhythmic, and cardioprotective properties that prevent post-reperfusion myocardial injury, angina pectoris, and cardiovascular-related diseases.</p>Formula:C22H26N2O4SPurezza:99.51% - 99.83%Colore e forma:White Crystalline Powder SolidPeso molecolare:414.52Amlodipine maleate
CAS:<p>Amlodipine maleate (Amvaz) is an oral dihydropyridine calcium blocker for hypertension and cancer studies.</p>Formula:C24H29ClN2O9Purezza:99.4%Colore e forma:White To Pale Yellow Crystalline PowderPeso molecolare:524.95Equilin
CAS:<p>Equilin (7-Dehydroestrone) is a neurotrophic estrogenic steroid with vasodilatory activity used in the study of hypertension.</p>Formula:C18H20O2Purezza:98.57% - 99.72%Peso molecolare:268.35Apinocaltamide
CAS:<p>Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.</p>Formula:C22H18F3N5OPurezza:99.80%Colore e forma:SolidPeso molecolare:425.41N6-(2-Hydroxyethyl)adenosine
CAS:<p>N6-(2-Hydroxyethyl)adenosine is a sedative, Ca2+ antagonist, and anti-inflammatory, affecting brain and heart blood flow.</p>Formula:C12H17N5O5Purezza:99.4%Colore e forma:SolidPeso molecolare:311.29N-Methyl-L-leucin
CAS:<p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>Formula:C7H15NO2Purezza:99.87%Colore e forma:SolidPeso molecolare:145.2Bupivacaine-d9
CAS:<p>Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.</p>Formula:C18H19D9N2OColore e forma:SolidPeso molecolare:297.48Gabapentin enacarbil
CAS:<p>Gabapentin enacarbil (XP-13512) is a prodrug for the anticonvulsant and analgesic gabapentin, offering sustained dose-proportional exposure and predictable bioavailability.</p>Formula:C16H27NO6Purezza:99.31%Colore e forma:SolidPeso molecolare:329.391-tert-Butyl 3-Ethyl 5-methyl 2-((2-((tert-Butoxycarbonyl)amino)ethoxy)methyl)-4-(2-chlorophenyl)-6-methylpyridine-1,3,5(4H)-tricarboxylate
CAS:Prodotto controllato<p>Applications 1-tert-Butyl 3-Ethyl 5-methyl 2-((2-((tert-Butoxycarbonyl)amino)ethoxy)methyl)-4-(2-chlorophenyl)-6-methylpyridine-1,3,5(4H)-tricarboxylate is an intermediate in the synthesis of 3-O-Desethyl-5-O-desmethyl Amlodipine (D291305). 3-O-Desethyl-5-O-desmethyl Amlodipine is an impurity of Amlodipine (A633495), which is a dihydropyridine calcium channel blocker.<br>References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)<br></p>Formula:C30H41ClN2O9Colore e forma:NeatPeso molecolare:609.1074-(2-Chlorophenyl)-2-methyl-5-oxo-4,4a,5,7,8,10-hexahydro-1H-pyrido[2',3':2,3]azeto[2,1-c][1,4]oxazine-3-carboxylic Acid
Prodotto controllato<p>Applications 4-(2-Chlorophenyl)-2-methyl-5-oxo-4,4a,5,7,8,10-hexahydro-1H-pyrido[2',3':2,3]azeto[2,1-c][1,4]oxazine-3-carboxylic Acid is an intermediate in the synthesis of 3-O-Desethyl-5-O-desmethyl Amlodipine (D291305). 3-O-Desethyl-5-O-desmethyl Amlodipine is an impurity of Amlodipine (A633495), which is a dihydropyridine calcium channel blocker.<br>References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)<br></p>Formula:C17H17ClN2O4Colore e forma:NeatPeso molecolare:348.781Cinepazide
CAS:<p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>Formula:C22H31N3O5Colore e forma:White PowderPeso molecolare:417.5Amlodipine besilate impurity G
CAS:<p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>Formula:C17H18ClNO4Purezza:98%Colore e forma:SolidPeso molecolare:335.78Amlodipine hydrochloride
CAS:<p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>Formula:C20H26Cl2N2O5Colore e forma:SolidPeso molecolare:445.34Topiramate D12
CAS:<p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>Formula:C12H21NO8SPurezza:98%Colore e forma:SolidPeso molecolare:351.44Nifedipine-d6
CAS:<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Formula:C17H18N2O6Purezza:98%Colore e forma:SolidPeso molecolare:352.37Cinnarizine D8
CAS:<p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>Formula:C26H28N2Purezza:98%Colore e forma:SolidPeso molecolare:376.573Maresin 1
CAS:<p>Maresin 1 is biosynthesized by macrophages (MΦ) and possesses significant anti-inflammatory activity that attenuates LPS-induced lung injury in mice.</p>Formula:C22H32O4Colore e forma:SolidPeso molecolare:360.49ORM-10103
CAS:<p>ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nM</p>Formula:C20H16N2O4Purezza:99.9%Colore e forma:SolidPeso molecolare:348.35Ionomycin calcium
CAS:<p>Ionomycin calcium (SQ23377 calcium) is an effective and selective calcium ionophore, exhibiting high specificity for calcium ions. Cost-effective and quality-assured.</p>Formula:C41H70CaO9Purezza:98% - 98.11%Colore e forma:SolidPeso molecolare:747.07R-(-)-Niguldipine hydrochloride
CAS:<p>R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.</p>Formula:C36H40ClN3O6Colore e forma:SolidPeso molecolare:646.17(R)-Lercanidipine Hydrochloride
CAS:Prodotto controllatoFormula:C36H41N3O6·ClHColore e forma:NeatPeso molecolare:648.19(S)-Lercanidipine Hydrochloride
CAS:Prodotto controllatoFormula:C36H41N3O6·ClHColore e forma:NeatPeso molecolare:648.19Dihydrocinnamyl Cilnidipine
Prodotto controllato<p>Applications Dihydrocinnamyl Cilnidipine is a metabolite of Cilnidipine (C441375); a dihydropyridine calcium channel blocker.<br>References Ikeda, K., et al.: Oyo Yakuri, 44, 433 (1992); Hosono, M., et al.: J. Pharmacobio-Dyn., 15, 547, (1992); Ishii, M.: Japan Pharmacol. Ther., 21, 59 (1993)<br></p>Formula:C27H30N2O7Colore e forma:NeatPeso molecolare:494.543-Desethyl-3-(2-phthalimidoethyl) Phthaloyl Amlodipine
Prodotto controllato<p>Stability Light and Temperature Sensitive<br>Applications 3-Desethyl-3-(2-phthalimidoethyl) Phthaloyl Amlodipine is a derivative of Amlodipine (A633495); a dihydropyridine calcium channel blocker where activity mainly resides in the (-)-isomer.<br>References Arrowsmith, J.E., et al.: J. Med. Chem., 29, 1696 (1986); Burges, R.A., et al.: J. Cardiovasc. Pharmacol., 9, 110 (1987); Haria, M., et al.: Drugs, 50, 560 (1995)<br></p>Formula:C36H30ClN3O9Colore e forma:NeatPeso molecolare:684.091Falipamil
CAS:Prodotto controllato<p>Applications Falipamil is a specific bradycardic agent and a calcium channel blocker.<br>References Boucher, M., et al.: Eur. J. Pharmacol., 306, 93 (1996), Mubagwa, K., et al.: Arch. Int. Pharmacodyn. Ther., 286, 71 (1987), Chaudhry, A., et al.: Development Cardiovascular Medicine, 46, 196 (1985), Ogiwara, Y., et al.: Jpn Heart J., 29, (1988)<br></p>Formula:C24H32N2O5Colore e forma:NeatPeso molecolare:428.52Halofuginone
CAS:<p>Halofuginone (RU-19110) inhibits prolyl-tRNA synthetase (Ki=18.3 nM), down-regulates Smad3, and blocks TGF-β at 10 ng/ml.</p>Formula:C16H17BrClN3O3Purezza:99.53%Colore e forma:Off-White SolidPeso molecolare:414.68Verapamil
CAS:<p>Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.</p>Formula:C27H38N2O4Purezza:99.61% - 99.93%Colore e forma:OilPeso molecolare:454.6SCH00013
CAS:<p>SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.</p>Formula:C18H20N4O2Purezza:98%Colore e forma:SolidPeso molecolare:324.38GZ4
CAS:<p>GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.</p>Formula:C11H17NO2Purezza:98%Colore e forma:SolidPeso molecolare:195.26BN 50341
CAS:<p>BN 50341 is an inhibitor of antithrombotic platelet activating factor.</p>Formula:C32H41ClN2O4Purezza:98%Colore e forma:SolidPeso molecolare:553.13EO-122
CAS:<p>EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.</p>Formula:C16H23ClN2OColore e forma:SolidPeso molecolare:294.82Gallopamil HCl, (-)-
CAS:<p>Gallopamil HCl, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>Formula:C28H41ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:521.09Hns 32
CAS:<p>Hns 32 possesses antiarrhythmic properties in dog and guinea pig hearts. It also has vasodilator action.</p>Formula:C24H29N3Purezza:98%Colore e forma:SolidPeso molecolare:359.51A 80b
CAS:<p>A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.</p>Formula:C16H17N7Purezza:98%Colore e forma:SolidPeso molecolare:307.35Methsuximide
CAS:<p>Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].</p>Formula:C12H13NO2Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:203.24
![4-(2-Chlorophenyl)-2-methyl-5-oxo-4,4a,5,7,8,10-hexahydro-1H-pyrido[2',3':2,3]azeto[2,1-c][1,4]oxa…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FC609788.webp&w=3840&q=75)
