Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColore e forma:SolidPeso molecolare:179.2Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Formula:C8H17NOPurezza:98%Colore e forma:SolidPeso molecolare:143.23NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurezza:99.44% - 99.86%Colore e forma:SolidPeso molecolare:353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purezza:99.72% - 99.99%Colore e forma:Solid PowderPeso molecolare:556.29ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formula:C21H21FN6Purezza:99.43%Colore e forma:SolidPeso molecolare:376.43Ref: TM-TQ0040
1mg60,00€5mg126,00€10mg170,00€25mg376,00€50mg562,00€100mg802,00€1mL*10mM (DMSO)140,00€Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formula:C15H17N3O3Colore e forma:SolidPeso molecolare:287.31Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurezza:99.17%Colore e forma:White Crystalline SolidPeso molecolare:249.71Ref: TM-T4440
1mg56,00€5mg119,00€10mg187,00€25mg359,00€50mg582,00€100mg908,00€200mg1.225,00€1mL*10mM (DMSO)114,00€Imepitoin
CAS:<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formula:C13H14ClN3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:279.72(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Formula:C6H9NO2Colore e forma:SolidPeso molecolare:127.1436-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purezza:99.69%Colore e forma:SolidPeso molecolare:236.27Thiocolchicoside
CAS:<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Formula:C27H33NO10SPurezza:99.11% - 99.39%Colore e forma:SolidPeso molecolare:563.62(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purezza:99.58% - 99.87%Colore e forma:SolidPeso molecolare:217.26DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurezza:99.74%Colore e forma:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecolare:156.272'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28Ref: TM-TN1217
1mg115,00€5mg274,00€10mg455,00€25mg730,00€50mgPrezzo su richiesta1mL*10mM (DMSO)378,00€(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formula:C10H12ClNO2Purezza:97.20% - 98.94%Colore e forma:SolidPeso molecolare:213.666-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurezza:99.03%Colore e forma:SolidPeso molecolare:201.22Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurezza:99.09% - 99.77%Colore e forma:White To Off-White SolidPeso molecolare:412.01Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purezza:99.69% - ≥95%Colore e forma:SolidPeso molecolare:177.63Ref: TM-T5799
2mg35,00€5mg50,00€10mg71,00€25mg105,00€50mg158,00€100mg225,00€200mg334,00€1mL*10mM (DMSO)51,00€Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:250.122SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Colore e forma:SolidPeso molecolare:335.44Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Formula:C20H24O9Purezza:98.76% - 99.81%Colore e forma:White PowderPeso molecolare:408.4Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurezza:99.81%Colore e forma:SolidPeso molecolare:301.3U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purezza:99.65% - 99.76%Colore e forma:SolidPeso molecolare:299.37Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formula:C53H90O22Purezza:98.83% - 99.56%Colore e forma:White PowderPeso molecolare:1079.27Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formula:C20H15FN4O2SPurezza:99.12% - 99.19%Colore e forma:SolidPeso molecolare:394.42Pipequaline hydrochloride
CAS:Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formula:C22H25ClN2Purezza:99.46%Colore e forma:SolidPeso molecolare:352.9Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purezza:98.51% - 99.24%Colore e forma:SolidPeso molecolare:368.23Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purezza:99.8%Colore e forma:SolidPeso molecolare:198.22Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formula:C6H9ClN2O2Purezza:99.39%Peso molecolare:176.601Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purezza:99.93%Colore e forma:White Crystalline PowderPeso molecolare:215.68Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Formula:C24H46N6O14Purezza:99.8%Colore e forma:Crystals IndicationPeso molecolare:642.65Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:1207.35SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormula:C22H26ClNO2Purezza:98.02%Colore e forma:SolidPeso molecolare:371.9Ref: TM-T12930
1mg35,00€5mg69,00€10mg95,00€25mg170,00€50mg279,00€100mg432,00€200mg622,00€1mL*10mM (DMSO)74,00€(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purezza:99.47%Colore e forma:SolidPeso molecolare:340.37α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurezza:97.02% - 98.41%Colore e forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecolare:152.23Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55Fipronil
CAS:Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurezza:97.21%Colore e forma:Solid PowderPeso molecolare:437.15Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formula:C41H72O2Purezza:99.65%Colore e forma:SolidPeso molecolare:597.01Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formula:C17H24O4Purezza:98.22%Colore e forma:SolidPeso molecolare:292.37α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purezza:99.64% - 99.64%Colore e forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecolare:208.25Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purezza:99.22% - 99.66%Colore e forma:SolidPeso molecolare:282.38Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46Ref: TM-T3417
2mg35,00€5mg52,00€10mg85,00€25mg133,00€50mg227,00€100mg369,00€200mg540,00€1mL*10mM (DMSO)63,00€AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purezza:98.99%Colore e forma:SolidPeso molecolare:366.41Ref: TM-T7136
1mg227,00€5mg464,00€10mg677,00€25mg1.074,00€50mg1.501,00€100mg2.043,00€1mL*10mM (DMSO)510,00€CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formula:C13H9F3N4Purezza:99.92%Colore e forma:SolidPeso molecolare:278.23p-Hydroxybenzaldehyde
CAS:1.Formula:C7H6O2Purezza:99.05% - 99.86%Colore e forma:SolidPeso molecolare:122.12Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:357.49Cyclothiazide
CAS:Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Formula:C14H16ClN3O4S2Purezza:98.23% - 99.49%Colore e forma:Crystals From Dilute Alcohol SolidPeso molecolare:389.882'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purezza:99.28% - 99.63%Colore e forma:SolidPeso molecolare:266.29Ref: TM-T8887
1mg51,00€5mg107,00€10mg160,00€25mg255,00€50mg359,00€100mg485,00€200mg662,00€1mL*10mM (DMSO)101,00€Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Colore e forma:SolidPeso molecolare:430.02
