Ricettore GABA
I recettori GABA sono i principali recettori dei neurotrasmettitori inibitori nel sistema nervoso centrale, svolgendo un ruolo cruciale nella regolazione dell'eccitabilità neuronale e nel mantenimento dell'equilibrio tra eccitazione e inibizione. La disfunzione dei recettori GABA è implicata in vari disturbi neurologici e psichiatrici, tra cui epilessia, ansia e depressione. Presso CymitQuimica, offriamo una gamma completa di modulatori dei recettori GABA per supportare la tua ricerca in neurobiologia, salute mentale e sviluppo terapeutico.
Trovati 365 prodotti di "Ricettore GABA"
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Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purezza:98.21% - 99.22%Colore e forma:Odourless Whitish SolidPeso molecolare:538.46Ref: TM-T3417
2mg35,00€5mg52,00€10mg85,00€25mg133,00€50mg227,00€100mg369,00€200mg540,00€1mL*10mM (DMSO)63,00€Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purezza:99.25% - 99.67%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:375.55Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formula:C6H9ClN2O2Purezza:99.39%Peso molecolare:176.601SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Colore e forma:SolidPeso molecolare:335.44Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purezza:98.51% - 99.24%Colore e forma:SolidPeso molecolare:368.236-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurezza:99.03%Colore e forma:SolidPeso molecolare:201.222'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purezza:98.75%Colore e forma:SolidPeso molecolare:270.28Ref: TM-TN1217
1mg115,00€5mg274,00€10mg455,00€25mg730,00€50mgPrezzo su richiesta1mL*10mM (DMSO)378,00€Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purezza:99.55%Colore e forma:SolidPeso molecolare:250.1226-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purezza:99.69%Colore e forma:SolidPeso molecolare:236.27DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurezza:99.74%Colore e forma:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Peso molecolare:156.27Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurezza:99.17%Colore e forma:White Crystalline SolidPeso molecolare:249.71Ref: TM-T4440
1mg56,00€5mg119,00€10mg187,00€25mg359,00€50mg582,00€100mg908,00€200mg1.225,00€1mL*10mM (DMSO)114,00€Imepitoin
CAS:<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formula:C13H14ClN3O2Purezza:99.82%Colore e forma:SolidPeso molecolare:279.72U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purezza:99.65% - 99.76%Colore e forma:SolidPeso molecolare:299.37Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purezza:99.72% - 99.99%Colore e forma:Solid PowderPeso molecolare:556.29Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formula:C53H90O22Purezza:98.83% - 99.56%Colore e forma:White PowderPeso molecolare:1079.27NS11394
CAS:NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formula:C23H19N3OPurezza:99.44% - 99.86%Colore e forma:SolidPeso molecolare:353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formula:C21H21FN6Purezza:99.43%Colore e forma:SolidPeso molecolare:376.43Ref: TM-TQ0040
1mg60,00€5mg126,00€10mg170,00€25mg376,00€50mg562,00€100mg802,00€1mL*10mM (DMSO)140,00€Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:1207.35Suritozole
CAS:<p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>Formula:C10H10FN3SPurezza:99.25%Colore e forma:SolidPeso molecolare:223.27Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFormula:C21H20FN3O5SPurezza:99.21% - 99.42%Colore e forma:SolidPeso molecolare:445.46Ref: TM-T7165
2mg38,00€5mg56,00€10mg79,00€25mg123,00€50mg197,00€100mg376,00€500mg847,00€1mL*10mM (DMSO)52,00€Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurezza:99.39% - ≥95%Colore e forma:SolidPeso molecolare:423.53Bicuculline
CAS:Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Formula:C20H17NO6Purezza:98% - 99.99%Colore e forma:Light Yellow PowderPeso molecolare:367.35Ref: TM-T2850
10mgPrezzo su richiesta25mgPrezzo su richiesta50mg69,00€100mgPrezzo su richiesta1mL*10mM (DMSO)55,00€Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Formula:C10H6Cl3N3Purezza:99.78%Colore e forma:SolidPeso molecolare:274.53Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formula:C16H14FN3OPurezza:99.72%Colore e forma:SolidPeso molecolare:283.3Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C21H31F3O2Purezza:98%Colore e forma:SolidPeso molecolare:372.46Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:364.8(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Formula:C10H12ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:213.66ABP-700
CAS:ABP-700 is a positive allosteric modulator of the GABAA receptor.Formula:C17H18N2O4Purezza:98%Colore e forma:SolidPeso molecolare:314.34CGP 46381
CAS:CGP 46381 is a GABAB receptor antagonist.Formula:C10H22NO2PPurezza:98%Colore e forma:White SolidPeso molecolare:219.26PF-0713
CAS:PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formula:C14H22OPurezza:98%Colore e forma:SolidPeso molecolare:206.32DAA-1097
CAS:DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Formula:C24H24ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:group I metabotropic glutamate receptor antagonist and group II mGlu agonistFormula:C9H9NO5Purezza:98%Colore e forma:SolidPeso molecolare:211.17CP-409092 hydrochloride
CAS:CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.Formula:C17H20ClN3O2Colore e forma:SolidPeso molecolare:333.81Arbaclofen placarbil
CAS:Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purezza:98%Colore e forma:SolidPeso molecolare:358.87Ethyl dirazepate
CAS:Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Formula:C18H14Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:377.22Ro 41-3290
CAS:Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Formula:C24H21ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:420.89GS 39783
CAS:GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormula:C15H23N5O2SPurezza:99.92%Colore e forma:SolidPeso molecolare:337.44SCH 50911
CAS:SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formula:C8H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:173.21U-7524
CAS:U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.Formula:C2H5NO3Colore e forma:SolidPeso molecolare:91.07Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purezza:98.61%Colore e forma:SolidPeso molecolare:337.33Ref: TM-T23445
1mg64,00€2mg96,00€5mg115,00€10mg150,00€25mg330,00€50mg472,00€100mg655,00€500mg1.293,00€Y 23684
CAS:Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.Formula:C18H13ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:356.83Ciclotizolam
CAS:Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formula:C20H18BrClN4SColore e forma:SolidPeso molecolare:461.81Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Formula:C13H25NO2Colore e forma:SolidPeso molecolare:227.34Ref: TM-T72977
1mg38,00€5mg75,00€10mg105,00€25mg172,00€50mg242,00€100mg337,00€200mg498,00€1mL*10mM (DMSO)84,00€DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Formula:C18H10Br2ClN3OSColore e forma:SolidPeso molecolare:511.62SH-053-S-CH3-2'F
CAS:SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Formula:C23H18FN3O2Colore e forma:SolidPeso molecolare:387.41Alfadolone
CAS:Alfadolone is an anesthetic derivative of pregnanedione.Formula:C21H32O4Colore e forma:SolidPeso molecolare:348.483-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Formula:C20H30N2O10S2Purezza:98%Colore e forma:SolidPeso molecolare:522.59
